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Cyclophilin A Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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Cyclosporin AIC509.6 [1]
Cyclosporin AKi12.2 [1]
2-[[(2R,5S,8S,11S,14S,17S,23S,26S,29S,32S)-17-Ethyl-14-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-4,7,10,13,19,22,28,32-octamethyl-5,8,23,29-tetrakis(2-methylpropyl)-3,6,9,12,15,18,21,24,27,30,33-undecaoxo-11,26-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacont-2-yl]methoxy]-N-[4-[[4-[[2-[[(2R,5S,8S,11S,14S,17S,23S,26S,29S,32S)-17-ethyl-14-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-4,7,10,13,19,22,28,32-octamethyl-5,8,23,29-tetrakis(2-methylpropyl)-3,6,9,12,15,18,21,24,27,30,33-undecaoxo-11,26-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacont-2-yl]methoxy]acetyl]amino]phenyl]diazenyl]phenyl]acetamideIC5030.0 [1], 206.0 [2], 266.0 [3], 487.0 [4]
2-[[(2R,5S,8S,11S,14S,17S,23S,26S,29S,32S)-17-Ethyl-14-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-4,7,10,13,19,22,28,32-octamethyl-5,8,23,29-tetrakis(2-methylpropyl)-3,6,9,12,15,18,21,24,27,30,33-undecaoxo-11,26-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacont-2-yl]methoxy]-N-(4-phenyldiazenylphenyl)acetamideIC502.79 [1], 4.75 [2], 147.0 [3], 227.0 [4]
Scy-635IC509.48 [1], 1549.0 [2]
Scy-635Ki1.84 [1]
GeclosporinIC50130.0 [1], 310.0 [2]
4-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[2-[(2S)-2-[[(2S,3S)-1-[[(2S)-1-Amino-1-oxopropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-2-oxoethyl]amino]-1-oxopropan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-4-oxobutanoic acidIC501000000.0 [1]
1-(4-Chlorophenyl)-3-[4-(thiazol-2-ylsulfamoyl)phenyl]thioureaIC50130.0 [1]
1-(3-Chlorophenyl)-3-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]phenyl]thioureaIC50330.0 [1]
1-(3-Chloro-4-methylphenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thioureaIC50590.0 [1]
1-(3-Chloro-4-methylphenyl)-3-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]phenyl]thioureaIC50650.0 [1]
1-(2-Fluorobenzoyl)-3-(9H-fluoren-9-yl)-ureaIC50159.0 [1]
1-(2,6-Difluorobenzoyl)-3-(9H-fluoren-9-yl)-ureaIC50263.0 [1]
1-(3-Fluorophenyl)-3-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]phenyl]thioureaIC50380.0 [1], 880.0 [2]
1-[4-[(5-Methylisoxazol-3-yl)sulfamoyl]phenyl]-3-(o-tolyl)thioureaIC50600.0 [1]
1-(3-Bromophenyl)-3-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]phenyl]thioureaIC50450.0 [1]
(3R,6R,9R,12S,15R,18R,21R,24R,27S,30R,33R)-27-(Hydroxymethyl)-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-30-propyl-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC5048.0 [1], 93.0 [2]
(3R,6R,9R,12S,15R,18R,21R,24R,30R,33R)-33-[(E,1R,2R)-1-Hydroxy-2-methylhex-4-enyl]-30-(3-hydroxypropyl)-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50256.0 [1], 450.0 [2]
(3S,6S,9R,10R,11S,12S,13E,15E,18S)-18-[(2E,4E,8S,9S)-10-[(2S,3R,4S,5S,6R,9S,11S)-9-Ethyl-4-hydroxy-3,5,11-trimethyl-8-oxo-1-oxa-7-azaspiro[5.5]undecan-2-yl]-9-hydroxy-8-methyldeca-2,4-dien-2-yl]-10,12-dihydroxy-3-[(3-hydroxyphenyl)methyl]-11-methyl-9-(3-oxobutyl)-6-propan-2-yl-19-oxa-1,4,7,25-tetrazabicyclo[19.3.1]pentacosa-13,15-diene-2,5,8,20-tetroneIC502.4 [1], 350.0 [2]
