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Caspase-9 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC503330.0 [1], 10000.0 [2]
3-((S)-2-(((Benzyloxy)carbonyl)amino)-3-methylbutanamido)-5-fluoro-4-oxopentanoic acidIC505.0 [1]
(S)-5-(2-Phenoxymethyl-pyrrolidine-1-sulfonyl)-1H-indole-2,3-dioneKi1200.0 [1]
Caspase-3/7 Inhibitor IKi1100.0 [1]
Isatin Sulfonamide 34Ki120.0 [1]
Grassystatin AIC505000.0 [1]
1-Methyl-5-nitroindoline-2,3-dioneKi7200.0 [1]
5-(Pyrrolidin-1-ylsulfonyl)indoline-2,3-dioneKi12000.0 [1]
4-(Ethoxycarbonylmethoxy)-1-hydroxy-naphthalene-2-carboxylic AcidIC5093000.0 [1]
5-(2-((Methyl(phenyl)amino)methyl)pyrrolidin-1-ylsulfonyl)indoline-2,3-dioneKi50000.0 [1]
(S)-3-((S)-2-(Benzyloxycarbonylamino)-3-methylbutanamido)-5-(methylsulfonyl)pent-4-enoic acidIC503330.0 [1]
2-[4-[4-[(2R)-4-[(2-Ethylphenyl)carbamoyl]-2-methyl-2,3-dihydro-1,4-benzoxazin-7-yl]phenyl]cyclohexyl]acetic acidIC505000.0 [1]
1-Benzyl-5-nitro-2,3-dihydro-1H-indole-2,3-dioneKi5000.0 [1]
5-Fluoro-3-((S)-3-methyl-2-phenylcarbamoyloxy-butyrylamino)-4-oxo-pentanoic acidIC5030.0 [1]
Caspase inhibitor-bp-22471IC509.0 [1]
4-Fluoro-2-[[2-[[(2S)-3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]benzoyl]amino]-3-oxobutanoic acidIC506.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-6-ethoxy-6-oxohex-4-enoic acidIC501000.0 [1]
(E,3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3,3-dimethylbutanoyl]azetidine-2-carbonyl]amino]-5-methylsulfonylpent-4-enoic acidIC501100.0 [1]
(E,3S)-3-[[(2S,3S)-2-[[(2S)-5-Amino-2-[[(2S)-3-(1H-indol-3-yl)-2-(phenylmethoxycarbonylamino)propanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC501740.0 [1]
(E,3S)-3-[[(2S,3S)-2-[[(2S)-5-Amino-2-[[(2S)-3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC50800.0 [1]
(E,3S)-3-[[(2S)-1-[(2R)-2-[(4-Amino-3-chlorobenzoyl)amino]-3,3-dimethylbutanoyl]pyrrolidine-2-carbonyl]amino]-5-methylsulfonylpent-4-enoic acidIC502300.0 [1]
5-[(2S)-2-(Anilinomethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dioneKi850.0 [1]
(S)-3-{(S)-4-Methyl-2-[2-(naphthalen-1-ylamino)-acetylamino]-pentanoylamino}-4-oxo-butyric acidIC50160.0 [1]
(S)-3-{(S)-4-Methyl-2-[2-(naphthalen-1-yloxy)-acetylamino]-pentanoylamino}-4-oxo-butyric acidIC502720.0 [1]
(3S)-3-[[(2S)-4-Methyl-2-[[2-(naphthalen-1-ylamino)-2-oxoacetyl]amino]pentanoyl]amino]-4-oxobutanoic acidIC50230.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-(2,3-dihydro-1H-inden-2-yl)acetyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
(Z,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-quinolin-2-ylpropanoyl]amino]-3-methylbutanoyl]amino]-5-chloro-5-methylsulfonylpent-4-enoic acidIC501200.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-quinolin-2-ylpropanoyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
(4S)-5-[[(2S)-1-[[(E,2S)-1-Carboxy-4-methylsulfonylbut-3-en-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-4-[[(2S)-3-carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-5-oxopentanoic acidIC50500.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-(1H-indol-3-yl)propanoyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
Methyl (E,3S)-3-[[(2S)-2-[[(2S)-2-(2,3-dihydro-1H-inden-2-yl)-2-[[(2S)-4-methoxy-4-oxo-2-(phenylmethoxycarbonylamino)butanoyl]amino]acetyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoateIC503000.0 [1]
