![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_c1303ad3101dce1e315ea55e799cd202.svg) | Etoposide | IC50 | 56000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_98a04b67a851c3bf4ca1fd9476597cf5.svg) | Doxorubicin | IC50 | 880.0 [1], 1000.0 [2], 3000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_fc414cacc72e2ed688da77f786d8de1f.svg) | Merbarone | IC50 | 32000.0 [1], 40000.0 [2], 120000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_2a3ab5989d8438a1e7cd0ac6ebb13d7d.svg) | 3-[(E)-4-Hydroxybenzylidene]-6-hydroxybenzofuran-2(3H)-one | IC50 | 400000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_acc869bf5b76dce971037f71afa3bf1c.svg) | 3-[3-[3-(4-Aminobutylamino)propylamino]-2-hydroxypropoxy]-1-hydroxyxanthen-9-one;2,2,2-trifluoroacetic acid | IC50 | 2500.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_1816df2dc49c11e622026cae2c8dc356.svg) | Camptothecin | IC50 | 300000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_f10d31b59c64b652ca2647081c7ffe43.svg) | Methyl 2'-(2-hydroxyphenyl)-(2,4'-bibenzoxazole)-4-carboxylate | IC50 | 32000.0 [1], 50000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_d0c8a71a5f3f48badd0d5657b46fafef.svg) | Topostatin | IC50 | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_62421dcdcf9705f1ef1c538db9e63b6b.svg) | 6-Chloro-14-[2-[2-hydroxyethyl(methyl)amino]ethyl]-14,15-diazatetracyclo[7.6.1.02,7.013,16]hexadeca-1(15),2(7),3,5,9(16),10,12-heptaen-8-one | IC50 | 7200.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_2fcfcd937657b1868746614fa0e93d8c.svg) | 1-[(2R,4S,5S)-5-[[Tert-butyl(dimethyl)silyl]oxymethyl]-4-[2-(3,4-dimethoxyphenyl)-1,3-dithian-2-yl]oxolan-2-yl]-5-methylpyrimidine-2,4-dione | IC50 | 8100.0 [1], 19100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_e27619235281d6093e5049d0804cb3a1.svg) | 4-[3-(Tert-Butylamino)imidazo[1,2-a]pyridine-2-yl]benzoic acid | IC50 | 52660.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_e27619235281d6093e5049d0804cb3a1.svg) | 4-[3-(Tert-Butylamino)imidazo[1,2-a]pyridine-2-yl]benzoic acid | Ki | 75000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_28737c7de0737e548547284a3a5402a4.svg) | 3-[3-(Butylamino)-2-hydroxypropoxy]-1-hydroxyxanthen-9-one | IC50 | 9000.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_8e925918740657eb46152966681bbb5f.svg) | 6-Amino-7-(1H-benzimidazol-2-yl)-5-[4-(dimethylamino)butyl]pyrrolo[2,3-b]pyrazine-2,3-dicarbonitrile | IC50 | 900.0 [1], 16500.0 [2] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_82002b165b2dabb5aad18f17908b3c07.svg) | 2-[4-(1,3-Benzoxazol-2-yl)-1,3-benzoxazol-2-yl]phenol | IC50 | 20000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_41399b75fff6cc36d8a967f8d44f4161.svg) | 3-[3-[3-[4-(3-Aminopropylamino)butylamino]propylamino]-2-hydroxypropoxy]-1-hydroxyxanthen-9-one;tetrahydrochloride | IC50 | 1000.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_15976e9843386a991246a922e8b855ad.svg) | Ciprofloxacin | IC50 | 256000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_53f760ea7e3000ebe6c3039afb4e3733.svg) | Spermine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_48579a303d998b0dc4f0d4b548fef913.svg) | Spermidine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_926035c06d9d341c1f456b3b189f3e17.svg) | Mitoxantrone | IC50 | 5300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_da5136da44515a73895b9fa711d3d6a4.svg) | Novobiocin | IC50 | 256000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_e4b95cfb6ae5b332d20673553d0a4833.svg) | Pibenzimol | IC50 | 28920.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_e25c9d2f82c5eda0b783aad009b4d224.svg) | Myricetin | IC50 | 390.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_07992946abda58514c65c68057ac00b7.svg) | Amsacrine | IC50 | 9940.