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Cysteinyl leukotriene receptor 2 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
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▼
Standard Values (in nM)
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▼
3-[(3-Carboxycyclohexyl)carbamoyl]-4-[3-[4-(4-cyclohexyloxybutoxy)phenyl]propoxy]benzoic AcidIC503.8 [1], 38.0 [2]
4-(3-Carboxypropyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC502.3 [1], 2.5 [2]
ZafirlukastIC507397.0 [1], 58000.0 [2]
BayCysLT2IC5053.0 [1]
4-[3-(Carboxymethyl)-4-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]indol-1-yl]butanoic acidIC5025.0 [1], 27.0 [2]
MontelukastIC5010000.0 [1]
Montelukast sodiumIC5027000.0 [1]
PranlukastIC503620.0 [1]
Pranlukast hemihydrateIC5043000.0 [1]
4-[(4S,5R,6E,8E,10Z,13Z)-1-Carboxy-4-hydroxynonadeca-6,8,10,13-tetraen-5-yl]sulfanylbenzoic acidIC50300.0 [1]
GemilukastIC5025.0 [1]
4-[2-(Methylsulfonylcarbamoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acidIC5016.0 [1]
4-(3-Carboxypropyl)-8-[[4-(4-phenylbutoxy)phenyl]methoxy]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC5030.0 [1]
4-[8-[(E)-2-[4-(4-Phenylbutoxy)phenyl]ethenyl]-2-(2H-tetrazol-5-yl)-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acidIC503.4 [1]
4-(3-Carboxypropyl)-8-[[4-(4-phenoxybutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC5017.0 [1]
4-(3-Carboxypropyl)-8-[[4-(5-phenylpentoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC500.62 [1]
4-[8-[2-[4-(4-Phenylbutoxy)phenyl]ethyl]-2-(2H-tetrazol-5-yl)-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acidIC5015.0 [1]
(2R)-4-(3-Carboxypropyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC5055.0 [1]
(2S)-4-(3-Carboxypropyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC500.87 [1]
4-[8-[[4-(4-Phenylbutoxy)benzoyl]amino]-2-(2H-tetrazol-5-yl)-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acidIC500.49 [1]
4-(3-Carboxypropyl)-8-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC500.31 [1]
4-(1-Carboxymethyl-7-(4-(4-phenoxybutyloxy)styryl)-1H-indole-3-yl)butyric acidIC506.0 [1]
4-Acetyl-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC503600.0 [1]
8-[[4-(4-Phenylbutoxy)benzoyl]amino]-4-propanoyl-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC505200.0 [1]
4-Butanoyl-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC503700.0 [1]
4-(4-Carboxybutyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC50170.0 [1]
4-[8-[[4-(4-Phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acidIC504300.0 [1]
4-[2-(Hydroxymethyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acidIC50410.0 [1]
1-(3-Carboxypropyl)-4-oxo-5-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]quinoline-3-carboxylic acidIC50370.0 [1]
3-(3-Carboxypropoxy)-8-[(E)-2-[4-(4-phenoxybutoxy)phenyl]ethenyl]quinoxaline-2-carboxylic acidIC5075.0 [1]
4-[1-(Carboxymethyl)-7-[(E)-2-[4-[4-(3-chlorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acidIC5023.0 [1]
4-[1-(Carboxymethyl)-7-[(E)-2-[4-[4-(2,3,6-trifluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acidIC502.1 [1]
4-[1-(Carboxymethyl)-7-[(E)-2-[4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acidIC5014.0 [1]
4-[1-(Carboxymethyl)-7-[(E)-2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acidIC504.6 [1]
4-[1-(Carboxymethyl)-2-methyl-7-[(E)-2-[4-(4-phenylbutoxy)phenyl]ethenyl]indol-3-yl]butanoic acidIC504.7 [1]
4-[1-(Carboxymethyl)-7-[(E)-2-[4-[4-(2-methoxyphenyl)butoxy]phenyl]ethenyl]-2-methylindol-3-yl]butanoic acidIC5015.0 [1]
4-[1-(Carboxymethyl)-2-methyl-7-[(E)-2-[4-[4-(2,3,6-trifluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acidIC501.0 [1]
4-[1-(Carboxymethyl)-2-methyl-7-[(E)-2-[4-[4-(2,3,5,6-tetrafluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acidIC503.7 [1]
4-[1-(Carboxymethyl)-2-methyl-7-[(E)-2-[4-[4-(2,3,4,5-tetrafluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acidIC501.5 [1]
4-[1-(Carboxymethyl)-7-[(E)-2-[4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl]ethenyl]-2-methylindol-3-yl]butanoic acidIC507.2 [1]
2-[1-(Carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]acetic acidIC500.89 [1]
3-[1-(Carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]propanoic acidIC505.7 [1]
4-[1-(Carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acidIC500.88 [1]
3-[3-(Carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]propanoic acidIC5096.0 [1]
3-[1-(2-Carboxyethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]propanoic acidIC5078.0 [1]
4-[1-(2-Carboxyethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acidIC5022.0 [1]
4-[3-(Carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]butanoic acidIC5055.0 [1]
4-[3-(2-Carboxyethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]butanoic acidIC5015.0 [1]
5-[3-(Carboxymethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]pentanoic acidIC50248.0 [1]
5-[3-(2-Carboxyethyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]pentanoic acidIC5060.0 [1]
5-[3-(3-Carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-1-yl]pentanoic acidIC5030.0 [1]
4-[1-(3-Carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-5-fluoro-2-methylindol-3-yl]butanoic acidIC5031.0 [1]
