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Cytochrome P450 51 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
KetoconazoleIC50190.0 [1]
KetoconazoleKi24.5 [1], 63.5 [2]
4-{2-[2-(4-Chloro-phenyl)-ethyl]-2-imidazol-1-ylmethyl-[1,3]dioxolan-4-ylmethylsulfanyl}-phenylamineKi17.7 [1], 40.4 [2]
CholesterolIC50200000.0 [1]
TestosteroneIC5050000.0 [1]
ProgesteroneIC50200000.0 [1]
RifampicinIC5030000.0 [1]
Arachidonic acidIC50200000.0 [1]
ErythromycinIC50200000.0 [1]
FluconazoleIC50200000.0 [1]
MetronidazoleIC50200000.0 [1]
LovastatinIC50200000.0 [1]
TolbutamideIC50200000.0 [1]
SporanoxIC503600.0 [1]
PregnenoloneIC50200000.0 [1]
MethimazoleIC50200000.0 [1]
BenzimidazoleIC50200000.0 [1]
GriseofulvinIC5050000.0 [1]
MiconazoleIC50200.0 [1]
ClotrimazoleIC50130.0 [1]
AnandamideIC50200000.0 [1]
PropafenoneIC50200000.0 [1]
ChlorpropamideIC50200000.0 [1]
SulfinpyrazoneIC50200000.0 [1]
EconazoleIC5050.0 [1]
SulfaphenazoleIC50200000.0 [1]
BifonazoleIC50342.0 [1]
TolnaftateIC5050000.0 [1]
TerconazoleIC503000.0 [1]
5-Chloro-1H-indole-2-carboxylic acid [1-(4-fluorobenzyl)-2-(4-hydroxypiperidin-1YL)-2-oxoethyl]amideIC504000.0 [1]
AzaconazoleIC5010000.0 [1]
TriarimolIC5010000.0 [1]
(S)-5-Chloro-N-(1-(4-hydroxypiperidin-1-yl)-1-oxo-3-phenylpropan-2-yl)-1H-indole-2-carboxamideIC503100.0 [1]
2-[(5-Chloro-1H-indole-2-carbonyl)-amino]-3-phenyl-propionic acidIC50200000.0 [1]
5-Chloro-N-[(2S)-1-(4-hydroxypiperidin-1-yl)-3-(4-methoxyphenyl)-1-oxopropan-2-yl]-1H-indole-2-carboxamideIC504500.0 [1]
5-Chloro-N-[(2S)-3-(4-hydroxyphenyl)-1-(4-hydroxypiperidin-1-yl)-1-oxopropan-2-yl]-1H-indole-2-carboxamideIC502500.0 [1]
N-[1-(4-Hydroxypiperidin-1-yl)-1-oxo-3-phenylpropan-2-yl]-1H-pyrrole-2-carboxamideIC50200000.0 [1]
N-[(2S)-1-(4-Hydroxypiperidin-1-yl)-1-oxo-3-phenylpropan-2-yl]-4,5,6,7-tetrahydro-1H-indole-2-carboxamideIC50200000.0 [1]
5-Chloro-N-[(2R)-1-(4-hydroxypiperidin-1-yl)-1-oxo-3-phenylpropan-2-yl]-1H-indole-2-carboxamideIC50100000.0 [1]
5-Chloro-N-[(2S)-1-(4-hydroxypiperidin-1-yl)-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]-1H-indole-2-carboxamideIC501300.0 [1]
5-Chloro-N-[1-(4-hydroxypiperidine-1-carbonyl)cyclopentyl]-1H-indole-2-carboxamideIC50100000.0 [1]
N-[(2S)-1-(4-Hydroxypiperidin-1-yl)-1-oxo-3-phenylpropan-2-yl]-1H-indole-2-carboxamideIC50910.0 [1]
5-Fluoro-N-[(2S)-1-(4-hydroxypiperidin-1-yl)-1-oxo-3-phenylpropan-2-yl]-1H-indole-2-carboxamideIC5075000.0 [1]
Analogue AIC50300.0 [1]
5-Chloro-N-[(2S)-1-(4-hydroxypiperidin-1-yl)-1-oxo-3-pyridin-3-ylpropan-2-yl]-1H-indole-2-carboxamideIC5026000.0 [1]
5-Chloro-N-[(2S)-3-(4-chlorophenyl)-1-(4-hydroxypiperidin-1-yl)-1-oxopropan-2-yl]-1H-indole-2-carboxamideIC509700.0 [1]
5-Chloro-N-[(2S)-3-(2-fluorophenyl)-1-(4-hydroxypiperidin-1-yl)-1-oxopropan-2-yl]-1H-indole-2-carboxamideIC50800.0 [1]
Items per page: 1 - 10 of 47
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cytochrome P450 51 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 30 Mar. 2025, https://www.aatbio.com/data-sets/cytochrome-p450-51-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, March 30). Quest Database™ Cytochrome P450 51 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cytochrome-p450-51-inhibitors-ic50-ki.
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