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Dual-specificity tyrosine-phosphorylation regulated kinase 2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
HarmineIC50900.0 [1]
Leucettine L41IC5035.0 [1], 73.0 [2], 220.0 [3]
Leucettamine BIC501500.0 [1], 2000.0 [2]
SeliciclibIC501700.0 [1]
6-Bromoindirubin-3'-oximeIC502100.0 [1]
HarmolIC501500.0 [1]
5-Quinoxalin-6-ylmethylene-thiazolidine-2,4-dioneIC50100.0 [1]
7-Bromo-3-[3-(hydroxyamino)-1H-indol-2-yl]indol-2-oneIC501300.0 [1]
JNK Inhibitor VIC50300.0 [1]
CID 59604787IC5010000.0 [1]
3-(4-Methoxy-benzylidene)-dihydro-furan-2-oneIC5010000.0 [1]
2-(3-Hydroxy-4-methoxystyryl)-8-hydroxyquinoline-7-carboxylic acidIC501100.0 [1]
CID 72716071IC50190000.0 [1]
3-(1,3-Benzodioxol-5-ylmethylene)dihydro-2(3H)-furanoneIC50990.0 [1]
7-Bromo-1-methyl-3-(3-nitroso-1H-indol-2-yl)indol-2-olIC5010000.0 [1]
4-[3-(4-Hydroxyphenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenolIC50166.0 [1]
2-(7-Bromo-2-hydroxy-1H-indol-3-yl)-3-nitroso-1H-indole-6-carboxylic acidIC501700.0 [1]
3-(3-Nitroso-1H-indol-2-yl)-7-(trifluoromethyl)-1H-indol-2-olIC5010000.0 [1]
Methyl 2-(7-bromo-2-hydroxy-1H-indol-3-yl)-3-nitroso-1H-indole-5-carboxylateIC5010000.0 [1]
2-(2,4-Dihydroxybenzylcarbamoyl)-8-hydroxyquinoline-7-carboxylic acidIC506300.0 [1]
2-N-(4-Aminocyclohexyl)-8-propan-2-yl-4-N-[(4-pyridin-2-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazine-2,4-diamineIC50120.0 [1]
2-(7-Bromo-2-hydroxy-1-methylindol-3-yl)indol-3-oneIC5010000.0 [1]
(2z,3e)-7'-Bromo-3-(Hydroxyimino)-2'-Oxo-1,1',2',3-Tetrahydro-2,3'-Biindole-5-Carboxylic AcidIC50130.0 [1]
2-[2-Hydroxy-7-(trifluoromethyl)-1H-indol-3-yl]-3-nitroso-1H-indole-5-carbonitrileIC5010000.0 [1]
(4Z)-2-[4-[2-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]ethoxy]anilino]-4-(1,3-benzodioxol-5-ylmethylidene)-1H-imidazol-5-oneIC50130.0 [1]
Methyl 2-(7-bromo-2-hydroxy-1H-indol-3-yl)-3-oxoindole-5-carboxylateIC5010000.0 [1]
Methyl 2-[2-hydroxy-7-(trifluoromethyl)-1H-indol-3-yl]-3-oxoindole-5-carboxylateIC5010000.0 [1]
2-[2-Hydroxy-7-(trifluoromethyl)-1H-indol-3-yl]-3-oxoindole-5-carbonitrileIC5010000.0 [1]
Methyl 2-(7-bromo-2-hydroxy-1-methylindol-3-yl)-3-oxoindole-5-carboxylateIC5010000.0 [1]
Methyl 2-(7-bromo-2-hydroxy-1H-indol-3-yl)-3-oxoindole-6-carboxylateIC5010000.0 [1]
Methyl 2-[2-hydroxy-7-(trifluoromethyl)-1H-indol-3-yl]-3-oxoindole-6-carboxylateIC5010000.0 [1]
2-(7-Bromo-2-hydroxy-1H-indol-3-yl)-3-oxoindole-6-carboxylic acidIC501300.0 [1]
2-(2-Hydroxy-1H-indol-3-yl)-3-nitroso-1H-indole-5-carboxylic acidIC50350.0 [1]
Methyl 2-[2-hydroxy-7-(trifluoromethyl)-1H-indol-3-yl]-3-nitroso-1H-indole-5-carboxylateIC5010000.0 [1]
Methyl 2-(7-bromo-2-hydroxy-1H-indol-3-yl)-3-nitroso-1H-indole-6-carboxylateIC5010000.0 [1]
2-[2-Hydroxy-7-(trifluoromethyl)-1H-indol-3-yl]-3-nitroso-1H-indole-6-carboxylic acidIC5010000.0 [1]
2-(2-Hydroxy-1H-indol-3-yl)-3-oxoindole-5-carboxylic acidIC501800.0 [1]
2-[2-Hydroxy-7-(trifluoromethyl)-1H-indol-3-yl]-5-(2H-tetrazol-5-yl)indol-3-oneIC5010000.0 [1]
