![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_beb7f72e73f61c5a9e1bf58b6572d39a.svg) | Cyclosporin A | IC50 | 400.0 [1], 500.0 [2], 900.0 [3], 10000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_beb7f72e73f61c5a9e1bf58b6572d39a.svg) | Cyclosporin A | Ki | 9500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_7678391665350c8597f29638df219c3b.svg) | Glyburide | IC50 | 1500.0 [1], 5000.0 [2], 5300.0 [3], 6100.0 [4], 10000.0 [5] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_7678391665350c8597f29638df219c3b.svg) | Glyburide | Ki | 27500.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_e386e75fd7c80f00255fc04b52e51041.svg) | Flutamide | IC50 | 75000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_a7e11d7bcee94c9af8c42c557a082c25.svg) | Chlorpromazine | IC50 | 90970.0 [1], 133000.0 [2], 135000.0 [3], 147600.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_a69f1db31ed30d6a63db389cb16202f2.svg) | Ketoconazole | IC50 | 2900.0 [1], 3400.0 [2], 4100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_fef79222ea6630efa6d072c722a2f0c2.svg) | Troglitazone | IC50 | 2700.0 [1], 3000.0 [2], 5900.0 [3], 6900.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_71acea9a6dfc0e4dac7865946b73384c.svg) | Paclitaxel | IC50 | 15000.0 [1], 24400.0 [2], 26800.0 [3], 28900.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_f28ce47318433f5c984060ce11c4a797.svg) | Tamoxifen | IC50 | 10000.0 [1], 15400.0 [2], 23300.0 [3], 133000.0 [4], 135000.0 [5] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_eeff5a96588de62beccbf378609f1809.svg) | Furosemide | IC50 | 133000.0 [1], 135000.0 [2], 964800.0 [3], 1000000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_75de8bb67a0e2555d13e845be859468c.svg) | Rosiglitazone | IC50 | 2800.0 [1], 3750.0 [2], 4400.0 [3], 6362.0 [4], 6400.0 [5] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_bb59a4ec4c1de9921ef616765123dce2.svg) | Flumazenil | IC50 | 100000.0 [1], 133000.0 [2], 135000.0 [3], 733500.0 [4], 1000000.0 [5] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_2abc8a1f0ee77ee021577efb9cbf0b7a.svg) | Pioglitazone | IC50 | 262.1 [1], 300.0 [2], 400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_575acb7546adcaf4c25ef5e411968354.svg) | Bosentan | IC50 | 22000.0 [1], 23000.0 [2], 25300.0 [3], 29000.0 [4], 38100.0 [5] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_65b961c9d10d3a8cf619bd052d84c672.svg) | Nefazodone | IC50 | 4200.0 [1], 6100.0 [2], 6110.0 [3], 7000.0 [4], 10000.0 [5] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_cddbf6b3255ab7e6c7ab2f39633ddb3f.svg) | Rifamycin | IC50 | 6300.0 [1], 9500.0 [2], 12200.0 [3], 206500.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_cddbf6b3255ab7e6c7ab2f39633ddb3f.svg) | Rifamycin | Ki | 31000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_651f4cfbe9aa97adaf2f12469bdbaf84.svg) | Sodium | IC50 | 10000.0 [1], 133000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_84be4cdb308fb643cf288980a1c24c41.svg) | Progesterone | IC50 | 10000.0 [1], 17300.0 [2], 224600.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_1d64f7b51ed811e6ea11101a6c1d74e3.svg) | Dexamethasone | IC50 | 101700.0 [1], 133000.0 [2], 135000.0 [3], 137400.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_1cc257bab28d3e85f276bcae9f111347.svg) | Methotrexate | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_c70f5b79af37726016ec15cea0b55e94.svg) | Propranolol | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_2417c7be24e5d7debb18533147580339.svg) | Acetaminophen | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_0cca37e8532dc6f7bb6fa13f5708ab01.svg) | Isoniazid | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_01814a6086009d7440d5f435a324c600.svg) | Verapamil | IC50 | 79100.0 [1], 133000.0 [2], 135000.0 [3], 178900.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_b2d54f313fd6fae3559ad99a1d264705.svg) | Imatinib | IC50 | 10000.0 [1], 25100.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_93ff81dbb74065f6358ff2946a8ae8ed.svg) | Rifampicin | IC50 | 11300.0 [1], 18700.0 [2], 25300.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_1232c84d43d4865ebdc5de8d7663a19f.svg) | Nifedipine | IC50 | 18650.0 [1], 30700.0 [2], 64000.0 [3], 69000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_8eea222a1bcb2e74405ba02fe4c3db74.svg) | Reserpine | IC50 | 8350.0 [1], 8400.0 [2], 10000.0 [3], 10200.