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Dual specificity protein kinase CLK3 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
▲
▼
SilmitasertibIC5041.0 [1]
9H-Purine-2,6-diamine, N2-(2-aminocyclohexyl)-N6-(3-chlorophenyl)-9-ethyl-, cis-IC501000.0 [1]
Cdk1/2 Inhibitor IIIIC5029.2 [1]
6-(1,3-Benzodioxol-5-yl)-N-(thiophen-2-ylmethyl)-4-quinazolinamineIC506936.0 [1]
CID 46926514IC5010000.0 [1]
Ethyl 3-[(E)-2-Amino-1-Cyanoethenyl]-6,7-Dichloro-1-Methyl-1h-Indole-2-CarboxylateIC50530.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(2-furanylmethyl)-N-methyl-4-quinazolinamineIC508744.0 [1]
[5-[4-[(5-Methyl-2-furanyl)methylamino]-6-quinazolinyl]-2-furanyl]methanolIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-[(2-methyl-4-thiazolyl)methyl]-4-quinazolinamineIC507448.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-[(2-methyl-4-thiazolyl)methyl]-4-quinazolinamineIC501924.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)quinazolin-4-amineIC504655.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-(thiophen-2-ylmethyl)-4-quinazolinamineIC504949.0 [1]
6-(Benzo[d][1,3]dioxol-5-yl)-N-(furan-3-ylmethyl)quinazolin-4-amineIC504650.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(3-oxolanylmethyl)-4-quinazolinamineIC503642.0 [1]
CID 46926513IC5010000.0 [1]
(Z)-3-Pyridin-3-yl-2-(1H-pyrrolo[2,3-b]pyridin-3-yl)prop-2-enenitrileIC5010000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
(5Z)-5-(Quinolin-6-ylmethylidene)-2-sulfanylidene-1,3-thiazolidin-4-oneIC5086.6 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
11H-Pyrido[3,4-a]carbazole-6-carbonitrileIC501800.0 [1]
Clk1-IN-1IC505590.0 [1]
N-(4-Morpholin-4-ylcyclohexyl)-5-(oxan-4-yl)-7H-pyrrolo[2,3-d]pyrimidin-4-amineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(3R)-piperidin-3-yl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(1R,2S)-2-aminocyclohexyl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
N-[3-[[2-[[(1R,2S)-2-Aminocyclohexyl]amino]-9-propan-2-ylpurin-6-yl]amino]-5-chlorophenyl]acetamideIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(1S,2S)-2-aminocyclohexyl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(1R,2R)-2-aminocyclohexyl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
N-[3-[[2-[[(1S,2R)-2-Aminocyclohexyl]amino]-9-propan-2-ylpurin-6-yl]amino]-5-chlorophenyl]acetamideIC501000.0 [1]
2-N-[(1S,2R)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
2-N-[(1R,2R)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
2-N-[(1S,2S)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(1S,2R)-2-aminocyclohexyl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
2-N-[(1R,2S)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-9-propan-2-yl-2-N-[(3S)-pyrrolidin-3-yl]purine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-2-N-[(3S)-piperidin-3-yl]-9-propan-2-ylpurine-2,6-diamineIC501000.0 [1]
6-N-(3-Amino-5-chlorophenyl)-9-propan-2-yl-2-N-[(3R)-pyrrolidin-3-yl]purine-2,6-diamineIC501000.0 [1]
1-[4-[4-[[5-(Oxan-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]cyclohexyl]piperazin-1-yl]ethanoneIC5010000.0 [1]
1-[4-[4-[(5-Propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]cyclohexyl]piperazin-1-yl]ethanoneIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-[(3-methylthiophen-2-yl)methyl]quinazolin-4-amineIC506555.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-[2-(1H-imidazol-5-yl)ethyl]quinazolin-4-amineIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(2-oxolanylmethyl)-4-quinazolinamineIC503294.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]quinazolin-4-amineIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-[2-(2-furanyl)ethyl]-4-quinazolinamineIC502017.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-[(5-methylfuran-2-yl)methyl]quinazolin-4-amineIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(1H-imidazol-2-ylmethyl)quinazolin-4-amineIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-[(5-methylthiophen-2-yl)methyl]quinazolin-4-amineIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-[(2-methyl-3-furanyl)methyl]-4-quinazolinamineIC506450.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-[(3-methylthiophen-2-yl)methyl]quinazolin-4-amineIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-ethyl-N-(thiophen-2-ylmethyl)-4-quinazolinamineIC506172.0 [1]
