Brain glycogen phosphorylase Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	D-Glucose	Ki	1700000.0 [1], 7400000.0 [2], 125893000000.0 [3]
	N-[(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide	Ki	32000.0 [1], 31622800000000.0 [2]
	N-[(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl]benzamide	Ki	81000.0 [1], 12589300000000.0 [2]
	(5S,8S,9S)-8,9,10-Trihydroxy-7-(hydroxymethyl)-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione	Ki	3100.0 [1], 12800.0 [2], 16500.0 [3], 26000.0 [4]
	Urea, alpha-D-glucopyranosyl-	Ki	140000.0 [1], 7943280000000.0 [2]
	2-Chloro-N-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide	Ki	45000.0 [1], 25118900000000.0 [2]
	1-Deoxy-1-methoxycarbamido-beta-D-gluco-2-heptulopyranosonamide	Ki	16000.0 [1], 3162280000000.0 [2], 63095700000000.0 [3]
	N-[(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl]butanamide	Ki	94000.0 [1], 10000000000000.0 [2]
	N-[(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl]propanamide	Ki	39000.0 [1], 25118900000000.0 [2]
	2-[(2R,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide	Ki	21100000.0 [1], 50118723363.0 [2]
	2-Acetamido-N-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide	Ki	990000.0 [1], 1000000000000.0 [2]
	N-Phenyl-2-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide	Ki	3600000.0 [1], 251189000000.0 [2]
	(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)-N'-methyloxane-2-carbohydrazide	Ki	1800000.0 [1], 501187000000.0 [2]
	N-(2,4-Difluorophenyl)-2-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]sulfanylacetamide	Ki	18900000.0 [1], 50118723363.0 [2]
	alpha-D-Glucopyranose, 5-thio-	Ki	2000000.0 [1], 501187000000.0 [2]
	8,9,10-Trihydroxy-7-hydroxymethyl-2-thioxo-6-oxa-1,3-diaza-spiro[4.5]decan-4-one	Ki	5100.0 [1], 7000.0 [2]
	3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid hydrazide	Ki	3000000.0 [1], 2511890000000.0 [2]
	(5S,7S,8S,9S,10S)-8,9,10-Trihydroxy-7-(hydroxymethyl)-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione	Ki	3000.0 [1], 316228000000000.0 [2]
	(5S,7S,8S,9S,10S)-3-Amino-8,9,10-trihydroxy-7-(hydroxymethyl)-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione	Ki	146000.0 [1], 6309570000000000.0 [2]
	(3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetonitrile	Ki	9000000.0 [1], 100000000000.0 [2]
	(6S,8S,9S,10S,11S)-9,10,11-Trihydroxy-8-(hydroxymethyl)-7-oxa-1,4-diazaspiro[5.5]undecane-2,5-dione	Ki	59700.0 [1], 15848900000000.0 [2]
	(2S,3R,4R,5S,6R)-2-(Azidomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol	Ki	15200000.0 [1], 63095734448.0 [2]
	Benzyl N-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]carbamate	Ki	350000.0 [1], 3162280000000.0 [2]
	(2R,3R,4R,5S,6R)-2-(Azidomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol	Ki	22400000.0 [1], 39810717055.0 [2]
	2-[(2S,3R,4S,5S,6R)-2,3,4,5-Tetrahydroxy-6-(hydroxymethyl)oxan-2-yl]acetonitrile	Ki	7600000.0 [1], 125893000000.0 [2]
	1-Deoxy-1-methoxycarbamido-beta-D-glucopyranose	Ki	11749000000000.0 [1], 12589300000000.0 [2]
	(5S,7S,8S,9S,10S)-3,8,9,10-Tetrahydroxy-7-(hydroxymethyl)-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione	Ki	25118900000000.0 [1], 25704000000000.0 [2]
	N-[(5S,7S,8S,9S,10S)-8,9,10-Trihydroxy-7-(hydroxymethyl)-2,4-dioxo-6-oxa-1,3-diazaspiro[4.5]decan-3-yl]acetamide	Ki	1819700000000.0 [1], 1995260000000.0 [2]
	(2R,3S,4S,5R,6S)-2-(Hydroxymethyl)-6-(1H-indol-2-yloxy)oxane-3,4,5-triol	Ki	2600000.0 [1], 398107000000.0 [2]
