 | Methyl N-[4-[5-chloro-2-[(1S)-1-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-2-phenylethyl]-1H-imidazol-4-yl]phenyl]carbamate | Ki | 2.7 [1], 3.7 [2], 5.8 [3] |
 | Methyl N-[(14S)-14-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-9-oxo-8,16,18-triazatricyclo[13.2.1.02,7]octadeca-1(17),2(7),3,5,15-pentaen-5-yl]carbamate | Ki | 1.0 [1], 5.0 [2] |
 | (2S)-2-[[(2R)-2-(3-Chlorophenyl)-2-hydroxyacetyl]amino]-N-[(2S)-5-(diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]-3-methylbutanamide | IC50 | 116.0 [1], 120.0 [2] |
 | 4-[[(1S)-2-[(E)-3-[3-Chloro-2-fluoro-6-(tetrazol-1-yl)phenyl]prop-2-enoyl]-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]benzoic acid | Ki | 3.7 [1], 5.0 [2] |
 | 4-[[(3S)-2-[(E)-3-[5-Chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-3,4-dihydro-1H-isoquinoline-3-carbonyl]amino]benzoic acid | Ki | 1700.0 [1], 1737.0 [2] |
 | 4-[[(1S)-2-[(E)-3-[5-Chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]benzoic acid | Ki | 10.32 [1], 11.0 [2] |
 | 4-[[6-[(E)-3-[5-Chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-7,8-dihydro-5H-1,6-naphthyridine-5-carbonyl]amino]benzoic acid | Ki | 51.0 [1], 51.2 [2] |
 | Methyl N-[[4-[[(1S)-2-[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]phenyl]methyl]carbamate | Ki | 886.4 [1], 890.0 [2] |
 | Razaxaban | Ki | 12000.0 [1] |
 | Bms-262084 | IC50 | 2.8 [1] |
 | alpha-Ketothiazole analogue 36 | IC50 | 30.0 [1] |
 | 6-Chloro-2-hydroxyquinoline | IC50 | 140000.0 [1] |
 | 6-Chloro-2-hydroxyquinoline | Ki | 70000.0 [1] |
 | (2S)-N-[(2S)-1-[[(2S)-5-(Diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-2-[(3,4-dichlorophenyl)methylcarbamoylamino]-4-methylpentanamide | IC50 | 63.0 [1] |
 | N-[1-[4-(3-Amino-1H-indazol-6-yl)pyridin-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexane-1-carboxamide | Ki | 13.0 [1] |
 | N-[(1S)-1-[4-(3-Amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexane-1-carboxamide | Ki | 0.31 [1] |
 | N-[(2S)-1-[(6-Chloro-2-oxo-1H-quinolin-4-yl)methylamino]-1-oxo-3-phenylpropan-2-yl]-4-hydroxy-2-oxo-1H-quinoline-6-carboxamide | IC50 | 1.0 [1] |
 | N-[(2S)-1-[(6-Chloro-2-oxo-1H-quinolin-4-yl)methylamino]-1-oxo-3-phenylpropan-2-yl]-4-hydroxy-2-oxo-1H-quinoline-6-carboxamide | Ki | 0.5 [1] |
 | (2S)-N-[(2S)-1-[[(2S)-5-(Diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-2-[(2,4-dichlorophenyl)methylcarbamoylamino]-4-methylpentanamide | IC50 | 45.0 [1] |
 | (2S)-2-[[(2S)-2-[[(1R)-1-(4-Bromophenyl)ethyl]carbamoylamino]-3-(4-hydroxyphenyl)propanoyl]amino]-N-[(2S)-5-(diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]-3-methylbutanamide | IC50 | 6.0 [1] |
 | N-[(2S)-1-[[(2S)-5-(Diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]-4-methylpentanamide | IC50 | 850.0 [1] |
 | (2S)-N-[(2S)-5-(Diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]-2-[(3,4-dichlorophenyl)methylcarbamoylamino]-3-methylbutanamide | IC50 | 480.0 [1] |
