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Coagulation factor XIII Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
▲
▼
Standard Values (in nM)
▲
▼
CeruleninIC504000.0 [1], 18000.0 [2]
N-(4-Bromophenyl)acrylamideIC502400.0 [1]
N-[(5S)-6-[4-(6-Methylpyridin-2-yl)piperazin-1-yl]-6-oxo-5-[(2-phenylacetyl)amino]hexyl]prop-2-enamideIC5035000.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-hexyl]-2-nitro-benzenesulfonamideIC50130.0 [1]
Ethyl (E,6S)-7-[[(2S)-1-[(2S)-2-[[(2S)-1-methoxy-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-methyl-1-oxobutan-2-yl]amino]-7-oxo-6-(phenylmethoxycarbonylamino)hept-2-enoateIC5050000.0 [1]
Ethyl (E,6S)-7-[[(2S)-5-amino-1-[(2S)-2-[[(2S)-1-methoxy-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-1,5-dioxopentan-2-yl]amino]-7-oxo-6-(phenylmethoxycarbonylamino)hept-2-enoateIC5050000.0 [1]
Benzyl N-[(2S)-1-[4-(2-chlorophenyl)piperazin-1-yl]-1-oxo-6-(prop-2-enoylamino)hexan-2-yl]carbamateIC5067000.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-hexyl]-3-nitro-benzenesulfonamideIC501900.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-hexyl]-4-nitro-benzenesulfonamideIC50910.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-hexyl]-4-methyl-benzenesulfonamideIC502200.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-hexyl]-benzenesulfonamideIC502300.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-ylamino)-hexyl]-2-methyl-benzenesulfonamideIC50700.0 [1]
{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitro-benzenesulfonylamino)-hexyl]-amino}-acetic acidIC50620.0 [1]
2-{Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-[6-(2-nitro-benzenesulfonylamino)-hexyl]-amino}-acetamideIC50420.0 [1]
N'-Imidazo[1,2-d][1,2,4]thiadiazol-3-ylhexane-1,6-diamineIC5011000.0 [1]
2-Nitro-N-[6-(3-nitro-pyridin-2-ylamino)-hexyl]-benzenesulfonamideIC50170000.0 [1]
N-[6-(Imidazo[1,2-d][1,2,4]thiadiazol-3-yl-methyl-amino)-hexyl]-2-nitro-benzenesulfonamideIC50110.0 [1]
CID 118722679IC501700.0 [1]
(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-4-Amino-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-5-amino-2-[[(2S)-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-6-amino-2-[[(2S,3S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-hydroxypropanoyl]amino]-4-carboxybutanoyl]amino]-4-methylpentanoyl]amino]-3-methylpentanoyl]amino]hexanoyl]pyrrolidine-2-carbonyl]amino]-4-methylsulfanylbutanoyl]amino]-3-carboxypropanoyl]amino]-3-carboxypropanoyl]amino]-3-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-5-oxopentanoyl]amino]-5-carbamimidamidopentanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-4-carboxybutanoyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carbonyl]amino]-4-oxobutanoyl]amino]-4-methylpentanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoic acidIC501900.0 [1]
CID 118722681IC502200.0 [1]
(2R,3S)-2-N-(4-Butylphenyl)oxirane-2,3-dicarboxamideIC50220.0 [1]
(2R,3S)-2-N-(4-Phenoxyphenyl)oxirane-2,3-dicarboxamideIC5055.0 [1]
(2R,3S)-2-N-(3-Chlorophenyl)oxirane-2,3-dicarboxamideIC5048.0 [1]
(2R,3S)-2-N-(3-Phenoxyphenyl)oxirane-2,3-dicarboxamideIC504.0 [1]
(2S,3R)-2-N-Phenyloxirane-2,3-dicarboxamideIC50720.0 [1]
(2S,3R)-2-N-(4-Bromophenyl)oxirane-2,3-dicarboxamideIC50130.0 [1]
(2S,3R)-2-N-(4-Bromo-3-chlorophenyl)oxirane-2,3-dicarboxamideIC504.0 [1]
(2S,3R)-2-N-(3,4-Dimethylphenyl)oxirane-2,3-dicarboxamideIC50110.0 [1]
(2S,3R)-2-N-[4-[2-[(2-Nitrophenyl)sulfonylamino]ethyl]phenyl]oxirane-2,3-dicarboxamideIC5090.0 [1]
