 | (R)-2,3,4,5-Tetrahydro-8-chloro-3-methyl-5-phenyl-1H-3-benzazepin-7-ol | IC50 | 0.66 [1], 0.74 [2], 0.82 [3], 1.4 [4], 520.0 [5] |
| (R)-2,3,4,5-Tetrahydro-8-chloro-3-methyl-5-phenyl-1H-3-benzazepin-7-ol | Ki | 0.15 [1] |
 | Haloperidol | Ki | 107.0 [1] |
 | 7-Methyl-6,7,8,9,14,15-hexahydro-5H-benz[d]indolo[2,3-g]azecine | Ki | 60.4 [1] |
 | Sch-23390 maleate | IC50 | 0.22 [1], 0.27 [2], 1.7 [3], 30.0 [4] |
| Sch-23390 maleate | Ki | 0.1 [1] |
 | 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-6-ol | Ki | 1.35 [1] |
 | (13As)-3,9,11-trimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-2-ol | IC50 | 9.85 [1], 1380.0 [2], 1400.0 [3] |
| (13As)-3,9,11-trimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-2-ol | Ki | 2.5 [1], 2.53 [2] |
 | Quetiapine | Ki | 214.6 [1], 390.0 [2], 1000.0 [3], 1300.0 [4], 4240.0 [5] |
 | 7-Chloro-3-methyl-1-phenyl-1,2,4,5-tetrahydro-3-benzazepin-8-ol | IC50 | 0.31 [1], 2.52 [2], 740.0 [3] |
| 7-Chloro-3-methyl-1-phenyl-1,2,4,5-tetrahydro-3-benzazepin-8-ol | Ki | 1.2 [1] |
 | l-Stepholidine | Ki | 3.4 [1], 5.9 [2], 6.23 [3], 12.29 [4] |
 | (+)-Dihydrexidine | Ki | 6.2 [1], 33.0 [2], 35.7 [3], 1200.0 [4] |
 | 1H-3-Benzazepine-7,8-diol, 2,3,4,5-tetrahydro-1-phenyl-, (1R)- | Ki | 5.1 [1], 56.0 [2], 73.0 [3], 130.0 [4], 320.0 [5] |
 | 6-Methoxy-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaene | Ki | 22.91 [1], 24.1 [2], 28.5 [3] |
 | 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3,5,7,14,16-hexaene | Ki | 3.47 [1], 4.5 [2], 40.4 [3] |
 | Ecopipam | Ki | 1.2 [1], 1.9 [2] |
 | (13As)-3-methoxy-9,11-dimethyl-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-2-ol | IC50 | 56.37 [1] |
| (13As)-3-methoxy-9,11-dimethyl-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-2-ol | Ki | 28.9 [1], 28.91 [2] |
 | Ziprasidone | Ki | 9.5 [1], 130.0 [2], 330.0 [3] |
 | 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine | Ki | 190.0 [1], 393.0 [2] |
 | N-Propylnorapomorphine | Ki | 1.0 [1], 490.0 [2], 1510.0 [3] |
 | (6Ar)-6-propyl-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-11-ol | Ki | 45.0 [1], 4300.0 [2], 10000.0 [3] |
 | 7-Chloro-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-6-ol | Ki | 0.46 [1], 0.81 [2], 0.83 [3] |
 | 12-Methyl-12,22-diazatetracyclo[13.7.0.03,8.016,21]docosa-1(15),3,5,7,16,18,20-heptaene | Ki | 2.04 [1], 2.2 [2], 2.8 [3] |
 | 11-Methyl-11,22-diazatetracyclo[13.7.0.03,8.016,21]docosa-1(15),3,5,7,16,18,20-heptaene | Ki | 158.49 [1], 163.5 [2], 304.0 [3] |
 | 10-Methyl-6-thia-10-azatricyclo[11.4.0.03,7]heptadeca-1(17),3(7),4,13,15-pentaene | Ki | 4.0 [1], 10.7 [2], 207.0 [3] |
 | (1S)-16,18-Dimethoxy-5,7-dioxa-13-azapentacyclo[11.8.0.02,10.04,8.015,20]henicosa-2,4(8),9,15(20),16,18-hexaene | IC50 | 141.58 [1] |
| (1S)-16,18-Dimethoxy-5,7-dioxa-13-azapentacyclo[11.8.0.02,10.04,8.015,20]henicosa-2,4(8),9,15(20),16,18-hexaene | Ki | 64.12 [1], 74.51 [2] |