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_1bfbaa18e3d29ff3836441853c767b54.svg) | Lupeol | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_3609fc3031c075e99b2a994d4c0a33b2.svg) | Ellipticine | IC50 | 3300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_419927d6fcebf01d0c36867edf5cb8bd.svg) | Ginsenoside rb1 | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_9ebd760982b58afe3bd72607ffec4a4f.svg) | Ginsenoside Rg3 | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_ac539ec1473267b3ea601e275753ac34.svg) | (1E,4Z,6E)-5-Hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one | IC50 | 15000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_713e666d1bf021e529e44920ca8b248a.svg) | 4,4'-(1,2-Dimethyl-1,2-ethanediyl)bis-2,6-piperazinedione | IC50 | 13900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_a488830c3ad35bcbad36e099ebc05a4b.svg) | Ginsenoside Re | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_fa5912ee40422074d089d53a997b7111.svg) | Gypenoside VIII | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_8f6c88ca778074869b46bffcb66852a2.svg) | alpha-Amyrin | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_e451cf08622b1140f6bb3d4a9219b729.svg) | Piroxantrone | IC50 | 4600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_f5c318e223e6f756c5e892b9863851e4.svg) | Losoxantrone | IC50 | 7300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_a264e3d54afb17928bcece90068391c7.svg) | Ginsenoside F2 | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_5b06b24da7a22932194db7fc6403b9cf.svg) | Ascididemin | IC50 | 1376.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_1351a848213aef394896b44405abc45d.svg) | 2-Pyridinecarboxaldehyde thiosemicarbazone | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_8464f2ab2fd3fadfc159225b17ac4491.svg) | N-[(Benzyloxy)carbonyl]-L-aspartic acid | IC50 | 26950.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_74b470319dd9a8bc1aad5a90379591ce.svg) | 1,3-Dihydroxy-9H-xanthen-9-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_429c760b0cb6e5d680a0c024d73265e1.svg) | Ganoderiol F | IC50 | 17000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_274d3e2cb9d813d3af159602adda1f3a.svg) | Mansonone E | IC50 | 18600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_063445299090c50226c4d70b0b62461b.svg) | Olivetolic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_8f276e6d77009dee9ec3023d2b896fb2.svg) | (20R)-Ginsenoside Rg3 | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_e33f671cca88f6e7d0dc8a4179853c6b.svg) | 4-Methyl-1-(1-(2-pyridyl)ethylidene)-3-thiosemicarbazide | IC50 | 92000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_0c975f2c6bd3261735e7b909db02d33d.svg) | Unii-W6V49A8fjq | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_a0c463a27aac6d1df0f56afea78c4a1e.svg) | {4-Amino-6-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}methyl morpholine-4-carbodithioate | IC50 | 229000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_ac0500a6806603b4ba5fc9fc67f2dc8f.svg) | 5,7-Dioxa-12-azoniapentacyclo[10.6.1.02,10.04,8.015,19]nonadeca-1(18),2,4(8),9,11,15(19),16-heptaen-17-olate | IC50 | 25800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_d270cf63ecc93463628d319f03066778.svg) | 4-Allyl-1-(1-(2-pyridyl)ethylidene)-3-thio-semicarbazide | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_ed2163d5042e8d4dd8553d74abef40d7.svg) | Gypenoside XVII | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_ff7763fa932bd8362e34a5013e8eafa7.svg) | {4-Amino-6-[(4-fluorophenyl)amino]-1,3,5-triazin-2-yl}methyl 4-methylpiperazine-1-carbodithioate | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_322d66ad34b3d7a64a35ee92623041de.svg) | {4-Amino-6-[(4-methoxyphenyl)amino]-1,3,5-triazin-2-yl}methyl piperidine-1-carbodithioate | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_2203ecd79760bdeacdb99b79b63ea8e8.svg) | {4-Amino-6-[(4-fluorophenyl)amino]-1,3,5-triazin-2-yl}methyl morpholine-4-carbodithioate | IC50 | 139000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_b1c712f2162e1d8b65f757dc495da6ef.svg) | N-[[4-(3,4-Dichlorophenyl)-5-sulfanylidene-1H-1,2,4-triazol-3-yl]methyl]-3-methoxybenzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_2a5632354e0d74598ad8e2837ee6c3f2.svg) | N-Cyclohexyl-[1,2,4]triazolo[4,3-a]quinoxalin-4-amine | IC50 | 680.