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Catenin beta-1 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
ToxoflavinIC5010000.0 [1], 30000.0 [2], 34000.0 [3], 340000.0 [4]
ToxoflavinKi3650.0 [1], 3800.0 [2], 5820.0 [3]
CercosporinIC5010000.0 [1], 41000.0 [2], 130000.0 [3], 150000.0 [4]
CercosporinKi5900.0 [1], 35560.0 [2]
4-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanoic acidIC5015000.0 [1], 170000.0 [2], 340000.0 [3]
4-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanoic acidKi1000.0 [1], 17000.0 [2], 59000.0 [3]
N-(4-Amino-1,2,5-oxadiazol-3-yl)-2-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetamideIC5031000.0 [1], 550000.0 [2], 630000.0 [3]
N-(4-Amino-1,2,5-oxadiazol-3-yl)-2-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetamideKi2700.0 [1], 31000.0 [2], 88000.0 [3]
8-[2-(2H-Tetrazol-5-yl)ethyl]-13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaeneIC5076000.0 [1], 770000.0 [2], 850000.0 [3]
8-[2-(2H-Tetrazol-5-yl)ethyl]-13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaeneKi18000.0 [1], 53000.0 [2], 180000.0 [3]
4-Amino-N-(13-oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-ylimino)-1,2,5-oxadiazole-3-carboxamideIC5030000.0 [1], 52000.0 [2], 60000.0 [3]
4-Amino-N-(13-oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-ylimino)-1,2,5-oxadiazole-3-carboxamideKi1200.0 [1], 20000.0 [2], 36000.0 [3]
[(2R)-1-[3,10-Dihydroxy-12-[(2R)-2-(4-hydroxyphenoxy)carbonyloxypropyl]-2,6,7,11-tetramethoxy-4,9-dioxoperylen-1-yl]propan-2-yl] benzoateIC5010000.0 [1], 38000.0 [2], 77000.0 [3], 110000.0 [4]
[(2R)-1-[3,10-Dihydroxy-12-[(2R)-2-(4-hydroxyphenoxy)carbonyloxypropyl]-2,6,7,11-tetramethoxy-4,9-dioxoperylen-1-yl]propan-2-yl] benzoateKi17780.0 [1]
1-Hydroxy-5-[2-(2H-tetrazol-5-yl)ethyl]indazoleIC5013000.0 [1], 300000.0 [2], 350000.0 [3]
1-Hydroxy-5-[2-(2H-tetrazol-5-yl)ethyl]indazoleKi3140.0 [1], 3800.0 [2]
(4S)-4-[[(2S)-3-Carboxy-2-[[(2S)-2-[[2-(5-chloro-1H-indol-2-yl)acetyl]amino]-3-naphthalen-2-ylpropanoyl]amino]propanoyl]amino]-5-methoxy-5-oxopentanoic acidIC506300.0 [1], 210000.0 [2], 680000.0 [3]
(4S)-4-[[(2S)-3-Carboxy-2-[[(2S)-2-[[2-(5-chloro-1H-indol-2-yl)acetyl]amino]-3-naphthalen-2-ylpropanoyl]amino]propanoyl]amino]-5-methoxy-5-oxopentanoic acidKi1300.0 [1], 1360.0 [2]
2-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetic acidIC5025000.0 [1], 280000.0 [2], 450000.0 [3]
2-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetic acidKi4100.0 [1]
3-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)propanoic acidIC5048000.0 [1], 580000.0 [2], 790000.0 [3]
3-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)propanoic acidKi3300.0 [1]
