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Dual-specificity tyrosine-phosphorylation regulated kinase 3 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
▲
▼
HarmineIC50210.0 [1], 410.0 [2], 800.0 [3]
Leucettine L41IC50320.0 [1], 700.0 [2]
SeliciclibIC5010000.0 [1]
N3-(4-Fluorophenyl)-1h-pyrazolo[3,4-d]pyrimidine-3,4-diamineIC503200.0 [1]
Leucettamine BIC501400.0 [1]
CID 72163809IC5070.0 [1]
7-Chloro-3-oxo-8-(1,3-thiazol-5-ylmethylamino)-11,16-dioxa-2,4,19,21-tetrazatricyclo[15.3.1.05,10]henicosa-1(20),5,7,9,17(21),18-hexaene-18-carbonitrileKi5804.0 [1]
2-N-(4-Aminocyclohexyl)-8-propan-2-yl-4-N-[(4-pyridin-2-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazine-2,4-diamineIC50380.0 [1]
(4Z)-2-[4-[2-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]ethoxy]anilino]-4-(1,3-benzodioxol-5-ylmethylidene)-1H-imidazol-5-oneIC50180.0 [1]
N-[2-[2-Aminoethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]acetamideIC5040.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
4-[[4-Cyclopentyloxy-5-(2-methyl-1,3-benzoxazol-6-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-N-methylbenzamideIC5099.0 [1]
10-Chloro-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC50100000.0 [1]
10-Bromo-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC50100000.0 [1]
10-Fluoro-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC502300.0 [1]
10-Chloro-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Bromo-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC501400.0 [1]
10-Iodo-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Chloro-3-ethoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Fluoro-2-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Chloro-2-(3-methoxyphenyl)-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5030.0 [1]
10-Bromo-11H-indolo[3,2-c][1,5]naphthyridine-6-carboxylic acidIC5010000.0 [1]
Clk1-IN-1IC5010000.0 [1]
4-[6-[6-(Propan-2-ylamino)indazol-1-yl]pyrazin-2-yl]benzoic acidIC5054.0 [1]
(4Z)-2-Anilino-4-benzylidene-1H-imidazol-5-oneIC5010000.0 [1]
(4Z)-2-[4-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]anilino]-4-(1,3-benzodioxol-5-ylmethylidene)-1H-imidazol-5-oneIC50200.0 [1]
(4Z)-2-[4-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]anilino]-4-benzylidene-1H-imidazol-5-oneIC5010000.0 [1]
(2S)-2-[[3-[3-[(E)-Hydroxyiminomethyl]phenyl]imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC50920.0 [1]
6-Methylsulfanyl-3-[3-(trifluoromethyl)phenyl]imidazo[1,2-b]pyridazineIC503000.0 [1]
(2S)-2-[[3-(2-Amino-5-chlorophenyl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC5017000.0 [1]
6-Methoxy-3-(2-methylsulfanylpyrimidin-4-yl)imidazo[1,2-b]pyridazineIC507900.0 [1]
(2S)-2-[[3-(1H-Indol-2-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC50120.0 [1]
6-Methoxy-3-(2-methylsulfinylpyrimidin-4-yl)imidazo[1,2-b]pyridazineIC5010000.0 [1]
6-Methoxy-3-[4-(trifluoromethyl)phenyl]imidazo[1,2-b]pyridazineIC504900.0 [1]
3-(3-Chlorophenyl)-6-(4-piperidin-1-ylpiperidin-1-yl)imidazo[1,2-b]pyridazineIC501100.0 [1]
(2S)-2-[[3-(2-Methylsulfonylpyrimidin-4-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC5010000.0 [1]
