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Bromodomain-containing protein 9 Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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N-[(2R,3S)-2-(4-Chlorophenyl)-1-(1,4-dimethyl-2-oxoquinolin-7-yl)-6-oxopiperidin-3-yl]-2-methylpropane-1-sulfonamideIC503300.0 [1], 5100.0 [2], 6200.0 [3]
4-Cyano-N-(1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50310.0 [1], 1100.0 [2]
4-Cyano-N-(1,3-diethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC5020000.0 [1], 100000.0 [2]
N'-(1,1-Dioxothian-4-yl)-5-ethyl-4-oxo-7-[3-(trifluoromethyl)phenyl]thieno[3,2-c]pyridine-2-carboximidamideIC5050.12 [1], 79.43 [2], 158.49 [3]
(4R)-4-Methyl-6-[1-methyl-3-(1-methylpyrazol-4-yl)indazol-5-yl]-1,3,4,5-tetrahydro-1,5-benzodiazepin-2-oneIC50730.0 [1]
CID 91827373IC50520.0 [1], 4400.0 [2]
4-Cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50910.0 [1]
N-(1-Methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50220.0 [1], 2200.0 [2]
1-Methyl-2-quinoloneIC5014000.0 [1]
Sgc-cbp30IC5020000.0 [1]
4-[(2s,4r)-1-Acetyl-4-[(4-Chlorophenyl)amino]-2-Methyl-1,2,3,4-Tetrahydroquinolin-6-Yl]benzoic AcidIC5031622.78 [1]
1-(7-(2-Methylsulfonyl-phenyl)-4-propoxy-1-aza-bicyclo[4.3.0]nona-2,4,6,8-tetraen-9-yl)-ethanoneIC5050000.0 [1]
4-[4-[(Dimethylamino)methyl]-2,5-Dimethoxy-Phenyl]-2-Methyl-2,7-Naphthyridin-1-OneIC5075.0 [1]
4-[4-[(Dimethylamino)methyl]-3,5-Dimethoxy-Phenyl]-2-Methyl-2,7-Naphthyridin-1-OneIC5019.0 [1]
3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-N-methyl-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridine-5-carboxamideIC5020000.0 [1]
5-{4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl}-1,3,6-trimethyl-1,2-dihydro-pyridin-2-oneIC5057.0 [1]
4-{4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl}-2-methyl-1,2-dihydroisoquinolin-1-oneIC5030.0 [1]
4-Bromo-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC507943.28 [1]
4-Bromo-2-methyl-5-[[(3S,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5031622.78 [1]
N,2-Dimethyl-5-(3-methyl[1,2,4]triazolo[3,4-a]phthalazin-6-yl)benzenesulfonamideIC501258.93 [1]
N-(1,4-Dimethyl-7-morpholin-4-yl-2,3-dioxoquinoxalin-6-yl)-4-(2-methylpropyl)benzenesulfonamideIC50204000.0 [1]
N-[5-(3-Methyl-[1,2,4]triazolo[3,4-a]phthalazin-6-yl)-2-morpholin-4-ylphenyl]methanesulfonamideIC50316.23 [1]
1-(3-Phenylazanyl-1,4,6,7-Tetrahydropyrazolo[4,3-C]pyridin-5-Yl)ethanoneIC5020000.0 [1]
4-Chloro-2-methyl-5-[(1-methylpiperidin-4-yl)amino]pyridazin-3-oneIC5050118.72 [1]
4-Chloro-2-methyl-5-(propan-2-ylamino)pyridazin-3-oneIC5050118.72 [1]
4-Chloro-2-methyl-5-[(1-methylpiperidin-3-yl)amino]pyridazin-3-oneIC5050118.72 [1]
5-[3,5-Dimethoxy-4-[(3-Oxidanylazetidin-1-Yl)methyl]phenyl]-1,3-Dimethyl-Pyridin-2-OneIC5021.0 [1]
4-(1,5-Dimethyl-6-Oxidanylidene-Pyridin-3-Yl)benzamideIC509338.0 [1]
4-Cyano-2-methoxy-N-(7-methoxy-1,3-dimethyl-2-oxoquinolin-6-yl)benzenesulfonamideIC50170.0 [1]
3-Chloro-4-cyano-N-(1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC502500.0 [1]
4-Cyano-N-(7-methoxy-1-methyl-2-oxoquinolin-6-yl)benzenesulfonamideIC502700.0 [1]
4-Cyano-N-(7-Methoxy-1,4-Dimethyl-2-Oxo-1,2-Dihydroquinolin-6-Yl)benzene-1-SulfonamideIC50890.0 [1]
(4R)-6-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-4-methyl-1,3,4,5-tetrahydro-1,5-benzodiazepin-2-oneIC5020000.0 [1]
N,6-Dimethyl-7-oxo-N-[1-(1-phenylethyl)piperidin-4-yl]-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC5011000.0 [1]
N-Methyl-7-oxo-6-prop-2-enyl-N-[1-(6-pyrazol-1-ylpyrimidin-4-yl)piperidin-4-yl]-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC506900.0 [1]
