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CDK12/Cyclin K Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
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Standard Values (in nM)
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▼
3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-(1-methylpyrazol-4-yl)phenyl]ureaIC5063.0 [1], 30000.0 [2]
N-[4-[(5-Cyanopyridin-2-yl)amino]cyclohexyl]-N-[4-(1-methylpyrazol-4-yl)phenyl]acetamideIC50130.0 [1], 30000.0 [2]
StaurosporineIC5053.0 [1]
CDK12 inhibitor 2IC5052.0 [1]
N-[4-(1-Methylpyrazol-4-yl)phenyl]-N-[4-(quinazolin-2-ylamino)cyclohexyl]acetamideIC5013.0 [1]
3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-(1-methyl-2-oxopyridin-4-yl)phenyl]ureaIC5044.0 [1]
N-[4-[(5-Cyanopyridin-2-yl)amino]cyclohexyl]-N-[4-(1-methylpyrazol-4-yl)phenyl]methanesulfonamideIC50110.0 [1]
Benzyl N-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-N-[4-(1-methylpyrazol-4-yl)phenyl]carbamateIC50640.0 [1]
1-[4-[(5-Cyanopyridin-2-yl)amino]cyclohexyl]-3-ethyl-1-[4-(1-methylpyrazol-4-yl)phenyl]ureaIC50460.0 [1]
6-[[1-[4-(1-Methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]amino]pyridine-3-carbonitrileIC50360.0 [1]
N-[1-[4-(1-Methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]pyridin-2-amineIC5030000.0 [1]
3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-(4-pyridin-3-ylphenyl)ureaIC5059.0 [1]
3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-phenylureaIC5063.0 [1]
Methyl N-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-N-[4-(1-methylpyrazol-4-yl)phenyl]carbamateIC50200.0 [1]
6-[[1-[4-(1-Methylpyrazol-4-yl)benzoyl]piperidin-4-yl]amino]pyridine-3-carbonitrileIC5023000.0 [1]
2-[[1-[4-(1-Methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]amino]pyridine-4-carbonitrileIC5030000.0 [1]
4-[[1-[4-(1-Methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]amino]benzonitrileIC5030000.0 [1]
6-[[1-[[4-(1-Methylpyrazol-4-yl)phenyl]methyl]piperidin-4-yl]amino]pyridine-3-carbonitrileIC5016000.0 [1]
3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-(1-methyl-6-oxopyridin-2-yl)phenyl]ureaIC50310.0 [1]
6-[[4-[4-(1-Methylpyrazol-4-yl)anilino]cyclohexyl]amino]pyridine-3-carbonitrileIC508600.0 [1]
[(2S,3S,4S,5R)-5-(6-Bromo-5-carbamoyl-4-imino-7H-pyrrolo[2,3-d]pyrimidin-1-yl)-3,4-dihydroxyoxolan-2-yl]methyl 2-methylpropanoateIC50110.0 [1]
1-[4-[(5-Cyanopyridin-2-yl)amino]cyclohexyl]-3-(cyclohexylmethyl)-1-[4-(1-methylpyrazol-4-yl)phenyl]ureaIC5099.0 [1]
6-[[1-[4-(1-Methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]amino]pyridine-2-carbonitrileIC5030000.0 [1]
N-[4-[(5-Cyanopyridin-2-yl)amino]cyclohexyl]-N-[4-(1-methylpyrazol-4-yl)phenyl]-3-phenylpropanamideIC50160.0 [1]
3-Benzyl-1-[4-[(5-cyanopyridin-2-yl)amino]cyclohexyl]-1-[4-(1-methyl-2-oxopyridin-3-yl)phenyl]ureaIC50250.0 [1]
5-Methoxy-N-[1-[4-(1-methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]pyridin-2-amineIC5030000.0 [1]
6-[Methyl-[1-[4-(1-methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]amino]pyridine-3-carbonitrileIC5030000.0 [1]
N-[1-[4-(1-Methylpyrazol-4-yl)phenyl]sulfonylpiperidin-4-yl]-5-(trifluoromethyl)pyridin-2-amineIC501800.0 [1]
Items per page: 1 - 10 of 28
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References

This online tool may be cited as follows

MLA

"Quest Database™ CDK12/Cyclin K Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Dec. 2024, https://www.aatbio.com/data-sets/cdk12-cyclin-k-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 22). Quest Database™ CDK12/Cyclin K Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cdk12-cyclin-k-inhibitors-ic50-ki.
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