![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_156565d24a79d6ccf50f85f1a835d892.svg) | L-Cysteine | IC50 | 116000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_156565d24a79d6ccf50f85f1a835d892.svg) | L-Cysteine | Ki | 59000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_57cea72581ed62f370a1571595f9b9ad.svg) | (S)-4-Carboxyphenylglycine | IC50 | 5000.0 [1], 15000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_3ff4237bb7209c39f00b225c2a55dea5.svg) | 4-[(E)-N-(2,4-Dinitroanilino)-C-methylcarbonimidoyl]-5-methyl-1,2-oxazole-3-carboxylic acid | IC50 | 290000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_3ff4237bb7209c39f00b225c2a55dea5.svg) | 4-[(E)-N-(2,4-Dinitroanilino)-C-methylcarbonimidoyl]-5-methyl-1,2-oxazole-3-carboxylic acid | Ki | 147000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_57bb29a82ee675c3652631961e42b74c.svg) | 5-Methyl-4-[(E)-C-methyl-N-(4-nitroanilino)carbonimidoyl]-1,2-oxazole-3-carboxylic acid | IC50 | 127000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_57bb29a82ee675c3652631961e42b74c.svg) | 5-Methyl-4-[(E)-C-methyl-N-(4-nitroanilino)carbonimidoyl]-1,2-oxazole-3-carboxylic acid | Ki | 60000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_87dbe0fc1b9a752e218231251de4880e.svg) | 4-[(E)-N-[3,5-Bis(trifluoromethyl)anilino]-C-methylcarbonimidoyl]-5-methyl-1,2-oxazole-3-carboxylic acid | IC50 | 129000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_87dbe0fc1b9a752e218231251de4880e.svg) | 4-[(E)-N-[3,5-Bis(trifluoromethyl)anilino]-C-methylcarbonimidoyl]-5-methyl-1,2-oxazole-3-carboxylic acid | Ki | 64000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_e8407d671771c537ba99d02a929eaa28.svg) | 4-[(E)-N-(2,4-Dinitroanilino)-C-methylcarbonimidoyl]-5-(2-naphthalen-2-ylethyl)-1,2-oxazole-3-carboxylic acid | IC50 | 225000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_e8407d671771c537ba99d02a929eaa28.svg) | 4-[(E)-N-(2,4-Dinitroanilino)-C-methylcarbonimidoyl]-5-(2-naphthalen-2-ylethyl)-1,2-oxazole-3-carboxylic acid | Ki | 113000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_6f2d0353355712e90231bdc33101bd30.svg) | Sulfasalazine | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_49543e9ac68f02347552797a6c469047.svg) | Mesalamine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_322ce77d20ed5ad4ae592a8570841ccc.svg) | Quisqualic acid | IC50 | 5000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_139b71606eae1367f4d37269e321dff8.svg) | Sulfapyridine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_d67a5f6b87b236a6abf7cdd467f7bf2c.svg) | L-Homocysteic acid | IC50 | 35000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_1d7bcf138427816910c2610eeceef367.svg) | Erastin | IC50 | 200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_efd54eb6669abc3e02bb9cbd7ae40aea.svg) | L-Serine O-sulfate | IC50 | 26000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_ca8f7408587acad006760311abe79994.svg) | Susalimod | IC50 | 70000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_2edd3e60ad3d7fdbd63a2ec1c223c72f.svg) | 2-Hydroxy-5-[2-[4-(pyridin-2-ylsulfamoyl)phenyl]ethynyl]benzoic acid | IC50 | 30000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_ec6bcf8709df3556a0a4bf5eb212d0f1.svg) | 3-Phenylethynyl-benzoic acid | IC50 | 270000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_4f576aa5c84127aa1b36f4d50bcc3fd0.svg) | 5-(Phenylazo)salicylic acid | IC50 | 200000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_da49f80787c1d7fce6f61b4e892ca3af.svg) | Imidazole ketone erastin | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_5f4c2688b6d4cd2752c9b53e05cf54fe.svg) | 3-(5-Acetyl-2-propan-2-yloxyphenyl)-2-[[4-[2-(4-chlorophenoxy)acetyl]piperazin-1-yl]methyl]quinazolin-4-one | IC50 | 30.