 | (S)-N-[(S)-4-Guanidino-1-(thiazole-2-carbonyl)-butyl]-3-methyl-2-ureido-butyramide | IC50 | 500.0 [1], 502.0 [2] |
 | Methyl N-[4-[2-[(1S)-1-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-2-phenylethyl]pyridin-4-yl]phenyl]carbamate | Ki | 23.0 [1] |
 | Methyl N-[4-[2-[(1S)-1-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-2-phenylethyl]-1H-imidazol-5-yl]phenyl]carbamate | Ki | 6.7 [1] |
 | 2-[3-[(2S,4R)-6-Carbamimidoyl-4-methyl-4-phenyl-2,3-dihydro-1H-quinolin-2-yl]-5-(3-methylbutanoylamino)phenyl]-5-carbamoylbenzoic acid | Ki | 0.2 [1], 0.59 [2] |
 | Methyl N-[(12E,15S)-18-chloro-15-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-9-oxo-8,17,19-triazatricyclo[14.2.1.02,7]nonadeca-1(18),2(7),3,5,12,16(19)-hexaen-5-yl]carbamate | Ki | 0.03 [1] |
 | Methyl N-[(15S)-15-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-9-oxo-8,17,19-triazatricyclo[14.2.1.02,7]nonadeca-1(18),2(7),3,5,16-pentaen-5-yl]carbamate | Ki | 3.2 [1] |
 | Methyl N-[(12E,15S)-15-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-9-oxo-8,17,19-triazatricyclo[14.2.1.02,7]nonadeca-1(18),2(7),3,5,12,16-hexaen-5-yl]carbamate | Ki | 0.16 [1] |
 | Methyl N-[(15S)-18-chloro-15-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-9-oxo-8,17,19-triazatricyclo[14.2.1.02,7]nonadeca-1(18),2(7),3,5,16(19)-pentaen-5-yl]carbamate | Ki | 0.47 [1] |
 | (2S)-2-[[2-(3-Chlorophenyl)-2-oxoacetyl]amino]-N-[(2S)-5-(diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]-3-methylbutanamide | IC50 | 250.0 [1], 254.0 [2] |
 | CID 76328755 | IC50 | 580.0 [1] |
 | CID 76328755 | Ki | 300.0 [1] |
 | N-[(1S)-1-[4-(3-Amino-1H-indazol-6-yl)pyridin-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexane-1-carboxamide | Ki | 7.2 [1], 8.4 [2] |
 | 2-[[(1R)-2-[[2-[(4-Carbamimidoylphenyl)methylcarbamoyl]-1,3-dihydroinden-2-yl]amino]-1-cyclohexyl-2-oxoethyl]amino]acetic acid | IC50 | 44000.0 [1] |
 | 2-[[(1R)-2-[[2-[(4-Carbamimidoylphenyl)methylcarbamoyl]-1,3-dihydroinden-2-yl]amino]-1-cyclohexyl-2-oxoethyl]amino]acetic acid | Ki | 19000.0 [1] |
 | N-[(1S)-1-[4-(3-Amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexane-1-carboxamide;2,2,2-trifluoroacetic acid | Ki | 0.3 [1], 0.8 [2] |
 | Methyl N-[(11E,14S)-14-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-16,18-diazatricyclo[13.2.1.02,7]octadeca-1(17),2(7),3,5,11,15-hexaen-5-yl]carbamate | Ki | 636.0 [1] |
 | Methyl N-[(14S)-14-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-16,18-diazatricyclo[13.2.1.02,7]octadeca-1(17),2(7),3,5,15-pentaen-5-yl]carbamate | Ki | 34.0 [1], 87.0 [2] |
 | Methyl N-[(14S)-17-chloro-14-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-8-oxa-16,18-diazatricyclo[13.2.1.02,7]octadeca-1(17),2(7),3,5,15(18)-pentaen-5-yl]carbamate | Ki | 249.0 [1], 250.0 [2] |