N-[1-(6-Methoxypyrimidin-4-yl)piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC508500.0 [1]
N-Methyl-7-oxo-6-prop-2-enyl-N-(1-pyrimidin-4-ylpiperidin-4-yl)-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC505000.0 [1]
6-Methyl-N-(1-methylpiperidin-4-yl)-7-oxo-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC502400.0 [1]
N,6-Dimethyl-7-oxo-N-(1-propan-2-ylpiperidin-4-yl)-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC5017800.0 [1]
N,6-Dimethyl-N-(1-methylpiperidin-4-yl)-7-oxo-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC5020000.0 [1]
N-Methyl-7-oxo-6-prop-2-enyl-N-[1-[6-(trifluoromethyl)pyrimidin-4-yl]piperidin-4-yl]-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC5011400.0 [1]
1-[3-[7-(Difluoromethyl)-6-(1-methylpyrazol-4-yl)-3,4-dihydro-2H-quinolin-1-yl]-1-(oxan-4-yl)-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5020000.0 [1]
1-[3-[2-Fluoro-4-(1-methylpyrazol-4-yl)anilino]-1-[(3R)-oxolan-3-yl]-6,7-dihydro-4H-pyrazolo[4,3-c]pyridin-5-yl]ethanoneIC5020000.0 [1]
4-Chloro-2-methyl-5-[[(3S)-1-methylpiperidin-3-yl]amino]pyridazin-3-oneIC5050118.72 [1]
4-Chloro-2-methyl-5-[[(3R)-1-methylpiperidin-3-yl]amino]pyridazin-3-oneIC5050118.72 [1]
7-(3,4-Dimethoxyphenyl)-N',5-dimethyl-4-oxothieno[3,2-c]pyridine-2-carboximidamideIC5079.43 [1]
7-(3,4-Dimethoxyphenyl)-N'-(1,1-dioxothian-4-yl)-5-methyl-4-oxothieno[3,2-c]pyridine-2-carboximidamideIC507.94 [1]
7-[3-(Dimethylamino)phenyl]-N'-(1,1-dioxothian-4-yl)-5-methyl-4-oxothieno[3,2-c]pyridine-2-carboximidamideIC5010.0 [1]
7-(3-Cyanophenyl)-N'-(1,1-dioxothian-4-yl)-5-methyl-4-oxothieno[3,2-c]pyridine-2-carboximidamideIC5039.81 [1]
7-(3,4-Dimethoxyphenyl)-5-methyl-2-(piperidine-1-carbonyl)thieno[3,2-c]pyridin-4-oneIC503981.07 [1]
7-(3,4-Dimethoxyphenyl)-N,N,5-trimethyl-4-oxothieno[3,2-c]pyridine-2-carboxamideIC505011.87 [1]
7-(3,4-Dimethoxyphenyl)-N,5-dimethyl-4-oxothieno[3,2-c]pyridine-2-carboxamideIC50125.89 [1]
1-[1-[2-(Hydroxymethyl)phenyl]indolizin-3-yl]ethanoneIC5023700.0 [1]
1-[1-(2-Methylsulfonylphenyl)indolizin-3-yl]ethanoneIC5017900.0 [1]
1-[7-Methoxy-1-(2-methylsulfonylphenyl)indolizin-3-yl]ethanoneIC5050000.0 [1]
N'-(1,1-Dioxothian-4-yl)-4-oxo-5-propan-2-yl-7-[3-(trifluoromethyl)phenyl]thieno[3,2-c]pyridine-2-carboximidamideIC503162.28 [1]
N'-(1,1-Dioxothian-4-yl)-5-methyl-4-oxo-7-phenylthieno[3,2-c]pyridine-2-carboximidamideIC5039.81 [1]
N'-(1,1-Dioxothian-4-yl)-7-(3-methoxyphenyl)-5-methyl-4-oxothieno[3,2-c]pyridine-2-carboximidamideIC5012.59 [1]
Tert-butyl N-[[3-acetyl-1-(2-methylsulfonylphenyl)indolizin-7-yl]methyl]carbamateIC501400.0 [1]
5-[4-[(Dimethylamino)methyl]-2,5-dimethoxyphenyl]-1,3,6-trimethylpyridin-2-oneIC50134.0 [1]
5-[4-[(Dimethylamino)methyl]-2,5-dimethoxyphenyl]-1,3,4-trimethylpyridin-2-oneIC50507.0 [1]
4-[4-[(Dimethylamino)methyl]-2,5-dimethoxyphenyl]-2-methylisoquinolin-1-oneIC50134.0 [1]
5-[4-[(Dimethylamino)methyl]phenyl]-1,3-dimethylpyridin-2-oneIC501147.0 [1]
5-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-1,3-dimethylpyridin-2-oneIC5054.0 [1]
5-[4-[(Dimethylamino)methyl]-3-methoxy-5-methylphenyl]-1,3-dimethylpyridin-2-oneIC50656.0 [1]
5-[4-[(Dimethylamino)methyl]-3-ethyl-5-methoxyphenyl]-1,3-dimethylpyridin-2-oneIC50195.0 [1]
5-[4-[(Dimethylamino)methyl]-2,5-dimethoxyphenyl]-1,3-dimethylpyridin-2-oneIC50468.0 [1]
5-[4-[(3-Aminoazetidin-1-yl)methyl]-3,5-dimethoxyphenyl]-1,3-dimethylpyridin-2-oneIC509.0 [1]
5-[4-[(Dimethylamino)methyl]-3-methoxyphenyl]-1,3-dimethylpyridin-2-oneIC50470.0 [1]
