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Cathepsin F Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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TelaprevirIC5010000.0 [1]
BoceprevirIC501100.0 [1]
OdanacatibIC50795.0 [1]
(1R,21S,24S)-21-Tert-butyl-N-[(1R,2S)-1-(cyclopropylsulfonylcarbamoyl)-2-ethenylcyclopropyl]-16,16-dimethyl-3,19,22-trioxo-2,18-dioxa-4,20,23-triazatetracyclo[21.2.1.14,7.06,11]heptacosa-6(11),7,9-triene-24-carboxamideIC5010000.0 [1]
N-[(2S)-3-Cyclohexyl-1-[2-(4-methoxyanilino)ethylamino]-1-oxopropan-2-yl]-5-[3-(trifluoromethyl)phenyl]furan-2-carboxamideKi20000.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC500.3 [1]
N-[(2R)-1-[[Cyano(methyl)amino]-methylamino]-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]benzamideKi21.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]thiophene-2-carboxamideKi40000.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]-5-phenylthiophene-2-carboxamideKi4000.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]-4-phenylthiophene-2-carboxamideKi4000.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]-5-thiophen-3-ylthiophene-2-carboxamideKi4000.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]-5-(2H-tetrazol-5-yl)thiophene-2-carboxamideKi4000.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]-4-thiophen-2-ylbenzamideKi4000.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]-5-thiophen-2-ylthiophene-2-carboxamideKi3200.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]-1-benzothiophene-2-carboxamideKi4000.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]thieno[2,3-b]thiophene-5-carboxamideKi4000.0 [1]
(3R,4R)-4-(2,3-Dimethylphenoxy)piperidin-3-olIC50100000.0 [1]
(4S,5R)-4-(2,3-Dimethylphenoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC50331.0 [1]
(4S,5S)-4-(2,3-Dimethylphenoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC505908.0 [1]
(4S,5R)-4-Phenoxy-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC50487.0 [1]
(4S,5R)-4-Phenylmethoxy-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC503760.0 [1]
(4S,5R)-4-(2-Methylpropoxy)-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC501826.0 [1]
(4S,5S)-4-Bromo-6-oxa-1-azabicyclo[3.2.1]octan-7-oneIC5010000.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-3-cyclopropyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]propanamideIC50147.0 [1]
(2S)-N-[(1R)-1-Cyano-2-(4-cyano-2-fluorophenyl)ethyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC5076.0 [1]
(2S)-N-[(1S)-1-Cyano-2-(4-cyano-2-fluorophenyl)ethyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC504.0 [1]
1-[4-[4-[(1S)-1-[[(2S)-1-[[(1S)-1-Cyano-2-(4-cyano-2-fluorophenyl)ethyl]amino]-3-methyl-1-oxobutan-2-yl]amino]-2,2,2-trifluoroethyl]phenyl]phenyl]cyclopropane-1-carboxamideIC5016.0 [1]
(2S)-N-[(1S)-1-Cyano-2-(4-cyano-2-fluorophenyl)ethyl]-2-[[(1S)-1-[4-[4-[(1R)-2,2-difluoro-1-hydroxyethyl]phenyl]phenyl]-2,2,2-trifluoroethyl]amino]-3-methylbutanamideIC5056.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-2-[[(1S)-1-[4-[4-[(1R)-2,2-difluoro-1-hydroxyethyl]phenyl]phenyl]-2,2,2-trifluoroethyl]amino]-4-fluoro-4-methylpentanamideIC5064.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC5067.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-[4-[1-(morpholine-4-carbonyl)cyclopropyl]phenyl]phenyl]ethyl]amino]pentanamideIC5022.0 [1]
1-[4-[4-[(1S)-1-[[(2S)-1-[[(1S)-1-Cyano-2-phenylethyl]amino]-4-fluoro-4-methyl-1-oxopentan-2-yl]amino]-2,2,2-trifluoroethyl]phenyl]phenyl]cyclopropane-1-carboxamideIC5037.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-3-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]butanamideIC50174.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-pyridin-4-ylphenyl)phenyl]ethyl]amino]pentanamideIC5051.0 [1]
(2S)-N-[(1S)-1-Cyano-2-(4-cyano-2-fluorophenyl)ethyl]-3-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]butanamideIC5023.0 [1]
(2S)-N-[(1S)-1-Cyano-2-pyridin-4-ylethyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC5012.0 [1]
4-[3-[3-[4-Chloro-3-[2-(4-chlorophenyl)ethynyl]phenyl]-5-methylsulfonyl-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-1-yl]propyl]morpholineIC5020000.0 [1]
(4S,5R)-4-Phenoxy-6-oxa-1-azabicyclo[3.2.1]octane-7-thioneIC5010000.0 [1]
5-((2,3-Dimethylphenoxy)methyl)-3-methyloxazolidin-2-oneIC50100000.0 [1]
(2S)-4,4-Dichloro-N-[(1S)-1-cyano-2-phenylethyl]-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]butanamideIC504.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-2-cyclopropyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]acetamideIC5080.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-3-phenyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]propanamideIC50769.0 [1]
(2S)-N-(Cyanomethyl)-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC50547.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-3,3-dimethyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]butanamideIC5010000.0 [1]
(2S)-N-[(S)-Cyano-(1-phenylcyclopropyl)methyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC5010000.0 [1]
(2S)-N-[(1S)-1-Cyano-2-phenylethyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(1H-pyrazol-4-yl)phenyl]ethyl]amino]pentanamideIC5024.0 [1]
(2S)-N-[(1S)-1-Cyano-3-phenylpropyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC503242.0 [1]
(2S)-N-[(1S)-1-Cyano-3,3,3-trifluoropropyl]-4-fluoro-4-methyl-2-[[(1S)-2,2,2-trifluoro-1-[4-(4-methylsulfonylphenyl)phenyl]ethyl]amino]pentanamideIC50654.0 [1]
N-[(2R)-1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]benzamideKi40000.0 [1]
N-[1-(Cyanomethylamino)-3-(2-methylpropylsulfonyl)-1-oxopropan-2-yl]benzamideKi40000.0 [1]
(3S,4R)-4-(2,3-Dimethylphenoxy)piperidin-3-olIC50100000.0 [1]
N-[(2R)-3-Benzylsulfonyl-1-oxo-1-[[(2S)-1-[4-(trifluoromethoxy)anilino]propan-2-yl]amino]propan-2-yl]morpholine-4-carboxamideKi30000.0 [1]
Items per page: 1 - 10 of 52
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References

This online tool may be cited as follows

MLA

"Quest Database™ Cathepsin F Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Nov. 2024, https://www.aatbio.com/data-sets/cathepsin-f-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 20). Quest Database™ Cathepsin F Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/cathepsin-f-inhibitors-ic50-ki.
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