 | Methyl N-[(15S)-15-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-12-methyl-9-oxo-8,17,19-triazatricyclo[14.2.1.02,7]nonadeca-1(18),2(7),3,5,16-pentaen-5-yl]carbamate | Ki | 5.0 [1], 18.0 [2] |
 | Methyl N-[(3S)-6-chloro-3-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-5,23-diazatetracyclo[16.3.1.14,7.08,13]tricosa-1(21),4(23),6,8(13),9,11,18(22),19-octaen-11-yl]carbamate | Ki | 8.16 [1], 8.2 [2] |
 | 3-[[(2R)-1-[[(2S)-1-[(4-Carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]propanoic acid | IC50 | 44000.0 [1] |
 | 3-[[(2R)-1-[[(2S)-1-[(4-Carbamimidoylphenyl)methylamino]-5-(diaminomethylideneamino)-1-oxopentan-2-yl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]propanoic acid | Ki | 19000.0 [1] |
 | 2-[[(2R)-1-[[3-[4-(Aminomethyl)phenyl]-1-[(4-carbamimidoylphenyl)methylamino]-1-oxopropan-2-yl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]acetic acid | IC50 | 43000.0 [1] |
 | 2-[[(2R)-1-[[3-[4-(Aminomethyl)phenyl]-1-[(4-carbamimidoylphenyl)methylamino]-1-oxopropan-2-yl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]acetic acid | Ki | 19000.0 [1] |
 | 2-[[(2R)-1-[[(2S)-1-[(4-Carbamimidoylphenyl)methylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]acetic acid | IC50 | 1900.0 [1] |
 | 2-[[(2R)-1-[[(2S)-1-[(4-Carbamimidoylphenyl)methylamino]-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]acetic acid | Ki | 800.0 [1] |
 | 2-[[(2R)-1-[[(1S)-2-[(4-Carbamimidoylphenyl)methylamino]-2-oxo-1-piperidin-4-ylethyl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]acetic acid | IC50 | 44000.0 [1] |
 | 2-[[(2R)-1-[[(1S)-2-[(4-Carbamimidoylphenyl)methylamino]-2-oxo-1-piperidin-4-ylethyl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]acetic acid | Ki | 19000.0 [1] |
 | 2-[[(2R)-1-[[1-[(4-Carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]acetic acid | IC50 | 44000.0 [1] |
 | 2-[[(2R)-1-[[1-[(4-Carbamimidoylphenyl)methylamino]-1-oxo-4-piperidin-4-ylbutan-2-yl]amino]-3-cyclohexyl-1-oxopropan-2-yl]amino]acetic acid | Ki | 19000.0 [1] |
 | (E)-N-[(1S)-1-[5-Chloro-4-(4-hydroxy-2-oxo-1H-quinolin-6-yl)-1H-imidazol-2-yl]-3-(4-methylpiperazin-1-yl)-3-oxopropyl]-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enamide | Ki | 0.04 [1], 0.1 [2] |
 | Methyl N-[(3S)-6-chloro-3-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-16-oxo-5,15,22-triazatetracyclo[15.2.2.14,7.08,13]docosa-1(20),4(22),6,8(13),9,11,17(21),18-octaen-11-yl]carbamate | Ki | 8100.0 [1], 8117.0 [2] |
 | Methyl N-[(3S)-3-[[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]amino]-5,23-diazatetracyclo[16.2.2.14,7.08,13]tricosa-1(21),4,6,8(13),9,11,18(22),19-octaen-11-yl]carbamate | Ki | 71.0 [1] |
 | 4-[[5-Acetamido-2-[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]benzoic acid | Ki | 21.0 [1], 21.43 [2] |
 | 4-[[3-[(4-Chlorophenyl)carbamoylamino]-6-[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-7,8-dihydro-5H-1,6-naphthyridine-5-carbonyl]amino]benzoic acid | Ki | 258.0 [1] |
