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Calpain 2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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Benzyl N-[1-[[1-(ethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi210.0 [1]
Benzyl N-[1-[[1-(cyclohexylmethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi44.0 [1]
Benzyl N-[1-[[1,2-dioxo-1-(2-phenylethylamino)pentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi22.0 [1]
Benzyl N-[1-[[4-(ethylamino)-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi39.0 [1]
Benzyl N-[1-[[3,4-dioxo-1-phenyl-4-(2-phenylethylamino)butan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi24.0 [1]
Benzyl N-[1-[[3,4-dioxo-1-phenyl-4-(propylamino)butan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi50.0 [1]
Benzyl N-[1-[[1,2-dioxo-1-(3-phenylpropylamino)pentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi43.0 [1]
Benzyl N-[1-[[1-(benzylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi22.0 [1], 350.0 [2]
Benzyl N-[1-[[1,2-dioxo-1-(propylamino)pentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi250.0 [1]
Benzyl N-[1-[[4-(benzylamino)-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi46.0 [1]
[(S)-1-(1-Ethylcarbamoyl-butylcarbamoyl)-3-methyl-butyl]-carbamic acid benzyl esterKi42.0 [1], 73.0 [2]
Benzyl N-[(2S)-1-[[1-(ethylamino)-1-oxo-3-phenylpropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi35.0 [1], 51.0 [2]
[(S)-1-(3-Ethylcarbamoyl-propylcarbamoyl)-3-methyl-butyl]-carbamic acid benzyl esterKi122.0 [1], 138.0 [2]
Z-Leu-leu-leu-alKi653.0 [1]
CID 11199915IC50350.0 [1]
3-(4-Iodophenyl)-2-mercapto-(Z)-2-propenoic acidKi370.0 [1]
Z-FY-ChoIC50184.0 [1]
CID 5353866Ki5330.0 [1]
3-Phenyl-N-(3-phenyl-N-((phenylmethoxy)carbonyl)-L-alanyl)-L-alanineIC50104.0 [1]
Z-Leu-Abu-CONH-CH2-CHOH-PhKi15.0 [1]
(R)-N-((S)-1-Benzyl-2-oxo-ethyl)-3-benzyloxy-2-methanesulfonylamino-propionamideKi5.0 [1]
(2R)-2-(Methanesulfonamido)-N-[(2S)-1-oxo-3-(4-phenylmethoxyphenyl)propan-2-yl]-3-phenylmethoxypropanamideKi5.0 [1]
(2R)-2-(Methanesulfonamido)-N-[(2S)-1-oxo-3-phenylpropan-2-yl]-3-phenylpropanamideKi13.0 [1]
(R)-N-((S)-1-Benzyl-2-oxo-ethyl)-3-benzyloxy-2-ethanesulfonylamino-propionamideKi9.0 [1]
(2R)-2-(Methanesulfonamido)-N-[(2S)-1-oxo-3-phenylpropan-2-yl]-3-thiophen-2-ylpropanamideKi11.0 [1]
(2S)-3-Benzylsulfanyl-2-(methanesulfonamido)-N-[(2S)-1-oxo-3-phenylpropan-2-yl]propanamideKi7.0 [1]
Benzyl N-[1-[[4-[3-(3,4-dihydro-1H-isoquinolin-2-yl)propylamino]-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi200.0 [1]
Benzyl N-[1-[[4-[3-(3,4-dihydro-2H-quinolin-1-yl)propylamino]-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi260.0 [1]
Benzyl N-[(9S,12S,15S)-15-[[(2S)-4-methyl-1-oxopentan-2-yl]carbamoyl]-12-(2-methylpropyl)-4-nitro-10,13-dioxo-2-oxa-11,14-diazatricyclo[15.2.2.13,7]docosa-1(19),3,5,7(22),17,20-hexaen-9-yl]carbamateKi2028.0 [1]
Benzyl N-[(9S,12S,15S)-12-[(4-methoxyphenyl)methyl]-15-[[(2S)-4-methyl-1-oxopentan-2-yl]carbamoyl]-4-nitro-10,13-dioxo-2-oxa-11,14-diazatricyclo[15.2.2.13,7]docosa-1(19),3,5,7(22),17,20-hexaen-9-yl]carbamateKi2983.0 [1]
Benzyl N-[(2S)-1-[[(2S)-3-(4-methoxyphenyl)-1-[[(2S)-1-[[(2S)-4-methyl-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]carbamateKi1708.0 [1]
Calpain Inhibitor XIIKi120.0 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-pentanoic acid ethyl esterKi400.0 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-4-phenyl-butyric acid ethyl esterKi400.0 [1]
Benzyl N-[1-[(1-amino-1,2-dioxopentan-3-yl)amino]-4-methyl-1-oxopentan-2-yl]carbamateKi19.0 [1]
Benzyl N-[4-methyl-1-[[1-(octylamino)-1,2-dioxopentan-3-yl]amino]-1-oxopentan-2-yl]carbamateKi19.0 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-4-phenyl-butyric acidKi5.7 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-pentanoic acidKi22.0 [1]
