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CDK9/Cyclin K Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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StaurosporineIC5013.0 [1]
4-[[[4-[5-Chloro-2-[[4-(2-methoxyethylamino)cyclohexyl]amino]pyridin-4-yl]-1,3-thiazol-2-yl]amino]methyl]oxane-4-carbonitrileIC506.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC5038.9 [1]
2-[(E)-2-(2,6-Dichlorophenyl)ethenyl]-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-oneIC50412.0 [1]
4-[[[4-[5-Chloro-2-[[4-[[(2S)-1-methoxypropan-2-yl]amino]cyclohexyl]amino]pyridin-4-yl]-1,3-thiazol-2-yl]amino]methyl]oxane-4-carbonitrileIC5010.0 [1]
4-[[[4-[5-Chloro-2-[[4-[[(2R)-1-methoxypropan-2-yl]amino]cyclohexyl]amino]pyridin-4-yl]-1,3-thiazol-2-yl]amino]methyl]oxane-4-carbonitrileIC509.0 [1]
N-[4-[[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]amino]cyclohexyl]acetamideIC50101.0 [1]
N-[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-4-fluorobenzamideIC502300.0 [1]
Tert-butyl N-[4-(5-chloro-2-fluoropyridin-4-yl)-1,3-thiazol-2-yl]carbamateIC5010000.0 [1]
4-N-[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-ethoxyethyl)cyclohexane-1,4-diamineIC5051.0 [1]
4-N-[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]cyclohexane-1,4-diamineIC5022.0 [1]
4-N-[5-Chloro-4-[2-(oxan-4-ylmethylsulfanyl)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5014.0 [1]
4-[5-Chloro-2-(2-methoxyethylamino)pyridin-4-yl]-N-(oxan-4-ylmethyl)-1,3-thiazol-2-amineIC501040.0 [1]
N-[4-[[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]amino]cyclohexyl]-2-methoxyacetamideIC501890.0 [1]
1-N-(2-Methoxyethyl)-4-N-[4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]cyclohexane-1,4-diamineIC50114.0 [1]
4-N-[5-Chloro-4-[2-(2,2,2-trifluoroethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5017.0 [1]
4-N-[4-[2-(Benzylamino)-1,3-thiazol-4-yl]-5-chloropyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5014.0 [1]
4-N-[5-Chloro-4-[2-(cyclopropylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5096.0 [1]
4-N-[5-Chloro-4-[2-(oxolan-3-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5090.0 [1]
4-(5-Chloro-2-fluoropyridin-4-yl)-N-(oxan-4-ylmethyl)-1,3-thiazol-2-amineIC50557.0 [1]
1-N-(2-Methoxyethyl)-4-N-[5-methyl-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]cyclohexane-1,4-diamineIC50253.0 [1]
4-N-[5-Chloro-4-[2-(cyclohexylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5027.0 [1]
4-[2-[(4-Aminocyclohexyl)methylamino]-5-chloropyridin-4-yl]-N-(oxan-4-ylmethyl)-1,3-thiazol-2-amineIC5084.0 [1]
4-N-[5-Chloro-4-[2-(methylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC50101.0 [1]
4-N-[4-[2-(2-Adamantylmethylamino)-1,3-thiazol-4-yl]-5-chloropyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5094.0 [1]
4-N-[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC502.0 [1]
4-N-[5-Chloro-4-[2-(oxan-4-ylmethoxy)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5028.0 [1]
4-[5-Chloro-2-[4-(2-methoxyethylamino)cyclohexyl]oxypyridin-4-yl]-N-(oxan-4-ylmethyl)-1,3-thiazol-2-amineIC501670.0 [1]
4-N-[5-Chloro-4-[2-(cyclopentylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC5080.0 [1]
4-N-[5-Chloro-4-[2-[(4-fluorophenyl)methylamino]-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC502.0 [1]
1-N-[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-4-N-[(2R)-1-methoxypropan-2-yl]cyclohexane-1,4-diamineIC50733.0 [1]
4-(2-Anilino-5-chloropyridin-4-yl)-N-(oxan-4-ylmethyl)-1,3-thiazol-2-amineIC50238.0 [1]
4-N-[5-Chloro-4-[2-(cyclobutylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(2-methoxyethyl)cyclohexane-1,4-diamineIC50107.0 [1]
4-N-[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-1-N-(3-methoxypropyl)cyclohexane-1,4-diamineIC5012.0 [1]
N-[4-[[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]amino]cyclohexyl]cyclopropanecarboxamideIC50150.0 [1]
1-N-[5-Chloro-4-[2-(oxan-4-ylmethylamino)-1,3-thiazol-4-yl]pyridin-2-yl]-4-N-[(2S)-1-methoxypropan-2-yl]cyclohexane-1,4-diamineIC5010000.0 [1]
4-{[4-Amino-5-(2-Nitrobenzoyl)-1,3-Thiazol-2-Yl]amino}benzenesulfonamideIC5013.0 [1]
Items per page: 1 - 10 of 38
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References

This online tool may be cited as follows

MLA

"Quest Database™ CDK9/Cyclin K Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/cdk9-cyclin-k-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ CDK9/Cyclin K Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk9-cyclin-k-inhibitors-ic50-ki.
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