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_347b1b64f072d35207a2dcbef37b1046.svg) | Azathioprine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_8159b09a6bebd9e5751360e57f770ab8.svg) | Clozapine | IC50 | 75140.0 [1], 126100.0 [2], 133000.0 [3], 135000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_b03a82411601ac2483b9406eae5a6277.svg) | Simvastatin | IC50 | 10000.0 [1], 24700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_2eb69008645ff5a1555c94aa65edac97.svg) | Acyclovir | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_a52107dd1a21bc400717c7e02e2e0f04.svg) | Tolbutamide | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_9f0a93e7b9951df86a7799cacbfb6848.svg) | Dapsone | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_f2beac4f632265172541ae8f16f89706.svg) | Nicardipine | IC50 | 7870.0 [1], 7900.0 [2], 10000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_922e591df45814020ba0e2ba5eca1f5b.svg) | Tacrine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_c71bb870afd3132ff8414544fb890815.svg) | Chlorpropamide | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_6c4785b8db910babcddc2fdbba6d440e.svg) | Iproniazid | IC50 | 133000.0 [1], 135000.0 [2], 952600.0 [3], 1000000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_ba6229a8df4deed4ea9c20524a02ee80.svg) | Glimepiride | IC50 | 10000.0 [1], 15700.0 [2], 34000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_07ef2b6946f6c72e3282969244c05e27.svg) | Clofazimine | IC50 | 12900.0 [1], 28700.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_051772800ae57850275d4fa2a21f5489.svg) | Sulindac | IC50 | 63690.0 [1], 133000.0 [2], 135000.0 [3], 226000.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_e92b9426ec3ed0b62b36d44608851ece.svg) | Dicloxacillin | IC50 | 10000.0 [1], 45000.0 [2], 56400.0 [3], 69700.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_4144082d3c34f90f55de601b70b12855.svg) | Tolcapone | IC50 | 33920.0 [1], 34500.0 [2], 36600.0 [3], 119600.0 [4] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_eb212ff63ed7fef055dc658629968c96.svg) | 5-Fluorouracil | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_cd9b5820bcad56865f8364f10caaf311.svg) | Prednisolone | IC50 | 91470.0 [1], 133000.0 [2], 135000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_bec8eaadb51e755de26c3660866564ee.svg) | Caffeine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_ef61fa49423965b00cafb173f3e07a26.svg) | Indomethacin | IC50 | 42000.0 [1], 49320.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_038301bf66445c6984ca669e09912730.svg) | Methylprednisolone | IC50 | 33030.0 [1], 133000.0 [2], 135000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_be4971788168689ef3407413c05b03d8.svg) | Chloramphenicol | IC50 | 133000.0 [1], 135000.0 [2], 957900.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_86630ba4a7e4889b44175ac812cce53f.svg) | Nicotine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_15976e9843386a991246a922e8b855ad.svg) | Ciprofloxacin | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_393a6636008719cf0eb93219e05af350.svg) | Metformin | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_db4ac60c18b24b7bd003d4edf05f0d21.svg) | Naloxone | IC50 | 133000.0 [1], 135000.0 [2], 549000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_2d46cd64b612bada34966bcfba251b25.svg) | Carbamazepine | IC50 | 133000.0 [1], 1000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_7ce5c90b273b41810bee3170ac9401d3.svg) | Haloperidol | IC50 | 22760.0 [1], 133000.0 [2], 135000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_5498b28ac748aa1a1c2a1db363e8d2d0.svg) | Amoxicillin | IC50 | 133000.0 [1], 1000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_693b10fcf0f1bf3ce26f73cb27aee812.svg) | Fluoxetine | IC50 | 133000.0 [1], 135000.0 [2], 143800.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_94fca8d3b15a98bf35a0a3961e7494ec.svg) | Midazolam | IC50 | 41700.0 [1], 41740.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_48f03bbeea35e7522fbad39cfe44c9eb.svg) | Ibuprofen | IC50 | 135000.0 [1], 598600.0 [2], 789000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_2f6aa077265088f9306897fbb768392e.svg) | Salbutamol | IC50 | 133000.0 [1], 1000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_7e646fe532894c3595457245499402ac.svg) | Colchicine | IC50 | 133000.0 [1], 135000.0 [2], 298700.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_be4565ca8c20c1d9804fa640fd1584d5.svg) | Risperidone | IC50 | 10250.0 [1], 133000.0 [2], 135000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_81af8877c0a8c32165f86d729092ee41.svg) | Amiodarone | IC50 | 10000.0 [1], 25000.0 [2], 43000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_3e94330ba1527a829fecddbee5acde55.svg) | Apomorphine | IC50 | 133000.0 [1], 135000.0 [2], 211500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_ebac36f7213da3162d29205ab4152aca.svg) | Prazosin | IC50 | 133000.0 [1], 135000.0 [2], 171800.