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Caspase-4 Inhibitors (IC50, Ki)

Structure
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▼
Compound Name
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Standard Type
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Standard Values (in nM)
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▼
CID 104934Ki337.0 [1]
(S)-5-(2-Phenoxymethyl-pyrrolidine-1-sulfonyl)-1H-indole-2,3-dioneKi33000.0 [1]
Caspase-3/7 Inhibitor IKi25000.0 [1]
Isatin Sulfonamide 34Ki5000.0 [1]
Grassystatin AIC505000.0 [1]
Cruzain-IN-1IC5033113.11 [1]
1-Methyl-5-nitroindoline-2,3-dioneKi4000.0 [1]
5-(Pyrrolidin-1-ylsulfonyl)indoline-2,3-dioneKi50000.0 [1]
5-(2-((Methyl(phenyl)amino)methyl)pyrrolidin-1-ylsulfonyl)indoline-2,3-dioneKi50000.0 [1]
1-Benzyl-5-nitro-2,3-dihydro-1H-indole-2,3-dioneKi5000.0 [1]
Inhibitor 62bKi22000.0 [1]
4-[4-[[3,5-Bis(trifluoromethyl)phenyl]methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineIC505000.0 [1]
4-[4-[(2-Nitrophenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi267.0 [1]
4-[4-(Pyridin-3-ylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi870.0 [1]
4-(4-Benzylpiperazin-1-yl)-2,6-dipyrrolidin-1-ylpyrimidineIC505000.0 [1]
4-[4-[(3,5-Dimethoxyphenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi148.0 [1]
4-[4-(2-Phenylethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi8.0 [1]
4-[4-[(3-Methoxyphenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi276.0 [1]
4-[4-(Pyridin-4-ylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi393.0 [1]
2,4-Dipyrrolidin-1-yl-6-[4-[[4-(trifluoromethyl)phenyl]methyl]piperazin-1-yl]pyrimidineKi563.0 [1]
4-[4-(Cyclohexylmethyl)piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi306.0 [1]
[4-[[4-(2,6-Dipyrrolidin-1-ylpyrimidin-4-yl)piperazin-1-yl]methyl]phenyl]-phenylmethanoneKi119.0 [1]
4-[4-[(4-Nitrophenyl)methyl]piperazin-1-yl]-2,6-dipyrrolidin-1-ylpyrimidineKi215.0 [1]
4-(Piperazin-1-yl)-2,6-di(pyrrolidin-1-yl)pyrimidineKi207.0 [1]
5-[[5-[[(2S)-1-Carboxy-4-(2-chlorophenyl)sulfanyl-3-oxobutan-2-yl]carbamoyl]pyridin-2-yl]methylsulfamoyl]-2-hydroxybenzoic acidKi38000.0 [1]
4-(Cyclopentylamino)-6-(3,5-difluorophenylamino)-1,3,5-triazine-2-carbonitrileIC508128.31 [1]
3-[2-[5-Tert-butyl-3-[(4-methyl-1,2,5-oxadiazol-3-yl)methylamino]-2-oxopyrazin-1-yl]butanoylamino]-5-[hexyl(methyl)amino]-4-oxopentanoic acid;hydrochlorideIC500.3 [1]
Inhibitor 47cKi96000.0 [1]
(3S)-3-[4-(3-Carboxy-4-hydroxyphenylsulfonylaminomethyl)benzoylamino]-4-oxobutanoic acidKi21000.0 [1]
CID 5327304Ki92000.0 [1]
Inhibitor 64bKi13000.0 [1]
Inhibitor 66aKi38000.0 [1]
Inhibitor 66bKi100000.0 [1]
Inhibitor 69bKi27000.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-6-ethoxy-6-oxohex-4-enoic acidIC50510.0 [1]
(E,3S)-3-[[(2S)-1-[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3,3-dimethylbutanoyl]azetidine-2-carbonyl]amino]-5-methylsulfonylpent-4-enoic acidIC505600.0 [1]
(E,3S)-3-[[(2S,3S)-2-[[(2S)-5-Amino-2-[[(2S)-3-(1H-indol-3-yl)-2-(phenylmethoxycarbonylamino)propanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC50180.0 [1]
(E,3S)-3-[[(2S,3S)-2-[[(2S)-5-Amino-2-[[(2S)-3-methyl-2-(phenylmethoxycarbonylamino)butanoyl]amino]-5-oxopentanoyl]amino]-3-methylpentanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC50370.0 [1]
(E,3S)-3-[[(2S)-1-[(2R)-2-[(4-Amino-3-chlorobenzoyl)amino]-3,3-dimethylbutanoyl]pyrrolidine-2-carbonyl]amino]-5-methylsulfonylpent-4-enoic acidIC5090.0 [1]
5-[(2S)-2-(Anilinomethyl)pyrrolidin-1-yl]sulfonyl-1H-indole-2,3-dioneKi30000.0 [1]
3-[[4-(2,6-Dipyrrolidin-1-ylpyrimidin-4-yl)piperazin-1-yl]methyl]-2,5,7,8-tetramethyl-3,4-dihydro-2H-chromen-6-olKi248.0 [1]
3-[2-[5-Tert-butyl-3-[(4-methyl-1,2,5-oxadiazol-3-yl)methylamino]-2-oxopyrazin-1-yl]butanoylamino]-5-[methyl(pentyl)amino]-4-oxopentanoic acidIC500.5 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC502800.0 [1]
(E,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-3-naphthalen-1-ylpropanoyl]amino]-3-methylbutanoyl]amino]-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
(Z,3S)-3-[[(2S)-2-[[(2S)-2-[[(2S)-3-Carboxy-2-(phenylmethoxycarbonylamino)propanoyl]amino]-2-phenylacetyl]amino]-3-methylbutanoyl]amino]-5-chloro-5-methylsulfonylpent-4-enoic acidIC503330.0 [1]
Items per page: 1 - 10 of 45
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References

This online tool may be cited as follows

MLA

"Quest Database™ Caspase-4 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/caspase-4-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Caspase-4 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/caspase-4-inhibitors-ic50-ki.
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