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C-C motif chemokine 2 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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Cyclohexanecarboxamide, 4-[(1R)-1-aminoethyl]-N-4-pyridinyl-, trans-IC502630.27 [1]
FasudilIC506918.31 [1]
HydroxyfasudilIC506918.31 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-(2,3-dihydro-1H-inden-1-ylamino)-1-propan-2-ylcyclopentane-1-carboxamideKi50.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-(cyclohexylamino)-1-propan-2-ylcyclopentane-1-carboxamideKi110.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-(oxan-4-ylamino)-1-propan-2-ylcyclopentane-1-carboxamideKi6.8 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-1-propan-2-yl-3-(thian-4-ylamino)cyclopentane-1-carboxamideKi31.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-1-propan-2-yl-3-(1,2,3,4-tetrahydronaphthalen-1-ylamino)cyclopentane-1-carboxamideKi33.0 [1]
(1S,3R)-3-(Benzylamino)-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1-propan-2-ylcyclopentane-1-carboxamideKi437.0 [1]
6-[(2-Phenylethylamino)methyl]isoquinolin-1-amineIC5031622.78 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(5-methoxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi6.1 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(5-hydroxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi29.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(5-chloro-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi18.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(5-bromo-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi289.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(6-methyl-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi55.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(6-cyano-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi54.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(4,5-dimethoxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi130.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(5,6-dimethoxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi3.9 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-(6,7-dihydro-5H-cyclopenta[f][1,3]benzodioxol-7-ylamino)-1-propan-2-ylcyclopentane-1-carboxamideKi6.3 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi27.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(5-hydroxy-1,2,3,4-tetrahydronaphthalen-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi35.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-(2-phenylethylamino)-1-propan-2-ylcyclopentane-1-carboxamideKi2400.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-(3-phenylpropylamino)-1-propan-2-ylcyclopentane-1-carboxamideKi134.0 [1]
(1S,3R)-3-[(4-Amino-2,3-dihydro-1H-inden-1-yl)amino]-N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-1-propan-2-ylcyclopentane-1-carboxamideKi43.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(4-hydroxy-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi86.0 [1]
(1S,3R)-N-[[3,5-Bis(trifluoromethyl)phenyl]methyl]-3-[(4-cyano-2,3-dihydro-1H-inden-1-yl)amino]-1-propan-2-ylcyclopentane-1-carboxamideKi70.0 [1]
Items per page: 1 - 10 of 26
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References

This online tool may be cited as follows

MLA

"Quest Database™ C-C motif chemokine 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/c-c-motif-chemokine-2-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ C-C motif chemokine 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/c-c-motif-chemokine-2-inhibitors-ic50-ki.
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