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_5d3455a39368409e8cda7d4eed2d0fef.svg) | Demethylzeylasterone | IC50 | 17600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_fe03cb346064924ad1ddb5274c2c1f0c.svg) | Kaempferol 3-O-beta-D-glucopyranosyl-7-O-alpha-L-rhamnopyranoside | IC50 | 600000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_063920cd305f9707fac4a2de9ac876be.svg) | 6-Phenyl-4-sulfanylidene-1H-1,3,5-triazin-2-one | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_733338340740c909a0ff912244476907.svg) | Bakuchicin | IC50 | 404000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_78593ef995750090730d8c001205aa6f.svg) | Dehydrotrametenonic acid | IC50 | 37500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_519bfaecd3d1a706e11cec8927c15d97.svg) | Ginsenoside F3 | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_9a353ffc7d7b96ebae585d4a496c56d6.svg) | 1-Methyl-3-[(E)-1-pyrazin-2-ylethylideneamino]thiourea | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_30f2e68f51af5e4052affc53bcbbac99.svg) | 6-(4-Methylpiperazin-1-yl)-2-[2-(4-prop-2-ynoxyphenyl)-3H-benzimidazol-5-yl]-1H-benzimidazole | IC50 | 51600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_81698274800470f5b1e17678c62cd508.svg) | 4-Ethyl-1-(1-(2-pyridyl)ethylidene)-3-thiosemicarbazide | IC50 | 79000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_5e93d6fc2f108b865761d74917c2df30.svg) | 6-Phenethylsulfanyl-7H-purin-2-amine | IC50 | 85000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_b8febd9ef4bf0e4c18397dc6bfbf210b.svg) | N2-(2-(Diethylamino)ethyl)-N9-phenylthiazolo[5,4-b]quinoline-2,9-diamine | IC50 | 168900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_d65ce65c0d82c0b01b4643b3b04e5069.svg) | Bengacarboline | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_e4bb0012f940ec8673f5ce731b8ba487.svg) | 6-Methyl-5-methylidene-2-[(5R,10S,13R,14R,17R)-4,4,10,13,14-pentamethyl-3-oxo-1,2,5,6,12,15,16,17-octahydrocyclopenta[a]phenanthren-17-yl]heptanoic acid | IC50 | 4600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_1a9928a2116a6686083b6cdbeacfc944.svg) | Anziaic acid | IC50 | 35000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_f82e7e8c0e7bd8fa3d588715b1479dbe.svg) | (2R,3S,4S,5R,6S)-2-[[(2S,3S,4S,5R)-3,4-Dihydroxy-5-(hydroxymethyl)oxolan-2-yl]oxymethyl]-6-[(2S)-6-methyl-2-[(3S,5R,6S,8R,9R,10R,12R,13R,14R,17S)-3,6,12-trihydroxy-4,4,8,10,14-pentamethyl-2,3,5,6,7,9,11,12,13,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-17-yl]hept-5-en-2-yl]oxyoxane-3,4,5-triol | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_a5c15013ad37d1297a5a94a8ba46ef15.svg) | 1-Benzyl-3-[(E)-2-pyridylmethyleneamino]thiourea | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_84a76465ccdb8e87fec89719b3bed36d.svg) | (E,6R)-6-[(3S,5R,10S,13R,14R,15S,17R)-15-Acetyloxy-3-hydroxy-4,4,10,13,14-pentamethyl-2,3,5,6,12,15,16,17-octahydro-1H-cyclopenta[a]phenanthren-17-yl]-2-methylhept-2-enoic acid | IC50 | 25000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_87982ba23af3b670d9f360420900675e.svg) | N-(3-(2-(Methylthio)thiazolo[5,4-b]quinolin-9-ylamino)phenyl)acetamide | IC50 | 29560.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_06fd052a637794d2cc714d8954402522.svg) | 4,6-Dichloro-[1,3,5]triazin-2-yl-4-methoxy-benzyl-amine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_40c3818dffdcb57483f5c6531452eafa.svg) | N1-(2-(Methylthio)thiazolo[5,4-b]quinolin-9-yl)benzene-1,3-diamine | IC50 | 16740.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_480a4cbf14009e7759e9fc71a25660f3.svg) | (3-Amino-5-(2-(methylthio)thiazolo[5,4-b]quinolin-9-ylamino)phenyl)methanol | IC50 | 18040.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_96ab335c33239674dad49aa5ada20630.svg) | (3E)-3-[(3-Hydroxy-4-methoxyphenyl)methylidene]-1-benzofuran-2-one | IC50 | 400000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_484730d839f3bd0057de0ef42fea333f.svg) | Indeno[1,2-c]cinnolin-11-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_709706f16b7d8901f1d0522b1c8dc7f2.svg) | 6-(4-Methylphenyl)-4-sulfanylidene-1H-1,3,5-triazin-2-one | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_f6bf51b1014364fd5f43312a450aab71.svg) | 20(S)-Ginsenoside Rg2 | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_a6fb9372b78a9add80ea56c9890b86a9.svg) | 4-Methylamino-[1,2,4]triazolo[4,3-a]quinoxaline | IC50 | 2090.