Ethyl 5-(4-(thiophen-2-ylmethylamino)quinazolin-6-yl)furan-2-carboxylateIC5010000.0 [1]
Ethyl 5-(4-((5-methylfuran-2-yl)methylamino)quinazolin-6-yl)furan-2-carboxylateIC5010000.0 [1]
6-(3-Furanyl)-N-methyl-N-[(3-methyl-2-thiophenyl)methyl]-4-quinazolinamineIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(1H-imidazol-2-ylmethyl)-N-methylquinazolin-4-amineIC5010000.0 [1]
(5-(4-(Methyl((3-methylthiophen-2-yl)methyl)amino)quinazolin-6-yl)furan-2-yl)methanolIC5010000.0 [1]
5-(4-((5-Methylfuran-2-yl)methylamino)quinazolin-6-yl)furan-2-carboxylic acidIC5010000.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(2-thiazolylmethyl)-4-quinazolinamineIC503527.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]quinazolin-4-amineIC503019.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(2,2-dimethylpropyl)quinazolin-4-amineIC50435.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(furan-2-ylmethyl)quinazolin-4-amineIC502556.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(cyclopentylmethyl)-4-quinazolinamineIC501320.0 [1]
6-(1,3-Benzodioxol-5-yl)-N-(3-oxanylmethyl)-4-quinazolinamineIC505461.0 [1]
4-(1,3-Benzodioxol-5-yl)-N-[3-(trifluoromethyl)phenyl]pyrimidin-2-amineIC5010000.0 [1]
4-(1,3-Benzodioxol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amineIC501473.0 [1]
N-[(3,4-Dichlorophenyl)methyl]-4-(2,3-dihydro-1,4-benzodioxin-6-yl)pyrimidin-2-amineIC5010000.0 [1]
4-(1,3-Benzodioxol-5-yl)-N-[(3,4-dichlorophenyl)methyl]pyrimidin-2-amineIC503634.0 [1]
4-(1,3-Benzodioxol-5-yl)-N-[(3,4-dibromophenyl)methyl]pyrimidin-2-amineIC503232.0 [1]
4-(1H-Indazol-5-yl)-N-(pyridin-3-ylmethyl)pyrimidin-2-amineIC502663.0 [1]
N-[(3,4-Dichlorophenyl)methyl]-4-(1H-indazol-5-yl)pyrimidin-2-amineIC502934.0 [1]
N2-[(1R,2S)-2-Aminocyclohexyl]-N6-(3-chlorophenyl)-9-ethyl-9H-purine-2,6-diamineIC501000.0 [1]
N-(2,2-Dimethylpropyl)-6-[5-(ethylaminomethyl)furan-2-yl]quinazolin-4-amineIC5010000.0 [1]
2-N-[(1S,2S)-2-Aminocyclohexyl]-6-N-(3-chlorophenyl)-9-ethylpurine-2,6-diamineIC501000.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC501000.0 [1]
(9-Methoxy-11H-pyrido[4,3-a]carbazol-6-yl)methanamineIC507000.0 [1]
(Z)-2-(6-Methoxy-1H-pyrrolo[2,3-b]pyridin-3-yl)-3-pyridin-3-ylprop-2-enenitrileIC5010000.0 [1]
9-Methoxy-11H-pyrido[4,3-a]carbazole-6-carbonitrileIC50190.0 [1]
1,9-Dimethoxy-11H-pyrido[4,3-a]carbazole-6-carbonitrileIC50320.0 [1]
N-[(9-Methoxy-11H-pyrido[4,3-a]carbazol-6-yl)methyl]acetamideIC508000.0 [1]
10-Methoxy-11H-pyrido[4,3-a]carbazole-6-carbonitrileIC50180.0 [1]
8-Fluoro-11H-pyrido[4,3-a]carbazole-6-carbonitrileIC5010000.0 [1]
7-Methoxy-11H-pyrido[4,3-a]carbazole-6-carbonitrileIC5010000.0 [1]
10-Methoxy-11H-pyrido[4,3-a]carbazole-6-carboxamideIC506100.0 [1]
8-Methoxy-11H-pyrido[4,3-a]carbazole-6-carbonitrileIC50710.0 [1]
N-[7-(5-Methoxy-1H-indol-3-yl)isoquinolin-6-yl]acetamideIC507000.0 [1]
6-Methoxy-3-pyridin-4-yl-1H-pyrrolo[2,3-b]pyridineIC506100.0 [1]
6-Methoxy-1-oxo-3-pyridin-3-yl-2,9-dihydropyrido[3,4-b]indole-4-carbonitrileIC5010000.0 [1]
14-Methoxy-5,15,17-triazatetracyclo[8.7.0.02,7.011,16]heptadeca-1,3,5,7,9,11(16),12,14-octaene-9-carbonitrileIC5010000.0 [1]
5,15,17-Triazatetracyclo[8.7.0.02,7.011,16]heptadeca-1,3,5,7,9,11(16),12,14-octaene-9-carbonitrileIC506800.0 [1]
6,10-Dihydroxy-11-methoxy-3,3-dimethyl-12H-pyrano[2,3-c]acridin-7-oneIC502300.0 [1]
Ethyl 3-[(Z)-2-amino-1-cyanoethenyl]-6,7-dichloro-1-methylindole-2-carboxylateIC50530.0 [1]
Items per page: 1 - 10 of 90
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References

This online tool may be cited as follows

MLA

"Quest Database™ Dual specificity protein kinase CLK3 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/dual-specificity-protein-kinase-clk3-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Dual specificity protein kinase CLK3 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dual-specificity-protein-kinase-clk3-inhibitors-ic50-ki.
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