3-[3-Nitroso-5-(2H-tetrazol-5-yl)-1H-indol-2-yl]-7-(trifluoromethyl)-1H-indol-2-olIC5010000.0 [1]
STO-609 acetateIC50950.0 [1]
N-[2-[2-Aminoethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]acetamideIC5040.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
(5Z)-5-(Quinolin-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-oneIC5060.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
10-Chloro-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5040.0 [1]
10-Bromo-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5016.0 [1]
10-Fluoro-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC508000.0 [1]
10-Chloro-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5033.0 [1]
10-Bromo-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5023.0 [1]
10-Iodo-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Chloro-3-ethoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Fluoro-2-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Chloro-2-(3-methoxyphenyl)-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5079.0 [1]
10-Bromo-11H-indolo[3,2-c][1,5]naphthyridine-6-carboxylic acidIC5010000.0 [1]
5-(4-Pyridin-3-ylthiophen-2-yl)-1,3-thiazoleIC5040.0 [1]
(3E)-3-[(4-Methoxyphenyl)methylidene]oxan-2-oneIC5010000.0 [1]
(5E)-2-Mercapto-5-(4-methoxybenzylidene)-1,3-thiazol-4(5H)-oneIC5010000.0 [1]
(3E)-3-(2,3-Dihydro-1-benzofuran-5-ylmethylidene)-5-methyloxolan-2-oneIC50430.0 [1]
(3E)-3-(2,3-Dihydro-1,4-benzodioxin-6-ylmethylidene)oxolan-2-oneIC502040.0 [1]
(3E)-3-(1,3-Benzothiazol-6-ylmethylidene)-5-methyloxolan-2-oneIC5010000.0 [1]
(5Z)-5-(1,3-Benzothiazol-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-oneIC50200.0 [1]
(3E)-3-(3,4-Dihydro-2H-chromen-6-ylmethylidene)oxolan-2-oneIC5010000.0 [1]
(3E)-3-(1,3-Benzothiazol-6-ylmethylidene)oxolan-2-oneIC5060.0 [1]
(5Z)-5-(1,3-Benzothiazol-6-ylmethylidene)-2-sulfanylideneimidazolidin-4-oneIC501500.0 [1]
(3E)-3-(2,3-Dihydro-1-benzofuran-5-ylmethylidene)oxolan-2-oneIC50820.0 [1]
Clk1-IN-1IC5010000.0 [1]
(4Z)-2-Anilino-4-benzylidene-1H-imidazol-5-oneIC5010000.0 [1]
(5Z)-2-(2-Aminoethylimino)-5-(1,3-benzodioxol-5-ylmethylidene)-3-methylimidazolidin-4-oneIC50710.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-3-methyl-2-(2-morpholin-4-ylethylimino)imidazolidin-4-oneIC501600.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-butylimino-3-methylimidazolidin-4-oneIC50610.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-(5-hydroxypentylimino)-3-methylimidazolidin-4-oneIC502000.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-3-methyl-2-methyliminoimidazolidin-4-oneIC502200.0 [1]
(4Z)-2-(1,3-Benzodioxol-5-ylamino)-4-(1,3-benzodioxol-5-ylmethylidene)-1H-imidazol-5-oneIC5040.0 [1]
(5Z)-5-[(2-Hydroxyphenyl)methylidene]-3-methyl-2-propyliminoimidazolidin-4-oneIC5010000.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-propyliminoimidazolidin-4-oneIC50120.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-(cyclopropylmethylimino)imidazolidin-4-oneIC5047.0 [1]
