Death-associated protein kinase 1 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Staurosporine	IC50	0.5 [1], 9.4 [2], 13.08 [3]
	Morin	IC50	1600.0 [1], 11000.0 [2]
	Quercetin	IC50	8900.0 [1]
	Cianidanol	IC50	300000.0 [1]
	Genistein	IC50	98000.0 [1]
	Apigenin	IC50	31000.0 [1]
	Kaempferol	IC50	10000.0 [1]
	Luteolin	IC50	21000.0 [1]
	Baicalein	IC50	120000.0 [1]
	Myricetin	IC50	23000.0 [1]
	Chrysin	IC50	300000.0 [1]
	Cyanidin	IC50	150000.0 [1]
	(-)-Epicatechin gallate	IC50	300000.0 [1]
	Pelargonidin	IC50	220000.0 [1]
	Doramapimod	IC50	30000.0 [1]
	Gossypetin	IC50	87000.0 [1]
	Sulfuretin	IC50	13150.0 [1]
	3',4',7-Trihydroxyisoflavone	IC50	280000.0 [1]
	4-(Pyridin-3-ylmethylene)-2-styryloxazol-5(4H)-one	IC50	1000.0 [1]
	(2e)-3-{3-[6-(4-Methyl-1,4-Diazepan-1-Yl)pyrazin-2-Yl]phenyl}prop-2-Enoic Acid	Ki	10000.0 [1]
	1-[5-Amino-4-(3,4-dichlorophenyl)-3-methylpyrazol-1-yl]ethanone	IC50	100000.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-2,2-dimethylpropanamide	IC50	700.0 [1]
	3-(6-Methoxy-1H-indol-2-yl)-1H-pyrazolo[4,3-b]pyridine	IC50	30000.0 [1]
	1-[5-Tert-butyl-3-[4-[2-(dimethylamino)ethyl]-5-oxo-1,4-diazepane-1-carbonyl]thiophen-2-yl]-3-(2,3-dichlorophenyl)urea	IC50	30000.0 [1]
	6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one	IC50	10000.0 [1]
	2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-one	IC50	10000.0 [1]
	2-[3-(3-Piperidin-4-ylpropoxy)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide	Ki	2000.0 [1]
	2-[3-(Methanesulfonamido)phenyl]-N-[4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1,3-thiazol-2-yl]acetamide	Ki	2000.0 [1]
	Drak2-IN-1	IC50	1800.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]cyclopropanecarboxamide	IC50	140.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3-methylbut-2-enamide	IC50	450.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]-3,3-dimethylbutanamide	IC50	10000.0 [1]
	6-Methoxy-7-(1-piperazin-1-ylethyl)-2-[(Z)-pyrazolo[3,4-b]pyridin-3-ylidenemethyl]-1-benzofuran-3-ol	IC50	12.0 [1]
	N-[2-Hydroxy-3-(3-nitroso-1H-indol-2-yl)-1H-indol-5-yl]butanamide	IC50	510.0 [1]
	2-Amino-7-methyl-4-[(4-methylphenyl)methylamino]-9H-pyrimido[4,5-b]indol-6-ol	IC50	100000.0 [1]
	N,N-Dicyclopropyl-7-[(4,5-dimethyl-1,3-thiazol-2-yl)amino]-10-ethyl-3-methyl-3,5,8,10-tetrazatricyclo[7.3.0.02,6]dodeca-1,4,6,8,11-pentaene-11-carboxamide	IC50	1400.0 [1]
	2-[3-(3-Piperazin-1-ylpropoxy)phenyl]-N-(4-pyridin-4-yl-1,3-thiazol-2-yl)acetamide	IC50	1000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 37 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Death-associated protein kinase 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/death-associated-protein-kinase-1-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 21). Quest Database™ Death-associated protein kinase 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/death-associated-protein-kinase-1-inhibitors-ic50-ki.
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