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Casein kinase II alpha Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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▼
SilmitasertibIC5014.7 [1]
4,5,6,7-TetrabromobenzotriazoleIC50320.0 [1], 500.0 [2], 900.0 [3], 1480.0 [4]
4,5,6,7-TetrabromobenzotriazoleKi400.0 [1]
4,5,6,7-TetrabromobenzimidazoleIC50170.0 [1], 1300.0 [2]
4,5,6,7-TetrabromobenzimidazoleKi45.0 [1], 315.0 [2], 462.0 [3], 1030.0 [4]
EmodinIC50890.0 [1], 2000.0 [2]
EmodinKi1850.0 [1], 40000.0 [2]
4,5,6,7-Tetrabromo-N,N-dimethyl-1H-benzimidazol-2-amineKi40.0 [1], 97.0 [2], 139.0 [3]
(5-Oxo-5,6-dihydro-indolo[1,2-A]quinazolin-7-YL)-acetic acidIC50390.0 [1]
(5-Oxo-5,6-dihydro-indolo[1,2-A]quinazolin-7-YL)-acetic acidKi170.0 [1]
4-[2-[(4-Methoxyphenyl)carbonylamino]-1,3-Thiazol-5-Yl]benzoic AcidIC5020.0 [1], 32.0 [2]
CID 72163809IC503.0 [1]
N-[1-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamideIC5010.0 [1]
N-[1-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]-N-methylacetamideIC5010.0 [1], 11.0 [2], 34.0 [3]
3-[5-Acetamido-3-[3-cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-1-yl]propanoic acidIC503.0 [1], 3000.0 [2], 3100.0 [3]
ApigeninIC50800.0 [1]
ApigeninKi740.0 [1]
5,6-Dichloro-1-beta-D-ribofuranosylbenzimidazoleIC5013000.0 [1]
5,6-Dichloro-1-beta-D-ribofuranosylbenzimidazoleKi4500.0 [1]
4-(7-Butyl-5H-pyrrolo[2,3-b]pyrazin-6-yl)phenolIC50100000.0 [1]
4,5,6,7-Tetraiodo-1H-benzimidazoleKi43.0 [1], 266.0 [2]
5-((3-Ethynylphenyl)amino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC506.0 [1], 98.0 [2]
[4,5,6,7-Tetrabromo-2-(Dimethylamino)-1h-Benzimidazol-1-Yl]acetic AcidKi83.0 [1], 88.0 [2]
3-(Cyclopropylamino)-5-{[3-(Trifluoromethyl)phenyl]amino}pyrimido[4,5-C]quinoline-8-Carboxylic AcidIC5010.0 [1], 750.0 [2]
((4,5,6,7-Tetrabromo-1H-benzimidazol-2-yl)sulfanyl)-acetic acidKi106.0 [1], 170.0 [2]
4,5,6,7-Tetrabromo-N,N,1-trimethylbenzimidazol-2-amineKi154.0 [1], 212.0 [2]
N-[3-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1H-indol-5-yl]acetamideIC5077.0 [1], 5000.0 [2]
2-[(4,5,6,7-Tetraiodo-1H-benzimidazol-2-yl)sulfanyl]acetic acidKi80.0 [1], 110.0 [2]
2-(4,5,6,7-Tetraiodobenzimidazol-1-yl)acetic acidKi261.0 [1], 378.0 [2]
(4,5,6,7-Tetrabromo-1h-Benzimidazol-1-Yl)acetic AcidKi670.0 [1], 798.0 [2]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
4-[(4,5,6,7-Tetrabromo-1H-benzimidazol-2-yl)sulfanyl]butanoic acidKi77.0 [1], 210.0 [2]
4-[6-[6-(Propan-2-ylamino)indazol-1-yl]pyrazin-2-yl]benzoic acidIC505.0 [1], 110.0 [2]
3-Chloro-4-[6-[6-(propan-2-ylamino)indazol-1-yl]pyrazin-2-yl]benzoic acidIC5015.0 [1], 3400.0 [2]
3-Fluoro-4-[6-[6-(propan-2-ylamino)indazol-1-yl]pyrazin-2-yl]benzoic acidIC505.0 [1], 340.0 [2]
6-[6-[6-(Propan-2-ylamino)indazol-1-yl]pyrazin-2-yl]pyridine-3-carboxylic acidIC507.0 [1], 1000.0 [2]
4-[6-[6-(Propan-2-ylamino)indazol-1-yl]pyrazin-2-yl]thiophene-2-carboxylic acidIC5026.0 [1], 3300.0 [2]
4-[6-[6-(Propan-2-ylamino)indol-1-yl]pyrazin-2-yl]benzoic acidIC503.0 [1], 96.0 [2]
2-Fluoro-4-[6-[6-(propan-2-ylamino)indazol-1-yl]pyrazin-2-yl]benzoic acidIC507.0 [1], 180.0 [2]
5-[6-[6-(Propan-2-ylamino)indazol-1-yl]pyrazin-2-yl]pyridine-2-carboxylic acidIC50297.0 [1], 4300.0 [2]