(2S)-3-Methyl-2-[[(2S)-2-[[(2S)-4-[(2-methylpropan-2-yl)oxy]-4-oxo-2-(phenylmethoxycarbonylamino)butanoyl]amino]-2-phenylacetyl]amino]butanoic acidIC503330.0 [1]
Tert-butyl (E,3S)-3-amino-5-(benzenesulfonyl)pent-4-enoateIC503330.0 [1]
Tert-butyl (E,3S)-3-amino-5-methylsulfonylpent-4-enoateIC503330.0 [1]
Tert-butyl (E,3S)-5-(benzenesulfonyl)-3-[(2-methylpropan-2-yl)oxycarbonylamino]pent-4-enoateIC503330.0 [1]
(E,3S)-3-Amino-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
(E,3S)-5-(Benzenesulfonyl)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]pent-4-enoic acidIC503330.0 [1]
(E,3S)-5-(Benzenesulfonyl)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-quinolin-2-ylpropanoyl]amino]-3-methylbutanoyl]amino]pent-4-enoic acidIC503330.0 [1]
(E,3S)-5-(Benzenesulfonyl)-3-[[(2S)-2-[[2-[[(2S)-3-carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-quinolin-2-ylpropanoyl]amino]-3-methylbutanoyl]amino]pent-4-enoic acidIC503330.0 [1]
(E,3S)-5-(Benzenesulfonyl)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-pyridin-2-ylpropanoyl]amino]-3-methylbutanoyl]amino]pent-4-enoic acidIC503330.0 [1]
(E,3S)-5-(Benzenesulfonyl)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-(4-hydroxyphenyl)-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-methylbutanoyl]amino]propanoyl]amino]pent-4-enoic acidIC5010000.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-(2,3-dihydro-1H-inden-2-yl)acetyl]amino]-3-methylbutanoyl]amino]-5-propan-2-ylsulfonylpent-4-enoic acidIC503330.0 [1]
Tert-butyl (E,3S)-3-[[(2S)-3-methyl-2-[[(2S)-2-[[(2S)-4-[(2-methylpropan-2-yl)oxy]-4-oxo-2-(phenylmethoxycarbonylamino)butanoyl]amino]-3-quinolin-2-ylpropanoyl]amino]butanoyl]amino]-5-morpholin-4-ylsulfonylpent-4-enoateIC503330.0 [1]
(4S)-5-[[(2S)-1-[[(E,2S)-1-Carboxy-4-methylsulfonylbut-3-en-2-yl]amino]-3-methyl-1-oxobutan-2-yl]amino]-4-[[(2S)-3-(4-hydroxyphenyl)-2-(phenylmethoxycarbonylamino)propanoyl]amino]-5-oxopentanoic acidIC501600.0 [1]
Methyl (E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-4-methoxy-4-oxo-2-(phenylmethoxycarbonylamino)butanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoateIC503330.0 [1]
(Z,3S)-5-Chloro-3-[[(2S)-3-methyl-2-[[(2S)-2-[(4-methylphenyl)sulfonylamino]-3-quinolin-2-ylpropanoyl]amino]butanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-naphthalen-1-ylpropanoyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-quinolin-2-ylpropanoyl]amino]-3-methylbutanoyl]amino]-5-phenoxysulfonylpent-4-enoic acidIC50300.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
(E,3S)-3-[[(2S)-2-[[2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-quinolin-2-ylpropanoyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC5010000.0 [1]
(Z,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-5-chloro-5-methylsulfonylpent-4-enoic acidIC502800.0 [1]
Items per page: 1 - 10 of 51
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References

This online tool may be cited as follows

MLA

"Quest Database™ Caspase-9 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/caspase-9-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Caspase-9 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/caspase-9-inhibitors-ic50-ki.
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