| 7-Methyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine | Ki | 12.7 [1] |
| 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-6-ol | Ki | 1.69 [1] |
| Haloperidol | Ki | 38.0 [1], 48.0 [2], 58.0 [3], 260.0 [4] |
| Clozapine | Ki | 198.0 [1], 235.0 [2], 780.0 [3], 1000.0 [4] |
| Aripiprazole | Ki | 1000.0 [1], 1051.0 [2], 1600.0 [3] |
| 6-Methoxy-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaene | Ki | 7.2 [1], 38.3 [2], 54.0 [3] |
| 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3,5,7,14,16-hexaene | Ki | 3.09 [1], 11.2 [2] |
| (R)-2,3,4,5-Tetrahydro-8-chloro-3-methyl-5-phenyl-1H-3-benzazepin-7-ol | IC50 | 1.1 [1] |
| (R)-2,3,4,5-Tetrahydro-8-chloro-3-methyl-5-phenyl-1H-3-benzazepin-7-ol | Ki | 2.8 [1], 8.1 [2] |
| 10-Methyl-6-thia-10-azatricyclo[11.4.0.03,7]heptadeca-1(17),3(7),4,13,15-pentaene | Ki | 15.0 [1], 33.7 [2], 79.1 [3] |
| Olanzapine | Ki | 90.0 [1], 100.0 [2] |
| 7-Chloro-3-methyl-1-phenyl-1,2,4,5-tetrahydro-3-benzazepin-8-ol | IC50 | 0.56 [1] |
| Sch-23390 maleate | IC50 | 0.15 [1], 0.37 [2] |
| Ecopipam | Ki | 2.0 [1] |
| 7-[4-[4-(2,3-Dichlorophenyl)-1,4-diazepan-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one | Ki | 615.0 [1], 1100.0 [2] |
| 7-Chloro-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-6-ol | Ki | 0.05 [1], 0.06 [2] |
| 12-Methyl-12,22-diazatetracyclo[13.7.0.03,8.016,21]docosa-1(15),3,5,7,16,18,20-heptaene | Ki | 0.61 [1], 2.8 [2] |
| 11-Methyl-11,22-diazatetracyclo[13.7.0.03,8.016,21]docosa-1(15),3,5,7,16,18,20-heptaene | Ki | 71.6 [1], 92.0 [2] |
| 2-[4-(4-Phenylpiperazin-1-yl)butyl]isoindolin-1-one | Ki | 80.0 [1], 10000.0 [2] |
| 2-(4-(4-Phenyl-1-piperazinyl)butyl)-1-isoindolinone | Ki | 75.4 [1], 137.0 [2] |
| 1-(4-(4-(2-Methoxyphenyl)-1-piperazinyl)butyl)-indolin-2-one | Ki | 313.0 [1], 10000.0 [2] |
| (8S)-N-[(3-Fluorophenyl)methyl]-N-methylpentacyclo[5.4.0.02,6.03,10.05,9]undecan-8-amine | Ki | 10000.0 [1] |
| 6,10-Dimethyl-6,10-diazatricyclo[11.4.0.03,7]heptadeca-1(17),3(7),4,13,15-pentaene | Ki | 337.0 [1], 361.0 [2] |
| 5-Amino-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3,5,7,14,16-hexaen-6-ol | Ki | 39.5 [1], 226.5 [2] |
| 6-Chloro-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3,5,7,14,16-hexaen-5-ol | Ki | 3.1 [1], 4.9 [2] |
| 6,16-Dimethoxy-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(14),3(8),4,6,15,17-hexaene | Ki | 11.5 [1], 12.6 [2] |
| 4-Chloro-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-5-ol | Ki | 0.98 [1], 1.6 [2] |
| 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(14),3(8),4,6,15,17-hexaene-6,16-diol | Ki | 0.54 [1], 1.68 [2] |