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_07a8490d2c41737dda5ad9e19567b446.svg) | 5-[3-(Dimethylamino)propyl]quinolino[4,3-b]quinoxalin-6-one | IC50 | 100000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_ca09564297ed13459ab0d23a0a1e14f2.svg) | Quinovic acid 3-O-beta-D-glucoside | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_929a2f501b505b38904f88fe403e4b7f.svg) | (1S,2R,4As,6aR,6aR,6bR,8aR,10S,12aR,14bS)-1,2,6b,9,9,12a-hexamethyl-10-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-4a-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxycarbonyl-2,3,4,5,6,6a,7,8,8a,10,11,12,13,14b-tetradecahydro-1H-picene-6a-carboxylic acid | IC50 | 250000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_df189e9f02a15efb85ffc0d75049bf14.svg) | Bis[2-[2-(6-chloro-8-oxo-14,15-diazatetracyclo[7.6.1.02,7.013,16]hexadeca-1(15),2(7),3,5,9(16),10,12-heptaen-14-yl)ethyl-methylamino]ethyl] pentanedioate | IC50 | 32000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_7fa53f5744d0bbc9b0786f19a2cbe860.svg) | N-(2-Ethylphenyl)-2-amino-4,6-dichloro-1,3,5-triazine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_5f5e497593a8ca65cff56be27bd60338.svg) | (3E)-3-[(4-Methoxyphenyl)methylidene]-1-benzofuran-2-one | IC50 | 400000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_69c5832b583ae1df543e2a006d538f77.svg) | N,N'-Bis[2-[2-(6-chloro-8-oxo-14,15-diazatetracyclo[7.6.1.02,7.013,16]hexadeca-1(15),2(7),3,5,9(16),10,12-heptaen-14-yl)ethyl-methylamino]ethyl]heptanediamide | IC50 | 22000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_3c9f46809d4b8b4cd9243ba28f893809.svg) | N-(2-Bromophenyl)-4,6-dichloro-1,3,5-triazin-2-amine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_ebf43a344f2052e72c5d11cea050bdf5.svg) | 18-[(3S)-3-Aminopyrrolidin-1-yl]-19-fluoro-22-oxo-16-oxa-1-azahexacyclo[15.7.1.02,15.05,14.06,11.021,25]pentacosa-2(15),3,5(14),6,8,10,12,17(25),18,20,23-undecaene-23-carboxylic acid | IC50 | 700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_04436fa44301f581e324eba625a913f9.svg) | 18-[(3R)-3-Aminopyrrolidin-1-yl]-19-fluoro-22-oxo-16-oxa-1-azahexacyclo[15.7.1.02,15.05,14.06,11.021,25]pentacosa-2(15),3,5(14),6,8,10,12,17(25),18,20,23-undecaene-23-carboxylic acid | IC50 | 60.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_5e42042e7513de7b358ca9909e050825.svg) | 2-(4,6-Dimethoxy-1,3,5-triazine-2-yloxy)benzoic acid methyl ester | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_e356be74ecbb0da1d511862599aebcc5.svg) | N-[(4-Phenyl-5-sulfanylidene-1H-1,2,4-triazol-3-yl)methyl]-2-(trifluoromethyl)benzamide | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_6401eaf7e24d67d20ef570d88a57ee5d.svg) | 3-[(E)-4-Hydroxybenzylidene]benzofuran-2(3H)-one | IC50 | 327000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_6042807b34bde6aae3ddeed65baeb3e2.svg) | 9-[[(4-Chloro)phenyl]amino]-2-(methylthio)thiazolo[5,4-b]quinoline | IC50 | 20490.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_5af84fc43de4196269e3f7b33821eecf.svg) | 9-[[(3-N-Methylamino)phenyl]amino]-2-(methylthio)-thiazolo[5,4-b]quinoline | IC50 | 12270.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_0105b1efce229ae87a21732045b5e958.svg) | 3-(2-(Methylthio)thiazolo[5,4-b]quinolin-9-ylamino)phenol | IC50 | 64340.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_ae5233e50f8ac5db0f8b7b37695c1ffe.svg) | 2-Methylsulfanyl-N-[3-(trifluoromethyl)phenyl]-[1,3]thiazolo[5,4-b]quinolin-9-amine | IC50 | 15420.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_a8bcac8dd3094a3a6484561c0e46d186.svg) | 9-[[(3-Chloro)phenyl]amino]-2-(methylthio)thiazolo[5,4-b]quinoline | IC50 | 21200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/dna-topoisomerase-ii-alpha_7742e4174a4c0ded18b963552a7da6d3.svg) | 9-N-(3-Chlorophenyl)-2-N-[3-(diethylamino)propyl]-[1,3]thiazolo[5,4-b]quinoline-2,9-diamine | IC50 | 40950.0 [1] |