Coagulation factor V Inhibitors (IC50, Ki)

Name: Coagulation factor V Inhibitors (IC50, Ki)
Creator: AAT Bioquest
License: https://www.aatbio.com/tou.html

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	2-[[[4-[[2-(2,4-Dichlorophenoxy)-1-oxoethyl]amino]phenyl]-oxomethyl]amino]benzoic acid	IC50	14070.0 ^[1], 16400.0 ^[2], 40570.0 ^[3]
	(2R)-1-(2,4-Dichlorophenoxy)-3-[2-imino-3-(2-piperidin-1-ylethyl)benzimidazol-1-yl]propan-2-ol	IC50	14000.0 ^[1], 15710.0 ^[2], 32400.0 ^[3]
	(4Z)-1-(3-Chlorophenyl)-4-[[5-(4,5-dimethyl-2-nitrophenyl)furan-2-yl]methylidene]pyrazolidine-3,5-dione	IC50	7400.0 ^[1], 8550.0 ^[2], 8950.0 ^[3]
	(5E)-1-(1,3-Benzodioxol-5-yl)-5-[[5-(2-methoxy-4-nitrophenyl)furan-2-yl]methylidene]-1,3-diazinane-2,4,6-trione	IC50	4800.0 ^[1], 5530.0 ^[2], 62900.0 ^[3]
	(5Z)-5-[[5-Chloro-2-[(4-nitrophenyl)methoxy]phenyl]methylidene]-1-(2-fluorophenyl)-1,3-diazinane-2,4,6-trione	IC50	14070.0 ^[1], 21920.0 ^[2], 38050.0 ^[3]
	3-[(4Z)-3-Methyl-4-[[5-(4-nitrophenyl)furan-2-yl]methylidene]-5-oxopyrazol-1-yl]benzoic acid	IC50	6710.0 ^[1], 8560.0 ^[2], 9190.0 ^[3]
	4-[[2-Ethoxy-4-[(E)-[1-[(2-fluorophenyl)methyl]-2,5-dioxoimidazolidin-4-ylidene]methyl]phenoxy]methyl]benzoic acid	IC50	2500.0 ^[1], 3510.0 ^[2], 18600.0 ^[3]
	Razaxaban	Ki	19700.0 ^[1]
	3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-[[4,5-dihydro-1,3-oxazol-2-yl(methyl)amino]methyl]thiophene-2-carboxamide	Ki	10000.0 ^[1]
	2-(3-Amino-1,2-benzoxazol-5-yl)-N-[4-[2-[(dimethylamino)methyl]phenyl]-2-fluorophenyl]-5-(trifluoromethyl)pyrazole-3-carboxamide	Ki	15000.0 ^[1]
	3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-(methylaminomethyl)thiophene-2-carboxamide	Ki	10000.0 ^[1]
	3-Chloro-N-[4-chloro-2-[(5-chloropyridin-2-yl)carbamoyl]-6-methoxyphenyl]-4-[[2-(methylamino)imidazol-1-yl]methyl]thiophene-2-carboxamide	Ki	5000.0 ^[1]
	(2R)-1-(3-Phenyl-4,5-dihydropyrazolo[4,3-a]carbazol-10-yl)-3-(propan-2-ylamino)propan-2-ol	IC50	3800.0 ^[1]
	2-(3-Amino-1,2-benzoxazol-5-yl)-N-[2-fluoro-4-[2-[[(3R)-3-hydroxypyrrolidin-1-yl]methyl]phenyl]phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamide	Ki	5700.0 ^[1]
	2-(3-Amino-1,2-benzoxazol-5-yl)-N-[2-fluoro-4-[2-(pyrrolidin-1-ylmethyl)phenyl]phenyl]-5-(trifluoromethyl)pyrazole-3-carboxamide	Ki	13000.0 ^[1]
	3-[5-[(E)-[1-(4-Bromophenyl)-3-methyl-5-oxopyrazol-4-ylidene]methyl]furan-2-yl]benzoic acid	IC50	1810.0 ^[1]

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MLA	"Quest Database™ Coagulation factor V Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 1 Apr. 2025, https://www.aatbio.com/data-sets/coagulation-factor-v-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, April 1). Quest Database™ Coagulation factor V Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/coagulation-factor-v-inhibitors-ic50-ki.
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Coagulation factor V Inhibitors (IC50, Ki)

References

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