| Danazol | IC50 | 12.0 [1], 19.0 [2], 77.0 [3], 100.0 [4] |
| Danazol | Ki | 20.0 [1] |
| Telmisartan | IC50 | 420.0 [1], 540.0 [2] |
| Telmisartan | Ki | 100.0 [1], 190.0 [2] |
| Flunarizine | IC50 | 760.0 [1], 940.0 [2], 950.0 [3] |
| Flunarizine | Ki | 100.0 [1], 130.0 [2] |
| Terfenadine | IC50 | 1130.0 [1], 1830.0 [2], 8100.0 [3] |
| N-(2,4-Dichlorobenzyl)-4-(pyrimidin-2-yloxy)piperidine-1-carboxamide | IC50 | 20000.0 [1] |
| Miconazole | IC50 | 580.0 [1], 640.0 [2] |
| Pimozide | IC50 | 30000.0 [1] |
| N-(2,4-Dichlorobenzyl)-4-phenoxypiperidine-1-carboxamide | IC50 | 1400.0 [1] |
| 4-(1-(2,4-Dichlorobenzylcarbamoyl)piperidin-4-yloxy)benzoic acid | IC50 | 20000.0 [1] |
| 3-(Pyridin-4-yl)-N-(2-(trifluoromethoxy)benzyl)pyrrolidine-1-carboxamide | IC50 | 10000.0 [1] |
| Hydrocortisone | IC50 | 50000.0 [1] |
| Dexamethasone | IC50 | 50000.0 [1] |
| Prednisolone | IC50 | 50000.0 [1] |
| Propranolol | IC50 | 50000.0 [1] |
| Acetaminophen | IC50 | 50000.0 [1] |
| Verapamil | IC50 | 22000.0 [1] |
| Naloxone | IC50 | 50000.0 [1] |
| Carbamazepine | IC50 | 50000.0 [1] |
| Chlorpromazine | IC50 | 24400.0 [1] |
| Haloperidol | IC50 | 4690.0 [1] |
| Amoxicillin | IC50 | 50000.0 [1] |
| Nifedipine | IC50 | 3060.0 [1] |
| Fluoxetine | IC50 | 50000.0 [1] |
| Furosemide | IC50 | 50000.0 [1] |
| Ticlopidine | IC50 | 21800.0 [1] |
| Ibuprofen | IC50 | 50000.0 [1] |
| Erythromycin | IC50 | 50000.0 [1] |
| Clozapine | IC50 | 14100.0 [1] |
| Omeprazole | IC50 | 50000.0 [1] |
| Diclofenac | IC50 | 50000.0 [1] |
| Acyclovir | IC50 | 50000.0 [1] |
| Imipramine | IC50 | 50000.0 [1] |
| Cimetidine | IC50 | 50000.0 [1] |
| Diltiazem | IC50 | 50000.0 [1] |
| Metoprolol | IC50 | 4870.0 [1] |
| Trimethoprim | IC50 | 50000.0 [1] |
| Naproxen | IC50 | 50000.0 [1] |
| Hydrochlorothiazide | IC50 | 50000.0 [1] |
| Sulfasalazine | IC50 | 50000.0 [1] |
| Ceftriaxone | IC50 | 27400.0 [1] |
| Minocycline | IC50 | 50000.0 [1] |
| Sertraline | IC50 | 18500.0 [1] |
| Desipramine | IC50 | 50000.0 [1] |
| Triamcinolone | IC50 | 9470.0 [1] |
| Antipyrine | IC50 | 50000.0 [1] |
| Sulpiride | IC50 | 50000.0 [1] |
| Diphenhydramine | IC50 | 50000.0 [1] |
| Ranitidine Base | IC50 | 50000.0 [1] |
| Ketoprofen | IC50 | 50000.0 [1] |
| Norfloxacin | IC50 | 2560.0 [1] |
| Piroxicam | IC50 | 50000.0 [1] |
| Nimodipine | IC50 | 3380.0 [1] |
| Phenacetin | IC50 | 50000.0 [1] |
| Nicardipine | IC50 | 1690.0 [1] |
| Amodiaquine | IC50 | 990.0 [1] |
| Lansoprazole | IC50 | 50000.0 [1] |
| Probucol | IC50 | 50000.0 [1] |
| Dextromethorphan | IC50 | 50000.0 [1] |
| Propafenone | IC50 | 50000.0 [1] |
| Flecainide | IC50 | 50000.0 [1] |
| Perphenazine | IC50 | 10600.0 [1] |