(2S,3R)-2-N-[4-(4-Nitrophenoxy)phenyl]oxirane-2,3-dicarboxamideIC50430.0 [1]
(2S,3R)-2-N-[4-(4-Aminophenoxy)phenyl]oxirane-2,3-dicarboxamideIC5086.0 [1]
(2S,3R)-2-N-[4-[4-[(4-Fluorobenzoyl)amino]phenoxy]phenyl]oxirane-2,3-dicarboxamideIC50100.0 [1]
(2S)-1-Acetyl-N-[(2S)-1-[[(2S)-1-[(2S)-2-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-methyl-1-oxopentan-2-yl]amino]-6-diazo-1,5-dioxohexan-2-yl]pyrrolidine-2-carboxamideIC5080000.0 [1]
N-Hexyl-2-nitrobenzenesulfonamideIC50100000.0 [1]
N-[4-(Pyrrolidine-1-sulfonyl)phenyl]prop-2-enamideIC50770.0 [1]
N-[4-[4-(Adamantane-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50180.0 [1]
(2,3-Difluorophenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50320.0 [1]
Cyclopentyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50240.0 [1]
N-[4-[4-(Piperidine-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50300.0 [1]
N-[4-[4-(Pyrrolidine-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50570.0 [1]
N-[4-[4-(3-Phenylpropyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC501200.0 [1]
Benzyl 4-[6-(prop-2-enoylamino)pyridin-3-yl]sulfonylpiperazine-1-carboxylateIC501300.0 [1]
N-[4-[4-(4-Phenylbutyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50980.0 [1]
N-[4-[4-(Cyclopropanecarbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50310.0 [1]
N-[4-[4-(Cyclopentanecarbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50280.0 [1]
N-[4-[4-(4,4-Difluoropiperidine-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50310.0 [1]
Tert-butyl 4-[6-(prop-2-enoylamino)pyridin-3-yl]sulfonylpiperazine-1-carboxylateIC501600.0 [1]
Benzyl 5-[4-(prop-2-enoylamino)phenyl]sulfonyl-1,3,3a,4,6,6a-hexahydropyrrolo[3,4-c]pyrrole-2-carboxylateIC50600.0 [1]
(3-Phenoxyphenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50670.0 [1]
Benzyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50420.0 [1]
Benzyl 4-[3-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50350.0 [1]
Benzyl 4-[4-(prop-2-enoylamino)phenyl]sulfonyl-1,4-diazepane-1-carboxylateIC50670.0 [1]
4-(4-Acryloylamino-benzenesulfonyl)-piperazine-1-carboxylic acid tert-butyl esterIC50430.0 [1]
4-(4-Acryloylamino-benzenesulfonylamino)-piperidine-1-carboxylic acid benzyl esterIC50480.0 [1]
[1-(4-Acryloylamino-benzenesulfonyl)-piperidin-4-yl]-carbamic acid benzyl esterIC50310.0 [1]
4-(4-Acryloylamino-benzenesulfonyl)-piperazine-1-carboxylic acid 2-chloro-benzyl esterIC50250.0 [1]
Benzyl (3R)-3-[[4-(prop-2-enoylamino)phenyl]sulfonylamino]pyrrolidine-1-carboxylateIC50410.0 [1]
4-(4-Acryloylamino-2-trifluoromethyl-benzenesulfonyl)-piperazine-1-carboxylic acid benzyl esterIC5039.0 [1]
Benzyl N-methyl-N-[2-[methyl-[4-(prop-2-enoylamino)phenyl]sulfonylamino]ethyl]carbamateIC50850.0 [1]
Benzyl 4-[[[4-(prop-2-enoylamino)phenyl]sulfonylamino]methyl]piperidine-1-carboxylateIC50520.0 [1]
Benzyl N-[[1-[4-(prop-2-enoylamino)phenyl]sulfonylpiperidin-4-yl]methyl]carbamateIC50440.0 [1]
[2-(Trifluoromethyl)phenyl]methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50340.0 [1]
Benzyl N-[(3R)-1-[4-(prop-2-enoylamino)phenyl]sulfonylpyrrolidin-3-yl]carbamateIC50960.0 [1]
N-(4-Piperazin-1-ylsulfonylphenyl)prop-2-enamideIC501100.0 [1]
N-[4-(4-Pyridin-2-ylpiperazin-1-yl)sulfonylphenyl]prop-2-enamideIC50500.0 [1]
N-[4-[4-(3-Methylpyridin-2-yl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50340.0 [1]
N-[4-[4-(6-Methylpyridin-2-yl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50220.0 [1]
