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C-C chemokine receptor type 10 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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4-Amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC5012.59 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamideIC500.4 [1], 1.0 [2], 1.26 [3], 10.0 [4], 25.12 [5], 3162.28 [6]
4-Amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-4-(2-nitroimidazol-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC5053.0 [1], 251.19 [2], 690.0 [3], 794.33 [4]
4-Amino-3,5-dichloro-N-[(2S)-1-(4-methylpiperidin-1-yl)-1-oxo-4-phenylbutan-2-yl]benzenesulfonamideIC5010000.0 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-6-sulfonamideIC507.94 [1], 15.85 [2]
N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-5-sulfonamideIC5012.59 [1], 199.53 [2]
4-Amino-3,5-dichloro-N-[(2R)-1-(4-methylpiperidin-1-yl)-1-oxo-4-phenylbutan-2-yl]benzenesulfonamideIC50501.19 [1], 630.96 [2]
4-Amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-(triazol-2-yl)butan-2-yl]benzenesulfonamideIC501258.93 [1], 3162.28 [2]
4-Amino-3,5-dichloro-N-[4-(2-chloroimidazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC50251.19 [1], 501.19 [2]
3-Amino-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-2,4-dimethylbenzenesulfonamideIC5079.43 [1], 100.0 [2]
4-Amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-pyrazol-1-ylbutan-2-yl]benzenesulfonamideIC501258.93 [1], 1584.89 [2]
CID 46861584IC5010000.0 [1]
4-Amino-3,5-dichloro-N-[(2R)-1-(4-methylpiperidin-1-yl)-4-(2-nitroimidazol-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC50501.19 [1]
2-[(4-Amino-3,5-dichlorophenyl)sulfonylamino]-4-(2-cyanopyrrol-1-yl)-N,N-dimethylbutanamideIC5010000.0 [1]
4-Amino-3,5-dichloro-N-[(2R)-4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC507.94 [1]
4-Amino-3,5-dichloro-N-[(2S)-1-(4-methylpiperidin-1-yl)-4-(2-nitroimidazol-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC5019952.62 [1]
4-Amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-oxo-1-pyrrolidin-1-ylbutan-2-yl]benzenesulfonamideIC5010000.0 [1]
4-Amino-3,5-dichloro-N-[4-imidazol-1-yl-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC5019952.62 [1]
4-Amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-(triazol-1-yl)butan-2-yl]benzenesulfonamideIC5019952.62 [1]
4-(2-Cyanopyrrol-1-yl)-2-(1H-indol-4-ylsulfonylamino)-N,N-dimethylbutanamideIC503981.07 [1]
4-Amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-(1,2,4-triazol-1-yl)butan-2-yl]benzenesulfonamideIC5019952.62 [1]
4-Amino-3,5-dichloro-N-[(2S)-4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC5015848.93 [1]
Methyl (2S)-1-[(2R)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2S)-1-[(2R)-2-hydroxy-3-methylbutanoyl]pyrrolidine-2-carbonyl]amino]acetyl]-methylamino]-4-methylpentanoyl]amino]propanoyl]-methylamino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC5020000.0 [1]
Methyl (2S)-1-[(2R)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2S)-1-[(2R,3S)-2-hydroxy-3-methylpentanoyl]pyrrolidine-2-carbonyl]amino]acetyl]-methylamino]-4-methylpentanoyl]amino]propanoyl]-methylamino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC5020000.0 [1]
Methyl (2S)-1-[(2R)-2-[methyl-[(2S)-2-[[(2S)-4-methyl-2-[methyl-[2-[[(2S)-1-[(2R,3S)-3-methyl-2-(3-phenylpropanoyloxy)pentanoyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]pentanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC503140.0 [1]
Methyl (2S)-1-[(2R)-2-[methyl-[(2S)-2-[[(2S)-4-methyl-2-[methyl-[2-[[(2S)-1-[(2R,3S)-3-methyl-2-[(E)-3-phenylprop-2-enoyl]oxypentanoyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]pentanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC50440.0 [1]
