 | 4-[5-(4-Fluorobenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]benzoic acid | IC50 | 4200.0 [1] |
 | 4-[(5Z)-5-Benzylidene-4-oxo-2-thioxo-1,3-thiazolidin-3-YL]benzoic acid | IC50 | 18000.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N,3-N-diethylpiperidine-1,3-dicarboxamide | IC50 | 12010.0 [1] |
 | 4-[(4-Cyclohexylphenyl)methyl-[2-[methyl(quinolin-8-ylsulfonyl)amino]acetyl]amino]-2-hydroxybenzoic acid | IC50 | 10000.0 [1] |
 | 6-Hydroxy-2-phenyl-3-[2-[3-(trifluoromethyl)phenyl]ethynyl]benzofuran-5-carboxylic acid | IC50 | 1400.0 [1] |
 | 3-[2-(3,5-Difluorophenyl)ethynyl]-6-hydroxy-2-phenyl-benzofuran-5-carboxylic acid | IC50 | 2900.0 [1] |
 | 6-Hydroxy-2-phenyl-3-[2-[4-(trifluoromethoxy)phenyl]ethynyl]benzofuran-5-carboxylic acid | IC50 | 1900.0 [1] |
 | 3-{4-Oxo-5-[1-phenyl-meth-(Z)-ylidene]-2-thioxo-thiazolidin-3-yl}-benzoic acid | IC50 | 7000.0 [1] |
 | 3-[(5Z)-5-(4-Nitrobenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]benzoic acid | IC50 | 2600.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-cyclohexylpiperidine-1,3-dicarboxamide | IC50 | 2250.0 [1] |
 | 3-[5-(4-Fluoro-benzylidene)-4-oxo-2-thioxo-thiazolidin-3-yl]-benzoic acid | IC50 | 1300.0 [1] |
 | 2-[4-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]phenyl]acetic acid | IC50 | 20000.0 [1] |
 | 5-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]benzene-1,3-dicarboxylic acid | IC50 | 103000.0 [1] |
 | 2-Thioxo-3-phenyl-5-benzylidenethiazolidine-4-one | IC50 | 200000.0 [1] |
 | 4-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-2-hydroxybenzoic acid | IC50 | 13000.0 [1] |
 | 5-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-2-hydroxybenzoic acid | IC50 | 13000.0 [1] |
 | 1-(2-Methyl-4,5-disulfophenyl)-5-oxo-4,5-dihydro-1H-pyrazole-3-carboxylic acid | IC50 | 100000.0 [1] |
 | 2-[3-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]phenyl]acetic acid | IC50 | 20000.0 [1] |
 | 4-[[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]methyl]benzoic acid | IC50 | 60000.0 [1] |
 | Methyl 4-[(5Z)-5-benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]benzoate | IC50 | 200000.0 [1] |
 | 2-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]benzoic acid | IC50 | 200000.0 [1] |
 | 4-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]-3-methylbenzoic acid | IC50 | 66000.0 [1] |
 | 4-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]benzenesulfonic acid | IC50 | 11000.0 [1] |
 | [4-[(5Z)-5-Benzylidene-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]phenyl]methylphosphonic acid | IC50 | 10000.0 [1] |
 | 3-[(5Z)-5-(Cyclohexylmethylidene)-4-oxo-2-sulfanylidene-1,3-thiazolidin-3-yl]benzoic acid | IC50 | 7300.0 [1] |
 | 3-[(5Z)-4-Oxo-5-propylidene-2-sulfanylidene-1,3-thiazolidin-3-yl]benzoic acid | IC50 | 59000.0 [1] |
 | 4-[(4Z)-4-[(4-Fluorophenyl)methylidene]-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoic acid | IC50 | 200000.0 [1] |
 | 4-[(4Z)-4-[(4-Fluorophenyl)methylidene]-3-methyl-5-oxo-2-sulfanylideneimidazolidin-1-yl]benzoic acid | IC50 | 200000.0 [1] |
 | 4-[(5Z)-5-[(4-Fluorophenyl)methylidene]-2,4-dioxo-1,3-thiazolidin-3-yl]benzoic acid | IC50 | 200000.0 [1] |
 | 4-[(5Z)-5-[(4-Fluorophenyl)methylidene]-4-oxo-2-sulfanylidene-1,3-oxazolidin-3-yl]benzoic acid | IC50 | 200000.0 [1] |
 | N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-(piperidine-1-carbonyl)piperidine-1-carboxamide | IC50 | 8390.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-cyclopentylpiperidine-1,3-dicarboxamide | IC50 | 3020.0 [1] |