 | (13As)-3,9,12-trimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-2-ol | IC50 | 7.22 [1], 1900.0 [2] |
| (13As)-3,9,12-trimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-2-ol | Ki | 3.7 [1] |
 | Chlorpromazine | Ki | 96.0 [1], 112.0 [2] |
 | Amitriptyline | Ki | 89.0 [1], 178.0 [2] |
 | Fluphenazine | Ki | 11.0 [1], 179.0 [2] |
 | Pergolide | Ki | 339.0 [1], 2020.0 [2] |
 | Maprotiline | Ki | 187.0 [1], 402.0 [2] |
 | Lisuride | Ki | 77.0 [1], 86.0 [2] |
 | Tetrahydropalmatine | Ki | 153.0 [1], 231.0 [2] |
 | Zotepine | Ki | 29.0 [1], 84.0 [2] |
 | GR-127935 | Ki | 10000.0 [1] |
 | Cariprazine | Ki | 2100.0 [1] |
 | 3-Methyl-6-chloro-2,3,4,5-tetrahydro-7,8-dihydroxy-1-(3-methylphenyl)-1H-3-benzazepine | Ki | 1.18 [1], 1.93 [2] |
 | 2-Naphthalenecarboxamide, N-(4-(4-(2-methoxyphenyl)-1-piperazinyl)butyl)- | Ki | 760.0 [1] |
 | 5-(4-Chlorophenyl)-N-(3,5-dimethoxyphenyl)furan-2-carboxamide | IC50 | 2000.0 [1], 7000.0 [2] |
 | (S)-Canadine | Ki | 48.6 [1], 66.0 [2] |
 | 4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochloride | IC50 | 10000.0 [1] |
| 4-Amino-5-chloro-N-((hexahydro-1H-pyrrolizin-1-yl)methyl)-2-methoxybenzamide hydrochloride | Ki | 10000.0 [1] |
 | N-[4-[4-(2,3-Dichlorophenyl)piperazin-1-yl]butyl]-1-benzothiophene-2-carboxamide | Ki | 1195.0 [1], 8800.0 [2] |
 | Di-deacetyl adrogolide | Ki | 49.0 [1] |
 | Corydalmine | Ki | 50.0 [1], 107.0 [2] |
 | N-[4-[4-(2-Methoxyphenyl)piperazin-1-yl]butyl]pyrazolo[1,5-a]pyridine-2-carboxamide | Ki | 1500.0 [1], 1600.0 [2] |
 | N-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)benzo[b]thiophene-2-carboxamide | Ki | 670.0 [1], 800.0 [2] |
 | (S)-Tetrahydrocolumbamine | Ki | 4.5 [1], 6.2 [2] |
 | 2-Methoxy-N-n-propylnorapomorphine | Ki | 8.1 [1], 5000.0 [2] |
 | N-(4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide | Ki | 1100.0 [1], 2000.0 [2] |
 | Corypalmine | Ki | 199.0 [1], 310.0 [2] |
 | N-(4-(4-(2,3-Dichlorophenyl)piperazin-1-yl)butyl)benzofuran-2-carboxamide | Ki | 2100.0 [1], 2900.0 [2] |
 | 7-[4-[4-(2,3-Dichlorophenyl)-1,4-diazepan-1-yl]butoxy]-3,4-dihydro-1H-quinolin-2-one | Ki | 340.0 [1], 825.0 [2] |
 | (6S)-6-[2-Phenylethyl(propyl)amino]-5,6,7,8-tetrahydronaphthalen-1-ol | Ki | 230.0 [1], 1200.0 [2] |
 | 5-[2-[4-(2,3-Dimethylphenyl)piperazin-1-yl]ethyl]-2H-benzotriazole | Ki | 4677.35 [1] |
 | (1R,11S)-5-Chloro-10-methyl-10-azatetracyclo[9.7.0.02,7.013,18]octadeca-2,4,6,13,15,17-hexaen-4-ol | Ki | 7.0 [1] |
 | 2-Chloro-N-[3-chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzodiazepin-11-yl]benzamide | Ki | 4.0 [1], 4.1 [2] |
 | 11-Methyl-11-azatricyclo[13.4.0.03,8]nonadeca-1(19),3(8),4,6,15,17-hexaen-6-ol | Ki | 2.67 [1], 3.2 [2] |
 | 17-Methoxy-11-methyl-11-azatricyclo[13.4.0.03,8]nonadeca-1(15),3,5,7,16,18-hexaene | Ki | 28.18 [1], 29.4 [2] |
 | 6-Methoxy-11-methyl-11-azatricyclo[13.4.0.03,8]nonadeca-1(19),3(8),4,6,15,17-hexaene | Ki | 18.5 [1], 21.88 [2] |
 | 5'-Chloro-N,N-dimethylspiro[cyclohex-2-ene-4,2'-tricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,9,11,13-heptaene]-1-amine | Ki | 0.3 [1], 3.1 [2] |