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_c3cb557f2cdaad45019276e00523fefb.svg) | 2-[[4-[2-(4-Chlorophenoxy)acetyl]piperazin-1-yl]methyl]-3-[5-(2-piperazin-1-ylacetyl)-2-propan-2-yloxyphenyl]quinazolin-4-one | IC50 | 100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_490969e52c733c5025873c5669409870.svg) | 2-[[4-[2-(4-Chlorophenoxy)acetyl]piperazin-1-yl]methyl]-3-[5-[2-(4-methylpiperazin-1-yl)acetyl]-2-propan-2-yloxyphenyl]quinazolin-4-one | IC50 | 300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_ef3aea0ee16c1c27d568d79b7c91f652.svg) | 2-[[4-[2-(4-Chlorophenoxy)acetyl]piperazin-1-yl]methyl]-3-[5-(2-morpholin-4-ylacetyl)-2-propan-2-yloxyphenyl]quinazolin-4-one | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_ae0f98147607dd4748427d9cfaf1b689.svg) | 2-[[4-[2-(4-Chlorophenoxy)acetyl]piperazin-1-yl]methyl]-3-[2-propan-2-yloxy-5-[2-(4-prop-2-enylpiperazin-1-yl)acetyl]phenyl]quinazolin-4-one | IC50 | 10.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_d36552d871c689efa263f22646643590.svg) | 2-[[4-[2-(4-Chlorophenoxy)acetyl]piperazin-1-yl]methyl]-3-[5-[2-[4-[(4-methoxyphenyl)methyl]piperazin-1-yl]acetyl]-2-propan-2-yloxyphenyl]quinazolin-4-one | IC50 | 4.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_99ff784d607900cf25ce0a481106ee48.svg) | 2-[[4-[2-(4-Chlorophenoxy)acetyl]piperazin-1-yl]methyl]-3-[5-(2-fluoroacetyl)-2-propan-2-yloxyphenyl]quinazolin-4-one | IC50 | 40.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_0e451ac7a026fa5d5ac39aae5c93993d.svg) | 2-[[4-[2-(4-Chlorophenoxy)acetyl]piperazin-1-yl]methyl]-3-[2-propan-2-yloxy-5-(2,2,2-trifluoroacetyl)phenyl]quinazolin-4-one | IC50 | 20.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_dfb4fec0177b7bf5603392ab9be791f0.svg) | Methyl 2-hydroxy-5-[[4-[(2-pyridinylamino)sulfonyl]phenyl]ethynyl]benzoate | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_920c441554b3a06cd512585ff438ed21.svg) | 2-Hydroxy-5-[(E)-2-[4-(pyridin-2-ylsulfamoyl)phenyl]ethenyl]benzoic acid | IC50 | 70000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_6722507f2d2cc1e378c0c865dc9b34fb.svg) | Methyl 2-hydroxy-5-[(E)-2-[4-(pyridin-2-ylsulfamoyl)phenyl]ethenyl]benzoate | IC50 | 900000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_c5d49dbcaea60b957344a1a37127e930.svg) | 2-Hydroxy-5-[2-[4-(pyridin-2-ylsulfamoyl)phenyl]ethyl]benzoic acid | IC50 | 700000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_7c8b44db8e6f71d7a2895e97c7d267e4.svg) | 2-Hydroxy-5-(phenylethynyl)benzoic acid | IC50 | 150000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_2fe513691a01a16e485e382a80f58f2f.svg) | 3-[3-Carboxy-5-[2-(1-naphthyl)ethyl]isoxazole-4-yl]-L-alanine | Ki | 117000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_e4d2a5c2ec9134c4cd97843633ab751e.svg) | 3-[3-Carboxy-5-[2-(2-naphthyl)ethyl]isoxazole-4-yl]-L-alanine | Ki | 52000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_2b0f4d5756c90ab5920c6386e954b4c7.svg) | 3-[2-[4-(Pyridin-2-ylsulfamoyl)phenyl]ethynyl]benzoic acid | IC50 | 75000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_11a76fe085d35ba80472800bdbeee00c.svg) | 3-[2-[4-(Pyridin-2-ylsulfamoyl)phenyl]ethyl]benzoic acid | IC50 | 920000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_2322d95f0eefd4d73db11fac13dda0a6.svg) | Methyl 2-hydroxy-5-[2-[4-(pyridin-2-ylsulfamoyl)phenyl]ethyl]benzoate | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_66e86b265baee69650566bc0b9121a53.svg) | (R)-4-Carboxyphenylglycine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_c9373e9767ab480dcc8ab0eca852b157.svg) | Piperazine Erastin | IC50 | 800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/cystine-glutamate-transporter_5a4de5bc6019c678aa1a3b339653e644.svg) | 3-[2-[[4-[2-(4-Chlorophenoxy)acetyl]piperazin-1-yl]methyl]-4-oxoquinazolin-3-yl]-4-propan-2-yloxybenzaldehyde | IC50 | 60.0 [1] |