8-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-6-methylpyrido[4,3-d]pyrimidin-5-oneIC5037.0 [1]
5-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-1,3,4-trimethylpyridin-2-oneIC5037.0 [1]
5-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-7-methyl-1,7-naphthyridin-8-oneIC50250.0 [1]
4-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-2-methyl-2,6-naphthyridin-1-oneIC50128.0 [1]
8-[4-[(Dimethylamino)methyl]-3,5-dimethoxyphenyl]-6-methyl-1,6-naphthyridin-5-oneIC50134.0 [1]
N,2-Dimethyl-7-oxo-N-[1-[(1S)-1-phenylethyl]piperidin-4-yl]-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC504400.0 [1]
4-Chloro-2-methyl-5-[(2-methyl-3,4-dihydro-1H-isoquinolin-5-yl)amino]pyridazin-3-oneIC502000.0 [1]
N-[1-(2,6-Dimethylpyrimidin-4-yl)piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC507600.0 [1]
N-[1-[6-(3-Methoxyphenyl)pyrimidin-4-yl]piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC501600.0 [1]
4-Cyano-2-methoxy-N-(1-methyl-2-oxo-3-propan-2-ylquinolin-6-yl)benzenesulfonamideIC509300.0 [1]
5-Anilino-4-chloro-2-methylpyridazin-3-oneIC502511.89 [1]
N-[1-(6-Tert-butylpyrimidin-4-yl)piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC505700.0 [1]
4-Chloro-2-methyl-5-[[(3S,5S)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5050118.72 [1]
1-Methyl-2-oxo-N-phenylquinoline-6-sulfonamideIC509800.0 [1]
N-Methyl-7-oxo-N-[1-(1-phenylethyl)piperidin-4-yl]-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC5020000.0 [1]
N-[1-(6-Cyclopropyl-2-methylpyrimidin-4-yl)piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC503500.0 [1]
4-Chloro-2-methyl-5-[[(3R,5R)-1-methyl-5-phenylpiperidin-3-yl]amino]pyridazin-3-oneIC5031622.78 [1]
N-[1-(6-Methoxy-2-methylpyrimidin-4-yl)piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC505800.0 [1]
N-[1-[6-(2-Methoxyphenyl)pyrimidin-4-yl]piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC502600.0 [1]
N-(1,3-Dimethyl-2-oxo-7-pyrrolidin-1-ylquinolin-6-yl)-2-methoxybenzamideIC50420.0 [1]
N-[1-[6-(2-Fluorophenyl)pyrimidin-4-yl]piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC501500.0 [1]
N,2-Dimethyl-7-oxo-N-[1-[(1R)-1-phenylethyl]piperidin-4-yl]-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC503500.0 [1]
N-[1-[6-(Furan-2-yl)pyrimidin-4-yl]piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC503300.0 [1]
4-Chloro-2-methyl-5-(3-methylanilino)pyridazin-3-oneIC501258.93 [1]
N-[1-(6-Cyclopropylpyrimidin-4-yl)piperidin-4-yl]-N-methyl-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC506100.0 [1]
N-Methyl-N-[1-[6-(2-methylphenyl)pyrimidin-4-yl]piperidin-4-yl]-7-oxo-6-prop-2-enyl-1H-pyrrolo[2,3-c]pyridine-4-carboxamideIC501700.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-5-(furan-2-yl)benzoic acidIC5020000.0 [1]
3-[(1-Acetyl-5-methoxyindole-3-carbonyl)amino]-4-fluoro-5-(1-methylpyrazol-4-yl)benzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-4-fluorobenzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]benzoic acidIC5020000.0 [1]
3-[(1-Acetylindole-3-carbonyl)amino]-5-(oxan-2-yloxymethyl)benzoic acidIC5020000.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Bromodomain-containing protein 9 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/bromodomain-containing-protein-9-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, November 21). Quest Database™ Bromodomain-containing protein 9 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bromodomain-containing-protein-9-inhibitors-ic50-ki.
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