| 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-5-ol | Ki | 37.5 [1], 42.3 [2] |
| 11-Ethyl-11,21-diazatetracyclo[12.7.0.03,8.015,20]henicosa-1(14),3,5,7,15,17,19-heptaene | Ki | 14.7 [1], 22.3 [2] |
| 1,1-Dioxo-2-[4-(4-phenylpiperazin-1-yl)butyl]-1,2-benzothiazol-3-one | Ki | 386.0 [1], 1629.0 [2] |
| 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-6-ol;hydrobromide | Ki | 1.5 [1], 1.69 [2] |
| 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3,5,7,14,16-hexaene-5,6-diol | Ki | 2.32 [1], 1078.0 [2] |
| Dopamine | Ki | 2440.0 [1] |
| Dopamine hydrochloride | Ki | 1023.29 [1] |
| Chlorpromazine | Ki | 172.0 [1] |
| Risperidone | Ki | 1000.0 [1] |
| Amitriptyline | Ki | 170.0 [1] |
| Quetiapine | Ki | 1000.0 [1] |
| Lysergide | Ki | 340.0 [1] |
| Fluphenazine | Ki | 21.0 [1] |
| 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine | Ki | 124.0 [1] |
| Maprotiline | Ki | 429.0 [1] |
| Ropinirole | Ki | 41211.0 [1] |
| Chlorprothixene | Ki | 9.0 [1] |
| Tetrahydropalmatine | Ki | 305.0 [1] |
| GR-127935 | Ki | 10000.0 [1] |
| Penfluridol | Ki | 125.0 [1] |
| Cariprazine | Ki | 7900.0 [1] |
| 3-((4-(4-Chlorophenyl)piperazin-1-yl)methyl)-1H-pyrrolo[2,3-b]pyridine | Ki | 10000.0 [1] |
| l-Stepholidine | Ki | 4.4 [1] |
| Cariprazine hydrochloride | IC50 | 1000.0 [1] |
| alpha-Methyltryptamine | Ki | 10000.0 [1] |
| 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide | IC50 | 10000.0 [1] |
| (S)-Canadine | Ki | 62.1 [1] |
| Phenyltoloxamine | Ki | 414.0 [1] |
| N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-9H-fluorene-2-carboxamide | Ki | 10000.0 [1] |
| 1H-3-Benzazepine-7,8-diol, 2,3,4,5-tetrahydro-1-phenyl-, (1R)- | Ki | 247.0 [1] |
| Benzonitrile, 3-fluoro-5-(2-(2-(fluoromethyl)-4-thiazolyl)ethynyl)- | Ki | 10000.0 [1] |
| Corydalmine | Ki | 242.0 [1] |
| N,N-Diallyl-5-methoxytryptamine | Ki | 10000.0 [1] |
| 3-(2-Aminopyrimidin-4-yl)-1H-indol-4-ol | Ki | 10000.0 [1] |
| N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide | Ki | 3700.0 [1] |
| (S)-Tetrahydrocolumbamine | Ki | 9.5 [1] |
| CID 11301655 | Ki | 8000.0 [1] |
| 6a,7,8,12b-Tetrahydro-6H-chromeno[3,4-c]isoquinoline-2,3-diol | Ki | 7.0 [1] |
| CID 11698643 | Ki | 939.0 [1] |
| Corypalmine | Ki | 313.0 [1] |
| Thalictruberine | Ki | 2397.0 [1] |
| N-[1-[(4-Iodophenyl)methyl]piperidin-4-yl]-N-methyl-3-propan-2-yloxypyridin-2-amine | Ki | 10000.0 [1] |
| 1,2,3,4,6,7,12,12b-Octahydroindolo[2,3-a]quinolizine | Ki | 10000.0 [1] |
| N-[2-(1H-Indol-3-yl)ethyl]-4-oxo-4-phenylbutanamide | Ki | 10000.0 [1] |
| N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]biphenylene-2-carboxamide | Ki | 10000.0 [1] |