(3S,6S,9R,10R,11S,12S,13E,15E,18S)-10,12-Dihydroxy-3-[(3-hydroxyphenyl)methyl]-11-methyl-18-[(2E,4E)-6-(oxazinan-2-yl)-6-oxohexa-2,4-dien-2-yl]-9-(3-oxobutyl)-6-propan-2-yl-19-oxa-1,4,7,25-tetrazabicyclo[19.3.1]pentacosa-13,15-diene-2,5,8,20-tetroneIC502.7 [1], 360.0 [2]
(2E,4E)-5-[(3S,6S,9R,10R,11S,12S,13E,15E,18S)-10,12-Dihydroxy-3-[(3-hydroxyphenyl)methyl]-11-methyl-2,5,8,20-tetraoxo-9-(3-oxobutyl)-6-propan-2-yl-19-oxa-1,4,7,25-tetrazabicyclo[19.3.1]pentacosa-13,15-dien-18-yl]-N-pyridin-2-ylhexa-2,4-dienamideIC504.1 [1], 390.0 [2]
(2E,4E)-5-[(3S,6S,9R,10R,11S,12S,13E,15E,18S)-10,12-Dihydroxy-3-[(3-hydroxyphenyl)methyl]-11-methyl-2,5,8,20-tetraoxo-9-(3-oxobutyl)-6-propan-2-yl-19-oxa-1,4,7,25-tetrazabicyclo[19.3.1]pentacosa-13,15-dien-18-yl]-N-methoxy-N-methylhexa-2,4-dienamideIC501.1 [1], 200.0 [2]
CyclosporineIC509.7 [1]
(Melle-4)cyclosporinKi2.11 [1]
AlisporivirKi0.34 [1]
[(40-OH)MeLeu]4-Cyclosporin AIC50166.0 [1]
Urea, N-(3-chlorophenyl)-N'-[3-(phenylmethoxy)-2-pyridinyl]-IC50316.0 [1]
(2S)-2-[[(2S,3S)-2-[[(2S)-1-[2-[[(2S)-2-[[(2S)-2-Amino-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-3-methylpentanoyl]amino]propanoic acidIC502000000.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-27-[2-(Diethylamino)ethylsulfanyl]-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC5015.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-24-(2-hydroxy-2-methylpropyl)-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18-tris(2-methylpropyl)-27-methylsulfanyl-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50110.0 [1]
Ethyl 4-[(3-benzyloxy-2-pyridyl)carbamoylamino]benzoateIC5020.0 [1]
Ethyl 3-[(3-benzyloxy-2-pyridyl)carbamoylamino]benzoateIC50951.0 [1]
Methyl 3-[(3-benzyloxy-2-pyridyl)carbamoylamino]benzoateIC50748.0 [1]
1-(3-Benzyloxy-2-pyridyl)-3-[4-(methylsulfamoyl)phenyl]ureaIC50320.0 [1]
4-[3-(3-Benzyloxy-pyridin-2-yl)-ureido]-benzamideIC50810.0 [1]
4-[(3-Benzyloxy-2-pyridyl)carbamoylamino]benzoic acidIC50140.0 [1]
3-[(3-Benzyloxy-2-pyridyl)carbamoylamino]benzoic acidIC5071.0 [1]
1-(3-Benzyloxy-2-pyridyl)-3-(3-nitrophenyl)ureaIC5060.0 [1]
1-(3-Benzyloxy-2-pyridyl)-3-(4-sulfamoylphenyl)ureaIC5060.0 [1]
1-(3-Benzyloxy-2-pyridyl)-3-(2-chlorophenyl)ureaIC50592.0 [1]
3-[3-(3-Benzyloxy-pyridin-2-yl)-ureido]-benzamideIC50361.0 [1]
1-(3-Benzyloxy-2-pyridyl)-3-(4-chlorophenyl)ureaIC50640.0 [1]
{3-[3-(3-Benzyloxy-pyridin-2-yl)-ureido]-phenyl}-ureaIC50528.0 [1]
Ethyl 2-[(3-benzyloxy-2-pyridyl)carbamoylamino]benzoateIC50880.0 [1]
N-{4-[3-(3-Benzyloxy-pyridin-2-yl)-ureido]-phenyl}-acetamideIC501437.0 [1]
1-(3-Benzyloxy-2-pyridyl)-3-(2,4-difluorophenyl)ureaIC50458.0 [1]
1-(3-Benzyloxy-2-pyridyl)-3-[4-(trifluoromethyl)phenyl]ureaIC50499.0 [1]
1-(4-Fluorophenyl)-3-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]phenyl]thioureaIC50350.0 [1]
N-(5-Methylisoxazol-3-yl)-4-(3-phenylthioureido)benzenesulfonamideIC50580.0 [1]
(2R,5S,11S,14S,21E)-2,11-Dimethyl-14-propan-2-yl-3-oxa-9,12,15,28-tetrazatricyclo[21.3.1.15,9]octacosa-1(26),21,23(27),24-tetraene-4,10,13,16-tetroneKi4.3 [1]
1-(3-Chloro-4-methylphenyl)-3-(4-methyl-3-nitrophenyl)thioureaIC50460.0 [1]
1-(4-Chlorophenyl)-3-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]phenyl]thioureaIC50690.0 [1]
1-(4-Methoxyphenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thioureaIC50920.0 [1]
1-(3-Benzyloxy-pyridin-2-yl)-3-phenyl-ureaIC50754.0 [1]
1-(4-Nitrophenyl)-3-(3-(phenylmethoxy)(2-pyridyl))ureaIC5014.0 [1]
1-(2,6-Dihydroxybenzoyl)-3-(9H-fluoren-9-yl)-ureaIC5032.0 [1]