N-[4-[4-[3-(Trifluoromethyl)pyridin-2-yl]piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50250.0 [1]
N-[4-[4-[5-(Trifluoromethyl)pyridin-2-yl]piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50570.0 [1]
N-[4-(4-Phenylpiperazin-1-yl)sulfonylphenyl]prop-2-enamideIC50370.0 [1]
N-[4-[4-[2-(Trifluoromethyl)phenyl]piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC501400.0 [1]
Benzyl (3S)-3-[[4-(prop-2-enoylamino)phenyl]sulfonylamino]pyrrolidine-1-carboxylateIC50500.0 [1]
Benzyl N-[(3S)-1-[4-(prop-2-enoylamino)phenyl]sulfonylpyrrolidin-3-yl]carbamateIC50720.0 [1]
(4-Fluorophenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50330.0 [1]
(3,5-Difluorophenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50500.0 [1]
(2-Methylphenyl)methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50230.0 [1]
Naphthalen-1-ylmethyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50380.0 [1]
Naphthalen-2-ylmethyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50720.0 [1]
Methyl 4-[4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50310.0 [1]
N-[4-[4-(3,4,4a,5,6,7,8,8a-Octahydro-1H-isoquinoline-2-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50280.0 [1]
N-[4-[4-(3,4,4a,5,6,7,8,8a-Octahydro-2H-quinoline-1-carbonyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50330.0 [1]
N-[4-[4-(3-Phenylpropanoyl)piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50760.0 [1]
N-[4-[4-[(1S,2S)-2-Phenylcyclopropanecarbonyl]piperazin-1-yl]sulfonylphenyl]prop-2-enamideIC50200.0 [1]
N-[5-[4-(Cyclopropanecarbonyl)piperazin-1-yl]sulfonylpyridin-2-yl]prop-2-enamideIC501500.0 [1]
N-[5-[4-(Adamantane-1-carbonyl)piperazin-1-yl]sulfonylpyridin-2-yl]prop-2-enamideIC502200.0 [1]
Tert-butyl 4-[2-(prop-2-enoylamino)pyrimidin-5-yl]sulfonylpiperazine-1-carboxylateIC503300.0 [1]
Benzyl 4-[2-(prop-2-enoylamino)pyrimidin-5-yl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
N-[5-[4-(Adamantane-1-carbonyl)piperazin-1-yl]sulfonylpyrimidin-2-yl]prop-2-enamideIC502500.0 [1]
Tert-butyl 4-[4-(2-fluoroprop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC508900.0 [1]
Tert-butyl 4-[4-(2-methylprop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 4-[4-[[(Z)-but-2-enoyl]amino]phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 4-[4-[[(E)-but-2-enoyl]amino]phenyl]sulfonylpiperazine-1-carboxylateIC5027000.0 [1]
Tert-butyl 4-[4-[[(E)-2-methylbut-2-enoyl]amino]phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Tert-butyl 4-[4-[[(Z)-3-chloroprop-2-enoyl]amino]phenyl]sulfonylpiperazine-1-carboxylateIC50870.0 [1]
4-[4-(1-Oxo-but-2-ynylamino)-benzenesulfonyl]-piperazine-1-carboxylic acid tert-butyl esterIC506700.0 [1]
Benzyl 4-[4-[(E)-4-ethoxy-4-oxobut-2-enyl]phenyl]sulfonylpiperazine-1-carboxylateIC506800.0 [1]
Benzyl 4-[3-[methyl(2-methylpropyl)amino]-4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5080000.0 [1]
Benzyl 4-[3-fluoro-4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC5016000.0 [1]
4-(4-Acryloylamino-2-methoxy-benzenesulfonyl)-piperazine-1-carboxylic acid tert-butyl esterIC50740.0 [1]
Tert-butyl 4-[2-methyl-4-(prop-2-enoylamino)phenyl]sulfonylpiperazine-1-carboxylateIC50210.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Coagulation factor XIII Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/coagulation-factor-xiii-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Coagulation factor XIII Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/coagulation-factor-xiii-inhibitors-ic50-ki.
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