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CDK2/Cyclin A1 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
StaurosporineIC500.5 [1]
CID 44814409IC5010000.0 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC505.85 [1]
4-[(6-Bromoquinolin-4-yl)amino]-N-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1H-pyrazole-5-carboxamideIC505.74 [1]
4-[(7-Methoxyquinolin-4-yl)amino]-N-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1H-pyrazole-5-carboxamideIC50697.0 [1]
4-[(2-Chloroquinazolin-4-yl)amino]-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamideIC5058.63 [1]
4-[(6-Bromoquinolin-4-yl)amino]-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamideIC5024.15 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(quinazolin-4-ylamino)-1H-pyrazole-5-carboxamideIC508.27 [1]
N-[4-(Morpholin-4-ylmethyl)phenyl]-4-(quinazolin-4-ylamino)-1H-pyrazole-5-carboxamideIC505.3 [1]
4-[(6-Ethylthieno[2,3-d]pyrimidin-4-yl)amino]-N-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1H-pyrazole-5-carboxamideIC501.87 [1]
4-[(6-Methoxyquinazolin-4-yl)amino]-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamideIC5029.8 [1]
4-[(6-Ethylthieno[2,3-d]pyrimidin-4-yl)amino]-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamideIC503.3 [1]
4-(Isoquinolin-1-ylamino)-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamideIC50287.19 [1]
N-[4-(Piperazin-1-ylmethyl)phenyl]-4-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC504.49 [1]
N-[4-[(Cyclopropylamino)methyl]phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC502.05 [1]
N-[4-(Diethylaminomethyl)phenyl]-4-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC5013.6 [1]
N-[4-(Diethylaminomethyl)phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC501.59 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-[(6-propan-2-ylthieno[2,3-d]pyrimidin-4-yl)amino]-1H-pyrazole-5-carboxamideIC503.89 [1]
N-[4-(Piperazin-1-ylmethyl)phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC502.08 [1]
N-[4-(Morpholin-4-ylmethyl)phenyl]-4-[(6-propan-2-ylthieno[2,3-d]pyrimidin-4-yl)amino]-1H-pyrazole-5-carboxamideIC509.85 [1]
N-[4-[(4-Methyl-1,4-diazepan-1-yl)methyl]phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC503.03 [1]
5-[(2,6-Dichlorobenzoyl)amino]-N-piperidin-4-yl-1H-pyrazole-4-carboxamideIC5057.2 [1]
(1S,3R)-3-Acetamido-N-[4-(4-fluoro-2-methoxyphenyl)pyridin-2-yl]cyclohexane-1-carboxamideIC5094.0 [1]
4-Benzamido-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamideIC50318.21 [1]
(1R,3S)-3-Acetamido-N-[4-(4-fluoro-2-methoxyphenyl)pyridin-2-yl]cyclopentane-1-carboxamideIC50913.0 [1]
4-{[4-Amino-5-(2-Nitrobenzoyl)-1,3-Thiazol-2-Yl]amino}benzenesulfonamideIC501.8 [1]
N-[4-(Morpholin-4-ylmethyl)phenyl]-4-(thieno[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC503.36 [1]
4-(Furo[2,3-d]pyrimidin-4-ylamino)-N-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1H-pyrazole-5-carboxamideIC5016.5 [1]
CID 72195175IC502.47 [1]
N-[4-(Morpholin-4-ylmethyl)phenyl]-4-(7H-pyrrolo[2,3-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC507.25 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-(thieno[3,2-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC509.32 [1]
N-[4-(Morpholin-4-ylmethyl)phenyl]-4-(thieno[3,2-d]pyrimidin-4-ylamino)-1H-pyrazole-5-carboxamideIC5011.64 [1]
4-[(5,6-Dimethylthieno[2,3-d]pyrimidin-4-yl)amino]-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamideIC507.34 [1]
4-[(5,6-Dimethylthieno[2,3-d]pyrimidin-4-yl)amino]-N-[4-[(4-methylpiperazin-1-yl)methyl]phenyl]-1H-pyrazole-5-carboxamideIC501.9 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-[(6-methylthieno[2,3-d]pyrimidin-4-yl)amino]-1H-pyrazole-5-carboxamideIC501.74 [1]
4-[(5-Methylthieno[2,3-d]pyrimidin-4-yl)amino]-N-[4-(morpholin-4-ylmethyl)phenyl]-1H-pyrazole-5-carboxamideIC501.08 [1]
N-[4-[(4-Methylpiperazin-1-yl)methyl]phenyl]-4-[(5-methylthieno[2,3-d]pyrimidin-4-yl)amino]-1H-pyrazole-5-carboxamideIC504.49 [1]
Items per page: 1 - 10 of 38
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References

This online tool may be cited as follows

MLA

"Quest Database™ CDK2/Cyclin A1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/cdk2-cyclin-a1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 22). Quest Database™ CDK2/Cyclin A1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk2-cyclin-a1-inhibitors-ic50-ki.
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