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Elastase 1 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
TelaprevirIC5030.0 [1]
BoceprevirIC5010000.0 [1]
Z-Pro-prolinalIC5051.6 [1]
PolyozellinIC502720.0 [1]
(1R,21S,24S)-21-Tert-butyl-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-16,16-dimethyl-3,19,22-trioxo-2,18-dioxa-4,20,23-triazatetracyclo[21.2.1.14,7.06,11]heptacosa-6(11),7,9-triene-24-carboxamideIC5010000.0 [1]
Kynapcin-12IC501250.0 [1]
Kynapcin-24Ki290.0 [1]
Methyl (3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-[(4-methoxy-4-oxobutanoyl)amino]propanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-4-methyl-2-oxopentanoateKi200.0 [1]
Methyl (3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-1-acetylpyrrolidine-2-carbonyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-2-oxobutanoateKi850.0 [1]
(2S)-1-[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S,3R)-2-[[(2S)-2-[[2-[[2-[[(2S)-2-[[(2S)-2-[[(3S,9S,12S,15S,18S,21S,24S,27S)-12-(3-Carbamimidamidopropyl)-18-(carboxymethyl)-3,15-bis[(4-hydroxyphenyl)methyl]-21,24-bis(1H-indol-3-ylmethyl)-2,5,8,11,14,17,20,23,26-nonaoxo-1,4,7,10,13,16,19,22,25-nonazabicyclo[25.3.0]triacontane-9-carbonyl]amino]-4-methylpentanoyl]amino]-3-phenylpropanoyl]amino]acetyl]amino]acetyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]-3-hydroxybutanoyl]amino]-3-phenylpropanoyl]amino]-3-methylpentanoyl]amino]-3-hydroxypropanoyl]pyrrolidine-2-carboxylic acidIC501100.0 [1]
Methyl 4-oxo-4-[[(2R)-1-oxo-3-phenyl-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]butanoateKi660.0 [1]
Tert-butyl N-[(2S)-1-oxo-3-phenyl-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]carbamateKi160.0 [1]
Benzyl N-[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]propan-2-yl]carbamateKi1.0 [1]
Methyl 4-oxo-4-[[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]propan-2-yl]amino]butanoateKi14.0 [1]
Methyl (3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-2-[(4-methoxy-4-oxobutanoyl)amino]propanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-2-oxo-4-phenylbutanoateKi1000000.0 [1]
Methyl 4-oxo-4-[[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[(2S)-2-[[(2S)-4,4,4-trifluoro-3-oxo-1-phenylbutan-2-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]propan-2-yl]amino]butanoateKi1500000.0 [1]
Acetyl-Pro-Ala-Pro-Ala-trifluoro methaneKi800000.0 [1]
Acetyl-Ala-Ala-Pro-Ala-trifluromethaneKi250.0 [1]
Ethyl (3S)-2-oxo-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-(phenylmethoxycarbonylamino)propanoyl]amino]propanoyl]amino]propanoyl]amino]butanoateKi300.0 [1]
Methyl 4-[[(5S)-5-(1-adamantylsulfonylamino)-6-oxo-6-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]hexyl]amino]-4-oxobutanoateKi0.58 [1]
Ethyl (4S)-2,2-difluoro-4-[[(2S)-1-[(2S)-2-[[(2S)-2-[(4-methoxy-4-oxobutanoyl)amino]propanoyl]amino]propanoyl]pyrrolidine-2-carbonyl]amino]-5-methyl-3-oxohexanoateKi4300.0 [1]
Tert-butyl N-[(2S)-1-oxo-1-[[(2S)-1-oxo-1-[(2S)-2-[[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]carbamoyl]pyrrolidin-1-yl]propan-2-yl]amino]propan-2-yl]carbamateKi44.0 [1]
2-[4-[Amino-[2-[(4R)-4-cyano-1,3-thiazolidin-3-yl]-2-oxoethyl]amino]piperidin-1-yl]-N-(5-chloropyridin-2-yl)acetamide;trihydrochlorideIC5010000.0 [1]
(2S)-1-[(2S)-2-[[(2S)-2-[[5-(Dimethylamino)naphthalen-1-yl]sulfonylamino]propanoyl]amino]propanoyl]-N-[(3S)-1,1,1-trifluoro-4-methyl-2-oxopentan-3-yl]pyrrolidine-2-carboxamideKi1000000.0 [1]
Items per page: 1 - 10 of 24
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References

This online tool may be cited as follows

MLA

"Quest Database™ Elastase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Dec. 2024, https://www.aatbio.com/data-sets/elastase-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 22). Quest Database™ Elastase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/elastase-1-inhibitors-ic50-ki.
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