![](https://images.aatbio.com/dataset/ic50/complement-c3_3e42afd532ca6df542c8a9b29bd43836.svg) | Compstatin | IC50 | 12000.0 [1], 63000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_20d3e5da2f24cc39fdb72e4ba6a506e4.svg) | 2-[(4R,7S,10S,13S,19S,22S,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-(3-carbamimidamidopropyl)-10-(1H-imidazol-5-ylmethyl)-19-(1H-indol-3-ylmethyl)-28-[(1-methylindol-3-yl)methyl]-13-(naphthalen-1-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 4000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_b16e1c0e7e3c1608d6204728a02d8e5a.svg) | 2-[(4R,7S,10S,13S,19S,22S,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-(3-carbamimidamidopropyl)-10-(1H-imidazol-5-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 1200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_0730f10a3468a5258fe02397faba4d25.svg) | (3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-3-sulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-5-amino-5-oxopentanoyl]amino]-4-[[(2S)-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(1S,2R)-1-carboxy-2-hydroxypropyl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-imidazol-4-yl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-3-(5-fluoro-1H-indol-3-yl)-1-oxopropan-2-yl]amino]-4-oxobutanoic acid | IC50 | 446.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_cd63c99f18169141e217c74c72ef6c03.svg) | (3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-3-sulfanylpropanoyl]amino]-3-methylbutanoyl]amino]-3-(1-methylindol-3-yl)propanoyl]amino]-5-amino-5-oxopentanoyl]amino]-4-[[(2S)-1-[[2-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(1S,2R)-1-carboxy-2-hydroxypropyl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-(1H-imidazol-4-yl)-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-2-oxoethyl]amino]-3-(5-fluoro-1H-indol-3-yl)-1-oxopropan-2-yl]amino]-4-oxobutanoic acid | IC50 | 205.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_ee2b51b3e552e3f56de6837f3f6e8393.svg) | 2-[(4R,7S,10S,13S,19S,22S,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3S)-1-amino-3-methyl-1-oxopentan-2-yl]-methylcarbamoyl]-25-(3-amino-3-oxopropyl)-7-(3-carbamimidamidopropyl)-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13,17-dimethyl-28-[(1-methylindol-3-yl)methyl]-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 62.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_c2132f7e4367bf007188747bc65575ba.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-28-[(1R)-1-hydroxyethyl]-10,13-bis(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_e4c2b654c2a1dc4df3bbe532051c1a72.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-28-(hydroxymethyl)-10,13-bis(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_a71e34abaea801475bd77fb55c3ba973.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10,13,28-tris(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 7000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_98f1db143ec660e722a6c5a484938df9.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-28-benzyl-7-[3-(diaminomethylideneamino)propyl]-10,13-bis(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_18aab50ebbb9a366eb9d426384fd21af.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-28-[(4-hydroxyphenyl)methyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 3000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_ff771365155cda0a41dd6c43cfc6059f.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-13,19,28-tris(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 6000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_f7f95c5c576d8999b0b783e81fdee3ab.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10,13-bis(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 7000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_dbb5a55a1018795129c0d2c2f444dce2.svg) | (2S,3R)-2-[[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 12000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_2a79cce4a18939824fabef1ca9be09bf.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-4-[[(2S,3R)-1-Amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-34-[[(2S,3S)-2-amino-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10,13-bis(1H-imidazol-5-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-28,31-di(propan-2-yl)-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 53600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_bee7514fd152bf6bcdc1be17d32dbf57.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10,13-bis(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-28,31-di(propan-2-yl)-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 32000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_85404349dad9e56f5a8e91263ff6eb32.svg) | Ac-I[CVVQDWGAHRC]T-NH2 | IC50 | 13000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_4fbbd38fafbc8697488c5b24ad32ac7b.svg) | (2S,3S)-2-[[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 2700.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_0c9e9aabdcbd5099114d5605218a9026.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-4-[[(2S,3R)-1-Amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-34-[[(2S,3S)-2-amino-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 55000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_352e900311e77553e1ecf7ea386d8cf8.svg) | (2S,3R)-2-[[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-29-cyclohexyl-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-5-ylmethyl)-19-(1H-indol-3-ylmethyl)-13,28-dimethyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 47800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_598b9ba70152aae166dc6ed810b7840c.svg) | (2S,3R)-2-[[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 10200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_805276e13e7c3953445d0bacbb43de44.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3S)-1-amino-3-methyl-1-oxopentan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-28-[(4-phosphonooxyphenyl)methyl]-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 9600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_b0b83a7d9fcf01bbf36596ac2e4745c4.svg) | (2S,3R)-2-[[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-28-(2,3-dihydro-1H-inden-1-yl)-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_3a72a6a7269478724138e255b8631d18.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-28-(2,3-dihydro-1H-inden-1-yl)-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_c9b85e7e13ff9f68e758ee1ccae6153b.svg) | (2S,3R)-2-[[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-28-(1-benzothiophen-3-yl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13,28-dimethyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_6679cd3bb75215ab7332fbf108a2ceb9.