5-Anilinobenzo[c][2,6]naphthyridine-8-carboxylic acidIC5010.0 [1], 7400.0 [2]
5-[2-(Dimethylamino)ethylamino]benzo[c][2,6]naphthyridine-8-carboxylic acidIC5019.0 [1], 50000.0 [2]
5-(2-Phenylethylamino)benzo[c][2,6]naphthyridine-8-carboxylic acidIC503.0 [1], 688.0 [2]
5-(3-Phenylpropylamino)benzo[c][2,6]naphthyridine-8-carboxylic acidIC5016.0 [1], 2500.0 [2]
5-(3-Methoxyanilino)benzo[c][2,6]naphthyridine-8-carboxylic acidIC507.0 [1], 2325.0 [2]
5-(3-Chloro-4-fluoroanilino)benzo[c][2,6]naphthyridine-8-carboxylic acidIC506.0 [1], 464.0 [2]
5-(3-Fluoroanilino)benzo[c][2,6]naphthyridine-8-carboxylic acidIC505.0 [1], 2933.0 [2]
5-(4-Chloroanilino)benzo[c][2,6]naphthyridine-8-carboxylic acidIC507.0 [1], 17.0 [2]
5-(3-Ethynylanilino)benzo[c][2,6]naphthyridine-8-carboxylic acidIC503.0 [1], 70.0 [2]
N-(3-Chlorophenyl)-8-(2H-tetrazol-5-yl)benzo[c][2,6]naphthyridin-5-amineIC5045.0 [1], 1016.0 [2]
5-(3-Chloroanilino)-3-(cyclopropylamino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC5010.0 [1], 13.0 [2]
5-(3,5-Difluoroanilino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC506.0 [1], 269.0 [2]
5-(3-Fluoroanilino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC506.0 [1], 26.0 [2]
5-(3-Chloro-4-fluoroanilino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC5010.0 [1], 1056.0 [2]
5-(3-Chloroanilino)-3-(ethylamino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC5010.0 [1], 30.0 [2]
5-[3-(Trifluoromethyl)anilino]pyrimido[4,5-c]quinoline-8-carboxylic acidIC5011.0 [1], 98.0 [2]
4-(4,5,6,7-Tetrabromobenzimidazol-1-yl)butyric acidKi368.0 [1], 472.0 [2]
4-[4,5,6,7-Tetrabromo-2-(dimethylamino)benzimidazol-1-yl]butanoic acidKi456.0 [1], 860.0 [2]
3-[(4,5,6,7-Tetrabromo-1H-benzimidazol-2-yl)sulfanyl]propanoic acidKi116.0 [1], 172.0 [2]
3-(4,5,6,7-Tetrabromo-1-methylbenzimidazol-2-yl)sulfanylpropanoic acidKi112.0 [1], 137.0 [2]
4-(4,5,6,7-Tetrabromo-1-methylbenzimidazol-2-yl)sulfanylbutanoic acidKi88.0 [1], 501.0 [2]
2-(4,5,6,7-Tetrabromo-1-methylbenzimidazol-2-yl)sulfanylacetic acidKi13.0 [1], 143.0 [2]
N-[3-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1-(3-hydroxypropyl)indol-5-yl]acetamideIC50210.0 [1], 3000.0 [2]
N-[1-[3-Cyano-7-[(1-methylpyrazol-3-yl)amino]pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamideIC5016.0 [1], 24.0 [2]
7-(Cyclopropylamino)-5-[6-(methylsulfonylmethyl)indol-1-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileIC507.0 [1], 83.0 [2]
N-[1-[3-Cyano-7-(3-pyrrolidin-1-ylpropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamideIC5018.0 [1], 860.0 [2]
N-[3-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1-methylindol-5-yl]acetamideIC5027.0 [1], 6000.0 [2]
N-[1-[3-Cyano-7-(oxetan-3-ylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamideIC504.0 [1], 57.0 [2]
N-[3-[3-Cyano-7-(cyclopropylamino)pyrazolo[1,5-a]pyrimidin-5-yl]-1-(2-hydroxyethyl)indol-5-yl]acetamideIC50500.0 [1], 3000.0 [2]
7-(Cyclopropylamino)-5-[6-(hydroxymethyl)indol-1-yl]pyrazolo[1,5-a]pyrimidine-3-carbonitrileIC50120.0 [1], 830.0 [2]
N-[1-[3-Cyano-7-(4-hydroxybutylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamideIC5030.0 [1], 190.0 [2]
N-[1-[3-Cyano-7-(2-morpholin-4-ylethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamideIC5030.0 [1], 460.0 [2]