2-[[2-(4-Ethylphenyl)-5-methyl-1,3-oxazol-4-yl]methylsulfanyl]-N-(2-phenylethyl)acetamideKi195470.0 [1], 364710.0 [2], 370000.0 [3]
(5Z)-5-{[2,5-Dimethyl-1-(3-pyridinyl)-1H-pyrrol-3-yl]methylene}-3-phenyl-1,3-thiazolidine-2,4-dioneKi40670.0 [1], 53510.0 [2], 54000.0 [3]
2-PhenoxybenzamideKi24390.0 [1], 180990.0 [2]
Ethyl 4-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanoateKi52000.0 [1], 120000.0 [2]
4-[5-(3,4-Dimethoxy-benzylidene)-4-oxo-2-thioxo-thiazolidin-3-yl]-butyric acidKi46810.0 [1], 80340.0 [2]
2,3-Bis(4-chlorophenyl)quinoxaline-6-carboxylic acidKi8800.0 [1], 13000.0 [2]
5-[4-(4-Chlorophenoxy)phenyl]-3-isoxazolecarboxylic acidKi21000.0 [1], 77000.0 [2]
Ethyl 2-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetateKi63000.0 [1], 150000.0 [2]
Methyl 3-(13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)propanoateKi100000.0 [1]
2-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)acetonitrileKi130000.0 [1], 240000.0 [2]
3-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)propanenitrileKi39000.0 [1], 47000.0 [2]
4-(13-Oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaen-8-yl)butanenitrileKi120000.0 [1], 160000.0 [2]
8-[3-(2H-Tetrazol-5-yl)propyl]-13-oxa-8,10,12,14,16-pentazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,9,11,14-heptaeneKi51000.0 [1], 74000.0 [2]
2,3-DI(1,3-Benzodioxol-5-YL)-7-hydroxy-6-quinoxalinecarboxylic acidKi8700.0 [1], 12000.0 [2]
5H-[1,2,5]Oxadiazolo[3',4':5,6]pyrazino[2,3-b]indoleKi120000.0 [1], 280000.0 [2]
3-[2-(1-Hydroxyindazol-5-yl)ethyl]-2H-1,2,4-oxadiazole-5-thioneKi7240.0 [1], 70370.0 [2]
3-[(1-Hydroxybenzotriazol-5-yl)methyl]-2H-1,2,4-oxadiazole-5-thioneKi42020.0 [1], 105900.0 [2]
1-Hydroxy-5-[2-(2H-tetrazol-5-yl)ethyl]benzotriazoleKi3830.0 [1], 7600.0 [2]
(4-Amino-1,2,5-oxadiazol-3-yl)(pyrrolidin-1-yl)methanoneKi1700000.0 [1]
3-Butanoyl-1,8-dihydroxy-2-methylphenanthrene-9,10-dioneIC5010000.0 [1]
N-[(E)-(5-Methylfuran-2-yl)methylideneamino]-2-phenoxybenzamideKi1800.0 [1]
9H-Indeno[1,2-b][1,2,5]oxadiazolo[3,4-E]pyrazin-9-oneKi310000.0 [1]
13-Oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-yliminothioureaKi240000.0 [1]
CID 1416323Ki80000.0 [1]
4-Amino-1,2,5-oxadiazole-3-carboxamideKi2000000.0 [1]
1-[12-[2-(2,4-Dihydroxy-6-methylbenzoyl)oxypropyl]-3,10-dihydroxy-2,6,7,11-tetramethoxy-4,9-dioxoperylen-1-yl]propan-2-yl 2,4-dihydroxy-6-methylbenzoateIC5010000.0 [1]
13-Oxa-10,12,14,16-tetrazatetracyclo[7.7.0.02,7.011,15]hexadeca-1(16),2,4,6,8,10,14-heptaen-8-yldiazeneKi230000.0 [1]
2-Hydroxy-5-({3-[(phenylsulfonyl)amino]quinoxalin-2-yl}amino)benzoic acidKi13000.0 [1]
4-Amino-N-isobutyl-1,2,5-oxadiazole-3-carboxamideKi2000000.0 [1]
4-Amino-N-benzyl-1,2,5-oxadiazole-3-carboxamideKi1700000.0 [1]
