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Disintegrin and metalloproteinase domain-containing protein 8 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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Unii-Q56UE7E40YIC501000.0 [1]
2-[(2S,5S,8S,11S,14S)-2,8-Bis(4-aminobutyl)-14-butyl-11-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50378.0 [1]
2-[(2S,5S,8S,11S,14S)-2,8-Bis(4-aminobutyl)-11-[3-(diaminomethylideneamino)propyl]-3,6,9,12,15,19-hexaoxo-14-propyl-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50452.0 [1]
2-[(2S,5S,8S,11S,14S)-2-(4-Aminobutyl)-8-(aminomethyl)-11-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC505000.0 [1]
2-[(2S,5S,8S,11S,14S)-2-(4-Aminobutyl)-8-(2-aminoethyl)-11-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC505000.0 [1]
2-[(2S,5S,8S,11S,14S,17R)-2,8-Bis(4-aminobutyl)-11-[3-(diaminomethylideneamino)propyl]-17-(hydroxymethyl)-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50157.0 [1]
2-[(2S,5S,8S,11S,14S)-2,8-Bis(4-aminobutyl)-11-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC501645.0 [1]
(2S,5S,8S,11S,14S,17S)-2,8-Bis(4-aminobutyl)-5-(carboxymethyl)-11-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadecane-17-carboxylic acidIC50420.0 [1]
2-[(2S,5S,8S,11S,14S)-2,8-Bis(4-aminobutyl)-11-[3-[[amino(nitramido)methylidene]amino]propyl]-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC502345.0 [1]
2-[(2S,5S,8S,11S,14S)-2,8-Bis(4-aminobutyl)-11-[3-(carbamoylamino)propyl]-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50890.0 [1]
2-[(2S,5S,8S,11S,14S,17R)-2,8-Bis(4-aminobutyl)-11-[3-(carbamoylamino)propyl]-17-(hydroxymethyl)-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50192.0 [1]
2-[(2S,5S,8S,11S,14S,17R)-2,8-Bis(4-aminobutyl)-11-[4-(diaminomethylideneamino)butyl]-17-(hydroxymethyl)-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50368.0 [1]
2-[(2S,5S,8S,11S,14S)-2,8-Bis(4-aminobutyl)-11-[3-(diaminomethylideneamino)propyl]-14-(2,2-dimethylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50256.0 [1]
2-[(2S,5S,8S,11S,14S)-2,8-Bis(4-aminobutyl)-11-[3-(diaminomethylideneamino)propyl]-14-(3-methylbutyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50220.0 [1]
2-[(2S,5S,8S,11S,14S,17R)-2,8-Bis(4-aminobutyl)-11-[3-(diaminomethylideneamino)propyl]-17-(hydroxymethyl)-14-(3-methylbutyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC50142.0 [1]
2-[(2S,5S,8S,11S,14R,17S)-5,17-Bis(4-aminobutyl)-8-[3-(diaminomethylideneamino)propyl]-14-(hydroxymethyl)-11-(2-methylpropyl)-3,6,9,12,15,18-hexaoxo-1,4,7,10,13,16-hexazacyclooctadec-2-yl]acetic acidIC50182.0 [1]
2-[(2S,5S,8S,11S,14S)-2-(4-Aminobutyl)-8-(3-aminopropyl)-11-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC505000.0 [1]
4-[(2S,5S,8S,11S,14S)-2-(4-Aminobutyl)-5-(carboxymethyl)-11-[3-(diaminomethylideneamino)propyl]-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-8-yl]butyl-trimethylazaniumIC5010000.0 [1]
2-[(2S,5S,8S,11S,14S,17R)-2,8-Bis(4-aminobutyl)-11-[3-[[amino(nitramido)methylidene]amino]propyl]-17-(hydroxymethyl)-14-(2-methylpropyl)-3,6,9,12,15,19-hexaoxo-1,4,7,10,13,16-hexazacyclononadec-5-yl]acetic acidIC501245.0 [1]
2-[(2S,5S,8S,11S,14S,17S)-5,17-Bis(4-aminobutyl)-8-[3-(diaminomethylideneamino)propyl]-14-(hydroxymethyl)-11-(2-methylpropyl)-3,6,9,12,15,18-hexaoxo-1,4,7,10,13,16-hexazacyclooctadec-2-yl]acetic acidIC50240.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Disintegrin and metalloproteinase domain-containing protein 8 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/disintegrin-and-metalloproteinase-domain-containing-protein-8-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Disintegrin and metalloproteinase domain-containing protein 8 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/disintegrin-and-metalloproteinase-domain-containing-protein-8-inhibitors-ic50-ki.
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