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Cell division cycle 7-related protein kinase Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-(Pyridin-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-oneIC5010.0 [1]
8-Chloro-2-[(2s)-Pyrrolidin-2-Yl][1]benzofuro[3,2-D]pyrimidin-4(3h)-OneIC503.4 [1], 118.0 [2], 140.0 [3]
N-[5-(1-Benzyltriazol-4-yl)-1H-indazol-3-yl]benzamideKi0.4 [1], 0.5 [2], 0.6 [3]
4-(4-Hydroxy-3-methylphenyl)-6-phenylpyrimidin-2(1H)-oneIC501.4 [1], 3.0 [2]
2-(2-Amino-pyrimidin-4-yl)-1,5,6,7-tetrahydro-pyrrolo[3,2-c]pyridin-4-oneIC507.0 [1]
8-Bromanyl-2-[[(3s)-3-Oxidanylpyrrolidin-1-Yl]methyl]-3h-[1]benzofuro[3,2-D]pyrimidin-4-OneIC507.7 [1], 1471.0 [2]
2-[[(3S)-3-Aminopyrrolidin-1-yl]methyl]-8-bromo-3H-[1]benzofuro[3,2-d]pyrimidin-4-oneIC5010.0 [1], 625.0 [2]
8-Bromo-2-(pyrrolidin-1-ylmethyl)[1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC503.7 [1], 353.0 [2]
8-Bromo-2-[[(3R)-3-hydroxypyrrolidin-1-yl]methyl]-3H-[1]benzofuro[3,2-d]pyrimidin-4-oneIC505.5 [1], 1805.0 [2]
1-(2-Aminopyrimidin-4-yl)indole-6-carbonitrileIC5075.0 [1], 5000.0 [2]
1-[(8-Bromo-4-oxo-3,4-dihydro[1]benzofuro[3,2-d]pyrimidin-2-yl)methyl]pyrrolidine-3-carboxylic acidIC5013.0 [1], 40000.0 [2]
8-Bromo-2-[(2S,4R)-4-hydroxypyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC509.1 [1], 440.0 [2]
2-Azetidin-3-yl-8-bromo[1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC507.7 [1], 2536.0 [2]
8-Bromo-2-{[(3S)-3-(methyloxy)pyrrolidin-1-yl]methyl}[1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC5011.0 [1], 362.0 [2]
8-Bromo-2-piperidin-4-yl[1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC506.2 [1], 1434.0 [2]
8-Bromo-2-piperidin-3-yl[1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC5015.0 [1], 2356.0 [2]
8-Bromo-2-[(2S,4S)-4-fluoropyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC5011.0 [1], 566.0 [2]
2-[(2S,4R)-4-Fluoropyrrolidin-2-yl]-8-(methyloxy)[1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC503.9 [1], 292.0 [2]
8-Chloro-2-[(2S,4R)-4-fluoropyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC504.0 [1], 167.0 [2]
2-(1-Aminoethyl)-8-bromo-3H-[1]benzofuro[3,2-d]pyrimidin-4-oneIC507.9 [1], 874.0 [2]
8-(Methyloxy)-2-[(2S)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC506.1 [1], 1374.0 [2]
8-Bromo-2-[(2R)-pyrrolidin-2-yl]-3H-[1]benzofuro[3,2-d]pyrimidin-4-oneIC5070.0 [1], 4592.0 [2]
8-Bromo-2-[(2S)-pyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC504.8 [1], 75.0 [2]
8-Bromo-2-[(2S,4R)-4-fluoropyrrolidin-2-yl][1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC503.7 [1], 82.0 [2]
8-Bromo-2-[(2S)-1-methylpyrrolidin-2-yl]-3H-[1]benzofuro[3,2-d]pyrimidin-4-oneIC507.3 [1], 802.0 [2]
4-(1H-Indol-1-yl)pyrimidin-2-amineIC504700.0 [1], 50000.0 [2]
5-(1-Benzyl-5-phenyltriazol-4-yl)-1H-indazol-3-amineKi1.2 [1], 2.1 [2]
5-[1-Benzyl-5-(4-fluorophenyl)triazol-4-yl]-1H-indazol-3-amineKi0.8 [1], 2.2 [2]
5-(1-Benzyl-5-methyltriazol-4-yl)-1H-indazol-3-amineKi17.0 [1], 23.0 [2]
N-[5-(1-Benzyltriazol-4-yl)-1H-indazol-3-yl]-3-fluorobenzamideKi0.5 [1], 1.0 [2]
1-(6-Aminopyrimidin-4-yl)pyrrolo[2,3-b]pyridine-6-carbonitrileIC509.0 [1], 1370.0 [2]
1-(2-Aminopyridin-4-yl)indole-6-carbonitrileIC509000.0 [1], 50000.0 [2]
