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Dual-specificity tyrosine-phosphorylation regulated kinase 1A Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
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▼
HarmineIC5056.0 [1]
HarmineKi33.0 [1]
SeliciclibIC503100.0 [1]
(Z)-1-(3-Ethyl-5-methoxy-2,3-dihydrobenzothiazol-2-ylidene)propan-2-oneIC50830.0 [1]
Leucettine L41IC5021.0 [1], 55.0 [2], 60.0 [3]
2-(4-Fluorophenyl)-N-[5-(4-pyridin-3-ylthiophen-2-yl)pyridin-3-yl]acetamideIC5014.3 [1], 79.0 [2]
(-)-Epigallocatechin gallateIC50330.0 [1], 13440.0 [2]
(1z)-1-(3-Ethyl-5-Hydroxy-1,3-Benzothiazol-2(3h)-Ylidene)propan-2-OneIC50240.0 [1]
4,5,6,7-TetrabromobenzotriazoleIC501000.0 [1], 4360.0 [2]
4,5,6,7-Tetrabromo-N,N-dimethyl-1H-benzimidazol-2-amineIC50120.0 [1], 400.0 [2]
5-Quinoxalin-6-ylmethylene-thiazolidine-2,4-dioneIC5030.0 [1], 1600.0 [2]
O6-Cyclohexylmethoxy-2-(4'-sulphamoylanilino) purineIC50900.0 [1]
Leucettamine BIC50600.0 [1], 950.0 [2]
6-(1,3-Benzodioxol-5-yl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineIC5027.0 [1], 62.0 [2]
PaprotrainIC505500.0 [1]
CID 46926514IC50282.0 [1], 2600.0 [2]
CID 71529770IC501.13 [1]
Ethyl 3-[(E)-2-Amino-1-Cyanoethenyl]-6,7-Dichloro-1-Methyl-1h-Indole-2-CarboxylateIC5055.0 [1]
CID 71529752IC500.16 [1], 3.6 [2]
1-Methyl-7-(pyridin-3-ylmethoxy)-9H-pyrido[3,4-b]indoleIC5010000.0 [1]
7-(2-Methoxyethoxy)-1-methyl-9H-pyrido[3,4-b]indoleIC5015500.0 [1], 16000.0 [2]
1-(6-Oxo-2,3,4,10b-tetrahydro-1H-pyrido[2,1-a]isoindol-10-yl)-3-pyridin-2-ylureaIC5010000.0 [1]
(7-Methoxy-9H-pyrido[3,4-b]indol-1-yl)methanolIC5054.8 [1], 106.0 [2]
5-(4-Pyridin-3-ylthiophen-2-yl)pyridin-3-amineIC50101.0 [1]
3-(4-Pyridin-3-ylthiophen-2-yl)pyridineIC50300.0 [1]
CID 46926513IC504.0 [1], 50.0 [2]
1-Methyl-7-cyclohexylmethyloxy-9-cyclohexylmethyl-beta-carbolineIC5010000.0 [1]
1-(6-Oxo-2,3,4,10b-tetrahydro-1H-pyrido[2,1-a]isoindol-10-yl)-3-pyrazin-2-ylureaIC5010000.0 [1]
Methyl 9-(2-bromo-4-fluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC500.16 [1], 3.6 [2]
1-Methyl-7-benzyloxy-9-benzyl-beta-carbolineIC5016000.0 [1], 16300.0 [2]
(5Z)-5-(Quinolin-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-oneIC5020.0 [1], 1400.0 [2]
(3E)-3-(2,3-Dihydro-1-benzofuran-5-ylmethylidene)-5-methyloxolan-2-oneIC50170.0 [1], 2100.0 [2]
(5Z)-5-(1,3-Benzothiazol-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-oneIC5040.0 [1], 2100.0 [2]
(3E)-3-(1,3-Benzothiazol-6-ylmethylidene)oxolan-2-oneIC50130.0 [1], 200.0 [2]
Methyl 9-(3-fluoro-4-hydroxyanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC508.63 [1]
Methyl 9-(4-hydroxy-3-nitroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC504.91 [1]
4-[5-(4-Aminophenyl)-1H-pyrrolo[2,3-b]pyridin-3-yl]phenolIC5043.0 [1], 711.0 [2]
5-(1,3-Benzodioxol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-4-amineIC5010000.0 [1], 26020.0 [2]
N-[(3,4-Dichlorophenyl)methyl]-4-(3-methoxyphenyl)pyrimidin-2-amineIC504654.0 [1], 5820.0 [2]
N-[(4-Chlorophenyl)methyl]-4-(3-methoxyphenyl)pyrimidin-2-amineIC506361.0 [1], 7330.0 [2]
N-[(3,4-Dichlorophenyl)methyl]-4-(4-methoxyphenyl)pyrimidin-2-amineIC50203.0 [1], 1160.0 [2]
N-[(4-Chlorophenyl)methyl]-4-(4-methoxyphenyl)pyrimidin-2-amineIC50558.0 [1], 2070.0 [2]
4-(1,3-Benzodioxol-5-yl)-N-[3-bromo-5-(trifluoromethyl)phenyl]pyrimidin-2-amineIC50107.0 [1], 520.0 [2]
4-(1,3-Benzodioxol-5-yl)-N-[3-(trifluoromethyl)phenyl]pyrimidin-2-amineIC5010.0 [1], 70.0 [2]
4-(1,3-Benzodioxol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amineIC507.0 [1], 40.0 [2]
N-[(3,4-Dichlorophenyl)methyl]-4-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrimidin-2-amineIC5018.0 [1], 210.0 [2]
5-(1,3-Benzodioxol-5-yl)-N-[(3,4-dichlorophenyl)methyl]pyrimidin-4-amineIC503454.0 [1], 4120.0 [2]
N,4-Bis(1,3-benzodioxol-5-yl)pyrimidin-2-amineIC5025.0 [1], 130.0 [2]
4-(1,3-Benzodioxol-5-yl)-N-[(3,5-dibromophenyl)methyl]pyrimidin-2-amineIC5011.0 [1], 70.0 [2]
4-(1,3-Benzodioxol-5-yl)-N-[(3,4-dichlorophenyl)methyl]pyrimidin-2-amineIC5026.0 [1], 160.0 [2]
5-(1,3-Benzodioxol-5-yl)-N-[(4-chlorophenyl)methyl]pyrimidin-4-amineIC504579.0 [1], 26020.0 [2]
4-(1,3-Benzodioxol-5-yl)-N-(4-chlorophenyl)pyrimidin-2-amineIC50273.0 [1], 520.0 [2]
