 | 1-Ethyl-3-[5-[6-(4-methoxy-2,6-dimethylphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]urea | IC50 | 455.0 [1] |
 | CID 58688563 | IC50 | 30000.0 [1] |
 | CID 58688690 | IC50 | 2198.0 [1] |
 | 5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamide | IC50 | 10000.0 [1] |
 | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
 | 3-Chloro-4-[6-[2-(propylamino)-1,3-thiazol-5-yl]-2-pyrazin-2-ylpyrimidin-4-yl]phenol | IC50 | 30000.0 [1] |
 | Methyl N-[5-[6-(2,6-dimethyl-4-pentan-3-yloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]carbamate | IC50 | 30000.0 [1] |
 | 5-[6-[2-Chloro-5-(2-cyclohexylethoxy)phenyl]-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | N-[5-[6-(2,6-Dimethyl-4-pentan-3-yloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]-2-methylpropanamide | IC50 | 12500.0 [1] |
 | Methyl N-[5-[6-(4-methoxy-2,6-dimethylphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]carbamate | IC50 | 11910.0 [1] |
 | 1-[5-[6-(2,6-Dichloro-4-methoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]-3-methylurea | IC50 | 30000.0 [1] |
 | 5-[6-(2,6-Dichloro-4-pentan-3-yloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | 5-[6-(2-Chloro-4-cyclopentyloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | 5-[6-(2,6-Dichloro-4-methoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | 5-[6-(2-Chloro-4-methoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | 5-[6-(2-Chloro-4-pentan-3-yloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | 5-[6-(2-Chloro-4-pentoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | 5-[6-(2,6-Dichloro-4-propoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | N-[5-[6-(2,6-Dimethyl-4-pentan-3-yloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]acetamide | IC50 | 30000.0 [1] |
 | 1-[5-[6-(4-Methoxy-2,6-dimethylphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]-3-methylurea | IC50 | 1133.0 [1] |
 | 5-[6-(2-Methyl-4-pentan-3-yloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | 5-[6-(2,6-Dichloro-4-cyclopentyloxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | N-[5-[6-(4-Methoxy-2,6-dimethylphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-1,3-thiazol-2-yl]acetamide | IC50 | 2265.0 [1] |
 | 5-[6-(2-Chloro-5-propoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |
 | 5-[6-(2-Chloro-5-methoxyphenyl)-2-pyrazin-2-ylpyrimidin-4-yl]-N-propyl-1,3-thiazol-2-amine | IC50 | 30000.0 [1] |