 | 4-[[2-[4-(5-Chloro-2-cyanophenyl)-5-methoxy-2-oxopyridin-1-yl]-3-(4-methoxycyclohexyl)propanoyl]amino]benzoic acid | IC50 | 2.4 [1], 600.0 [2] |
 | Methyl N-[3-[[(1S)-2-[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]phenyl]carbamate | Ki | 2795.0 [1] |
 | Ethyl 5-[[3-ethoxycarbonyl-5-[(6-ethoxy-3-ethoxycarbonyl-5-sulfooxy-1-benzofuran-2-yl)methoxy]-6-methoxy-1-benzofuran-2-yl]methoxy]-6-methoxy-2-methyl-1-benzofuran-3-carboxylate | IC50 | 820.0 [1], 49000.0 [2] |
 | 4-[[5-[(E)-3-[3-Chloro-2-fluoro-6-(tetrazol-1-yl)phenyl]prop-2-enoyl]-3-methyl-2,4,6,7-tetrahydropyrazolo[4,3-c]pyridine-4-carbonyl]amino]benzoic acid | Ki | 5.02 [1] |
 | 4-[[8-Bromo-2-[(E)-3-[5-chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-4,4-dimethyl-1,3-dihydroisoquinoline-1-carbonyl]amino]benzoic acid | Ki | 171.6 [1] |
 | 4-[[5-[(E)-3-[5-Chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-3-ethyl-1-methyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-4-carbonyl]amino]benzoic acid | Ki | 23.3 [1] |
 | 4-[[(1S)-2-[3-[5-Chloro-2-(tetrazol-1-yl)phenyl]prop-2-ynoyl]-3,4-dihydro-1H-isoquinoline-1-carbonyl]amino]benzoic acid | Ki | 7.08 [1] |
 | 4-[[2-[(E)-3-[3-Chloro-2-fluoro-6-(tetrazol-1-yl)phenyl]prop-2-enoyl]-5-morpholin-4-yl-3,4-dihydro-1H-2,6-naphthyridine-1-carbonyl]amino]benzoic acid | Ki | 5.0 [1] |
 | (1S)-2-[(E)-3-[5-Chloro-2-(tetrazol-1-yl)phenyl]prop-2-enoyl]-N-(4-pyrrolidin-2-ylphenyl)-3,4-dihydro-1H-isoquinoline-1-carboxamide | Ki | 6732.0 [1] |
 | 5-(4-Carbamoylphenyl)-2-[(E)-3-[3-chloro-2-fluoro-6-(tetrazol-1-yl)phenyl]prop-2-enoyl]-N-(1H-indazol-6-yl)-3,4-dihydro-1H-2,6-naphthyridine-1-carboxamide | Ki | 5.0 [1] |
 | Benzamidine hydrochloride | IC50 | 120000.0 [1] |
 | Melagatran | IC50 | 20000.0 [1] |
 | 5-(N,N-Hexamethylene)amiloride | IC50 | 50000.0 [1] |
 | Anabaenopeptin F | IC50 | 3900.0 [1] |
 | Anabaenopeptin B | IC50 | 24000.0 [1] |
 | (3R,8R,11S,14S,17S,20S,23S,26S,29S,32S)-3-Amino-11-(carboxymethyl)-20-[3-(diaminomethylideneamino)propyl]-23-(hydroxymethyl)-17,26-bis[(4-hydroxyphenyl)methyl]-29-methyl-14-(2-methylpropyl)-2,10,13,16,19,22,25,28,31-nonaoxo-5,6-dithia-1,9,12,15,18,21,24,27,30-nonazabicyclo[30.3.0]pentatriacontane-8-carboxylic acid | Ki | 1000000.0 [1] |
 | Grassystatin A | IC50 | 10000.0 [1] |
 | Cyanopeptolin 1020 | IC50 | 3.9 [1] |
 | Unii-vwj4vvz3OU | Ki | 0.71 [1] |
 | (2,4-Dibromo-3-{[(4-carbamimidamidobutyl)carbamoyl]oxy}-6-hydroxyphenyl)acetic acid | IC50 | 1300.0 [1] |
 | 3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-[[4,5-dihydro-1,3-oxazol-2-yl(methyl)amino]methyl]thiophene-2-carboxamide | Ki | 10000.0 [1] |
 | 5-Chloro-N-((1R,2S)-2-(4-(2-oxopyridin-1(2H)-YL)benzamido) cyclopentyl)thiophene-2-carboxamide | Ki | 15000.0 [1] |
 | 3-Chloro-N-((1R,2S)-2-(4-(2-oxopyridin-1(2H)-YL)benzamido)cyclohexyl)-1H-indole-6-carboxamide | Ki | 15000.0 [1] |
