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Dual specificity mitogen-activated protein kinase kinase 7 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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5Z-7-OxozeaenolIC50300.0 [1], 1300.0 [2]
AS-252424IC5010000.0 [1]
JNK Inhibitor VIC5010000.0 [1]
1-((2S,5R)-5-((7H-Pyrrolo[2,3-d]pyrimidin-4-yl)amino)-2-methylpiperidin-1-yl)prop-2-en-1-oneIC5050000.0 [1]
CID 59604787IC5010000.0 [1]
CID 72547959IC505000.0 [1]
JAK3 covalent inhibitor-1IC5010000.0 [1]
2-[[1-Cyclopentyl-5-[1-(Oxetan-3-Yl)piperidin-4-Yl]pyrazol-3-Yl]amino]pyridine-4-CarbonitrileIC505000.0 [1]
(13R,15S)-13-Methyl-16-oxa-8,9,12,22,24-pentazahexacyclo[15.6.2.16,9.112,15.02,7.021,25]heptacosa-1(24),2,4,6,17,19,21(25)-heptaene-23,27-dioneIC501000.0 [1]
3-[5-Chloro-4-[(2,4-difluorophenyl)methoxy]-6-oxopyrimidin-1-yl]-N-(2-hydroxyethyl)-4-methylbenzamideIC5010000.0 [1]
2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi2000.0 [1]
2-[3-[3-(4-Methylpiperazin-1-yl)propoxy]phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamideKi10000.0 [1]
5-(1,3-Benzodioxol-5-yl)-7-[[(2R)-1-ethenylsulfonylpyrrolidin-2-yl]methyl]pyrrolo[2,3-d]pyrimidin-4-amineIC50188.6 [1]
[(1S)-6-(7H-Pyrrolo[2,3-d]pyrimidin-4-yl)-2,3-dihydro-1H-inden-1-yl]cyanamideIC5010000.0 [1]
[(1S)-6-[5-[3-(Hydroxymethyl)phenyl]-7H-pyrrolo[2,3-d]pyrimidin-4-yl]-2,3-dihydro-1H-inden-1-yl]cyanamideIC5010000.0 [1]
4-(4-(2-(Cyclopentylamino)pyrimidin-4-yl)-1H-pyrazol-3-yl)cyclohexanolIC50860.0 [1]
2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamideIC5010000.0 [1]
2-Amino-4-(benzylamino)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[4-(Dimethylamino)phenyl]-9H-pyrimido[4,5-b]indole-6-carboxamideIC501000.0 [1]
4-(4-Benzyl-4-hydroxypiperidin-1-yl)-9H-pyrimido[4,5-b]indole-6-carboxamideIC501000.0 [1]
4-[4-(Hydroxymethyl)piperidin-1-yl]-9H-pyrimido[4,5-b]indole-6-carboxamideIC501000.0 [1]
Tert-butyl N-[1-(6-carbamoyl-9H-pyrimido[4,5-b]indol-4-yl)piperidin-3-yl]carbamateIC501000.0 [1]
4-(4-Fluorophenyl)-9H-pyrimido[4,5-b]indole-6-carboxamideIC501000.0 [1]
4-Phenyl-9H-pyrimido[4,5-b]indole-6-carboxamideIC501000.0 [1]
4-(4-Methoxyphenyl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(4-Fluorophenyl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-phenyl-9H-pyrimido[4,5-b]indole-6-carboxamideIC501000.0 [1]
4-[Benzyl(2-hydroxyethyl)amino]-9H-pyrimido[4,5-b]indole-6-carboxamideIC501000.0 [1]
1-(2-Amino-6-hydroxy-9H-pyrimido[4,5-b]indol-4-yl)piperidine-4-carboxylic acidIC501000.0 [1]
4-[(3R)-3-Hydroxypiperidin-1-yl]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(3-Aminopiperidin-1-yl)-9H-pyrimido[4,5-b]indole-6-carboxamide;dihydrochlorideIC501000.0 [1]
4-(6-Hydroxy-9H-pyrimido[4,5-b]indol-4-yl)piperazine-1-carbaldehydeIC501000.0 [1]
4-(2-Aminoethylamino)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[[(2R)-1-Hydroxypropan-2-yl]amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[[(2S)-1-Hydroxypropan-2-yl]amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(4-Aminopiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
Tert-butyl N-[2-[(6-carbamoyl-9H-pyrimido[4,5-b]indol-4-yl)amino]ethyl]carbamateIC501000.0 [1]
2-Amino-4-(4-benzylpiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
Acetic acid;2-amino-4-morpholin-4-yl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(3-Aminopiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-(1,4-dioxa-8-azaspiro[4.5]decan-8-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
Tert-butyl N-[1-(6-hydroxy-9H-pyrimido[4,5-b]indol-4-yl)piperidin-4-yl]carbamateIC501000.0 [1]
4-[3-(Hydroxymethyl)piperidin-1-yl]-2-methyl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[[(2S)-1-Hydroxy-3-phenylpropan-2-yl]amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[(2S)-2-(Hydroxymethyl)pyrrolidin-1-yl]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
Tert-butyl 4-[(6-hydroxy-9H-pyrimido[4,5-b]indol-4-yl)amino]piperidine-1-carboxylateIC501000.0 [1]
4-(3-Aminopropylamino)-9H-pyrimido[4,5-b]indole-6-carboxamide;dihydrochlorideIC501000.0 [1]
2-Amino-4-[cyclohexyl(methyl)amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(3-Aminopyrrolidin-1-yl)-9H-pyrimido[4,5-b]indole-6-carboxamide;dihydrochlorideIC501000.0 [1]
4-[4-(Hydroxymethyl)piperidin-1-yl]-2-methyl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(3-Hydroxypiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-ol;hydrochlorideIC501000.0 [1]