2-[(3S,6S,9S,12S,16Z,21S)-12-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-5-amino-5-oxopentanoyl]amino]-21-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-12,21-dimethyl-6-(2-methylpropyl)-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclohenicos-16-en-3-yl]acetic acidIC505000.0 [1]
2-[(3S,6S,9S,12S,16Z,21S)-12-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[(2S)-2-Acetamido-5-carbamimidamidopentanoyl]amino]-5-carbamimidamidopentanoyl]amino]-3-(1H-indol-3-yl)propanoyl]pyrrolidine-2-carbonyl]amino]-5-carbamimidamidopentanoyl]amino]-21-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-(1H-indol-3-yl)-1-oxopropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-5-carbamimidamido-1-oxopentan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-3-(1H-imidazol-5-yl)-1-oxopropan-2-yl]carbamoyl]-9-[(2S)-butan-2-yl]-12,21-dimethyl-6-(2-methylpropyl)-2,5,8,11-tetraoxo-1,4,7,10-tetrazacyclohenicos-16-en-3-yl]acetic acidIC505000.0 [1]
Methyl (6R,6aS,14aR)-1,6,8,14a-tetrahydroxy-11-[[(2R,3S,4S,5S,6R)-4-hydroxy-3,5-dimethoxy-6-methyloxan-2-yl]amino]-6a-methoxy-3-methyl-7,9,12,14-tetraoxo-5,6-dihydrobenzo[a]tetracene-2-carboxylateIC5010000.0 [1]
1-Hydroxy-5-[2-(2H-tetrazol-1-ium-1-yl)ethyl]benzotriazoleKi54200.0 [1]
1-Hydroxy-5-(2H-tetrazol-1-ium-1-ylmethoxymethyl)indazoleKi13550.0 [1]
3-[(1-Hydroxybenzotriazol-5-yl)methyl]-4H-1,2,4-oxadiazol-5-oneKi125100.0 [1]
3-[2-(1-Hydroxybenzotriazol-5-yl)ethyl]-4H-1,2,4-oxadiazol-5-oneKi551250.0 [1]
3-[2-(1-Hydroxyindazol-5-yl)ethyl]-4H-1,2,4-oxadiazol-5-oneKi97700.0 [1]
1-Hydroxy-5-(2H-tetrazol-5-ylmethyl)benzotriazoleKi94400.0 [1]
1-Hydroxy-5-(2H-tetrazol-5-ylmethoxymethyl)benzotriazoleKi155100.0 [1]
3-[2-(1-Hydroxybenzotriazol-5-yl)ethyl]-2H-1,2,4-oxadiazole-5-thioneKi24360.0 [1]
1-Hydroxy-5-(2H-tetrazol-5-ylmethoxy)benzotriazoleKi50400.0 [1]
5-[2-(2H-Tetrazol-5-yl)ethyl]-1H-indazoleKi179930.0 [1]
1-Hydroxy-N-(2H-tetrazol-5-ylmethyl)indazol-5-amineKi3380.0 [1]
3-Bromo-5-fluoro-N-(1-hydroxyindazol-5-yl)-N-(2H-tetrazol-5-ylmethyl)benzamideKi28740.0 [1]
3-Chloro-N-(1-hydroxyindazol-5-yl)-N-(2H-tetrazol-5-ylmethyl)benzamideKi33140.0 [1]
N-(1-Hydroxyindazol-5-yl)-N-(2H-tetrazol-5-ylmethyl)pyridine-3-carboxamideKi179930.0 [1]
N-(1-Hydroxyindazol-5-yl)-3,5-dimethyl-N-(2H-tetrazol-5-ylmethyl)-1,2-oxazole-4-carboxamideKi16570.0 [1]
Items per page: 1 - 10 of 70
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References

This online tool may be cited as follows

MLA

"Quest Database™ Catenin beta-1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/catenin-beta-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Catenin beta-1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/catenin-beta-1-inhibitors-ic50-ki.
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