N-[3-[6-[[(2S)-1-Hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]phenyl]acetamideIC50110.0 [1]
(2S)-2-[[3-(2-Methylsulfinylpyrimidin-4-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC5010000.0 [1]
(2S)-2-[[3-(3-Methylsulfonylphenyl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC502100.0 [1]
Ethyl 3-[6-[[(2S)-1-hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]benzoateIC50110.0 [1]
N-[(2S)-1-Hydroxybutan-2-yl]-3-[6-[[(2S)-1-hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]benzamideIC508100.0 [1]
2-[4-[3-(3-Chlorophenyl)imidazo[1,2-b]pyridazin-6-yl]piperazin-1-yl]ethanolIC50430.0 [1]
(2S)-2-[[3-[3-[[(2S)-1-Hydroxybutan-2-yl]iminomethyl]phenyl]imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC501400.0 [1]
(NE)-N-[[3-(6-methoxyimidazo[1,2-b]pyridazin-3-yl)phenyl]methylidene]hydroxylamineIC50140.0 [1]
(2S)-3-Methyl-2-[(3-pyridin-3-ylimidazo[1,2-b]pyridazin-6-yl)amino]butan-1-olIC50320.0 [1]
N-[3-[[3-(3-Chlorophenyl)imidazo[1,2-b]pyridazin-6-yl]amino]phenyl]acetamideIC505300.0 [1]
3-(1H-Indol-5-yl)-6-methylsulfanylimidazo[1,2-b]pyridazineIC501200.0 [1]
(2S)-2-[[3-(3-Methylsulfanylphenyl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC501300.0 [1]
4-Chloro-2-(6-chloroimidazo[1,2-b]pyridazin-3-yl)anilineIC5041000.0 [1]
(2S)-2-[[3-(3-Aminophenyl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC505100.0 [1]
(2S)-2-[[3-(1H-Indol-5-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC501800.0 [1]
(2S)-2-[[3-[3-(Trifluoromethyl)phenyl]imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC50100000.0 [1]
6-Methoxy-3-[(E)-2-[3-(trifluoromethyl)phenyl]ethenyl]imidazo[1,2-b]pyridazineIC5010000.0 [1]
(2S)-2-[[3-(2-Aminopyrimidin-4-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC50320.0 [1]
(2S)-2-[[3-[(E)-2-[3-(Trifluoromethyl)phenyl]ethenyl]imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC5010000.0 [1]
(2S)-2-[[3-(5-Bromo-1H-indol-2-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC50610.0 [1]
3-(6-Fluoroimidazo[1,2-b]pyridazin-3-yl)benzaldehydeIC5010000.0 [1]
(2R)-2-[[3-[3-[[(2R)-1-Hydroxybutan-2-yl]iminomethyl]phenyl]imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC503100.0 [1]
Ethyl N-(3-pyridin-3-ylimidazo[1,2-b]pyridazin-6-yl)carbamateIC5010000.0 [1]
(NE)-N-[[3-(6-chloroimidazo[1,2-b]pyridazin-3-yl)phenyl]methylidene]hydroxylamineIC50510.0 [1]
3-(6-Chloroimidazo[1,2-b]pyridazin-3-yl)-N-[(2R)-1-hydroxybutan-2-yl]benzamideIC5010000.0 [1]
N-[(2R)-1-Hydroxybutan-2-yl]-3-[6-[[(2R)-1-hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]benzamideIC5010000.0 [1]
3-(1H-Indol-5-yl)-6-methoxyimidazo[1,2-b]pyridazineIC50910.0 [1]
N-[(2S)-1-Hydroxybutan-2-yl]-3-[6-[[(2R)-1-hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]benzamideIC503900.0 [1]
4-(6-Methoxyimidazo[1,2-b]pyridazin-3-yl)pyrimidin-2-amineIC502300.0 [1]
Ethyl N-[3-(3-chlorophenyl)imidazo[1,2-b]pyridazin-6-yl]carbamateIC507100.0 [1]
3-[6-[[(2S)-1-Hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]benzoic acidIC506600.0 [1]
N-[3-[6-[Acetyl-[(2S)-1-hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]phenyl]acetamideIC50930.0 [1]
(2S)-2-[[3-(2-Methylsulfanylpyrimidin-4-yl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC5010000.0 [1]
