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C-X-C chemokine receptor type 7 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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2-[3-[(3S,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC50800.0 [1], 860.0 [2]
Cyclo(-D-Tyr-Arg-Arg-Nal-Gly-)IC5030000.0 [1]
(3-Amino-6-ethyl-7,8-dihydro-5H-thieno[2,3-b][1,6]naphthyridin-2-yl)-(3,4-dihydro-1H-isoquinolin-2-yl)methanoneIC5010000.0 [1]
N-[3-[Benzyl(ethyl)amino]propyl]-2-(4-methyl-1-oxo-[1]benzothiolo[2,3-d]pyridazin-2-yl)butanamideIC502780.0 [1]
N-(1-Benzylpiperidin-4-yl)-2-[(4,7-dimethyl-2-oxo-2H-chromen-5-yl)oxy]acetamideIC501490.0 [1]
N-[(1-Ethylpyrrolidin-2-yl)methyl]-5-indol-1-ylthiophene-2-carboxamideIC506750.0 [1]
2-[3-[(2S,5S,8S,11R,14R)-5-[3-(Diaminomethylideneamino)propyl]-14-[(4-hydroxyphenyl)methyl]-11-methyl-8-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidineIC5030000.0 [1]
2-[3-[(2S,5S,8S,11S,14R)-5-[3-(Diaminomethylideneamino)propyl]-14-[(4-hydroxyphenyl)methyl]-11-methyl-8-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidineIC5018000.0 [1]
2-[3-[(2R,5S,8S,11S)-8-[3-(Diaminomethylideneamino)propyl]-2-[(4-hydroxyphenyl)methyl]-11-(naphthalen-2-ylmethyl)-3,6,9,12,16-pentaoxo-1,4,7,10,13-pentazacyclohexadec-5-yl]propyl]guanidineIC5030000.0 [1]
N-[3-[Benzyl(methyl)amino]propyl]-5-methyl-4-oxothieno[3,2-c]quinoline-2-carboxamideIC502210.0 [1]
3,4,5-Trimethoxy-N-[(E)-2-methyl-3-phenylprop-2-enyl]-N-(3-morpholin-4-ylpropyl)benzamideKi398.11 [1]
3,4-Dimethoxy-N-[(E)-2-methyl-3-phenylprop-2-enyl]-N-[2-(1-methylpyrrolidin-2-yl)ethyl]benzamideKi25.12 [1]
1-[4-Chloro-2-hydroxy-3-[(3S)-3-methyloxolan-3-yl]sulfonylphenyl]-3-[(1R)-2-methylcyclopent-2-en-1-yl]ureaIC5010000.0 [1]
N-(3-Hydroxypropyl)-3,4,5-trimethoxy-N-[(E)-2-methyl-3-phenylprop-2-enyl]benzamideKi1584.89 [1]
2-[3-[(2S,5S,8S,11S,14R)-5-[3-(Diaminomethylideneamino)propyl]-14-[(4-hydroxyphenyl)methyl]-10,11-dimethyl-8-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidineIC5015000.0 [1]
2-[3-[(2S,5S,8S,11R,14R)-5-[3-(Diaminomethylideneamino)propyl]-14-[(4-hydroxyphenyl)methyl]-10,11-dimethyl-8-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propyl]guanidineIC5030000.0 [1]
2-[3-[(3S,6S,9S,12S,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5030000.0 [1]
2-[3-[(3S,6R,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5030000.0 [1]
2-[3-[(3R,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5030000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-13-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5018000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-10-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC502400.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-4-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC503400.0 [1]
2-[3-[(3S,6S,9S,12S,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-13-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5023000.0 [1]
2-[3-[(3S,6S,9R,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-10-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5013000.0 [1]
2-[3-[(3S,6R,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC504600.0 [1]
2-[3-[(3R,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-4-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5030000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-7,12-dimethyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5030000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-12-[(4-Hydroxyphenyl)methyl]-7,9-dimethyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC5016000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-12-[(4-Hydroxyphenyl)methyl]-6,7-dimethyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5011000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-3,7-dimethyl-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC5030000.0 [1]