1-(3-Chloro-4-methylphenyl)-3-[2-[[2-(diethylamino)-6-methyl-5-nitropyrimidin-4-yl]amino]ethyl]thioureaIC50740.0 [1]
1-(3-Bromophenyl)-3-(2-(2-(diethylamino)-6-methyl-5-nitropyrimidin-4-ylamino)ethyl)thioureaIC50810.0 [1]
1-(3-Fluorophenyl)-3-(3-oxo-1,3-dihydroisobenzofuran-5-yl)thioureaIC50740.0 [1]
1-(3-Chloro-4-methylphenyl)-3-[4-(1,3-thiazol-2-ylsulfamoyl)phenyl]thioureaIC50160.0 [1]
1-(p-Tolyl)-3-[4-(thiazol-2-ylsulfamoyl)phenyl]thioureaIC50450.0 [1]
(2S)-N-[(2S,3S)-1-(Benzylamino)-3-methyl-1-oxopentan-2-yl]-1-[2-[[(2S)-2-[[(2S)-3-(1H-imidazol-5-yl)-2-(3-methylbutanoylamino)propanoyl]amino]propanoyl]amino]acetyl]pyrrolidine-2-carboxamideIC506000.0 [1]
(2S)-N-[(2S,3S)-1-(Benzylamino)-3-methyl-1-oxopentan-2-yl]-1-[2-[[(2S)-2-[3-(1H-imidazol-5-yl)propanoylamino]propanoyl]amino]acetyl]pyrrolidine-2-carboxamideIC5010000000.0 [1]
CID 497076IC5090000.0 [1]
(2S)-N-[(2S,3S)-1-(Benzylamino)-3-methyl-1-oxopentan-2-yl]-1-[2-[[2-[[(2S)-3-(1H-imidazol-5-yl)-2-(3-methylbutanoylamino)propanoyl]amino]-2-methylpropanoyl]amino]acetyl]pyrrolidine-2-carboxamideIC5010000000.0 [1]
(2S)-N-[1-(Benzylcarbamoyl)cyclopentyl]-1-[2-[[2-[[(2S)-3-(1H-imidazol-5-yl)-2-(3-methylbutanoylamino)propanoyl]amino]-2-methylpropanoyl]amino]acetyl]pyrrolidine-2-carboxamideIC50500000.0 [1]
N-[3-(Benzyloxy)-2-pyridinyl]-N'-[3-(trifluoromethyl)phenyl]ureaIC50303.0 [1]
3-[3-(Benzyloxy)pyridin-2-yl]-1-(3-cyanophenyl)ureaIC505500.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-12-(Diethylaminomethyl)-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,15,19,25,28-octamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50140.0 [1]
(2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[1-[[(2S)-1-amino-1-oxopropan-2-yl]carbamoyl]cyclopentyl]pyrrolidine-2-carboxamideIC50680000.0 [1]
(2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Amino-3-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(2S,3S)-1-(benzylamino)-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideIC50260000.0 [1]
(2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(2S,3S)-1-(benzylamino)-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideIC50115000.0 [1]
(2S)-1-[2-[[(2S)-2-[[(2S)-2-Acetamido-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(2S,3S)-1-(benzylamino)-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideIC50280000.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-12-(4-Aminobutyl)-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,15,19,25,28-octamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC5011.1 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-27-methylsulfanyl-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC503.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-27-[2-(Dimethylamino)ethylsulfanyl]-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC5047.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-27-[2-[methyl(propan-2-yl)amino]ethylsulfanyl]-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC5061.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-27-[2-[Tert-butyl(methyl)amino]ethylsulfanyl]-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50277.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-27-(2-piperidin-1-ylethylsulfanyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC5097.