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Dual specificity tyrosine-phosphorylation-regulated kinase 1B Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
▲
▼
HarmineIC5028.0 [1], 160.0 [2], 166.0 [3], 180.0 [4]
HarmineKi166.0 [1]
Leucettine L41IC5044.0 [1], 77.0 [2]
CID 71529770IC504.74 [1]
CID 71529752IC500.24 [1], 6.55 [2]
CID 72716071IC503.0 [1], 42.0 [2]
3-(2-Methylpyrimidin-4-yl)-1H-pyrrolo[2,3-c]pyridineIC5017.0 [1], 3069.0 [2]
Methyl 9-(2-bromo-4-fluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC500.24 [1], 6.55 [2]
6-(1H-Indol-3-yl)-N-[4-(4-methylpiperazin-1-yl)phenyl]pyrimidin-4-amineIC5085.0 [1], 9965.0 [2]
N-[4-(4-Methylpiperazin-1-yl)phenyl]-6-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-4-amineIC502.0 [1], 453.0 [2]
N-[2-Methoxy-4-(4-methylpiperazin-1-yl)phenyl]-6-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-4-amineIC501.0 [1], 282.0 [2]
N-[2-Methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineIC504.0 [1], 85.0 [2]
N-[2-Methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(7-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineIC505.0 [1], 83.0 [2]
4-(1,7-Dimethylpyrrolo[2,3-c]pyridin-3-yl)-N-[2-methoxy-4-(4-methylpiperazin-1-yl)phenyl]pyrimidin-2-amineIC509.0 [1], 168.0 [2]
3-[2-(4-Methylsulfonylphenyl)pyrimidin-4-yl]-1H-pyrrolo[2,3-c]pyridineIC5021.0 [1], 898.0 [2]
1-Methyl-3-[2-(4-methylsulfonylphenyl)pyrimidin-4-yl]pyrrolo[2,3-c]pyridineIC5012.0 [1], 810.0 [2]
7-Methyl-3-[2-(4-methylsulfonylphenyl)pyrimidin-4-yl]-1H-pyrrolo[2,3-c]pyridineIC5014.0 [1], 2118.0 [2]
3-[2-[(E)-2-Phenylethenyl]pyrimidin-4-yl]-1H-pyrrolo[2,3-c]pyridineIC507.0 [1], 192.0 [2]
AZ Dyrk1B 33IC507.0 [1], 194.0 [2]
3-(1H-Pyrrolo[2,3-b]pyridin-4-yl)-1H-pyrrolo[2,3-c]pyridineIC503.0 [1], 378.0 [2]
Methyl 9-(3-fluoro-4-hydroxyanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5011.0 [1]
Methyl 9-(4-hydroxy-3-nitroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC505.68 [1]
Methyl 9-(2,4-dichloroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboxylateIC507.7 [1]
9-(2-Bromo-4-fluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboxamideIC5031.5 [1]
Methyl 9-(3,4,5-trimethoxyanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC50485.8 [1]
Methyl 9-(2,4-dimethoxyanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5011.13 [1]
Methyl 9-anilino-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC503.48 [1]
Methyl 9-(4-methylanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC502.83 [1]
Methyl 9-(4-fluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC509.64 [1]
Methyl 9-(3-cyanoanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5071.98 [1]
Methyl 9-(4-cyanoanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC507.69 [1]
Methyl 9-(2,4-dichloroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC500.28 [1]
Methyl 9-(4-tert-butylanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5093.84 [1]
Methyl 9-(3-chloroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5018.78 [1]
Methyl 9-[4-(dimethylamino)anilino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5064.28 [1]
Methyl 9-(2,4-difluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC501.07 [1]
Methyl 9-[4-(trifluoromethyl)anilino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5025.21 [1]
Ethyl 9-(1,3-benzodioxol-5-ylamino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC507.72 [1]
Benzyl 9-(1,3-benzodioxol-5-ylamino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5037.34 [1]
Methyl 9-(4-methoxyanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5019.22 [1]
Methyl 9-(1,3-benzodioxol-5-ylamino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC504.2 [1]
SeliciclibIC501200.0 [1]
SilmitasertibIC506.4 [1]
5-Quinoxalin-6-ylmethylene-thiazolidine-2,4-dioneIC5080.0 [1]
Leucettamine BIC504100.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineIC50697.0 [1]
CID 46926514IC501156.0 [1]
3-(4-Methoxy-benzylidene)-dihydro-furan-2-oneIC503800.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamineIC50452.0 [1]
(5Z)-5-(4-Methoxybenzylidene)imidazolidine-2,4-dioneIC5010000.0 [1]
3-(1,3-Benzodioxol-5-ylmethylene)dihydro-2(3H)-furanoneIC502630.0 [1]
[5-[4-[(5-Methyl-2-furanyl)methylamino]-6-quinazolinyl]-2-furanyl]methanolIC504420.0 [1]
4-[3-(4-Hydroxyphenyl)-1H-pyrrolo[2,3-b]pyridin-5-yl]phenolIC5015.0 [1]
Mirk-IN-1IC5068.0 [1]
N-Cyclopentyl-4-[4-(4-oxo-1,5,6,7-tetrahydropyrrolo[3,2-c]pyridin-2-yl)pyridin-2-yl]benzamideIC5043.0 [1]