CXCR7 modulator 2Ki13.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-9-(3-Aminopropyl)-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502600.0 [1]
[4-[[4-(7-Ethylimidazo[1,2-a]pyridin-8-yl)-1,4-diazepan-1-yl]methyl]piperidin-1-yl]-[(1S,2R,4R)-7-oxabicyclo[2.2.1]heptan-2-yl]methanoneKi760.0 [1]
3-[(3S,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propylureaIC503600.0 [1]
Cyclopentyl-[4-[[4-(7-methylimidazo[1,2-a]pyridin-8-yl)-1,4-diazepan-1-yl]methyl]piperidin-1-yl]methanoneKi950.0 [1]
3-[(3S,6S,9S,12R,15S)-9-[3-(Diaminomethylideneamino)propyl]-7-methyl-3,12-bis(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propylureaIC50690.0 [1]
4-[[4-(1,7-Naphthyridin-8-yl)-1,4-diazepan-1-yl]methyl]-2-phenyl-1,3-thiazoleKi1900.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-12,16-bis(3-phenylpropyl)-3-(pyridin-3-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi25.12 [1]
2-[3-[(3S,6S,9S,12R,15S)-9-[(1R)-1-Hydroxyethyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-12-[(4-Hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-9-propan-2-yl-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-9-[(2S)-Butan-2-yl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
2-[(3S,6S,9S,12R,15S)-9-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]acetamideIC504100.0 [1]
3-[(2S,5S,8S,11R,14S)-8-[(2S)-Butan-2-yl]-14-[3-(diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-1,7-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC502200.0 [1]
3-[(2S,5S,8S,11R,14S)-14-[3-(Diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-1,7-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-8-[(4-phenylphenyl)methyl]-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC504000.0 [1]
3-[(3S,6S,9S,12R,15S)-9-[3-(Diaminomethylideneamino)propyl]-7-methyl-3-(naphthalen-2-ylmethyl)-12-[(4-nitrophenyl)methyl]-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propylureaIC502000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-6-(3-Aminopropyl)-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC501300.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-9-[4-(Diaminomethylideneamino)butyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC50840.0 [1]
Cyclopentyl-[3-[[4-(7-methylimidazo[1,2-a]pyridin-8-yl)-1,4-diazepan-1-yl]methyl]piperidin-1-yl]methanoneKi8500.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-7-methyl-12,16-bis(3-phenylpropyl)-3-(pyridin-3-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi19.95 [1]
2-[3-[(3S,6S,9S,12R,15S)-12-[(4-Hydroxyphenyl)methyl]-9-(1H-indol-3-ylmethyl)-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
3-[(3S,6S,9S,12R,15S)-9-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazatricyclo[13.8.0.017,22]tricosa-17,19,21-trien-6-yl]propylureaIC504200.0 [1]
2-Phenyl-4-[[4-[7-(trifluoromethyl)imidazo[1,2-a]pyridin-8-yl]-1,4-diazepan-1-yl]methyl]-1,3-thiazoleKi760.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-16-[3-(2,4-difluorophenyl)propyl]-6,12-bis(2,2-dimethylpropyl)-3-(1,3-thiazol-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi100.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-9-(4-Aminobutyl)-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
3-[(2S,5S,8S,11R,14S)-8-(1-Benzothiophen-3-ylmethyl)-14-[3-(diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-1,7-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC501000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-6-[4-(Diaminomethylideneamino)butyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propyl]guanidineIC50560.0 [1]
[4-[[4-(7-Ethylimidazo[1,2-a]pyridin-8-yl)-1,4-diazepan-1-yl]methyl]piperidin-1-yl]-[(1R,2S,4S)-7-oxabicyclo[2.2.1]heptan-2-yl]methanoneKi13.0 [1]