N-[1-[3-Cyano-7-(2-pyrrolidin-1-ylethylamino)pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamideIC5040.0 [1], 780.0 [2]
N-[1-[3-Cyano-7-[3-(dimethylamino)propylamino]pyrazolo[1,5-a]pyrimidin-5-yl]indol-6-yl]acetamideIC5030.0 [1], 1200.0 [2]
4-[2-(Dimethylamino)ethylamino]thieno[3,2-c]quinoline-7-carboxylic acidIC50277.0 [1], 50000.0 [2]
4-(Phenylamino)thieno[3,2-c]quinoline-7-carboxylic acidIC50310.0 [1], 15700.0 [2]
4-(3-Fluoroanilino)thieno[3,2-c]quinoline-7-carboxylic acidIC5068.0 [1], 3564.0 [2]
4-(3-Ethynylanilino)thieno[3,2-c]quinoline-7-carboxylic acidIC5028.0 [1], 8360.0 [2]
N-(3-Chlorophenyl)-7-(2H-tetrazol-5-yl)thieno[3,2-c]quinolin-4-amineIC50181.0 [1], 9590.0 [2]
N-(3-Fluorophenyl)-7-(2H-tetrazol-5-yl)thieno[3,2-c]quinolin-4-amineIC5096.0 [1], 4426.0 [2]
3-(Cyclopropylmethylamino)-5-(3-ethynylanilino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC5027.0 [1], 50.0 [2]
4-(3,5-Dichloroanilino)thieno[3,2-c]quinoline-7-carboxylic acidIC5035.0 [1], 580.0 [2]
5-[2-(3-Fluorophenyl)ethylamino]benzo[c][2,6]naphthyridine-8-carboxylic acidIC507.0 [1], 3600.0 [2]
Methyl 5-anilinobenzo[c][2,6]naphthyridine-8-carboxylateIC50200.0 [1], 19870.0 [2]
4-(3-Fluoroanilino)-[1,3]thiazolo[4,5-c]quinoline-7-carboxylic acidIC50146.0 [1], 25800.0 [2]
5-(3-Chloro-4-fluoroanilino)-3-(2-methoxyethylamino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC5047.0 [1], 52.0 [2]
N-(4-Chloro-3-fluorophenyl)-8-(2H-tetrazol-5-yl)benzo[c][2,6]naphthyridin-5-amineIC5052.0 [1], 220.0 [2]
Methyl 5-(3-methoxyanilino)benzo[c][2,6]naphthyridine-8-carboxylateIC5025000.0 [1], 50000.0 [2]
5-(3,5-Difluoroanilino)benzo[c][2,6]naphthyridine-8-carboxylic acidIC505.0 [1], 1351.0 [2]
5-[2-(3-Chlorophenyl)ethylamino]benzo[c][2,6]naphthyridine-8-carboxylic acidIC505.0 [1], 640.0 [2]
4-(3,5-Difluoroanilino)thieno[3,2-c]quinoline-7-carboxylic acidIC5070.0 [1], 4338.0 [2]
5-(3-Ethynylanilino)-3-(2-methoxyethylamino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC5010.0 [1], 40.0 [2]
N-(3-Fluorophenyl)-8-(2H-tetrazol-5-yl)benzo[c][2,6]naphthyridin-5-amineIC5047.0 [1], 630.0 [2]
3-(2-Ethoxyethylamino)-5-(3-ethynylanilino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC50171.0 [1], 172.0 [2]
5-(3-Ethynylanilino)-3-(oxolan-2-ylmethylamino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC5011.0 [1], 114.0 [2]
4-(3-Cyanoanilino)thieno[3,2-c]quinoline-7-carboxylic acidIC5081.0 [1], 10660.0 [2]
N-Methyl-3-[[7-(2H-tetrazol-5-yl)thieno[3,2-c]quinolin-4-yl]amino]benzamideIC50283.0 [1], 37890.0 [2]
5-(3-Chloro-4-fluoroanilino)-3-(cyclopropylamino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC5030.0 [1], 83.0 [2]
3-Amino-5-(3-chloro-4-fluoroanilino)pyrimido[4,5-c]quinoline-8-carboxylic acidIC507.0 [1], 44.0 [2]
Methyl 5-(3-chloro-4-fluoroanilino)benzo[c][2,6]naphthyridine-8-carboxylateIC501661.0 [1], 7066.0 [2]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Casein kinase II alpha Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/casein-kinase-ii-alpha-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Casein kinase II alpha Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/casein-kinase-ii-alpha-inhibitors-ic50-ki.
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