![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_beb7f72e73f61c5a9e1bf58b6572d39a.svg) | Cyclosporin A | IC50 | 13600.0 [1], 14500.0 [2], 20000.0 [3], 25600.0 [4] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_beb7f72e73f61c5a9e1bf58b6572d39a.svg) | Cyclosporin A | Ki | 4700.0 [1], 8110.0 [2], 21000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_762429a93cd073a0fe051daeaab480c5.svg) | Verlukast | IC50 | 1000.0 [1], 4000.0 [2], 10000.0 [3], 133000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_762429a93cd073a0fe051daeaab480c5.svg) | Verlukast | Ki | 13100.0 [1], 26400.0 [2] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_651f4cfbe9aa97adaf2f12469bdbaf84.svg) | Sodium | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_16f499e9c486fb216537dd71b443728b.svg) | Calcium | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_c1303ad3101dce1e315ea55e799cd202.svg) | Etoposide | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_c1303ad3101dce1e315ea55e799cd202.svg) | Etoposide | Ki | 756000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_01814a6086009d7440d5f435a324c600.svg) | Verapamil | IC50 | 133000.0 [1], 200000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_8eea222a1bcb2e74405ba02fe4c3db74.svg) | Reserpine | IC50 | 68400.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_8eea222a1bcb2e74405ba02fe4c3db74.svg) | Reserpine | Ki | 295000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_b03a82411601ac2483b9406eae5a6277.svg) | Simvastatin | IC50 | 25000.0 [1], 133000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_ad6ccf602ee43f3992fdd4c89edf213b.svg) | Probenecid | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_ad6ccf602ee43f3992fdd4c89edf213b.svg) | Probenecid | Ki | 42200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_39f28c7db5b571077dbf34394d5beb87.svg) | Dolutegravir | IC50 | 90000.0 [1], 100000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_b1defc2de62c1df9aff680bcb93af1f1.svg) | (5S,6R,7E,9E,11Z,14Z)-6-[(2S)-2-[[(4S)-4-Amino-4-carboxybutanoyl]amino]-3-(carboxymethylamino)-3-oxopropyl]sulfanyl-5-hydroxyicosa-7,9,11,14-tetraenoic acid | IC50 | 150.0 [1], 3300.0 [2] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_fed013ffe1da597b6e1b4df2d54259d1.svg) | Potassium | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_5c516e5fa259eb4dabbdf74f9982ff4f.svg) | Testosterone | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_403ea7c4448257bf6b5ee38ec62638e7.svg) | Aspirin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_eb212ff63ed7fef055dc658629968c96.svg) | 5-Fluorouracil | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_98a04b67a851c3bf4ca1fd9476597cf5.svg) | Doxorubicin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_1d64f7b51ed811e6ea11101a6c1d74e3.svg) | Dexamethasone | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_cdc9bc215732b879638336c369906e58.svg) | Cyclophosphamide | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_cd9b5820bcad56865f8364f10caaf311.svg) | Prednisolone | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_1cc257bab28d3e85f276bcae9f111347.svg) | Methotrexate | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_c70f5b79af37726016ec15cea0b55e94.svg) | Propranolol | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_bec8eaadb51e755de26c3660866564ee.svg) | Caffeine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_4fafa8dfcd5b32e244e222d42d1d8a8e.svg) | Warfarin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_71acea9a6dfc0e4dac7865946b73384c.svg) | Paclitaxel | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_2417c7be24e5d7debb18533147580339.svg) | Acetaminophen | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_ef61fa49423965b00cafb173f3e07a26.svg) | Indomethacin | IC50 | 235000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_f49643c3e5855473bdcde726c343e778.svg) | Melatonin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_3767f0f3bff8c5bb3468fa4b71c82615.svg) | Cyclosporine | IC50 | 3100.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_038301bf66445c6984ca669e09912730.svg) | Methylprednisolone | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_dc3b519ae4da383d84a5502ee939a5d0.svg) | Lidocaine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_86630ba4a7e4889b44175ac812cce53f.svg) | Nicotine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_15976e9843386a991246a922e8b855ad.svg) | Ciprofloxacin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_0cca37e8532dc6f7bb6fa13f5708ab01.svg) | Isoniazid | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_29f872b26cb31380c7e625ee9fa67f34.svg) | Theophylline | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_fbb5de82454ad47fc51ee2ed6f17cfc3.svg) | Vincristine | Ki | 802000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_973775538a5e21510c22b2ace50dc811.svg) | Tretinoin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_3a6bba03ec052485bdc33dc1df003990.svg) | Vincristine sulfate | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_393a6636008719cf0eb93219e05af350.svg) | Metformin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_10cf6922bd91d0359571f946a414f827.svg) | Tetracycline | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_b2d54f313fd6fae3559ad99a1d264705.svg) | Imatinib | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_f28ce47318433f5c984060ce11c4a797.svg) | Tamoxifen | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_4ad269998f5e13425718a1af1458766f.svg) | Gemcitabine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_3b0dab840ef0bf1dc3cf420126b55e81.svg) | Cytarabine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_93ff81dbb74065f6358ff2946a8ae8ed.svg) | Rifampicin | IC50 | 53000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_1816df2dc49c11e622026cae2c8dc356.svg) | Camptothecin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_db4ac60c18b24b7bd003d4edf05f0d21.svg) | Naloxone | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_38f1e4a242c4d3e6c7e8d2105139bf5a.svg) | Somatostatin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_2d46cd64b612bada34966bcfba251b25.svg) | Carbamazepine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_a7e11d7bcee94c9af8c42c557a082c25.svg) | Chlorpromazine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_2016e1fb48c552930d228a3e7f6e1433.svg) | Quercetin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_4401a17c9674bce3d2939b7f54f885a2.svg) | Levodopa | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_7ce5c90b273b41810bee3170ac9401d3.svg) | Haloperidol | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_07b574dd4ce0922414319841c8c53da0.svg) | Tacrolimus | IC50 | 40300.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_5498b28ac748aa1a1c2a1db363e8d2d0.svg) | Amoxicillin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_1232c84d43d4865ebdc5de8d7663a19f.svg) | Nifedipine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_693b10fcf0f1bf3ce26f73cb27aee812.svg) | Fluoxetine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_eeff5a96588de62beccbf378609f1809.svg) | Furosemide | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_923918ca2b63f82fdc23b9aff249ab4c.svg) | Chloroquine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_347b1b64f072d35207a2dcbef37b1046.svg) | Azathioprine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_2f6aa077265088f9306897fbb768392e.svg) | Salbutamol | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_dd9d47a0f93bd51eb50e8b6e680776e7.svg) | Calcitriol | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_7e646fe532894c3595457245499402ac.svg) | Colchicine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_0bd0719e120d20528fc513a96e10413d.svg) | Erythromycin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_8159b09a6bebd9e5751360e57f770ab8.svg) | Clozapine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_b3b0b96fadcb6f14e4a9be2aec908180.svg) | Omeprazole | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_e26448bf7b64df856705b530202d4116.svg) | Fluconazole | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_2eb69008645ff5a1555c94aa65edac97.svg) | Acyclovir | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_fbcb4fa3ddad51bf7bb5ba0967dcba8f.svg) | Metronidazole | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_5359f5c5b8786f1ff331cf22d9c655e5.svg) | Vinblastine | IC50 | 21000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_a047ba0a887d642df2938965c5266c0d.svg) | Ketamine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_6ed002577e209d84253997afbcf211f8.svg) | Carbon tetrachloride | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_80e0a660787cb33d419c39e347aee962.svg) | Vincaleukoblastine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_be4565ca8c20c1d9804fa640fd1584d5.svg) | Risperidone | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_aa2e99d28a503d46358101ca36fad499.svg) | Hydroxyurea | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_a6c9efafa4ac79796554cef55030a830.svg) | Ribavirin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_81af8877c0a8c32165f86d729092ee41.svg) | Amiodarone | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_8871e5bc150daca600c47dd7893b11be.svg) | Ethinyl estradiol | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_105aa90f970fa13d88993e59627fb373.svg) | Argipressin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_f0ad53ee3776de5bbc76b6da2787fa14.svg) | Bupivacaine hydrochloride | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_8b78ef0953132cb6729f40caa0d6bbea.svg) | Olanzapine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_7c96aacd70e2a071d3ee5d7e2d852a1d.svg) | Zidovudine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_3e94330ba1527a829fecddbee5acde55.svg) | Apomorphine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_b54108840a699d11d2503d2c2029b01e.svg) | Clarithromycin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_1d5eba4b4bb57896dda18b1604bab021.svg) | Staurosporine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_01ae8b9629ab2f1b394fdd8173a950dd.svg) | Docetaxel | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_23fca591a36dc0b52f4af729424e9b97.svg) | Allopurinol | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_b251fb4eaa57c07f3154b5aed978a0dd.svg) | Ofloxacin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_6c3911c895bcf58e15c1ea316421d8fe.svg) | Imipramine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_2019d6686c0079c33ef9d229dcb67e59.svg) | Dipyridamole | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_4966566b510149ad787ec8422453983d.svg) | Ticlopidine hydrochloride | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_7d4bb2f53887bffc73ff65aad54e92db.svg) | Captopril | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_3fb59b292039fb68c21d347565286601.svg) | Quinine | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_b83ef9b45debeb15bb4aeb2f69070c06.svg) | Ganciclovir | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_bc5cdfcd6f06f10b41114065330f79d1.svg) | Leucovorin | IC50 | 133000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/canalicular-multispecific-organic-anion-transporter-1_ed21bd772e0ab6cdca3f2f3540dc656d.svg) | Doxycycline hydrochloride | IC50 | 133000.0 [1] |