3-[(2S,5S,8S,11R,14S)-14-[3-(Diaminomethylideneamino)propyl]-8,11-bis[(4-hydroxyphenyl)methyl]-1,7-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC501800.0 [1]
3-[(3S,6S,9S,12R,15S)-12-Benzyl-9-[3-(diaminomethylideneamino)propyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propylureaIC501100.0 [1]
2-[3-[(3R,9S,12S,15R,18S,21S)-15-Benzyl-12,18-bis(1H-indol-3-ylmethyl)-2,8,11,14,17,20-hexaoxo-1,7,10,13,16,19-hexazatetracyclo[19.8.0.03,7.023,28]nonacosa-23,25,27-trien-9-yl]propyl]guanidineKi2100.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-6-(1H-indol-3-ylmethyl)-12,16-bis(3-phenylpropyl)-3-(pyridin-3-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi23.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-9,12-Bis[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-6,12-bis(1H-indol-3-ylmethyl)-16-(3-phenylpropyl)-3-(1,3-thiazol-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi32.0 [1]
3-[(2S,5S,8S,11R,14S)-14-[3-(Diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-1,7-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-8-(sulfanylmethyl)-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC504600.0 [1]
4-[[4-(6-Methylimidazo[1,2-a]pyridin-8-yl)-1,4-diazepan-1-yl]methyl]-2-phenyl-1,3-thiazoleKi900.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-6-(2,2-dimethylpropyl)-12,16-bis(3-phenylpropyl)-3-(pyridin-3-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi31.62 [1]
4-[[4-(7-Methylimidazo[1,2-a]pyridin-8-yl)-1,4-diazepan-1-yl]methyl]-2-phenyl-1,3-thiazoleKi29.0 [1]
[4-[[4-(7-Methylimidazo[1,2-a]pyridin-8-yl)-1,4-diazepan-1-yl]methyl]piperidin-1-yl]-[(1R,2S,4S)-7-oxabicyclo[2.2.1]heptan-2-yl]methanoneKi520.0 [1]
3-[(3S,6S,9S,12R,15S)-6-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-9-yl]propanamideIC509500.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-12-(cyclohexylmethyl)-16-[3-(2,4-difluorophenyl)propyl]-6-(2,2-dimethylpropyl)-3-(1,3-thiazol-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi31.62 [1]
3-[(2S,5S,8S,11R,14S)-14-[3-(Diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-8-(1H-indol-3-ylmethyl)-1-methyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC50850.0 [1]
3-[(1S,4R,7S,10S,13S)-7-[3-(Diaminomethylideneamino)propyl]-4-[(4-hydroxyphenyl)methyl]-9-methyl-13-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-3,6,9,12,15-pentazatricyclo[13.7.0.016,21]docosa-16,18,20-trien-10-yl]propylureaIC50190.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-12-[(4-Hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-9-(sulfanylmethyl)-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC50250.0 [1]
3-[(3S,6S,9S,12R,15S)-9-[3-(Diaminomethylideneamino)propyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propylureaIC5013000.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-12-[(4-Hydroxyphenyl)methyl]-9-(1H-imidazol-5-ylmethyl)-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
3-[(2S,5S,8S,11R,14S)-14-[3-(Diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-1,7-dimethyl-8-(2-methylpropyl)-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC501900.0 [1]
(3S,6S,9R,12S,18R)-9,12-Dibenzyl-6-(2,2-dimethylpropyl)-16-(3-phenylpropyl)-3-(1,3-thiazol-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi501.19 [1]
2-[3-[(3S,6S,9R,12S,18R)-9-Benzyl-16-[3-(2,4-difluorophenyl)propyl]-6,12-bis(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-3-yl]propyl]guanidineKi8.0 [1]
3-[(2S,5S,8S,11R,14S)-14-[3-(Diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-1,7-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-8-propan-2-yl-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC504900.0 [1]
2-[3-[(3S,6S,9R,12S,18R)-9-Benzyl-6,12-bis(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-16-(2-phenylethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-3-yl]propyl]guanidineKi7700.0 [1]
