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CDK7/Cyclin H/MNAT1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
AbemaciclibIC503112.0 [1]
AbemaciclibKi3910.0 [1]
1-[4-[4-[[5-(Oxan-4-yl)pyrrolo[2,1-f][1,2,4]triazin-4-yl]amino]cyclohexyl]piperazin-1-yl]ethanoneIC50516.0 [1], 30000.0 [2]
1-[4-[4-[(5-Propan-2-ylpyrrolo[2,1-f][1,2,4]triazin-4-yl)amino]cyclohexyl]piperazin-1-yl]ethanoneIC502310.0 [1], 30000.0 [2]
StaurosporineIC50120.0 [1]
AlvocidibIC50514.0 [1]
DinaciclibIC50170.0 [1]
Sns-032IC5062.0 [1]
4-(2,6-Dichlorobenzamido)-N-(piperidin-4-yl)-1H-pyrazole-3-carboxamideKi2800.0 [1]
(16E)-14-Methyl-20-oxa-5,7,14,27-tetrazatetracyclo[19.3.1.12,6.18,12]heptacosa-1(25),2(27),3,5,8,10,12(26),16,21,23-decaeneIC503.0 [1]
BS-181IC50134.0 [1]
CID 23643976IC502870.0 [1]
(3-((6-(2-Methoxyphenyl)pyrimidin-4-yl)amino)phenyl)methanesulfonamideIC5020000.0 [1]
CID 78357764IC50246.0 [1]
CDK12 inhibitor 2IC5010000.0 [1]
4-[[[4-[5-Chloro-2-[[4-(2-methoxyethylamino)cyclohexyl]amino]pyridin-4-yl]-1,3-thiazol-2-yl]amino]methyl]oxane-4-carbonitrileIC501720.0 [1]
2-Anilino-7-[(1S)-4-hydroxy-2,3-dihydro-1H-inden-1-yl]-5,5-dimethylpyrrolo[2,3-d]pyrimidin-6-oneIC50793.0 [1]
1-[4-[4-Amino-3-[4-(2-morpholin-4-ylethoxy)phenyl]pyrazolo[3,4-d]pyrimidin-1-yl]phenyl]-3-(5-tert-butyl-1,2-oxazol-3-yl)ureaIC5010000.0 [1]
(2S,3R)-3-[2-[4-(Cyclopropylsulfonimidoyl)anilino]-5-(trifluoromethyl)pyrimidin-4-yl]oxybutan-2-olIC5025.0 [1]
2-[5-[[[2-[(4-Aminocyclohexyl)amino]-9-cyclopentylpurin-6-yl]amino]methyl]pyridin-2-yl]phenolIC50306.0 [1]
2-[3-[3-(1H-Pyrrolo[2,3-b]pyridin-3-yl)propyl]triazol-4-yl]-1H-pyrrolo[2,3-b]pyridineIC5050000.0 [1]
N-[3-[6-[(3-Bromophenyl)methylamino]purin-9-yl]cyclobutyl]-6-methylpyridine-2-carboxamideIC50359.0 [1]
N-[3-[6-[(3-Chlorophenyl)methylamino]purin-9-yl]cyclobutyl]-6-methylpyridine-2-carboxamideIC50319.0 [1]
3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-(1-methylpyrazol-4-yl)phenyl]ureaIC5010000.0 [1]
6-[[1-[4-(1-Methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]amino]pyridine-3-carbonitrileIC5010000.0 [1]
[(2S,3S,4S,5R)-5-(6-Bromo-5-carbamoyl-4-imino-7H-pyrrolo[2,3-d]pyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl 2-methylpropanoateIC501200.0 [1]
N-[1-[4-(4-Fluoroanilino)pyrimidin-2-yl]piperidin-4-yl]-4-methoxybenzamideIC5089.8 [1]
5-N-(2-Aminocyclohexyl)-7-N-benzyl-3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamineIC50100000.0 [1]
5-N-(4-Aminocyclohexyl)-7-N-benzyl-3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamineIC50100000.0 [1]
6-(Benzimidazol-1-yl)-N-[5-[2-(dimethylamino)ethoxy]pyridin-2-yl]pyrimidin-4-amineIC501100.0 [1]
Items per page: 1 - 10 of 30
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References

This online tool may be cited as follows

MLA

"Quest Database™ CDK7/Cyclin H/MNAT1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/cdk7-cyclin-h-mnat1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ CDK7/Cyclin H/MNAT1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk7-cyclin-h-mnat1-inhibitors-ic50-ki.
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