| Mefenamic acid | IC50 | 50000.0 [1] |
| Fexofenadine | IC50 | 50000.0 [1] |
| Mexiletine | IC50 | 50000.0 [1] |
| Alprenolol | IC50 | 50000.0 [1] |
| Mibefradil | IC50 | 2140.0 [1] |
| Bepridil | IC50 | 11500.0 [1] |
| Chlorzoxazone | IC50 | 50000.0 [1] |
| Olmesartan | IC50 | 50000.0 [1] |
| Troleandomycin | IC50 | 50000.0 [1] |
| Mephenytoin | IC50 | 50000.0 [1] |
| Benzbromarone | IC50 | 4260.0 [1] |
| Sulfaphenazole | IC50 | 50000.0 [1] |
| Tenoxicam | IC50 | 50000.0 [1] |
| Benzydamine | IC50 | 50000.0 [1] |
| Eletriptan | IC50 | 50000.0 [1] |
| Bufuralol | IC50 | 50000.0 [1] |
| 4-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-propylphenyl)butan-1-one | Ki | 160.0 [1] |
| 4'-Tert-Butyl-4-(4-(hydroxybenzhydryl)piperidino)butyrophenone | IC50 | 700.0 [1] |
| N-[3,3-Bis-(4-fluorophenyl)-propyl]-6-(2,2,2-trifluoro-ethoxy)-nicotinamide | IC50 | 2000.0 [1] |
| 1-(4-Pyridyl)-3-(3,4,5-trimethoxyphenyl)-2-propen-1-one | IC50 | 20000.0 [1] |
| 1-(4-Allylphenyl)-4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)butan-1-one | IC50 | 400.0 [1] |
| 2-[5-Chloro-4-[2-[(2-chloro-4-cyclopropylphenyl)sulfonylamino]-4-[(1-hydroxy-2-methylpropan-2-yl)carbamoyl]phenoxy]-2-fluorophenyl]acetic acid | Ki | 240100.0 [1] |
| 4-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-1-p-tolylbutan-1-one | IC50 | 700.0 [1] |
| 1-(4-Bromophenyl)-4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)butan-1-one | IC50 | 4200.0 [1] |
| 4-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-methoxyphenyl)butan-1-one | IC50 | 7600.0 [1] |
| 1-(4-Ethylphenyl)-4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)butan-1-one | IC50 | 600.0 [1] |
| 4-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-(2-hydroxyethyl)phenyl)butan-1-one | IC50 | 1300.0 [1] |
| 4-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)-1-(4-(3-hydroxypropyl)phenyl)butan-1-one | IC50 | 1900.0 [1] |
| 1-(4-Butylphenyl)-4-(4-(hydroxydiphenylmethyl)piperidin-1-yl)butan-1-one | IC50 | 700.0 [1] |
| 3-(4-(4-(4-(Hydroxydiphenylmethyl)piperidin-1-yl)butanoyl)phenyl)propyl acetate | IC50 | 2500.0 [1] |
| 1-[4-(2,2-Difluoroethyl)phenyl]-4-[4-[hydroxy(diphenyl)methyl]piperidin-1-yl]butan-1-one | IC50 | 2200.0 [1] |
| 1-(1,3-Benzodioxol-5-yl)-4-[4-[hydroxy(diphenyl)methyl]piperidin-1-yl]butan-1-one | IC50 | 6700.0 [1] |
| 4-Cyano-N-[3-(4-fluorophenyl)-3-(4-methylsulfonylphenyl)propyl]benzamide | IC50 | 3000.0 [1] |
| 4-(Pyrimidin-2-yloxy)-N-(2-(trifluoromethoxy)benzyl)piperidine-1-carboxamide | IC50 | 2000.0 [1] |
| 4-(Pyridin-4-yloxy)-N-(2-(trifluoromethoxy)benzyl)piperidine-1-carboxamide | IC50 | 10000.0 [1] |
| N-(2,4-Dichlorobenzyl)-4-(pyridin-4-yloxy)piperidine-1-carboxamide | IC50 | 2700.0 [1] |