 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-2,3-difluorobenzamide | IC50 | 32.59 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-3-fluoropyridine-4-carboxamide | IC50 | 20.37 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-4-methylthiadiazole-5-carboxamide | IC50 | 62.44 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-4-methyl-1,3-thiazole-5-carboxamide | IC50 | 206.7 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-5-methyl-1,2-oxazole-4-carboxamide | IC50 | 256.1 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-2-methylbenzamide | IC50 | 36.35 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-2-phenylacetamide | IC50 | 456.6 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-2-pyridin-2-ylacetamide | IC50 | 968.1 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-3-fluoropyridine-4-carboxamide | IC50 | 243.9 [1] |
 | 3,5-Dichloro-N-[4-(3,5-dicyclopropylpyrazol-1-yl)phenyl]pyridine-4-carboxamide | IC50 | 129.6 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]pyridine-4-carboxamide | IC50 | 141.3 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)-3-fluorophenyl]-2,6-difluorobenzamide | IC50 | 145.1 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)-3-fluorophenyl]pyridine-4-carboxamide | IC50 | 184.6 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-4-methylthiadiazole-5-carboxamide | IC50 | 183.6 [1] |
 | N-[6-(3,5-Dicyclopropylpyrazol-1-yl)pyridin-3-yl]-2,6-difluorobenzamide | IC50 | 436.1 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-4-methyl-1,3-thiazole-5-carboxamide | IC50 | 72.03 [1] |
 | 3,5-Dichloro-N-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]pyridine-4-carboxamide | IC50 | 65.49 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-5-methyl-1,2-oxazole-4-carboxamide | IC50 | 63.17 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-2-methylbenzamide | IC50 | 119.7 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-3,5-dimethyl-1,2-oxazole-4-carboxamide | IC50 | 124.5 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)-3-fluorophenyl]-4-methylpyrimidine-5-carboxamide | IC50 | 223.5 [1] |
 | N-[4-(4-Chloro-3,5-dicyclopropylpyrazol-1-yl)-3-fluorophenyl]-4-methylthiadiazole-5-carboxamide | IC50 | 181.1 [1] |
 | N-[4-(3,5-Dicyclopropylpyrazol-1-yl)-3-fluorophenyl]-4-methylthiadiazole-5-carboxamide | IC50 | 60.31 [1] |
 | 6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-N-(2,6-difluorophenyl)pyridine-3-carboxamide | IC50 | 72.11 [1] |
 | N-[4-[5-(Fluoromethyl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-4-methyl-1,3-thiazole-5-carboxamide | IC50 | 373.4 [1] |
 | N-[2-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyrimidin-5-yl]-2,6-difluorobenzamide | IC50 | 295.4 [1] |
 | N-[4-[5-(Difluoromethyl)-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-4-methyl-1,3-thiazole-5-carboxamide | IC50 | 52.62 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-2-methylbenzamide | IC50 | 147.2 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-5-methyl-1,2-oxazole-4-carboxamide | IC50 | 20.79 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-4-methyl-1,3-thiazole-5-carboxamide | IC50 | 48.17 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-2,6-difluorobenzamide | IC50 | 98.58 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]pyridine-4-carboxamide | IC50 | 254.7 [1] |
 | 1-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-3-(4-methyl-1,3-thiazol-5-yl)urea | IC50 | 269.0 [1] |
 | 4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-N-(4-methyl-1,3-thiazol-5-yl)benzamide | IC50 | 34.11 [1] |
 | 4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-N-(2,6-difluorophenyl)benzamide | IC50 | 123.8 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-4-methylthiadiazole-5-carboxamide | IC50 | 35.72 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]pyridine-3-carboxamide | IC50 | 205.7 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]pyridine-4-carboxamide | IC50 | 232.0 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-3-fluoropyridine-4-carboxamide | IC50 | 159.1 [1] |
 | 3,5-Dichloro-N-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]pyridine-4-carboxamide | IC50 | 159.3 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-4-methylpyrimidine-5-carboxamide | IC50 | 81.25 [1] |
 | 4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-N-(2,6-difluorophenyl)-3-fluorobenzamide | IC50 | 99.71 [1] |
 | N-[6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-3-yl]-4-methylthiadiazole-5-carboxamide | IC50 | 149.6 [1] |
 | N-[6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-3-yl]-2-methylbenzamide | IC50 | 22.96 [1] |
 | N-[6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-3-yl]-2-fluorobenzamide | IC50 | 60.0 [1] |
 | N-[6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-3-yl]-2,3-difluorobenzamide | IC50 | 70.32 [1] |
 | N-[6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-3-yl]-2,6-difluorobenzamide | IC50 | 50.58 [1] |
 | N-[6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-3-yl]pyridine-3-carboxamide | IC50 | 47.21 [1] |
 | N-[6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-3-yl]pyridine-4-carboxamide | IC50 | 62.56 [1] |
 | N-[6-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]pyridin-3-yl]-3-fluoropyridine-4-carboxamide | IC50 | 37.58 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-2-pyridin-3-ylacetamide | IC50 | 48.22 [1] |
 | N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-2-pyridin-2-ylacetamide | IC50 | 604.3 [1] |
 | N-[4-[4-Chloro-5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]-4-methyl-1,3-thiazole-5-carboxamide | IC50 | 194.0 [1] |
 | 4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-N-[(4-methyl-1,3-thiazol-5-yl)methyl]aniline | IC50 | 48.02 [1] |
 | 1-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]-3-(4-methylpyrimidin-5-yl)urea | IC50 | 600.3 [1] |
 | N-[3-Amino-4-(3,5-dicyclopropylpyrazol-1-yl)phenyl]-4-methyl-1,3-thiazole-5-carboxamide | IC50 | 851.4 [1] |