4-(1,3-Benzodioxol-5-yl)-N-[(3,4-dibromophenyl)methyl]pyrimidin-2-amineIC5079.0 [1], 820.0 [2]
N-[(3,4-Dichlorophenyl)methyl]-4-(1H-indazol-6-yl)pyrimidin-2-amineIC50169.0 [1], 1640.0 [2]
N-[(3,4-Dichlorophenyl)methyl]-2-(1H-indazol-5-yl)pyrimidin-4-amineIC502352.0 [1], 4630.0 [2]
2-(1H-Indazol-6-yl)-N-(pyridin-3-ylmethyl)pyrimidin-4-amineIC501434.0 [1], 2070.0 [2]
4-(1H-Indazol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amineIC5061.0 [1], 150.0 [2]
N-[(3,4-Dichlorophenyl)methyl]-4-(1H-indazol-5-yl)pyrimidin-2-amineIC50129.0 [1], 330.0 [2]
2-(1H-Indazol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-4-amineIC50349.0 [1], 650.0 [2]
Methyl 9-(2,4-dichloroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboxylateIC505.1 [1]
9-(4-Bromo-2-fluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboxamideIC50194.4 [1]
9-(2-Bromo-4-fluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboxamideIC5026.2 [1]
Methyl 9-(3,4,5-trimethoxyanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC50436.1 [1]
Methyl 9-(2,4-dimethoxyanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC509.53 [1]
Methyl 9-anilino-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC501.81 [1]
Methyl 9-(4-methylanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC500.98 [1]
Methyl 9-(4-fluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC506.06 [1]
Methyl 9-(3-cyanoanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5042.7 [1]
Methyl 9-(4-cyanoanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC503.89 [1]
Methyl 9-(2,4-dichloroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC500.22 [1]
Methyl 9-(4-tert-butylanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5039.03 [1]
Methyl 9-(3-chloroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5013.64 [1]
Methyl 9-[4-(dimethylamino)anilino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5035.64 [1]
Methyl 9-(2,4-difluoroanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC500.94 [1]
Methyl 9-[4-(trifluoromethyl)anilino]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5018.26 [1]
Ethyl 9-(1,3-benzodioxol-5-ylamino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC506.02 [1]
Benzyl 9-(1,3-benzodioxol-5-ylamino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5033.93 [1]
9-(1,3-Benzodioxol-5-ylamino)-N'-[2-(dimethylamino)ethyl]-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidamideIC50431.2 [1]
Methyl 9-(4-methoxyanilino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC5013.08 [1]
Methyl 9-(1,3-benzodioxol-5-ylamino)-[1,3]thiazolo[5,4-f]quinazoline-2-carboximidateIC501.65 [1]
10-Iodo-11h-Indolo[3,2-C]quinoline-6-Carboxylic AcidIC506.0 [1], 500.0 [2]
2,9-Dibenzyl-1-methyl-7-phenylmethoxypyrido[3,4-b]indol-2-iumIC5021000.0 [1], 21200.0 [2]
2-Benzyl-7-(cyclohexylmethoxy)-9-(cyclohexylmethyl)-1-methylpyrido[3,4-b]indol-2-iumIC5043000.0 [1]
StaurosporineIC5019.0 [1]
Ellagic acidIC5040000.0 [1]
6-Bromoindirubin-3'-oximeIC5052.0 [1]
SilmitasertibIC506.8 [1]
HarmolIC5090.0 [1]
Purvalanol AIC50300.0 [1]
4,5,6,7-TetrabromobenzimidazoleIC502100.0 [1]
1,4-DiaminoanthraquinoneIC503600.0 [1]
4-(1H-Indol-3-yl)pyrimidin-2-amineIC50588.0 [1]
4-[1-Ethyl-7-[(piperidin-4-ylamino)methyl]imidazo[4,5-c]pyridin-2-yl]-1,2,5-oxadiazol-3-amineIC504900.0 [1]
JNK Inhibitor VIIIKi6900.0 [1]
(5-Oxo-5,6-dihydro-indolo[1,2-A]quinazolin-7-YL)-acetic acidIC508000.0 [1]
(2S,3S)-3-((7-(Benzylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-5-yl)amino)butane-1,2,4-triolIC502100.0 [1]
4-(Pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-oneIC5010000.0 [1]
ButyrolactoneiIC50100000.0 [1]
3-(4-Methoxy-benzylidene)-dihydro-furan-2-oneIC501810.0 [1]
6-(3-Methoxyphenyl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineIC505697.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Dual-specificity tyrosine-phosphorylation regulated kinase 1A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/dual-specificity-tyrosine-phosphorylation-regulated-kinase-1a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ Dual-specificity tyrosine-phosphorylation regulated kinase 1A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dual-specificity-tyrosine-phosphorylation-regulated-kinase-1a-inhibitors-ic50-ki.
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