(4-Fluoro-3-hydroxyphenyl)-(5-hydroxy-1-benzothiophen-2-yl)methanoneIC50400.0 [1]
2-N-(4-Aminocyclohexyl)-8-propan-2-yl-4-N-[(4-pyridin-2-ylphenyl)methyl]pyrazolo[1,5-a][1,3,5]triazine-2,4-diamineIC50110.0 [1]
5-(1,3-Benzodioxol-5-Ylmethyl)-2-(Phenylamino)-4h-Imidazol-4-OneIC5037.0 [1]
(4Z)-2-[4-[2-[2-[2-(2-Aminoethoxy)ethoxy]ethoxy]ethoxy]anilino]-4-(1,3-benzodioxol-5-ylmethylidene)-1H-imidazol-5-oneIC5072.0 [1]
5-(4-Pyridin-3-ylthiophen-2-yl)pyridin-3-amineIC50154.3 [1]
2-(4-Fluorophenyl)-N-[5-(4-pyridin-3-ylthiophen-2-yl)pyridin-3-yl]acetamideIC50383.0 [1]
N-Propyl-4-({4-[(2,2,2-trifluoroethyl)amino]-1H-pyrrolo[2,3-d]pyrimidin-2-yl}amino)benzamideIC501530.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-[(2-methyl-4-thiazolyl)methyl]-4-quinazolinamineIC501510.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-[(2-methyl-4-thiazolyl)methyl]-4-quinazolinamineIC5025.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)quinazolin-4-amineIC50180.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-(thiophen-2-ylmethyl)-4-quinazolinamineIC5073.0 [1]
6-(Benzo[d][1,3]dioxol-5-yl)-N-(furan-3-ylmethyl)quinazolin-4-amineIC50938.0 [1]
3-(4-Pyridin-3-ylthiophen-2-yl)pyridineIC50300.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(3-oxolanylmethyl)-4-quinazolinamineIC50734.0 [1]
CID 46926513IC507.0 [1]
(Z)-3-Pyridin-3-yl-2-(1H-pyrrolo[2,3-b]pyridin-3-yl)prop-2-enenitrileIC50240.0 [1]
N-[2-[2-Aminoethyl(methyl)amino]-5-[[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]amino]phenyl]acetamideIC5040.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
(5Z)-5-(Quinolin-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-oneIC5060.0 [1]
4-[[4-Cyclopentyloxy-5-(2-methyl-1,3-benzoxazol-6-yl)-7H-pyrrolo[2,3-d]pyrimidin-2-yl]amino]-3-methoxy-N-methylbenzamideIC50157.0 [1]
(5-Hydroxy-1-benzothiophen-2-yl)-(3-hydroxyphenyl)methanoneIC50200.0 [1]
(5-Hydroxy-1-benzofuran-2-yl)-(3-hydroxyphenyl)methanoneIC506100.0 [1]
(5-Hydroxy-1-methylindol-2-yl)-(3-hydroxyphenyl)methanoneIC502700.0 [1]
(5-Hydroxy-1-benzothiophen-2-yl)-(4-hydroxyphenyl)methanoneIC50800.0 [1]
(5-Hydroxy-1-benzofuran-2-yl)-(4-hydroxyphenyl)methanoneIC501300.0 [1]
(5-Hydroxy-1-benzothiophen-2-yl)-(3-hydroxy-4-methylphenyl)methanoneIC50200.0 [1]
(5-Hydroxy-1-benzothiophen-2-yl)-(4-hydroxy-3-methylphenyl)methanoneIC507000.0 [1]
(2-Fluoro-5-hydroxyphenyl)-(5-hydroxy-1-benzothiophen-2-yl)methanoneIC50400.0 [1]
3-(5-Hydroxy-1-benzothiophene-2-carbonyl)benzonitrileIC502300.0 [1]
(5-Hydroxy-1-benzothiophen-2-yl)-phenylmethanoneIC501000.0 [1]
(6-Hydroxynaphthalen-2-yl)-(3-hydroxyphenyl)methanoneIC502300.0 [1]
1-[4-[3-Methoxy-4-[[6-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-4-yl]amino]phenyl]piperazin-1-yl]ethanoneIC5016.0 [1]
1-[4-[3-Methoxy-4-[[6-(1-methylpyrrolo[2,3-c]pyridin-3-yl)pyrimidin-4-yl]amino]phenyl]piperazin-1-yl]ethanoneIC5034.0 [1]
1-[4-[3-Methoxy-4-[[4-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-yl]amino]phenyl]piperazin-1-yl]ethanoneIC509.0 [1]
N-[2-Methoxy-4-(4-methylpiperazin-1-yl)phenyl]-4-(5-methyl-1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineIC504.0 [1]
5-Chloro-N-[4-(4-methylpiperazin-1-yl)phenyl]-4-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-amineIC5025.0 [1]
N-Cyclopentyl-4-[4-(1H-pyrrolo[2,3-c]pyridin-3-yl)pyrimidin-2-yl]benzamideIC5098.0 [1]
10-Chloro-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC50210.0 [1]
10-Bromo-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5080.0 [1]
10-Fluoro-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC503000.0 [1]
10-Chloro-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC501000.0 [1]
10-Bromo-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC50230.0 [1]
10-Iodo-3-methoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Chloro-3-ethoxy-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
10-Fluoro-2-iodo-11H-indolo[3,2-c]quinoline-6-carboxylic acidIC5010000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Dual specificity tyrosine-phosphorylation-regulated kinase 1B Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/dual-specificity-tyrosine-phosphorylation-regulated-kinase-1b-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Dual specificity tyrosine-phosphorylation-regulated kinase 1B Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dual-specificity-tyrosine-phosphorylation-regulated-kinase-1b-inhibitors-ic50-ki.
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