4-[(3S)-3-Aminopyrrolidin-1-yl]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-(4-pyrrolidin-1-ylpiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[2-(Hydroxymethyl)piperidin-1-yl]-2-methyl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-Morpholin-4-yl-9H-pyrimido[4,5-b]indole-6-carboxamide;hydrochlorideIC501000.0 [1]
4-(2-Aminoethylamino)-9H-pyrimido[4,5-b]indole-6-carboxamide;hydrochlorideIC501000.0 [1]
4-(3,4,4a,5,6,7,8,8a-Octahydro-1H-isoquinolin-2-yl)-2-amino-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[3-(Methylamino)pyrrolidin-1-yl]-9H-pyrimido[4,5-b]indole-6-carboxamide;dihydrochlorideIC501000.0 [1]
4-[Cyclohexyl(methyl)amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
Methyl 2-amino-4-piperidin-1-yl-9H-pyrimido[4,5-b]indole-6-carboxylateIC501000.0 [1]
Acetic acid;2-amino-4-piperidin-1-yl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[4-(4-Hydroxybutyl)piperazin-1-yl]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(4-Benzyl-4-hydroxypiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-Piperidin-1-yl-9H-pyrimido[4,5-b]indole-6-carboxamide;hydrochlorideIC501000.0 [1]
4-(1-Hydroxypropan-2-ylamino)-2-methyl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
Methyl 2-methyl-4-piperidin-1-yl-9H-pyrimido[4,5-b]indole-6-carboxylateIC501000.0 [1]
4-Piperidin-1-yl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Methyl-4-piperidin-1-yl-9H-pyrimido[4,5-b]indole-6-carboxylic acidIC501000.0 [1]
2-[(2-Methyl-6-phenylmethoxy-9H-pyrimido[4,5-b]indol-4-yl)amino]propan-1-olIC501000.0 [1]
2-Amino-4-(azepan-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-(2-methylpiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-(4-methoxypiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-[methyl(propan-2-yl)amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-(3-hydroxypiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-Morpholin-4-yl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(Cyclohexylamino)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-Pyrrolidin-1-yl-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[2-Hydroxyethyl(methyl)amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(4-Hydroxypiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(2-Hydroxyethylamino)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(4-Methylpiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(Azepan-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(3-Methylpiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(2-Methoxyethylamino)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[4-(Hydroxymethyl)piperidin-1-yl]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(4-Methoxypiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(Cycloheptylamino)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(3,5-Dimethylpiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(3-Hydroxypiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-(2-pyrrolidin-1-ylethylamino)-9H-pyrimido[4,5-b]indol-6-olIC5010000.0 [1]
4-(3-Hydroxypyrrolidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(2-Ethylpiperidin-1-yl)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
2-Amino-4-(dibenzylamino)-9H-pyrimido[4,5-b]indol-6-olIC5010000.0 [1]
4-[Methyl(propan-2-yl)amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-(1-Hydroxypropan-2-ylamino)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[2-(Hydroxymethyl)piperidin-1-yl]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[3-(Hydroxymethyl)piperidin-1-yl]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
1-(6-Hydroxy-9H-pyrimido[4,5-b]indol-4-yl)piperidin-4-oneIC501000.0 [1]
2-Amino-4-(cyclohexylamino)-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
4-[(4-Hydroxycyclohexyl)amino]-9H-pyrimido[4,5-b]indol-6-olIC501000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Dual specificity mitogen-activated protein kinase kinase 7 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/dual-specificity-mitogen-activated-protein-kinase-kinase-7-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Dual specificity mitogen-activated protein kinase kinase 7 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/dual-specificity-mitogen-activated-protein-kinase-kinase-7-inhibitors-ic50-ki.
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