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_3fb59b292039fb68c21d347565286601.svg) | Quinine | IC50 | 98830.0 [1], 133000.0 [2], 135000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_35003ced678586a25de172e3d06d122a.svg) | Cimetidine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_3bd5dcd12d2ef57fd5cbefabf7849aa3.svg) | Gefitinib | IC50 | 10900.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_c8494007663098abb5d227cb27cc738b.svg) | Sorafenib | IC50 | 8000.0 [1], 10000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_3f59bab9b954f7e2737294dc8b7f1b51.svg) | Trimethoprim | IC50 | 133000.0 [1], 135000.0 [2], 833100.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_9eea3482ccbd85339d3c08d99095be33.svg) | Ritonavir | IC50 | 1740.0 [1], 2200.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_74e5f3770fba46d28349ec72450a0138.svg) | Levofloxacin | IC50 | 133000.0 [1], 1000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_3eb3a5b1dcd4c8d28eded74657153a42.svg) | Naproxen | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_a34616d3de075a93790bddad07a71c2d.svg) | Sulfamethoxazole | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_5e0cec3bd7dc255f04fcd00c5dba41c3.svg) | Nevirapine | IC50 | 133000.0 [1], 135000.0 [2], 294600.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_0aa07f27faeb9f6a511108b5adb9f577.svg) | Busulfan | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_a14f1dfe550f843a4d18cc55574220bb.svg) | Praziquantel | IC50 | 60270.0 [1], 67100.0 [2], 96800.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_c70118dba6fb13f8f3e2091ee27ddd79.svg) | Trimethyl glycine | IC50 | 1000000.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_a421ce3b176dfb4b05941f1c1476b9e3.svg) | Papaverine | IC50 | 10000.0 [1], 133000.0 [2], 135000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_b2f3218cdbd5f04949eaaf044a21d56f.svg) | Desipramine | IC50 | 133000.0 [1], 135000.0 [2], 150400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_b57a4c933cfa9b7d739e976f2180d4a0.svg) | Antipyrine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_83a1f5cdeed2a8c8b0248d33d27539f1.svg) | Carmustine | IC50 | 97210.0 [1], 133000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_48a4213adc65d3ea6cd72259c7aa7e02.svg) | Venlafaxine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_2a26b13bc4676a12b69e95c9aa8b738a.svg) | Fenofibrate | IC50 | 15300.0 [1], 41000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_2393a08407e73e5fc381a2b27c1e0625.svg) | Donepezil | IC50 | 78000.0 [1], 145600.0 [2], 205700.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_22ba1cf70b75274f542c287569ff1448.svg) | Neostigmine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_f8b479996e8e0acb73005bd3a3bf5a1b.svg) | Rofecoxib | IC50 | 95360.0 [1], 133000.0 [2], 135000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_4e0841d9168e98e6e1a9831cb8b4f704.svg) | Methimazole | IC50 | 133000.0 [1], 1000000.0 [2] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_fcf0bc9f27e280b269d420fa8a3dc69d.svg) | Sulfadiazine | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_3b2da37f0b0ee76d72c81525a0edc58c.svg) | Clomipramine | IC50 | 37400.0 [1], 133000.0 [2], 135000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_855cc535c493e26b0a86aed64af61585.svg) | Diazoxide | IC50 | 133000.0 [1], 135000.0 [2], 1000000.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_2dbbe179cee38c655ac88c7d09ddeb01.svg) | Finasteride | IC50 | 28200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_c9960c7f038fe75af1672de453506a31.svg) | Indinavir | IC50 | 21200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_ad6ccf602ee43f3992fdd4c89edf213b.svg) | Probenecid | IC50 | 133000.0 [1], 564800.0 [2], 586800.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_5e73a1ef8d0e8c863280cb26b68ae8b5.svg) | Telmisartan | IC50 | 16200.0 [1] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_91ef444c9cb25042f17ad02e275ab775.svg) | Leflunomide | IC50 | 110000.0 [1], 133000.0 [2], 177400.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_47eddd337dafa05fe9d237d27dca82c1.svg) | Buspirone | IC50 | 59630.0 [1], 100000.0 [2], 104500.0 [3] |
![](https://images.aatbio.com/dataset/ic50/bile-salt-export-pump_755000a88f2651809d912de0f446bcfe.svg) | Lapatinib | IC50 | 6500.0 [1], 10000.0 [2] |