	alpha-D-Gluco-2-Heptulopyranose	Ki	15800000.0 [1], 63095734448.0 [2]
	Methyl alpha-D-glucopyranoside	Ki	79432823472.0 [1]
	Methyl beta-D-glucopyranoside	Ki	39810717055.0 [1]
	1-Thio-beta-D-glucopyranose	Ki	1000000000000.0 [1]
	3,4,5-Trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide	Ki	370000.0 [1]
	2-Aminomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol	Ki	34500000.0 [1]
	2-Amino-N-[(2S,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide	Ki	370000.0 [1]
	3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methyl ester	Ki	24200000.0 [1]
	2-Hydroxymethyl-6-mercapto-tetrahydro-pyran-3,4,5-triol	Ki	1000000.0 [1]
	Methanesulfonic acid 3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-ylmethyl ester	Ki	4800000.0 [1]
	N-Methyl-6-(hydroxymethyl)-3,4,5-trihydroxy-tetrahydro-2H-pyran-2-carboxamide	Ki	160000.0 [1]
	2,6-Bis-hydroxymethyl-tetrahydro-pyran-3,4,5-triol	Ki	1500000.0 [1]
	2-Bromo-N-[(2S,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide	Ki	44000.0 [1]
	3,4,5-Trihydroxy-6-(hydroxymethyl)-N-phenyloxane-2-carboxamide	Ki	5400000.0 [1]
	(2R,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide	Ki	2511890000000.0 [1]
	(2R,3S,4S,5S,6S)-2-(Azidomethyl)-6-(hydroxymethyl)oxane-2,3,4,5-tetrol	Ki	7400000.0 [1]
	(2S,3S,4S,5S,6S)-N-Cyclopropyl-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide	Ki	1300000.0 [1]
	(2S,3S,4S,5S,6S)-3,4,5-Trihydroxy-N-(2-hydroxyethyl)-6-(hydroxymethyl)oxane-2-carboxamide	Ki	2600000.0 [1]
	3,4,5-Trihydroxy-6-(hydroxymethyl)-N-(4-hydroxyphenyl)oxane-2-carboxamide	Ki	4400000.0 [1]
	2-(2-Aminoethyl)-6-(hydroxymethyl)oxane-3,4,5-triol	Ki	4500000.0 [1]
	alpha-D-Glucopyranosyl-2-carboxylic acid amide	Ki	2511890000000.0 [1]
	N-Bromoacetylglucopyranosylamine	Ki	25118900000000.0 [1]
	[(2S,3S,4S,5S,6S)-2,3,4,5-Tetrahydroxy-6-(hydroxymethyl)oxan-2-yl]methyl methanesulfonate	Ki	3700000.0 [1]
	(2S,3S,4S,5S,6S)-2,6-Bis(hydroxymethyl)oxane-2,3,4,5-tetrol	Ki	15800000.0 [1]
	(2S,3S,4S,5S,6S)-3,4,5-Trihydroxy-6-(hydroxymethyl)-N-(2,2,2-trifluoroethyl)oxane-2-carboxamide	Ki	8100000.0 [1]
	N-Benzyloxycarbonyl-glycyl-glycyl-hydroxamsaeure	Ki	4.0 [1]
	(2R,3R,4S,5S,6R)-2-(2-Hydroxyethoxy)-6-(hydroxymethyl)oxane-3,4,5-triol	Ki	39810717055.0 [1]
	(2S)-2-[[(2S)-2-(Phosphonoamino)propanoyl]amino]propanoic acid	Ki	4.0 [1]
	(2R,3S,4S,5R,6R)-2-(Hydroxymethyl)-6-[2-(hydroxymethyl)phenoxy]oxane-3,4,5-triol	Ki	125893000000.0 [1]
	(2S)-2-[Acetyl(hydroxy)amino]-N-[(2S)-1-[(2-amino-2-oxoethyl)amino]-1-oxopropan-2-yl]-4-methylpentanamide	Ki	4.0 [1]
	(2S)-N-[(2S)-1-[(2-Amino-2-oxoethyl)amino]-1-oxopropan-2-yl]-N'-hydroxy-2-methylpropanediamide	Ki	4.0 [1]
	Z-Gly-leu-NH2	Ki	4.0 [1]
	(2S,3R,4S,5S,6R)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxane-2-carbohydrazide	Ki	316228000000.0 [1]
	(2S,3R,4S,5S,6R)-N-[(2,4-Difluorophenyl)methyl]-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide	Ki	39810717055.0 [1]
	(2S,3R,4R,5S,6R)-2-(Aminomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol	Ki	63095734448.0 [1]
	2,2,2-Trifluoro-N-[(2R,3S,4S,5S,6S)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide	Ki	710000.0 [1]
	alpha-Isomaltose	Ki	63095734448.0 [1]
	(R)-2-Hydroxymethyl-6-methoxy-tetrahydro-pyran-3,4,5-triol	Ki	24700000.0 [1]
	Methyl (2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxylate	Ki	39810717055.0 [1]
	2-Deoxy-2-fluoro-alpha-d-glucopyranosyl fluoride	Ki	5011870000000.0 [1]