 | N1-(2,3-Diphenylquinoxalin-6-yl)-N3,N3-diethylpiperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | N-(2,3-Diphenylquinoxalin-6-yl)-3-(piperidine-1-carbonyl)piperidine-1-carboxamide | IC50 | 40000.0 [1] |
 | 1-N-[2,3-Bis(4-methylphenyl)quinoxalin-6-yl]-3-N,3-N-diethylpiperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | N3-Cyclopentyl-N1-(2,3-dip-tolylquinoxalin-6-yl)piperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | 1-N-[2,3-Bis(4-fluorophenyl)quinoxalin-6-yl]-3-N,3-N-diethylpiperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | 1-N-[2,3-Bis(4-fluorophenyl)quinoxalin-6-yl]-3-N-cyclohexylpiperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | 1-N-[2,3-Bis(4-bromophenyl)quinoxalin-6-yl]-3-N,3-N-diethylpiperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | N-[2,3-Bis(4-bromophenyl)quinoxalin-6-yl]-3-(pyrrolidine-1-carbonyl)piperidine-1-carboxamide | IC50 | 40000.0 [1] |
 | N-(2,3-Dimethoxyquinoxalin-6-yl)-3-(piperidine-1-carbonyl)piperidine-1-carboxamide | IC50 | 100000.0 [1] |
 | N3-Cyclohexyl-N1-(2,3-dimethoxyquinoxalin-6-yl)piperidine-1,3-dicarboxamide | IC50 | 100000.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N,3-N-dimethylpiperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-butyl-3-N-methylpiperidine-1,3-dicarboxamide | IC50 | 5550.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-butyl-3-N-ethylpiperidine-1,3-dicarboxamide | IC50 | 2350.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N,3-N-dipropylpiperidine-1,3-dicarboxamide | IC50 | 2500.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-ethylpiperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-propan-2-ylpiperidine-1,3-dicarboxamide | IC50 | 40000.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-tert-butylpiperidine-1,3-dicarboxamide | IC50 | 8050.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-(2-methylpropyl)piperidine-1,3-dicarboxamide | IC50 | 8360.0 [1] |
 | 1-N-[2,3-Bis(furan-2-yl)quinoxalin-6-yl]-3-N-butylpiperidine-1,3-dicarboxamide | IC50 | 2790.0 [1] |
 | 5-[(E)-[4-[3-[Difluoro(phosphono)methyl]phenyl]phenyl]methoxyiminomethyl]furan-2-carboxylic acid | IC50 | 400000.0 [1] |
 | 4-[(4-Cyclohexylphenyl)methyl-[2-[methyl(naphthalen-1-ylsulfonyl)amino]acetyl]amino]-2-hydroxybenzoic acid | IC50 | 10000.0 [1] |
 | CID 56680468 | IC50 | 10000.0 [1] |
 | 3-[(5Z)-5-(4-Methylbenzylidene)-4-oxo-2-thioxo-1,3-thiazolidin-3-yl]benzoic acid | IC50 | 16000.0 [1] |
 | 3-{5-[(4-Methoxyphenyl)methylene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl}benzoic acid | IC50 | 26000.0 [1] |
 | 3-{5-[(4-Hydroxyphenyl)methylene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl}benzoic acid | IC50 | 157000.0 [1] |
 | 3-{5-[(4-Carboxyphenyl)methylene]-4-oxo-2-thioxo-1,3-thiazolidin-3-yl}benzoic acid | IC50 | 200000.0 [1] |
 | 2-Hydroxy-4-[[4-[4-(3-methoxycarbonylphenyl)phenyl]phenyl]methyl-[2-[methyl-(4-methylphenyl)sulfonylamino]acetyl]amino]benzoic acid | IC50 | 10000.0 [1] |
 | N-(4-Fluoro-1,3-benzothiazol-2-yl)-5-(4-methoxyphenyl)-1,3,4-oxadiazol-2-amine | IC50 | 26000.0 [1] |
 | 4-[[4-[4-(3-Carbamoylphenyl)phenyl]phenyl]methyl-[2-[methyl-(4-methylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | IC50 | 10000.0 [1] |
 | 4-[[4-[4-(3-Cyanophenyl)phenyl]phenyl]methyl-[2-[methyl-(4-methylphenyl)sulfonylamino]acetyl]amino]-2-hydroxybenzoic acid | IC50 | 10000.0 [1] |