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Calcium release-activated calcium channel protein 1 Inhibitors (IC50, Ki)

Structure
Compound Name
Standard Type
Standard Values (in nM)
MiconazoleIC5027000.0 [1], 100000.0 [2]
MibefradilIC5052100.0 [1], 100000.0 [2]
EconazoleIC5017000.0 [1], 94000.0 [2]
N-[4-(2,5-Dimethoxyphenyl)phenyl]-3-fluoro-N-methylpyridine-4-carboxamideIC5026.0 [1], 1300.0 [2]
1-[2-(4-Methoxyphenyl)-2-[4-(4-methoxyphenyl)butoxy]ethyl]imidazoleIC5042000.0 [1], 67000.0 [2]
3,5-Dichloro-2-(2-pyridin-3-yloxyethoxy)benzaldehydeIC50100000.0 [1]
CRAC Channel Inhibitor, BTP2IC502800.0 [1]
2-(4-Methoxyphenoxy)-1-[4-(4-phenylcyclohexyl)piperazin-1-yl]ethanoneIC5075000.0 [1]
4-Chloro-4'-[3,5-bis(trifluoromethyl)-1H-pyrazol-1-yl]benzanilideIC5057000.0 [1]
1-[5-Hydroxy-3-(3-nitrophenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5089000.0 [1]
2-(4-Chlorophenyl)-1-[5-hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanoneIC5047000.0 [1]
2-(3-Chlorophenyl)-1-[5-hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanoneIC5075000.0 [1]
1-[5-Hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(4-methoxyphenyl)ethanoneIC5033000.0 [1]
1-[5-Hydroxy-5-(trifluoromethyl)-3-[3-(trifluoromethyl)phenyl]-4H-pyrazol-1-yl]-2-phenylethanoneIC5029000.0 [1]
1-[3-(2,5-Dichlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5054000.0 [1]
2-(3-Chlorophenyl)-1-[5-hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanoneIC5079000.0 [1]
1-[5-Hydroxy-3-(trifluoromethyl)-5-[2-(trifluoromethyl)phenyl]-4H-pyrazol-1-yl]-2-phenylethanoneIC5049000.0 [1]
1-[5-Hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(3-methylphenyl)ethanoneIC5045000.0 [1]
2-(2-Chlorophenyl)-1-[5-hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanoneIC5042000.0 [1]
1-[5-Hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(3-methylphenyl)ethanoneIC5042000.0 [1]
1-[3-(2-Bromophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5030000.0 [1]
2-(2-Chlorophenyl)-1-[5-hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanoneIC5040000.0 [1]
1-[3-(3-Chlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5048000.0 [1]
1-[5-Hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(3-methoxyphenyl)ethanoneIC5032000.0 [1]
1-[3-(2,3-Difluorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5055000.0 [1]
2-(4-Chlorophenyl)-1-[5-hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]ethanoneIC5060000.0 [1]
1-[3-(2-Chlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5033000.0 [1]
1-[5-Hydroxy-3-(3-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5036000.0 [1]
1-[5-Hydroxy-3-(2-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenoxyethanoneIC50105000.0 [1]
1-[5-Hydroxy-3-(5,6,7,8-tetrahydronaphthalen-2-yl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5089000.0 [1]
1-[5-Hydroxy-3-(4-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(2-methylphenyl)ethanoneIC5055000.0 [1]
1-[3-(2,4-Dichlorophenyl)-5-hydroxy-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-phenylethanoneIC5058000.0 [1]
1-[5-Hydroxy-3-(4-methylphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-2-(3-methylphenyl)ethanoneIC5042000.0 [1]
Chembl4128571IC5047000.0 [1]
N-[6-(Benzimidazol-1-yl)pyridin-3-yl]-3-(dimethylamino)benzamideIC5048000.0 [1]
2-(2-Chloro-6-fluorophenyl)-5-[2-methyl-5-(trifluoromethyl)pyrazol-3-yl]-1H-pyrrolo[2,3-b]pyridineIC50100.0 [1]
2-(2-Chloro-6-fluorophenyl)-5-(6-methoxy-4-methylpyridin-3-yl)-1H-pyrrolo[2,3-b]pyridineIC50104.0 [1]
2-(2-Chloro-6-fluorophenyl)-5-(4,6-dimethoxypyridin-3-yl)-1H-pyrrolo[2,3-b]pyridineIC50440.0 [1]
(E)-1-[2-[2-(4-Butan-2-ylphenoxy)ethoxy]-3,5-dichlorophenyl]-N-(1,2,4-triazol-4-yl)methanimineIC5069900.0 [1]
N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-2H-benzotriazole-5-carboxamideIC50182.5 [1]
2-(Benzimidazol-1-yl)-N-[4-(3,5-dicyclopropylpyrazol-1-yl)phenyl]acetamideIC50383.1 [1]
2-(Benzotriazol-1-yl)-N-[4-(3,5-dicyclopropylpyrazol-1-yl)phenyl]acetamideIC5051.31 [1]
N-[4-(3,5-Dicyclopropylpyrazol-1-yl)phenyl]-2-quinolin-6-ylacetamideIC50146.7 [1]
2-(Benzotriazol-1-yl)-N-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]acetamideIC5039.17 [1]
2-(Benzotriazol-2-yl)-N-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]acetamideIC50139.0 [1]
N-[4-(3,5-Dicyclopropylpyrazol-1-yl)-3-fluorophenyl]-2-quinolin-6-ylacetamideIC50263.2 [1]
N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]quinoline-6-carboxamideIC5086.12 [1]
2-(Benzotriazol-1-yl)-N-[4-[5-cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]-3-fluorophenyl]acetamideIC50160.5 [1]
N-[4-[5-Cyclopropyl-3-(trifluoromethyl)pyrazol-1-yl]phenyl]quinoxaline-6-carboxamideIC5053.36 [1]



References

This online tool may be cited as follows

MLA

"Quest Database™ Calcium release-activated calcium channel protein 1 Inhibitors (IC50, Ki)." AAT Bioquest, Inc.22 Dec2024https://www.aatbio.com/data-sets/calcium-release-activated-calcium-channel-protein-1-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024December 22). Quest Database™ Calcium release-activated calcium channel protein 1 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/calcium-release-activated-calcium-channel-protein-1-inhibitors-ic50-ki.
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