3-(6-Chloroimidazo[1,2-b]pyridazin-3-yl)-N-[(2S)-1-hydroxybutan-2-yl]benzamideIC501900.0 [1]
3-[6-[[(2S)-1-Hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]benzaldehydeIC50460.0 [1]
N-[3-[6-(3-Acetamidoanilino)imidazo[1,2-b]pyridazin-3-yl]phenyl]acetamideIC50520.0 [1]
(2S)-2-[[3-[4-(Trifluoromethyl)phenyl]imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC502100.0 [1]
(2S)-2-[[3-(3-Chlorophenyl)imidazo[1,2-b]pyridazin-6-yl]amino]butan-1-olIC5081.0 [1]
(2S)-2-[(3-Thiophen-3-ylimidazo[1,2-b]pyridazin-6-yl)amino]butan-1-olIC501700.0 [1]
N-[(2R)-1-Hydroxybutan-2-yl]-3-[6-[[(2S)-1-hydroxybutan-2-yl]amino]imidazo[1,2-b]pyridazin-3-yl]benzamideIC5010000.0 [1]
(2S)-2-[(3-Pyridin-3-ylimidazo[1,2-b]pyridazin-6-yl)amino]butan-1-olIC50950.0 [1]
6-Fluoro-3-[3-(trifluoromethyl)phenyl]imidazo[1,2-b]pyridazineIC5010000.0 [1]
6-Chloro-3-[(E)-2-[3-(trifluoromethyl)phenyl]ethenyl]imidazo[1,2-b]pyridazineIC5010000.0 [1]
6-Methoxy-3-[3-(trifluoromethyl)phenyl]imidazo[1,2-b]pyridazineIC505300.0 [1]
6-Chloro-3-(pyridin-3-yl)imidazo[1,2-b]pyridazineIC5016000.0 [1]
6-Chloro-3-(3-chlorophenyl)imidazo[1,2-b]pyridazineIC503000.0 [1]
3-(6-Chloroimidazo[1,2-b]pyridazin-3-yl)anilineIC5015000.0 [1]
6-Chloro-3-(3-(trifluoromethyl)phenyl)imidazo[1,2-b]pyridazineIC5010000.0 [1]
(2S)-N-[5-(6-Aminopyridin-3-yl)-4-methyl-1,3-thiazol-2-yl]-4,4,4-trifluoro-2-methylbutanamideIC5010000.0 [1]
[3-(2-Aminopyrimidin-4-yl)-5-bromoindol-1-yl]-morpholin-4-ylmethanoneIC502200.0 [1]
6,10-Dihydroxy-11-methoxy-3,3-dimethyl-12H-pyrano[2,3-c]acridin-7-oneIC501200.0 [1]
6-Chloro-3-[4-(trifluoromethyl)phenyl]imidazo[1,2-b]pyridazineIC5010000.0 [1]
3-(6-Chloroimidazo[1,2-b]pyridazin-3-yl)benzaldehydeIC501700.0 [1]
CID 90388565IC504700.0 [1]
10-Iodo-11h-Indolo[3,2-C]quinoline-6-Carboxylic AcidIC5010000.0 [1]
10-Chloro-2-Iodo-11h-Indolo[3,2-C]quinoline-6-Carboxylic AcidIC5010000.0 [1]
10-Bromo-2-Iodo-11h-Indolo[3,2-C]quinoline-6-Carboxylic AcidIC5010000.0 [1]
2-(2-(2-Aminoethoxy)ethoxy)ethanolIC5010000.0 [1]
(5Z)-2-(2-Chlorophenyl)imino-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-oneIC5010.0 [1]
(5Z)-2-[2-(Dimethylamino)ethylimino]-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-oneIC501000.0 [1]
(5Z)-5-(2,3-Dihydro-1-benzofuran-5-ylmethylidene)-2-[2-(trifluoromethyl)phenyl]imino-1,3-thiazolidin-4-oneIC50100.0 [1]
(5Z)-2-(5-Amino-2-chlorophenyl)imino-5-(quinolin-6-ylmethylidene)-1,3-thiazolidin-4-oneIC501.0 [1]
(5Z)-2-[(2-Bromophenyl)amino]-5-(6-quinolinylmethylidene)-1,3-thiazol-4(5H)-oneIC501.0 [1]
Items per page: 1 - 10 of 99
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References

This online tool may be cited as follows

MLA

"Quest Database™ Dual-specificity tyrosine-phosphorylation regulated kinase 3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/dual-specificity-tyrosine-phosphorylation-regulated-kinase-3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Dual-specificity tyrosine-phosphorylation regulated kinase 3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dual-specificity-tyrosine-phosphorylation-regulated-kinase-3-inhibitors-ic50-ki.
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