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Bone morphogenetic protein receptor type-1A Inhibitors (IC50, Ki)

Structure
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Compound Name
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Standard Type
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Standard Values (in nM)
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4-(6-(4-(Piperazin-1-yl)phenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinolineIC502.15 [1], 5.0 [2], 19.0 [3]
StaurosporineIC504288.0 [1]
DorsomorphinIC5095.0 [1]
VactosertibIC5010000.0 [1]
5-[6-[4-(1-Piperazinyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinolineIC50539.0 [1]
1-(4-(6-Methyl-5-(3,4,5-trimethoxyphenyl)pyridin-3-yl)phenyl)piperazineIC501171.0 [1]
5-[6-(4-Methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineIC5010800.0 [1]
4-[6-(4-Propan-2-yloxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]quinolineIC505.0 [1]
4-(6-(4-Methoxyphenyl)pyrazolo[1,5-a]pyrimidin-3-yl)quinolineIC506.78 [1]
5-(2-Amino-[1,2,4]triazolo[1,5-a]pyridin-7-yl)-N-tert-butylpyridine-3-sulfonamideIC5010000.0 [1]
CID 60182364IC505.0 [1]
CID 60182389IC505.0 [1]
4-(4-(3-(1H-Pyrazol-4-yl)pyrazolo[1,5-a]pyrimidin-6-yl)phenyl)morpholineIC5010.4 [1]
6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-oneIC5010000.0 [1]
4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]quinolineIC507.0 [1]
3-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]benzenesulfonamideIC502534.0 [1]
4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-2-methylbenzenesulfonamideIC5016550.0 [1]
2-Amino-4-[6-[4-[(2R,6S)-2,6-dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]benzenesulfonamideIC5010000.0 [1]
4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC503466.0 [1]
4-[6-[4-(2-Piperidin-1-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-N,N-dimethylnaphthalene-1-sulfonamideIC5064750.0 [1]
4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]-N-methylnaphthalene-1-sulfonamideIC5010000.0 [1]
4-[6-[4-(2-Methyl-1-piperidin-1-ylpropan-2-yl)oxyphenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]-3-(4-methylsulfonylphenyl)pyrazolo[1,5-a]pyrimidineIC5010000.0 [1]
4-[6-(6-Piperazin-1-ylpyridin-3-yl)pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
4-[6-[4-(2-Aminopropan-2-yl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
4-[6-[6-(2-Piperidin-1-ylethoxy)pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
N-[4-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalen-1-yl]methanesulfonamideIC508897.0 [1]
4-[6-[4-(Pyrrolidin-1-ylmethyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
4-[6-[4-(2-Pyrrolidin-1-ylethoxy)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
4-[6-[4-(1-Aminocyclobutyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC508195.0 [1]
4-[6-[6-[2-(Dimethylamino)ethoxy]pyridin-3-yl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
5-[6-[4-[(2S,6R)-2,6-Dimethylpiperazin-1-yl]phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC50444.0 [1]
4-[6-(4-Piperidin-4-ylphenyl)pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5010000.0 [1]
4-[6-[4-(1-Aminoethyl)phenyl]pyrazolo[1,5-a]pyrimidin-3-yl]naphthalene-1-sulfonamideIC5012830.0 [1]
(4S,9S,10S)-9,10,18-Trihydroxy-16-methoxy-4-methyl-3-oxabicyclo[12.4.0]octadeca-1(14),15,17-triene-2,8-dioneIC506267.0 [1]
Alk2-IN-2IC506439.0 [1]
6-(4-Methoxyphenyl)-3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidineIC5041.0 [1]
4-[[(3S,4R)-1-(5-Cyanopyridin-2-yl)-3-fluoropiperidin-4-yl]amino]-1H-pyrrolo[2,3-b]pyridine-5-carboxamideIC501000.0 [1]
6-(4-Piperazin-1-ylphenyl)-3-(1H-pyrazol-4-yl)pyrazolo[1,5-a]pyrimidineIC5055.0 [1]
N-[4-[(6-Chloro-[1,3]dioxolo[4,5-B]pyridin-7-Yl)amino]-2-Pyridyl]cyclopropanecarboxamideIC502.4 [1]
Items per page: 1 - 10 of 41
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References

This online tool may be cited as follows

MLA

"Quest Database™ Bone morphogenetic protein receptor type-1A Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 20 Feb. 2025, https://www.aatbio.com/data-sets/bone-morphogenetic-protein-receptor-type-1a-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 20). Quest Database™ Bone morphogenetic protein receptor type-1A Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/bone-morphogenetic-protein-receptor-type-1a-inhibitors-ic50-ki.
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