2-Pyrimidinamine, 4-(1H-pyrrolo[2,3-b]pyridin-1-yl)-IC5026700.0 [1], 50000.0 [2]
2-Pyrimidinamine, 4-(6-chloro-1H-pyrrolo[3,2-c]pyridin-1-yl)-IC50360.0 [1], 50000.0 [2]
4-[3-(2-Chloropyridin-3-yl)pyrrolo[3,2-c]pyridin-1-yl]pyrimidin-2-amineIC507.0 [1], 850.0 [2]
4-[6-Chloro-3-(2-chloropyridin-3-yl)pyrrolo[3,2-c]pyridin-1-yl]pyrimidin-2-amineIC5030.0 [1], 2300.0 [2]
N-[5-(1-Benzyl-5-phenyltriazol-4-yl)-1H-indazol-3-yl]benzamideKi0.8 [1], 0.9 [2]
N-[5-(1-Benzyl-5-cyclopropyltriazol-4-yl)-1H-indazol-3-yl]-3-fluorobenzamideKi0.9 [1], 2.4 [2]
MilciclibIC5010000.0 [1]
Pha-793887IC5010000.0 [1]
CID 59604787IC503500.0 [1]
5-[2,4-Dihydroxy-6-(4-Nitrophenoxy)phenyl]-N-(1-Methylpiperidin-4-Yl)-1,2-Oxazole-3-CarboxamideIC5010.0 [1]
8-[2-Methoxy-5-(4-methylpiperazin-1-yl)anilino]-1-methyl-4,5-dihydropyrazolo[4,3-h]quinazoline-3-carboxamideIC5010000.0 [1]
5-(2-Aminopyrimidin-4-yl)-2-phenyl-1H-pyrrole-3-carboxamideIC5022.0 [1]
8-Bromo[1]benzofuro[3,2-d]pyrimidin-4(3H)-oneIC502000.0 [1]
4-(1H-Indazol-5-yl)-6-phenylpyrimidin-2(1H)-oneIC5010.0 [1]
2-(2-Chloropyridin-4-yl)-6,7-dihydro-1H-pyrrolo[3,2-c]pyridin-4(5H)-oneIC50147.0 [1]
(7S)-2-(2-Aminopyrimidin-4-yl)-7-(2-fluoroethyl)-1,5,6,7-tetrahydro-4H-pyrrolo[3,2-c]pyridin-4-oneIC502.0 [1]
1H,4H,5H,6H,7H-Pyrrolo[3,2-c]pyridin-4-oneIC505000.0 [1]
2,2-Dimethyl-7-(2-oxo-3H-imidazo[4,5-b]pyridin-1-yl)-1-[(1R)-1-phenylethyl]-3H-quinazolin-4-oneIC501000.0 [1]
3-[(4-Morpholin-4-ylbenzoyl)amino]-N-[(1S)-1-phenyl-2-pyrrolidin-1-ylethyl]-1H-thieno[3,2-c]pyrazole-5-carboxamideIC501970.0 [1]
2-[[(3R)-3-Aminopyrrolidin-1-yl]methyl]-8-bromo-3H-[1]benzofuro[3,2-d]pyrimidin-4-oneIC50207.0 [1]
5-(1-Benzyl-1h-1,2,3-triazol-4-yl)-1h-indazol-3-amineKi12.0 [1]
4-[[4-Chloro-6-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-yl]amino]cyclohexan-1-olKi0.16 [1]
1-N-[4-Chloro-6-(1H-pyrrolo[2,3-b]pyridin-3-yl)pyrimidin-2-yl]-4-N,4-N-dimethylcyclohexane-1,4-diamineKi0.32 [1]
N-[5-(1-Benzyltriazol-4-yl)-1H-indazol-3-yl]-3-chlorobenzamideKi0.79 [1]
3-Amino-6-{4-Chloro-3-[(2,3-Difluorophenyl)sulfamoyl]phenyl}-N-Methylpyrazine-2-CarboxamideIC503600.0 [1]
6-(Cyclohexylamino)-4-(1H-pyrrolo[2,3-b]pyridin-3-yl)-1H-pyridin-2-oneKi0.28 [1]
3-Amino-6-[4-chloro-3-[(3-fluoro-2-methylphenyl)sulfamoyl]phenyl]-N-methylpyrazine-2-carboxamideIC503600.0 [1]
4-(6-Chloro-1H-indol-1-yl)pyrimidin-2-amineIC5066.0 [1]
4-(6-Bromoindol-1-yl)pyrimidin-2-amineIC50350.0 [1]
N-[5-(2,2-Dimethylpropanoyl)-6,6-dimethyl-1,4-dihydropyrrolo[3,4-c]pyrazol-3-yl]-3,5-difluorobenzamideIC5010000.0 [1]
2-(9H-Purin-6-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC50178.0 [1]
2-(2-Aminopyrimidin-4-yl)-7-methyl-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC506.0 [1]
2-(2-Aminopyrimidin-4-yl)-7-phenyl-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC5019.0 [1]
2-(2-Aminopyrimidin-4-yl)-6,6-dimethyl-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC5064.0 [1]
2-[2-(Benzylamino)pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC50220.0 [1]
2-[2-(Phenylamino)pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC507.0 [1]
2-(2-Aminopyrimidin-4-yl)-6-(propan-2-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC5012.0 [1]