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-27-(2-morpholin-4-ylethylsulfanyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50128.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-27-(2-hydroxyethylsulfanyl)-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC5019.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-27-(2-imidazol-1-ylethylsulfanyl)-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18,24-tetrakis(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50165.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-27-[2-(Diethylamino)ethylsulfanyl]-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-24-(2-hydroxy-2-methylpropyl)-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18-tris(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC506047.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-27-[2-[Tert-butyl(methyl)amino]ethylsulfanyl]-30-ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-24-(2-hydroxy-2-methylpropyl)-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18-tris(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC501572.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-24-(2-hydroxy-2-methylpropyl)-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18-tris(2-methylpropyl)-27-(2-piperidin-1-ylethylsulfanyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50882.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-30-Ethyl-27-(2-hydroxyethylsulfanyl)-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-24-(2-hydroxy-2-methylpropyl)-1,4,7,10,12,15,19,25,28-nonamethyl-6,9,18-tris(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50959.0 [1]
(3S,6S,9S,12R,15S,18S,21S,24S,30S,33S)-30-Ethyl-33-[(E,1R,2R)-1-hydroxy-2-methylhex-4-enyl]-1,4,7,10,12,15,19,25,28-nonamethyl-24-[(2S)-2-methylbutyl]-6,9,18-tris(2-methylpropyl)-3,21-di(propan-2-yl)-1,4,7,10,13,16,19,22,25,28,31-undecazacyclotritriacontane-2,5,8,11,14,17,20,23,26,29,32-undeconeIC50934.0 [1]
(3S,6S,13E,15E,21S)-3-[(3-Hydroxyphenyl)methyl]-6-propan-2-yl-19-oxa-1,4,7,25-tetrazabicyclo[19.3.1]pentacosa-13,15-diene-2,5,8,20-tetroneKi795.0 [1]
(2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-3-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(2S,3S)-1-(benzhydrylamino)-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamideIC501500000.0 [1]
N-(4-Bromophenyl)-N-[2-(cyclohexylamino)-1-(4-nitrophenyl)-2-oxoethyl]-3-(4-methoxyphenyl)propanamideIC5011.2 [1]
N-(9H-Fluoren-9-ylcarbamoyl)-2,4-dihydroxybenzamideIC5010000.0 [1]
N-(9H-Fluoren-9-ylcarbamoyl)-5-fluoro-2-hydroxybenzamideIC5010000.0 [1]
N-(9H-Fluoren-9-ylcarbamoyl)-2-(2-fluorophenyl)acetamideIC5010000.0 [1]
N-[(1-Fluoro-9H-fluoren-9-yl)carbamoyl]-2,6-dihydroxybenzamideIC50940.0 [1]
2-Fluoro-N-[(3-methyl-9H-fluoren-9-yl)carbamoyl]benzamideIC5010000.0 [1]
N-[(3-Fluoro-9H-fluoren-9-yl)carbamoyl]-2,6-dihydroxybenzamideIC502760.0 [1]
2-Fluoro-N-[(1-fluoro-9H-fluoren-9-yl)carbamoyl]benzamideIC5010430.0 [1]
2-Fluoro-N-[(3-fluoro-9H-fluoren-9-yl)carbamoyl]benzamideIC5010260.0 [1]
1-[(2,6-Dihydroxyphenyl)methyl]-3-(9H-fluoren-9-yl)ureaIC5010000.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cyclophilin A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/cyclophilin-a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Cyclophilin A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cyclophilin-a-inhibitors-ic50-ki.
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