 | (1S)-16-Methoxy-5,7-dioxa-13-azapentacyclo[11.8.0.02,10.04,8.015,20]henicosa-2,4(8),9,15(20),16,18-hexaen-17-ol | Ki | 6.3 [1], 6.5 [2] |
 | 10-[2-[(2R)-1-Methylpiperidin-2-yl]ethyl]-2-methylsulfinylphenothiazine | IC50 | 137.0 [1] |
| 10-[2-[(2R)-1-Methylpiperidin-2-yl]ethyl]-2-methylsulfinylphenothiazine | Ki | 103.0 [1] |
 | N-[3-Chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzodiazepin-11-yl]-4-methoxybenzamide | Ki | 47.0 [1] |
 | N-[3-Chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzodiazepin-11-yl]benzamide | Ki | 157.0 [1] |
 | N-[3-Chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzodiazepin-11-yl]-2,6-dimethoxybenzamide | Ki | 1.6 [1] |
 | N-[3-Chloro-6-(4-methylpiperazin-1-yl)benzo[b][1,4]benzodiazepin-11-yl]-2,6-dimethylbenzamide | Ki | 3.0 [1] |
 | 11-Methyl-11,21-diazatetracyclo[12.7.0.03,8.015,20]henicosa-1(14),3,5,7,15(20),16,18-heptaen-17-ol | Ki | 0.56 [1] |
 | (4As,5R,10bR)-5-phenyl-1,2,3,4,4a,5,6,10b-octahydrobenzo[h]isoquinoline-7,8-diol | Ki | 47.0 [1], 18000.0 [2] |
 | 2-[[(2R)-2-Phenethylmorpholino]methyl]-1H-benzoimidazole | IC50 | 100000.0 [1] |
| 2-[[(2R)-2-Phenethylmorpholino]methyl]-1H-benzoimidazole | Ki | 100000.0 [1] |
 | (13As)-3,11-dimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-2-ol | Ki | 35.79 [1], 35.8 [2] |
 | (13As)-12-(hydroxymethyl)-3,9,11-trimethoxy-6,8,13,13a-tetrahydro-5H-isoquinolino[2,1-b]isoquinolin-2-ol | Ki | 17.29 [1], 17.3 [2] |
 | 6,10-Dimethyl-6,10-diazatricyclo[11.4.0.03,7]heptadeca-1(17),3(7),4,13,15-pentaene | Ki | 61.0 [1], 1000.0 [2] |
 | 4-[2-(1H-Benzotriazol-5-yl)ethyl]-1-(2-methoxyphenyl)piperazine | Ki | 812.83 [1] |
 | 4-[2-(1H-Benzotriazol-5-yl)ethyl]-1-(1-naphthyl)piperazine | Ki | 5754.4 [1] |
 | 5,7-Dichloro-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3,5,7,14,16-hexaen-6-ol | Ki | 3.2 [1], 3.8 [2] |
 | 5-Methoxy-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaene | Ki | 82.0 [1], 567.0 [2] |
 | 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-4-ol | Ki | 8.7 [1], 64.1 [2] |
 | 4-Methoxy-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaene | Ki | 7.6 [1], 37.6 [2] |
 | 5-Amino-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3,5,7,14,16-hexaen-6-ol | Ki | 9.3 [1], 20.9 [2] |
 | 6-Chloro-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3,5,7,14,16-hexaen-5-ol | Ki | 3.1 [1], 10.8 [2] |
 | 6,16-Dimethoxy-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(14),3(8),4,6,15,17-hexaene | Ki | 9.4 [1], 26.9 [2] |
 | 4-Chloro-11-methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-5-ol | Ki | 0.46 [1], 6.8 [2] |
 | 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(14),3(8),4,6,15,17-hexaene-6,16-diol | Ki | 2.0 [1], 3.3 [2] |
 | 11-Methyl-11-azatricyclo[12.4.0.03,8]octadeca-1(18),3(8),4,6,14,16-hexaen-5-ol | Ki | 2.6 [1], 8.9 [2] |
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