2-(Propylamino)-3-methyl-5-[(Z)-(1,3-benzodioxole-5-yl)methylene]-1-imidazoline-4-oneIC50550.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-3-methyl-2-(3-methylbutylimino)imidazolidin-4-oneIC50560.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-(3-hydroxypropylimino)-3-methylimidazolidin-4-oneIC50470.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-3-methyl-2-(2-methylpropylimino)imidazolidin-4-oneIC50210.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-3-methyl-2-prop-2-enyliminoimidazolidin-4-oneIC50620.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-(cyclopropylmethylimino)-3-methylimidazolidin-4-oneIC50340.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-cyclopentylimino-3-methylimidazolidin-4-oneIC506000.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-(2-methoxyethylimino)-3-methylimidazolidin-4-oneIC50770.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-benzylimino-3-methylimidazolidin-4-oneIC50560.0 [1]
(5Z)-3-Methyl-2-propylimino-5-[(3,4,5-trimethoxyphenyl)methylidene]imidazolidin-4-oneIC5010000.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-3-phenyl-2-propyliminoimidazolidin-4-oneIC5010000.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-ethyliminoimidazolidin-4-oneIC50160.0 [1]
(4Z)-4-(1,3-Benzodioxol-5-ylmethylidene)-2-(4-methylanilino)-1H-imidazol-5-oneIC5061.0 [1]
(4Z)-4-(1,3-Benzodioxol-5-ylmethylidene)-2-(4-hydroxyanilino)-1H-imidazol-5-oneIC5060.0 [1]
(4Z)-4-(1,3-Benzodioxol-5-ylmethylidene)-2-(4-methoxyanilino)-1H-imidazol-5-oneIC5080.0 [1]
(4Z)-4-(1,3-Benzodioxol-5-ylmethylidene)-2-(2,3-dihydro-1,4-benzodioxin-6-ylamino)-1H-imidazol-5-oneIC50110.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-3-propyl-2-propyliminoimidazolidin-4-oneIC502100.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-ethylimino-3-methylimidazolidin-4-oneIC50640.0 [1]
(5z)-5-(1,3-Benzodioxol-5-Ylmethylidene)-3-Methyl-2-(Propan-2-Ylamino)imidazol-4-OneIC50530.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-(2-hydroxyethylimino)-3-methylimidazolidin-4-oneIC5010000.0 [1]
(5Z)-5-(1,3-Benzodioxol-5-ylmethylidene)-2-(1,3-benzodioxol-5-ylmethylimino)-3-methylimidazolidin-4-oneIC503300.0 [1]
Methyl 2-(7-bromo-2-hydroxy-1-methylindol-3-yl)-3-nitroso-1H-indole-5-carboxylateIC5010000.0 [1]
(4Z)-2-[4-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]anilino]-4-(1,3-benzodioxol-5-ylmethylidene)-1H-imidazol-5-oneIC50150.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Dual-specificity tyrosine-phosphorylation regulated kinase 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Nov. 2024, https://www.aatbio.com/data-sets/dual-specificity-tyrosine-phosphorylation-regulated-kinase-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 20). Quest Database™ Dual-specificity tyrosine-phosphorylation regulated kinase 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dual-specificity-tyrosine-phosphorylation-regulated-kinase-2-inhibitors-ic50-ki.
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