	(5R,8R,9S)-8,9,10-Trihydroxy-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione	Ki	10000000.0 [1]
	(5S,8R,9S)-8,9,10-Trihydroxy-2-sulfanylidene-6-oxa-1,3-diazaspiro[4.5]decan-4-one	Ki	10000000.0 [1]
	(5S,8R,9S)-8,9,10-Trihydroxy-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione	Ki	11500000.0 [1]
	3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid amide	Ki	440000.0 [1]
	(5R,8S,9S)-8,9,10-Trihydroxy-7-(hydroxymethyl)-6-oxa-1,3-diazaspiro[4.5]decane-2,4-dione	Ki	320000.0 [1]
	(2S,4S,5S)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide	Ki	370000.0 [1]
	6-Hydroxymethyl-tetrahydro-pyran-2,3,4,5-tetraol	Ki	1700000.0 [1]
	2,3,4,5-Tetrahydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid amide	Ki	3100000.0 [1]
	Methyl N-[(2S)-2-carbamoyl-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]carbamate	Ki	16000.0 [1]
	(2R)-3,4,5-Trihydroxy-6-(hydroxymethyl)-N-methyloxane-2-carboxamide	Ki	160000.0 [1]
	(R)-2-Hydroxymethyl-6-methyl-tetrahydro-pyran-3,4,5-triol	Ki	53100000.0 [1]
	Benzyl N-[(2R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]carbamate	Ki	350000.0 [1]
	(2S)-2-(2-Aminoethyl)-6-(hydroxymethyl)oxane-3,4,5-triol	Ki	4500000.0 [1]
	((S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetonitrile	Ki	9000000.0 [1]
	(2R)-3,4,5-Trihydroxy-6-(hydroxymethyl)-N-(4-hydroxyphenyl)oxane-2-carboxamide	Ki	4400000.0 [1]
	(2S)-3,4,5-Trihydroxy-6-(hydroxymethyl)-N-methyloxane-2-carboxamide	Ki	36700000.0 [1]
	(2R)-2-(Aminomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol	Ki	34500000.0 [1]
	((S)-2,3,4,5-Tetrahydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetonitrile	Ki	7600000.0 [1]
	(S)-2-Azidomethyl-6-hydroxymethyl-tetrahydro-pyran-2,3,4,5-tetraol	Ki	7400000.0 [1]
	(2S)-3,4,5-Trihydroxy-N-(2-hydroxyethyl)-6-(hydroxymethyl)oxane-2-carboxamide	Ki	16900000.0 [1]
	(2S)-2-(Aminomethyl)-6-(hydroxymethyl)oxane-3,4,5-triol	Ki	16800000.0 [1]
	(2S)-3,4,5-Trihydroxy-6-(hydroxymethyl)oxane-2-carboxylic acid	Ki	15200000.0 [1]
	(S)-3,4,5-Trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-carboxylic acid methyl ester	Ki	24200000.0 [1]
	2-Bromo-N-[(2R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]acetamide	Ki	44000.0 [1]
	(R)-2-Azidomethyl-6-hydroxymethyl-tetrahydro-pyran-3,4,5-triol	Ki	22400000.0 [1]
	(S)-2-Hydroxymethyl-6-mercapto-tetrahydro-pyran-3,4,5-triol	Ki	1000000.0 [1]
	(2S)-3,4,5-Trihydroxy-6-(hydroxymethyl)-N-(4-hydroxyphenyl)oxane-2-carboxamide	Ki	5600000.0 [1]
	(2R)-3,4,5-Trihydroxy-6-(hydroxymethyl)-N-phenyloxane-2-carboxamide	Ki	5400000.0 [1]
	(R)-2,6-Bis-hydroxymethyl-tetrahydro-pyran-3,4,5-triol	Ki	1500000.0 [1]
	(2S)-N-[(2,4-Difluorophenyl)methyl]-3,4,5-trihydroxy-6-(hydroxymethyl)oxane-2-carboxamide	Ki	27200000.0 [1]
	(2R)-3,4,5-Trihydroxy-6-(hydroxymethyl)-N-(2,2,2-trifluoroethyl)oxane-2-carboxamide	Ki	8100000.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 100 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Brain glycogen phosphorylase Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 22 Feb. 2025, https://www.aatbio.com/data-sets/brain-glycogen-phosphorylase-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2025, February 22). Quest Database™ Brain glycogen phosphorylase Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/brain-glycogen-phosphorylase-inhibitors-ic50-ki.
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