Methyl (2S)-1-[(2R)-2-[methyl-[(2S)-2-[[(2S)-4-methyl-2-[methyl-[2-[[(2S)-1-[(2R,3S)-3-methyl-2-[(Z)-3-phenylprop-2-enoyl]oxypentanoyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]pentanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC502710.0 [1]
Methyl (2S)-1-[(2R)-2-[[(2S)-2-[[(2S)-2-[[2-[[(2S)-1-[(2R,3S)-2-[(2S)-2-(dimethylamino)-3-phenylpropanoyl]oxy-3-methylpentanoyl]pyrrolidine-2-carbonyl]amino]acetyl]-methylamino]-4-methylpentanoyl]amino]propanoyl]-methylamino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC5020000.0 [1]
Methyl (2S)-1-[(2R)-2-[methyl-[(2S)-2-[[(2S)-4-methyl-2-[methyl-[2-[[(2S)-1-[(2R,3S)-3-methyl-2-(3-phenylprop-2-ynoyloxy)pentanoyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]pentanoyl]amino]propanoyl]amino]-3-phenylpropanoyl]pyrrolidine-2-carboxylateIC5020000.0 [1]
4-Amino-3,5-dichloro-N-[4-(2-chlorophenyl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC50125.89 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1-methylindole-4-sulfonamideIC50125.89 [1]
4-Amino-3,5-dichloro-N-[1-(4-methylpiperidin-1-yl)-1-oxo-4-pyrrol-1-ylbutan-2-yl]benzenesulfonamideIC503981.07 [1]
4-Amino-3,5-dichloro-N-[4-(2-cyanoimidazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC50501.19 [1]
4-Amino-3,5-dichloro-N-[4-(5-cyanopyrazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC5063.1 [1]
4-Amino-N-[1-(azepan-1-yl)-4-(2-cyanopyrrol-1-yl)-1-oxobutan-2-yl]-3,5-dichlorobenzenesulfonamideIC50251.19 [1]
4-Amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-oxo-1-[4-(trifluoromethyl)piperidin-1-yl]butan-2-yl]benzenesulfonamideIC50398.11 [1]
4-Amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(3-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC50630.96 [1]
4-Amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-oxo-1-piperidin-1-ylbutan-2-yl]benzenesulfonamideIC50158.49 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(4-hydroxypiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamideIC50125.89 [1]
4-Amino-2,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC5063.1 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(2-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamideIC5019.95 [1]
2-Amino-4,6-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC5039.81 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(3-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamideIC5063.1 [1]
4-Amino-3,5-dichloro-N-[4-(2-cyanopyrrol-1-yl)-1-(2-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC50794.33 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC501258.93 [1]
4-Amino-3,5-dichloro-N-[4-(5-chloropyrazol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]benzenesulfonamideIC50251.19 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-oxo-1-[4-(trifluoromethyl)piperidin-1-yl]butan-2-yl]-1H-indole-4-sulfonamideIC5010.0 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-oxo-1-piperidin-1-ylbutan-2-yl]-1H-indole-4-sulfonamideIC5010.0 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]naphthalene-1-sulfonamideIC5050.12 [1]
N-[1-(Azepan-1-yl)-4-(2-cyanopyrrol-1-yl)-1-oxobutan-2-yl]-1H-indole-4-sulfonamideIC5025.12 [1]
N-[4-(2-Cyanopyrrol-1-yl)-1-(4-methylpiperidin-1-yl)-1-oxobutan-2-yl]-1H-indole-7-sulfonamideIC50251.19 [1]
Items per page: 1 - 10 of 51
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References

This online tool may be cited as follows

MLA

"Quest Database™ C-C chemokine receptor type 10 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/c-c-chemokine-receptor-type-10-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ C-C chemokine receptor type 10 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/c-c-chemokine-receptor-type-10-inhibitors-ic50-ki.
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