 | (2R,15R)-2-[(1-Aminoisoquinolin-6-yl)amino]-7-cyclopropylsulfonyl-4,15,17-trimethyl-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaene-3,12-dione | Ki | 2300.0 [1] |
 | 3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-(methylaminomethyl)thiophene-2-carboxamide | Ki | 10000.0 [1] |
 | 3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-[[2-(methylamino)imidazol-1-yl]methyl]thiophene-2-carboxamide | Ki | 5000.0 [1] |
 | 5-Chloro-N-[(1R,2S)-2-[[4-[1-(pyrrolidin-1-ylmethyl)cyclopropyl]benzoyl]amino]cyclopentyl]thiophene-2-carboxamide | Ki | 10000.0 [1] |
 | 5-[[3-Ethoxycarbonyl-5-[(3-ethoxycarbonyl-5-hydroxy-6-methoxy-1-benzofuran-2-yl)methoxy]-6-methoxy-1-benzofuran-2-yl]methoxy]-6-methoxy-2-methyl-1-benzofuran-3-carboxylic acid | IC50 | 384000.0 [1] |
 | 2-[3-(6-Carbamimidoyl-4-methyl-4-phenyl-2,3-dihydro-1H-quinolin-2-yl)phenyl]-5-carbamoylbenzoic acid | Ki | 0.39 [1] |
 | 2-[2-[(4-Carbamimidoylphenyl)carbamoyl]-6-methoxypyridin-3-yl]-5-(2,2-dimethylpropylcarbamoyl)benzoic acid | IC50 | 4600.0 [1] |
 | 5-(2-(2-Fluoro-4-(2-oxopyridin-1(2H)-yl)phenyl)acetyl)-1-(4-methoxyphenyl)-1H-pyrazole-3-carboxamide | Ki | 15000.0 [1] |
 | 2-[(1-Aminoisoquinolin-6-yl)amino]-N-benzyl-2-(3-ethoxy-4-propan-2-yloxyphenyl)acetamide | Ki | 3900.0 [1] |
 | 2-[3-(6-Carbamimidoyl-4-methyl-4-phenyl-2,3-dihydro-1H-quinolin-2-yl)-5-(3-methylbutanoylamino)phenyl]-5-carbamoylbenzoic acid | Ki | 230.0 [1] |
 | (3R,4R)-3-N-(5-Chloropyridin-2-yl)-4-N-[2-fluoro-4-(2-oxopyridin-1-yl)phenyl]-1-propan-2-ylpyrrolidine-3,4-dicarboxamide | Ki | 33000.0 [1] |
 | 5-Chloro-N-((1R,2S)-2-(4-(2-oxopiperidin-1-yl)benzamido)cyclopentyl)thiophene-2-carboxamide | Ki | 10000.0 [1] |
 | (2S)-2-[[(2S)-2-[[(1R)-1-(4-Bromophenyl)ethyl]carbamoylamino]-3-pyridin-3-ylpropanoyl]amino]-N-[(2S)-5-(diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]-3-methylbutanamide | IC50 | 12.0 [1] |
 | (2S)-N-[(2S)-5-(Diaminomethylideneamino)-1-oxo-1-(1,3-thiazol-2-yl)pentan-2-yl]-2-[[(2R)-2-hydroxy-2-phenylacetyl]amino]-3-methylbutanamide | IC50 | 425.0 [1] |
 | N-[1-[4-(3-Amino-1H-indazol-6-yl)-6-oxo-1H-pyridin-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexane-1-carboxamide | Ki | 3.7 [1] |
 | 1-Amino-N-[(1S)-1-[4-(3-amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl]-5,6,7,8-tetrahydroisoquinoline-6-carboxamide | Ki | 2.5 [1] |
 | 4-(Aminomethyl)-N-[(1S)-2-phenyl-1-(5-phenyl-1H-imidazol-2-yl)ethyl]cyclohexane-1-carboxamide | Ki | 120.0 [1] |
 | N-[(1S)-1-[4-(3-Amino-1H-indazol-6-yl)-5-chloro-1H-imidazol-2-yl]-2-phenylethyl]-4-(aminomethyl)benzamide | Ki | 1.16 [1] |
 | Methyl N-[4-[2-[1-[[4-(aminomethyl)cyclohexanecarbonyl]amino]-2-phenylethyl]pyridin-4-yl]phenyl]carbamate | Ki | 12.0 [1] |
 | N-[1-[4-(3-Amino-1,2-benzoxazol-6-yl)pyridin-2-yl]-2-phenylethyl]-4-(aminomethyl)cyclohexane-1-carboxamide | Ki | 9.2 [1] |