Benzyl N-[(7S,10S,13S)-7-formyl-10-(2-methylpropyl)-9,12-dioxo-2-oxa-8,11-diazabicyclo[13.2.2]nonadeca-1(17),15,18-trien-13-yl]carbamateIC5030.0 [1]
Benzyl N-[(6S,9S,12S)-6-formyl-9-(2-methylpropyl)-8,11-dioxo-2-oxa-7,10-diazabicyclo[12.2.2]octadeca-1(16),14,17-trien-12-yl]carbamateIC50850.0 [1]
Benzyl N-[(8S,11S,14S)-8-(hydroxymethyl)-11-(2-methylpropyl)-10,13-dioxo-2-oxa-9,12-diazabicyclo[14.2.2]icosa-1(18),16,19-trien-14-yl]carbamateIC501100.0 [1]
Benzyl N-[(9R,12S,15S)-9-(hydroxymethyl)-12-(2-methylpropyl)-11,14-dioxo-2-oxa-7-thia-10,13-diazabicyclo[15.2.2]henicosa-1(19),17,20-trien-15-yl]carbamateIC5028000.0 [1]
Benzyl N-[(6S,9S,12S)-6-(hydroxymethyl)-9-(2-methylpropyl)-8,11-dioxo-2-oxa-7,10-diazabicyclo[12.2.2]octadeca-1(16),14,17-trien-12-yl]carbamateIC5031000.0 [1]
Benzyl N-[(7S,10S,13S)-7-(hydroxymethyl)-10-(2-methylpropyl)-9,12-dioxo-2-oxa-8,11-diazabicyclo[13.2.2]nonadeca-1(17),15,18-trien-13-yl]carbamateIC50700.0 [1]
Benzyl N-[(8S,11S,14S)-8-formyl-11-(2-methylpropyl)-10,13-dioxo-2-oxa-9,12-diazabicyclo[14.2.2]icosa-1(18),16,19-trien-14-yl]carbamateIC50180.0 [1]
Benzyl N-[(9R,12S,15S)-9-formyl-12-(2-methylpropyl)-11,14-dioxo-2-oxa-7-thia-10,13-diazabicyclo[15.2.2]henicosa-1(19),17,20-trien-15-yl]carbamateIC501010.0 [1]
(R)-N-((S)-1-Benzyl-2-oxo-ethyl)-3-benzyloxy-2-methanesulfonylamino-butyramideKi7.0 [1]
Ethyl 4-(4-chlorophenyl)-3-[[4-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]amino]-2-oxobutanoateKi400.0 [1]
Ethyl 3-[[4-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]amino]-5-methylsulfanyl-2-oxopentanoateKi1500.0 [1]
Benzyl N-[1-[[1,2-dioxo-1-(2-phenylpropylamino)pentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi59.0 [1]
Benzyl N-[1-[(4-amino-3,4-dioxo-1-phenylbutan-2-yl)amino]-4-methyl-1-oxopentan-2-yl]carbamateKi760.0 [1]
Benzyl 3-[[4-methyl-2-(phenylmethoxycarbonylamino)pentanoyl]amino]-2-oxo-4-phenylbutanoateKi1600.0 [1]
Benzyl N-[1-[[1-(2,2-diphenylethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi63.0 [1]
Benzyl N-[1-[[1-(decylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi600.0 [1]
3-(2-Diphenylacetylamino-4-methyl-pentanoylamino)-2-oxo-pentanoic acid ethyl esterKi200.0 [1]
Ethyl 3-[[4-methyl-2-(3-phenylpropanoylamino)pentanoyl]amino]-2-oxopentanoateKi1200.0 [1]
Benzyl N-[1-[(1-amino-1,2-dioxohexan-3-yl)amino]-4-methyl-1-oxopentan-2-yl]carbamateKi78.0 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-hexanoic acid ethyl esterKi1200.0 [1]
Benzyl N-[1-[[4-(butylamino)-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi28.0 [1]
Benzyl N-[4-methyl-1-[[4-(2-methylpropylamino)-3,4-dioxo-1-phenylbutan-2-yl]amino]-1-oxopentan-2-yl]carbamateKi65.0 [1]
Benzyl N-[1-[[1-(ethylamino)-1,2-dioxohexan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi88.0 [1]
3-(2-Isobutoxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-pentanoic acid ethyl esterKi17000.0 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-pentanoic acid methyl esterKi500.0 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-pentanoic acid benzyl esterKi470.0 [1]
Benzyl N-[4-methyl-1-[[1-(2-methylpropylamino)-1,2-dioxopentan-3-yl]amino]-1-oxopentan-2-yl]carbamateKi140.0 [1]
Benzyl N-[1-[[1-(butylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi50.0 [1]
Ethyl 3-[[4-methyl-2-(4-phenylbutanoylamino)pentanoyl]amino]-2-oxopentanoateKi2900.0 [1]
Benzyl N-[1-[[1-(heptylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi67.0 [1]
Ethyl 3-[[4-methyl-2-[(4-methyl-5-phenylpentanoyl)amino]pentanoyl]amino]-2-oxopentanoateKi1600.0 [1]
Ethyl 3-[[4-methyl-2-(5-phenylpentanoylamino)pentanoyl]amino]-2-oxopentanoateKi1900.0 [1]