| 1-(4-Fluorophenyl)-4-(thiophen-2-ylmethyl)piperazine | Ki | 2059.0 [1] |
| N-[(3S)-1-Benzylpyrrolidin-3-yl]-5-chloro-4-(cyclopropanecarbonylamino)-2-methoxybenzamide | Ki | 10000.0 [1] |
| 1-(2,3-Dihydro-1,4-benzodioxin-6-yl)-4-(2,3-dihydro-1H-inden-2-ylmethyl)piperazine | Ki | 3000.0 [1] |
| Tetrahydro-6-phenylpyran-2-one | Ki | 10000.0 [1] |
| 3-((2-Fluorothiazol-4-yl)ethynyl)-5-fluorobenzonitrile | Ki | 10000.0 [1] |
| 7-[4-[4-(2,3-Dichlorophenyl)-1,4-diazepan-1-yl]butoxy]-3,4-dihydro-1H-1,8-naphthyridin-2-one | Ki | 513.0 [1] |
| 1-(4-(4-Phenyl-1-piperazinyl)butyl)indolin-2-one | Ki | 330.0 [1] |
| (6-Chloro-1,3-benzodioxol-5-yl)methyl 3-[2-(methylamino)-2-oxoethyl]-4-oxo-1-phenyl-1,3,8-triazaspiro[4.5]decane-8-carboxylate | IC50 | 3660.0 [1] |
| (6-Chloro-1,3-benzodioxol-5-yl)methyl 4-(2-oxo-3H-benzimidazol-1-yl)piperidine-1-carboxylate | IC50 | 4890.0 [1] |
| 1-[3-(2-Benzyl-phenoxy)-propyl]-pyrrolidine | Ki | 113.0 [1] |
| 2-[4-[4-(7-(111C)Methoxynaphthalen-1-yl)piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dione | Ki | 10000.0 [1] |
| 2-[4-[4-(3-Methoxyphenyl)piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dione | Ki | 10000.0 [1] |
| 3-Methoxy-6,8,9,13b-tetrahydro-5H-isoquinolino[1,2-a]isoquinoline | Ki | 10000.0 [1] |
| 3-(4-Amino-2-bromo-pyrimidin-5-yl)-1H-indol-4-ol | Ki | 10000.0 [1] |
| 2-Chloro-N-[3-chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzodiazepin-11-yl]benzamide | Ki | 73.0 [1] |
| 4-Fluoro-N-methyl-N-(4-(6-(methylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl)benzamide | Ki | 10000.0 [1] |
| 17-Methoxy-11,21-dimethyl-11,21-diazatetracyclo[12.7.0.03,8.015,20]henicosa-1(14),3,5,7,15(20),16,18-heptaene | Ki | 0.23 [1] |
| 11-Methyl-11-azatricyclo[13.4.0.03,8]nonadeca-1(19),3(8),4,6,15,17-hexaen-6-ol | Ki | 9.8 [1] |
| 17-Methoxy-11-methyl-11-azatricyclo[13.4.0.03,8]nonadeca-1(15),3,5,7,16,18-hexaene | Ki | 55.0 [1] |
| 6-Methoxy-11-methyl-11-azatricyclo[13.4.0.03,8]nonadeca-1(19),3(8),4,6,15,17-hexaene | Ki | 4.6 [1] |
| 1-[3-(p-Fluorophenoxy)-propyl]-4-(p-chlorophenyl)-4-hydroxypiperidine | Ki | 103.0 [1] |
| 4-(4-Chlorophenyl)-1-[3-[(4-fluorophenyl)thio]propyl]-4-piperidinol | Ki | 113.0 [1] |
| 1-Benzyl-4-(2-ethoxyphenyl)piperazine | Ki | 10000.0 [1] |
| 3-(4-(4-Phenyl-1-piperazinyl)butyl)quinazolin-4(3H)-one | Ki | 10000.0 [1] |
| (1S)-16-Methoxy-5,7-dioxa-13-azapentacyclo[11.8.0.02,10.04,8.015,20]henicosa-2,4(8),9,15(20),16,18-hexaen-17-ol | Ki | 15.1 [1] |
| 1-[3-(4-Fluorophenoxy)propyl]-4-pyridin-2-ylpiperazine | Ki | 2392.0 [1] |
| 1-[4-(4-Fluorophenyl)butyl]-4-pyridin-2-ylpiperazine | Ki | 1451.0 [1] |