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Breast cancer type 1 susceptibility protein Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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[(2S)-2-Acetamido-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC504600.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateKi1850.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC503200.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateKi1960.0 [1]
(2S)-2-[[(2S,3R)-2-[[(2S)-1-[(2S)-2-Acetamido-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]-3-hydroxybutanoyl]amino]-3-phenylpropanoic acidIC501000.0 [1]
(2S)-2-[[(2S,3R)-2-[[(2S)-1-[(2S)-2-Acetamido-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]-3-hydroxybutanoyl]amino]-3-phenylpropanoic acidKi270.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Acetamido-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoic acidIC501600.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-Acetamido-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoic acidKi200.0 [1]
3-(4-Methylpiperidin-1-yl)-10,10-dioxothioxanthen-9-oneKi39000.0 [1]
1-(9,10,10-Trioxothioxanthen-3-yl)piperidine-4-carboxamideKi30000.0 [1]
3-(4-Benzylpiperidin-1-yl)-10,10-dioxothioxanthen-9-oneKi38000.0 [1]
[(2S)-2-Amino-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC5010800.0 [1]
2-[(2S)-2-Acetamido-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl]propanedioic acidIC5052800.0 [1]
[(2R,3S)-3-Acetamido-4-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-4-oxobutan-2-yl] dihydrogen phosphateIC50250000.0 [1]
[(2S)-2-Acetamido-3-[[(2S)-1-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-oxopropyl] dihydrogen phosphateIC5015000.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC5035000.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxopropan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC5030100.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S,3S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC507100.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-4-methyl-1-oxopentan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC5018400.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-3-(4-hydroxyphenyl)-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC5014900.0 [1]
[(2S)-2-Acetamido-3-[[(2S)-1-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxopropan-2-yl]amino]-3-oxopropyl] dihydrogen phosphateIC5098400.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[(2S)-2-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]carbamoyl]pyrrolidine-1-carbonyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC50250000.0 [1]
[(2R)-2-[[(2R)-2-[[(2R,3S)-2-[[(2R)-2-Acetamido-3-phenylpropanoyl]amino]-3-hydroxybutanoyl]amino]propanoyl]amino]-3-amino-3-oxopropyl] dihydrogen phosphateIC50250000.0 [1]
(4S)-4-Acetamido-5-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-5-oxopentanoic acidIC50250000.0 [1]
(2S)-2-[[(2S)-3-Methyl-2-[[(2S)-1-[(2S)-2-(3-phenylpropanoylamino)-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]butanoyl]amino]-3-phenylpropanoic acidKi100.0 [1]
[(2S)-2-[[(2S)-2-Acetamido-3-naphthalen-2-ylpropanoyl]amino]-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateKi1240.0 [1]
(2S)-2-[[(2S)-3-Methyl-2-[[(2S)-1-[(2S)-2-(5-phenylpentanoylamino)-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]butanoyl]amino]-3-phenylpropanoic acidKi12050.0 [1]
(2S)-2-[[(2S)-3-Methyl-2-[[(2S)-1-[(2S)-2-[(2-naphthalen-1-ylacetyl)amino]-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]butanoyl]amino]-3-phenylpropanoic acidKi15670.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[3-(3,4-Dimethoxyphenyl)propanoylamino]-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoic acidKi4040.0 [1]
(2S)-2-[[(2S)-3-Methyl-2-[[(2S)-1-[(2S)-2-[(3-phenylbenzoyl)amino]-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]butanoyl]amino]-3-phenylpropanoic acidKi80.0 [1]
[(2S)-2-[[(2R)-2-Acetamido-3-naphthalen-2-ylpropanoyl]amino]-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateKi19440.0 [1]
[(2S)-2-[[(2S)-2-Acetamido-3-naphthalen-2-ylpropanoyl]amino]-3-[(2S)-2-[[(2S)-1-[[(2S)-1-amino-1-oxo-3-phenylpropan-2-yl]amino]-3-methyl-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateKi540.0 [1]
(2S)-2-[[(2S)-3-Methyl-2-[[(2S)-1-[(2S)-2-(4-phenylbutanoylamino)-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]butanoyl]amino]-3-phenylpropanoic acidKi500.0 [1]
(2S)-2-[[(2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-Acetamido-3-naphthalen-2-ylpropanoyl]amino]-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]-3-methylbutanoyl]amino]-3-phenylpropanoic acidKi130.0 [1]
(2S)-2-[[(2S)-3-Methyl-2-[[(2S)-1-[(2S)-2-[[(E)-4-phenylbut-3-enoyl]amino]-3-phosphonooxypropanoyl]pyrrolidine-2-carbonyl]amino]butanoyl]amino]-3-phenylpropanoic acidKi40.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-3-naphthalen-1-yl-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC50171700.0 [1]
[(2S)-2-Acetamido-3-[(2S)-2-[[(2S,3R)-1-[[(2S)-1-amino-3-naphthalen-2-yl-1-oxopropan-2-yl]amino]-3-hydroxy-1-oxobutan-2-yl]carbamoyl]pyrrolidin-1-yl]-3-oxopropyl] dihydrogen phosphateIC5017700.0 [1]
Items per page: 1 - 10 of 37
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References

This online tool may be cited as follows

MLA

"Quest Database™ Breast cancer type 1 susceptibility protein Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Dec. 2024, https://www.aatbio.com/data-sets/breast-cancer-type-1-susceptibility-protein-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2024, December 21). Quest Database™ Breast cancer type 1 susceptibility protein Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/breast-cancer-type-1-susceptibility-protein-inhibitors-ic50-ki.
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