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Caspase-5 Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
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▼
Standard Values (in nM)
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▼
4-[4-(Pyridin-3-ylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineIC50155.0 [1], 2560.0 [2]
4-[4-(Pyridin-3-ylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi59.0 [1]
CID 104934Ki210.0 [1]
Grassystatin AIC505000.0 [1]
N-[3-[1-[[(3S)-2-Hydroxy-5-oxooxolan-3-yl]carbamoyl]cyclopropyl]-2,4-dioxo-1-propan-2-ylpyrimidin-5-yl]-2-methyl-4-(naphthalen-2-ylamino)benzamideIC502980.0 [1]
Inhibitor 62bKi32000.0 [1]
4-[4-[[3,5-Bis(trifluoromethyl)phenyl]methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi48.0 [1]
4-[4-[(2-Nitrophenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi24.0 [1]
4-(4-Benzylpiperazin-1-yl)-2,6-dipyrrolidin-1-ylpyrimidineKi41.0 [1]
4-[4-[(3,5-Dimethoxyphenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi34.0 [1]
4-[4-(2-Phenylethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi16.0 [1]
4-[4-[(3-Methoxyphenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi111.0 [1]
4-[4-(Pyridin-4-ylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi34.0 [1]
2,4-Dipyrrolidin-1-yl-6-[4-[[4-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]pyrimidineKi135.0 [1]
4-[4-(Cyclohexylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi59.0 [1]
[4-[[4-(2,6-Dipyrrolidin-1-ylpyrimidin-4-yl)piperazin-1-yl]methyl]phenyl]-phenylmethanoneKi28.0 [1]
4-[4-[(4-Nitrophenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi99.0 [1]
4-(Piperazin-1-yl)-2,6-di(pyrrolidin-1-yl)pyrimidineKi47.0 [1]
5-[[5-[[(2S)-1-Carboxy-4-(2-chlorophenyl)sulfanyl-3-oxobutan-2-yl]carbamoyl]pyridin-2-yl]methylsulfamoyl]-2-hydroxybenzoic acidKi11000.0 [1]
4-(Cyclopentylamino)-6-(3,5-difluorophenylamino)-1,3,5-triazine-2-carbonitrileIC5013489.63 [1]
3-[2-[5-Tert-butyl-3-[(4-methyl-1,2,5-oxadiazol-3-yl)methylamino]-2-oxopyrazin-1-yl]butanoylamino]-5-[hexyl(methyl)amino]-4-oxopentanoic acid;hydrochlorideIC500.2 [1]
Inhibitor 47cKi98000.0 [1]
(3S)-3-[4-(3-Carboxy-4-hydroxyphenylsulfonylaminomethyl)benzoylamino]-4-oxobutanoic acidKi12000.0 [1]
CID 5327304Ki22000.0 [1]
Inhibitor 64bKi23000.0 [1]
Inhibitor 66aKi24000.0 [1]
Inhibitor 66bKi63000.0 [1]
Inhibitor 69bKi36000.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-6-ethoxy-6-oxohex-4-enoic acidIC50100000.0 [1]
(E,3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3,3-dimethylbutanoyl]azetidine-2-carbonyl]amino]-5-methylsulfonylpent-4-enoic acidIC5035200.0 [1]
(E,3S)-3-[[(2S,3S)-2-[[(2S)-5-Amino-2-[[(2S)-3-(1H-indol-3-yl)-2-(phenylmethoxycarbonylamino)propanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC50750.0 [1]
(E,3S)-3-[[(2S,3S)-2-[[(2S)-5-Amino-2-[[(2S)-3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC5019500.0 [1]
(E,3S)-3-[[(2S)-1-[(2R)-2-[(4-Amino-3-chlorobenzoyl)amino]-3,3-dimethylbutanoyl]pyrrolidine-2-carbonyl]amino]-5-methylsulfonylpent-4-enoic acidIC50560.0 [1]
3-[[4-(2,6-Dipyrrolidin-1-ylpyrimidin-4-yl)piperazin-1-yl]methyl]-2,5,7,8-tetramethyl-3,4-dihydro-2H-chromen-6-olKi81.0 [1]
3-[2-[5-Tert-butyl-3-[(4-methyl-1,2,5-oxadiazol-3-yl)methylamino]-2-oxopyrazin-1-yl]butanoylamino]-5-[methyl(pentyl)amino]-4-oxopentanoic acidIC500.81 [1]
Items per page: 1 - 10 of 35
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References

This online tool may be cited as follows

MLA

"Quest Database™ Caspase-5 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/caspase-5-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Caspase-5 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/caspase-5-inhibitors-ic50-ki.
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