2-{2-[(Cyclohexylmethyl)amino]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC50655.0 [1]
2-(2-Aminopyrimidin-4-yl)-7-(propan-2-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC504.0 [1]
7-Ethyl-2-(pyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC502.0 [1]
8,9,10,11-Tetrahydro-3,8,11-triaza-benzo[a]fluoren-7-oneIC502.0 [1]
N-[4-(4-Oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl)pyrimidin-2-yl]benzamideIC50262.0 [1]
2-(2-Aminopyrimidin-4-yl)-6-methyl-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC5026.0 [1]
2-[2-(Propylamino)pyrimidin-4-yl]-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC50259.0 [1]
2-(2-Aminopyrimidin-4-yl)-6-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC508.0 [1]
2-{2-[(2-Methylpropyl)amino]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC50636.0 [1]
2-(2-Aminopyrimidin-4-yl)-7,7-diethyl-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC505.0 [1]
3-Methyl-2-(pyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC5045.0 [1]
2-{1H-Pyrrolo[2,3-b]pyridin-4-yl}-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC5014.0 [1]
2-(3-Fluoropyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC509.0 [1]
7,7-Dimethyl-2-(pyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC503.0 [1]
7-Methyl-2-(pyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC5010.0 [1]
7,7-Diethyl-2-(pyridin-4-yl)-1H,4H,5H,6H,7H-pyrrolo[3,2-c]pyridin-4-oneIC506.0 [1]
2-(4-Piperazin-1-ylphenyl)-1H-pyrrolo[2,3-b]pyridine-4-carbonitrileIC5060.0 [1]
1-Methyl-2-(4-piperazin-1-ylphenyl)pyrrolo[2,3-b]pyridine-4-carbonitrileIC5010000.0 [1]
2-Phenyl-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5050.0 [1]
2-(2-Methylmorpholin-4-yl)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5066.0 [1]
2-(4-Methylpiperidin-1-yl)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC50105.0 [1]
2-(Cyclohexylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5021.0 [1]
2-(Benzylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5020.0 [1]
2-(2-Hydroxyethylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5037.0 [1]
2-(3,3-Dimethylbutylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5024.0 [1]
2-(Furan-2-ylmethylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5015.0 [1]
2-(Cyclopropylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5033.0 [1]
5-[(Z)-Pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-2-(thiophen-2-ylmethylamino)-1H-imidazol-4-olIC5018.0 [1]
2-(Oxolan-2-ylmethylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5021.0 [1]
2-(Pentylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC5035.0 [1]
2-(Heptylamino)-5-[(Z)-pyrrolo[2,3-b]pyridin-3-ylidenemethyl]-1H-imidazol-4-olIC50247.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cell division cycle 7-related protein kinase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/cell-division-cycle-7-related-protein-kinase-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Cell division cycle 7-related protein kinase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cell-division-cycle-7-related-protein-kinase-inhibitors-ic50-ki.
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