 | Abemaciclib | IC50 | 10.0 [1] |
 | Abemaciclib | Ki | 10.0 [1] |
 | N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamide | IC50 | 4.24 [1], 10.0 [2] |
 | Staurosporine | IC50 | 2.9 [1] |
 | Seliciclib | IC50 | 23500.0 [1] |
 | Palbociclib | IC50 | 3.76 [1] |
 | Fascaplysin | IC50 | 3400.0 [1] |
 | (2S,3S)-3-((7-(Benzylamino)-3-isopropylpyrazolo[1,5-a]pyrimidin-5-yl)amino)butane-1,2,4-triol | IC50 | 35500.0 [1] |
 | CID 56649281 | IC50 | 9.82 [1] |
 | N'-(Pyrrolidino[2,1-B]isoindolin-4-ON-8-YL)-N-(pyridin-2-YL)urea | IC50 | 71.0 [1] |
 | 2-Bromo-N-(2,5-dichlorothiophen-3-yl)sulfonyl-N-phenylacetamide | IC50 | 34900.0 [1] |
 | 6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one | IC50 | 10000.0 [1] |
 | 4-Methyl-N-[3-(trifluoromethyl)phenyl]benzenesulfonamide | IC50 | 208800.0 [1] |
 | 2-[(E)-2-(2,6-Dichlorophenyl)ethenyl]-5,7-dihydroxy-8-[(3S,4R)-3-hydroxy-1-methylpiperidin-4-yl]chromen-4-one | IC50 | 45.0 [1] |
 | 2,4,5-Trichloro-N-[3-(trifluoromethyl)phenyl]benzenesulfonamide | IC50 | 58800.0 [1] |
 | N-(6-Methoxyquinolin-8-yl)-N',N'-bis(3-methylbutyl)propane-1,3-diamine | IC50 | 325000.0 [1] |
 | (2S)-2-[Bis(2-methylpropyl)amino]-1-[(6-methoxy-2-methylquinolin-8-yl)amino]propan-2-ol | IC50 | 691000.0 [1] |
 | 5-N-(2-Aminocyclohexyl)-7-N-benzyl-3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamine | IC50 | 100000.0 [1] |
 | CID 49798457 | IC50 | 110400.0 [1] |
 | 2,5-Dichloro-N-p-tolylthiophene-3-sulfonamide | IC50 | 51300.0 [1] |
 | 2,5-Dichloro-N-(4-methylphenyl)-N-(trichloromethylsulfanyl)thiophene-3-sulfonamide | IC50 | 18000.0 [1] |
 | 5-N-(4-Aminocyclohexyl)-7-N-benzyl-3-propan-2-yl-2H-pyrazolo[4,3-d]pyrimidine-5,7-diamine | IC50 | 91000.0 [1] |
 | N-[(4-Methoxyphenyl)methyl]-[1]benzofuro[2,3-b]pyridin-4-amine | IC50 | 129000.0 [1] |
 | 4-Phenyl-[1]benzofuro[2,3-b]pyridine-3,6-diol | Ki | 773000.0 [1] |
 | 4-{[4-Amino-5-(2-Nitrobenzoyl)-1,3-Thiazol-2-Yl]amino}benzenesulfonamide | IC50 | 6.6 [1] |
 | N-[4-(Morpholin-4-ylmethyl)phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamide | IC50 | 3.88 [1] |
 | 4-(Furo[2,3-d]pyrimidin-4-ylamino)-N-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1H-pyrazole-5-carboxamide | IC50 | 5.09 [1] |
 | CID 72195175 | IC50 | 1.96 [1] |
 | N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(thieno[3,2-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamide | IC50 | 4.11 [1] |