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-28-(1-benzothiophen-3-yl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13,28-dimethyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_a127360970679cf6988b0623650c7cfc.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-28-[(4-benzoylphenyl)methyl]-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 600.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_ac15c6d99709f29c58ef7d155f69f7ee.svg) | (2S,3R)-2-[[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-28-(naphthalen-1-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 1800.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_6e3b522b495cbb3ef03710a6a254dc76.svg) | (2S,3R)-2-[[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-28-(naphthalen-2-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 1400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_f9b423a9e07dcc7c4a05c92e24b4621a.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2S,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-28-(naphthalen-2-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_9d567035d8f70a0d4ccc036e647c340d.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2R,3S)-1-amino-3-methyl-1-oxopentan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-28-[(4-hydroxyphenyl)methyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_3d9de29b318224fcb99a6e1a85378e77.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2R,3S)-1-amino-3-methyl-1-oxopentan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_bbf1316107ecebddd340d7666192d041.svg) | 2-[(4R,7R,10R,13S,19S,22R,25S,28R,31S,34R)-4-[[(2S,3R)-1-Amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-34-[[(2S,3S)-2-amino-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_c09e7ffe4bbc7edfac80cf1cd06c0596.svg) | 2-[(4R,7S,10R,13S,19S,22R,25R,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-4-carbamoyl-7-[3-(diaminomethylideneamino)propyl]-10,13-bis(1H-imidazol-5-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-28,31-di(propan-2-yl)-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_f90d020232d473f17c45674144a07113.svg) | 2-[(4S,7R,10S,13R,19R,22S,25S,28S,31R,34S,37R)-37-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-28-(3-amino-3-oxopropyl)-4-carbamoyl-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10,13-bis(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33,36-undecaoxo-31,34-di(propan-2-yl)-1,2-dithia-5,8,11,14,17,20,23,26,29,32,35-undecazacyclooctatriacont-25-yl]acetic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_69d95acc3a1c444a438dd8551c5f78e6.svg) | 2-[(4R,7S,10R,13S,19R,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-4-carbamoyl-7-[3-(diaminomethylideneamino)propyl]-10,13-bis(1H-imidazol-5-ylmethyl)-19-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-28,31-di(propan-2-yl)-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_7f6059286adcbeaf33393132f247ab80.svg) | (2R,3R)-2-[[(4R,7S,10S,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 136200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_3765da3296fdc5785fa2e5ccaeea0377.svg) | (2R,3R)-2-[[(4R,7S,10R,13R,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 132400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_f4ce86f90fbbf37f4d5101a374c9d2df.svg) | (2R,3R)-2-[[(4R,7S,10R,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[2-(diaminomethylideneamino)ethyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 23100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_2c5370e37c0c4534dffc96bec1957575.svg) | (3S)-3-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S,3R)-2-Amino-3-hydroxybutanoyl]amino]-3-sulfanylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-4-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S,3S)-1-methoxy-3-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-naphthalen-2-yl-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-4-oxobutanoic acid | IC50 | 545.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_656b7321ec38d0b5a0dd6fdbbf23f7c2.svg) | 2-[(4R,7S,10R,13S,19S,22R,25S,28R,31R,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-4-[[(2R,3R)-1-amino-3-hydroxy-1-oxobutan-2-yl]carbamoyl]-25-(3-amino-3-oxopropyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacont-22-yl]acetic acid | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_f98385ecab617f73b7d2338f0dac9ce7.svg) | (3S)-3-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S,3R)-2-Amino-3-hydroxybutanoyl]amino]-3-sulfanylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-4-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S,3S)-1-methoxy-3-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-(5-methyl-1H-indol-3-yl)-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-4-oxobutanoic acid | IC50 | 870.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_fe539219c10505b102efa9a2dcc3b9ef.svg) | (3S)-4-[[(2S)-5-Amino-1-[[(2S)-3-(5-fluoro-1H-indol-3-yl)-1-[[(2S)-1-[[(2R)-1-[[(2S,3S)-1-methoxy-3-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-3-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S,3R)-2-amino-3-hydroxybutanoyl]amino]-3-sulfanylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-4-oxobutanoic acid | IC50 | 1740.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_a041ac092f5319e9d66c3031765ab9c7.svg) | (3S)-3-[[(2S)-2-[[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2R)-2-[[(2S,3R)-2-Amino-3-hydroxybutanoyl]amino]-3-sulfanylpropanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]amino]-3-(1H-imidazol-4-yl)propanoyl]amino]propanoyl]amino]acetyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-4-[[(2S)-5-amino-1-[[(2S)-1-[[(2S)-1-[[(2R)-1-[[(2S,3S)-1-methoxy-3-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-sulfanylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-(1-methylindol-3-yl)-1-oxopropan-2-yl]amino]-1,5-dioxopentan-2-yl]amino]-4-oxobutanoic acid | IC50 | 205.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_691d6f92457692f389a82b47bef8a1f3.svg) | (2S,3R)-2-[[(4S,7R,10S,13S,19S,22R,25S,28R,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-13-ethyl-10-(1H-imidazol-4-ylmethyl)-19,28-bis(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 1500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/complement-c3_bfc048c57a79adcd18798af7718a7d7d.svg) | (2S,3R)-2-[[(4R,7S,10R,13S,19S,22S,25S,28S,31S,34R)-34-[[(2S,3S)-2-Acetamido-3-methylpentanoyl]amino]-25-(3-amino-3-oxopropyl)-28-[(4-benzoylphenyl)methyl]-22-(carboxymethyl)-7-[3-(diaminomethylideneamino)propyl]-10-(1H-imidazol-4-ylmethyl)-19-(1H-indol-3-ylmethyl)-13-methyl-6,9,12,15,18,21,24,27,30,33-decaoxo-31-propan-2-yl-1,2-dithia-5,8,11,14,17,20,23,26,29,32-decazacyclopentatriacontane-4-carbonyl]amino]-3-hydroxybutanoic acid | IC50 | 1100.0 [1] |