| 2-[[[4-[[2-(2,4-Dichlorophenoxy)-1-oxoethyl]amino]phenyl]-oxomethyl]amino]benzoic acid | IC50 | 14070.0 [1], 16400.0 [2], 40570.0 [3] |
| (2R)-1-(2,4-Dichlorophenoxy)-3-[2-imino-3-(2-piperidin-1-ylethyl)benzimidazol-1-yl]propan-2-ol | IC50 | 14000.0 [1], 15710.0 [2], 32400.0 [3] |
| (4Z)-1-(3-Chlorophenyl)-4-[[5-(4,5-dimethyl-2-nitrophenyl)furan-2-yl]methylidene]pyrazolidine-3,5-dione | IC50 | 7400.0 [1], 8550.0 [2], 8950.0 [3] |
| (5E)-1-(1,3-Benzodioxol-5-yl)-5-[[5-(2-methoxy-4-nitrophenyl)furan-2-yl]methylidene]-1,3-diazinane-2,4,6-trione | IC50 | 4800.0 [1], 5530.0 [2], 62900.0 [3] |
| (5Z)-5-[[5-Chloro-2-[(4-nitrophenyl)methoxy]phenyl]methylidene]-1-(2-fluorophenyl)-1,3-diazinane-2,4,6-trione | IC50 | 14070.0 [1], 21920.0 [2], 38050.0 [3] |
| 3-[(4Z)-3-Methyl-4-[[5-(4-nitrophenyl)furan-2-yl]methylidene]-5-oxopyrazol-1-yl]benzoic acid | IC50 | 6710.0 [1], 8560.0 [2], 9190.0 [3] |
| 4-[[2-Ethoxy-4-[(E)-[1-[(2-fluorophenyl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]phenoxy]methyl]benzoic acid | IC50 | 2500.0 [1], 3510.0 [2], 18600.0 [3] |
| Razaxaban | Ki | 19700.0 [1] |
| 3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-[[4,5-dihydro-1,3-oxazol-2-yl(methyl)amino]methyl]thiophene-2-carboxamide | Ki | 10000.0 [1] |
| 2-(3-Amino-1,2-benzoxazol-5-yl)-N-[4-[2-[(dimethylamino)methyl]phenyl]-2-fluorophenyl]-5-(trifluoromethyl)pyrazole-3-carboxamide | Ki | 15000.0 [1] |
| 3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-(methylaminomethyl)thiophene-2-carboxamide | Ki | 10000.0 [1] |
| 3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-[[2-(methylamino)imidazol-1-yl]methyl]thiophene-2-carboxamide | Ki | 5000.0 [1] |
| (2R)-1-(3-Phenyl-4,5-dihydropyrazolo[4,3-a]carbazol-10-yl)-3-(propan-2-ylamino)propan-2-ol | IC50 | 3800.0 [1] |
| 2-(3-Amino-1,2-benzoxazol-5-yl)-N-[2-fluoro-4-[2-[[(3R)-3-hydroxypyrrolidin-1-yl]methyl]phenyl]phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamide | Ki | 5700.0 [1] |
| 2-(3-Amino-1,2-benzoxazol-5-yl)-N-[2-fluoro-4-[2-(pyrrolidin-1-ylmethyl)phenyl]phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamide | Ki | 13000.0 [1] |
| 3-[5-[(E)-[1-(4-Bromophenyl)-3-methyl-5-oxopyrazol-4-ylidene]methyl]furan-2-yl]benzoic acid | IC50 | 1810.0 [1] |