Ethyl 3-[[4-methyl-2-(naphthalen-2-ylsulfonylamino)pentanoyl]amino]-2-oxopentanoateKi2200.0 [1]
Ethyl 3-[[4-methyl-2-(2-phenoxybutanoylamino)pentanoyl]amino]-2-oxopentanoateKi1400.0 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-4-phenyl-butyric acid butyl esterKi1100.0 [1]
3-(2-Benzyloxycarbonylamino-4-methyl-pentanoylamino)-2-oxo-pentanoic acid butyl esterKi400.0 [1]
N-[1-[[1-(Ethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]isoquinoline-1-carboxamideKi110.0 [1]
N-[1-[[1-(Ethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]quinoline-2-carboxamideKi300.0 [1]
N-[1-[[1-(Ethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]morpholine-4-carboxamideKi9900.0 [1]
N-[1-[[1-(Ethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]pyrazine-2-carboxamideKi480.0 [1]
Benzyl N-[1-[[1-[(2-hydroxy-2-phenylethyl)amino]-1,2-dioxohexan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi11000.0 [1]
N-[1-[[1-(Ethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]furan-2-carboxamideKi580.0 [1]
Benzyl N-[4-methyl-1-[[1-(3-morpholin-4-ylpropylamino)-1,2-dioxohexan-3-yl]amino]-1-oxopentan-2-yl]carbamateKi100.0 [1]
Benzyl N-[4-methyl-1-[[1-(methylamino)-1,2-dioxopentan-3-yl]amino]-1-oxopentan-2-yl]carbamateKi83.0 [1]
Benzyl N-[1-[[4-[[2-hydroxy-2-[3-(trifluoromethyl)phenyl]ethyl]amino]-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi290.0 [1]
Benzyl N-[1-[[4-[[2-hydroxy-2-(2,3,4,5,6-pentafluorophenyl)ethyl]amino]-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi350.0 [1]
Benzyl N-[1-[[4-[[2-[4-(dimethylamino)phenyl]-2-hydroxyethyl]amino]-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi310.0 [1]
Benzyl N-[1-[[4-[(2-hydroxy-2-phenylethyl)amino]-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi50.0 [1]
N-[1-[[1-(Ethylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]pyridine-3-carboxamideKi830.0 [1]
Benzyl N-[4-methyl-1-[[1-[2-(1-methylpyrrol-2-yl)ethylamino]-1,2-dioxopentan-3-yl]amino]-1-oxopentan-2-yl]carbamateKi76.0 [1]
2-[(2,2-Diphenylacetyl)amino]-N-[1-[(2-hydroxy-2-phenylethyl)amino]-1,2-dioxopentan-3-yl]-4-methylpentanamideKi200.0 [1]
Benzyl N-[1-[[1-(3-imidazol-1-ylpropylamino)-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi68.0 [1]
2-[(2,2-Diphenylacetyl)amino]-N-[1-(ethylamino)-1,2-dioxopentan-3-yl]-4-methylpentanamideKi1200.0 [1]
Benzyl N-[4-methyl-1-[[1-(2-morpholin-4-ylethylamino)-1,2-dioxopentan-3-yl]amino]-1-oxopentan-2-yl]carbamateKi160.0 [1]
Benzyl N-[1-[[1-[2-(4-methoxyphenyl)ethylamino]-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi46.0 [1]
Benzyl N-[1-[[1-[2-(3-methoxyphenyl)ethylamino]-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi86.0 [1]
Benzyl N-[1-[[1-[2-(2-methoxyphenyl)ethylamino]-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi160.0 [1]
N-[1-(Ethylamino)-1,2-dioxopentan-3-yl]-4-methyl-2-[(2-naphthalen-1-ylacetyl)amino]pentanamideKi250.0 [1]
Benzyl N-[1-[[1-[2-(2-hydroxyethoxy)ethylamino]-1,2-dioxopentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi160.0 [1]
Benzyl N-[1-[[1,2-dioxo-1-(2-pyridin-2-ylethylamino)pentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi470.0 [1]
Benzyl N-[1-[[1,2-dioxo-1-(pyridin-3-ylmethylamino)pentan-3-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi120.0 [1]
Benzyl N-[1-[[4-[2-[5-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]pentanoylamino]ethylamino]-3,4-dioxo-1-phenylbutan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamateKi160.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ Calpain 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/calpain-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Calpain 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/calpain-2-inhibitors-ic50-ki.
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