3-[(3S,6S,9S,12R,15S)-9-[3-(Diaminomethylideneamino)propyl]-12-[(2-fluorophenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propylureaIC50410.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-9-Benzyl-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
3-[(2S,5S,8S,11R,14S)-8-Benzyl-14-[3-(diaminomethylideneamino)propyl]-11-[(4-hydroxyphenyl)methyl]-1,7-dimethyl-5-(naphthalen-2-ylmethyl)-3,6,9,12,15-pentaoxo-1,4,7,10,13-pentazacyclopentadec-2-yl]propylureaIC50600.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-6,12-bis(1H-indol-3-ylmethyl)-3-[(1-methylimidazol-4-yl)methyl]-16-(3-phenylpropyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi410.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-6,12,16-tris(3-phenylpropyl)-3-(pyridin-3-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi71.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-12-[(4-Hydroxyphenyl)methyl]-7-methyl-9-(2-methylpropyl)-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502000.0 [1]
3-[(3S,6S,9S,12R,15S)-12-[(4-Chlorophenyl)methyl]-9-[3-(diaminomethylideneamino)propyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propylureaIC50790.0 [1]
[4-[[4-(7-Methylimidazo[1,2-a]pyridin-8-yl)-1,4-diazepan-1-yl]methyl]piperidin-1-yl]-(oxolan-3-yl)methanoneKi9700.0 [1]
CXCR7 modulator 1Ki10.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-7,10-dimethyl-12,16-bis(3-phenylpropyl)-3-(pyridin-3-ylmethyl)-6-(1,3-thiazol-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi199.53 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-6,12-bis(1H-indol-3-ylmethyl)-16-(3-phenylpropyl)-3-(pyridin-3-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi71.0 [1]
3-[(3S,6S,9S,12R,15S)-12-[(4-Benzoylphenyl)methyl]-9-[3-(diaminomethylideneamino)propyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propylureaIC50720.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-16-[3-(2,4-difluorophenyl)propyl]-6-(2,2-dimethylpropyl)-12-[(4-fluorophenyl)methyl]-3-(1,3-thiazol-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi39.81 [1]
3-[(3S,6S,9S,12R,15S)-12-(1-Benzothiophen-3-ylmethyl)-9-[3-(diaminomethylideneamino)propyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propylureaIC50540.0 [1]
2-Phenyl-4-[[4-[7-(trifluoromethoxy)quinolin-8-yl]-1,4-diazepan-1-yl]methyl]-1,3-thiazoleKi42.0 [1]
(3S,6S,9R,12S,18R)-9-Benzyl-6,12-bis(1H-indol-3-ylmethyl)-16-(3-phenylpropyl)-3-(pyridin-4-ylmethyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi189.0 [1]
2-[3-[(3S,6S,9R,12S,18R)-9,16-Dibenzyl-6,12-bis(1H-indol-3-ylmethyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosan-3-yl]propyl]guanidineKi4500.0 [1]
2-Phenyl-4-[[4-(6-propan-2-yl-1,7-naphthyridin-8-yl)-1,4-diazepan-1-yl]methyl]-1,3-thiazoleKi730.0 [1]
(3S,6S,9R,12S,18R)-3,9-Dibenzyl-6,12-bis(1H-indol-3-ylmethyl)-16-(3-phenylpropyl)-1,4,7,10,13,16-hexazabicyclo[16.3.0]henicosane-2,5,8,11,14,17-hexoneKi774.0 [1]
2-[3-[(3S,6S,9S,12R,15S)-9-[2-(Diaminomethylideneamino)ethyl]-12-[(4-hydroxyphenyl)methyl]-7-methyl-3-(naphthalen-2-ylmethyl)-2,5,8,11,14-pentaoxo-1,4,7,10,13-pentazabicyclo[13.3.0]octadecan-6-yl]propyl]guanidineIC502600.0 [1]
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References

This online tool may be cited as follows

MLA

"Quest Database™ C-X-C chemokine receptor type 7 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 19 Feb. 2025, https://www.aatbio.com/data-sets/c-x-c-chemokine-receptor-type-7-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 19). Quest Database™ C-X-C chemokine receptor type 7 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/c-x-c-chemokine-receptor-type-7-inhibitors-ic50-ki.
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