4-[1-(3-Carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-6-fluoro-2-methylindol-3-yl]butanoic acidIC5048.0 [1]
[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]phenyl]methyl (E)-3-(4,6-dichloro-1H-indol-3-yl)prop-2-enoateIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
3-[(E)-3-[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC5058000.0 [1]
4-Chloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC5036000.0 [1]
3-[(E)-3-[[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]phenyl]methoxy]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
3-[[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]phenyl]carbamoyl]-1H-indole-2-carboxylic acidIC5023000.0 [1]
3-[3-[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]anilino]-3-oxopropyl]-1H-indole-2-carboxylic acidIC5050000.0 [1]
5-Chloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
6-Chloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC5087000.0 [1]
7-Chloro-3-[(E)-3-[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
3-[(E)-3-[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-5-fluoro-1H-indole-2-carboxylic acidIC5046000.0 [1]
3-[(E)-3-[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-4,6-difluoro-1H-indole-2-carboxylic acidIC5076000.0 [1]
3-[(E)-3-[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-5-methoxy-1H-indole-2-carboxylic acidIC5046000.0 [1]
4,6-Dichloro-3-[(E)-3-[[3-[(E)-2-(7-chloroquinolin-2-yl)ethenyl]phenyl]methoxy]-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-oxo-3-phenoxyprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-oxo-3-phenylmethoxyprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-oxo-3-(2-phenylethoxy)prop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-oxo-3-(3-phenylpropoxy)prop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-oxo-3-(4-phenylbutoxy)prop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-cyclohexyloxy-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-oxo-3-pentoxyprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
3-[(E)-3-[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-6-methoxy-1H-indole-2-carboxylic acidIC50100000.0 [1]
3-[(E)-3-[3-[(E)-2-(7-Chloroquinolin-2-yl)ethenyl]anilino]-3-oxoprop-1-enyl]-7-methoxy-1H-indole-2-carboxylic acidIC5015000.0 [1]
4,6-Dichloro-3-[(E)-3-(4-methylpentoxy)-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-(cyclohexylmethoxy)-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4,6-Dichloro-3-[(E)-3-(4-cyanobutoxy)-3-oxoprop-1-enyl]-1H-indole-2-carboxylic acidIC50100000.0 [1]
4-(3-Carboxypropanoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC50890.0 [1]
4-(3-Carboxypropyl)-8-[[4-(3-phenylpropoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC5068.0 [1]
4-(5-Carboxypentanoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC50890.0 [1]
4-[2-(Benzenesulfonylcarbamoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazin-4-yl]butanoic acidIC505.7 [1]
4-(4-Carboxybutanoyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC501800.0 [1]
4-(3-Carboxypropyl)-8-[(E)-2-[4-(4-phenylbutoxy)phenyl]ethenyl]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC505.7 [1]
4-(3-Carboxypropyl)-8-[2-[4-(4-phenylbutoxy)phenyl]ethyl]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC5016.0 [1]
4-(3-Carboxypropyl)-8-[[4-(3-phenoxypropoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC5016.0 [1]
4-(3-Carboxypropyl)-8-[[4-(2-phenoxyethoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC501500.0 [1]
4-(5-Carboxypentyl)-8-[[4-(4-phenylbutoxy)benzoyl]amino]-2,3-dihydro-1,4-benzoxazine-2-carboxylic acidIC50290.0 [1]
4-[1-(3-Carboxypropyl)-2-methyl-7-[2-[4-[4-(2,3,4,6-tetrafluorophenyl)butoxy]phenyl]ethynyl]indol-3-yl]butanoic acidIC503.6 [1]
4-[1-(3-Carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-4-fluoro-2-methylindol-3-yl]butanoic acidIC5012.0 [1]
4-[1-(3-Carboxypropyl)-4-fluoro-2-methyl-7-[2-[4-[4-(2,3,4,6-tetrafluorophenyl)butoxy]phenyl]ethynyl]indol-3-yl]butanoic acidIC5013.0 [1]
4-[1-(3-Carboxypropyl)-7-[2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acidIC505.5 [1]
4-[1-(3-Carboxypropyl)-7-[2-[4-[4-(3-fluoro-2-methylphenyl)butoxy]phenyl]ethynyl]-2-methylindol-3-yl]butanoic acidIC508.8 [1]
(Z)-2-Cyano-N-[2-(4-cyanobenzoyl)-5-[(E)-4-(diethylamino)-4-oxobut-2-en-2-yl]-1-benzofuran-3-yl]-3-hydroxybut-2-enamideIC507700.0 [1]
4-[1-(Carboxymethyl)-7-[(E)-2-[4-[4-(3-chloro-2-methylphenyl)butoxy]phenyl]ethenyl]-2-methylindol-3-yl]butanoic acidIC505.1 [1]
4-(1-Carboxymethyl-7-(4-(4-phenylbutyloxy)styryl)-1H-indole-3-yl)butyric acidIC5025.0 [1]
4-[1-(Carboxymethyl)-2-methyl-7-[(E)-2-[4-[4-(2,3,4,6-tetrafluorophenyl)butoxy]phenyl]ethenyl]indol-3-yl]butanoic acidIC502.2 [1]
8-[[4-(4-Phenylbutoxy)benzoyl]amino]-3,4-dihydro-2H-1,4-benzoxazine-2-carboxylic acidIC504600.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cysteinyl leukotriene receptor 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/cysteinyl-leukotriene-receptor-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Cysteinyl leukotriene receptor 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cysteinyl-leukotriene-receptor-2-inhibitors-ic50-ki.
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