| gamma-Aminobutyric acid | IC50 | 9000.0 [1], 25000.0 [2], 36000.0 [3], 39000.0 [4], 181000.0 [5] |
| (S)-Snap 5114 | IC50 | 71700.0 [1], 140000.0 [2], 141253.75 [3] |
| N-(1-Benzylpiperidin-4-yl)-2,4-dichlorobenzamide | IC50 | 2000.0 [1], 13489.63 [2], 58000.0 [3], 1000000.0 [4] |
| 1-[3-(9H-Carbazol-9-yl)propyl]-4-(2-methoxyphenyl)piperidin-4-ol | IC50 | 5100.0 [1] |
| N-(1-Benzylpiperidin-4-yl)-2,6-dichloropyridine-3-carboxamide | IC50 | 44000.0 [1], 1000000.0 [2] |
| Tiagabine | IC50 | 1670000.0 [1] |
| Nipecotic acid | IC50 | 2370000.0 [1] |
| N-(4,4-Diphenyl-3-butenyl)nipecotic acid | IC50 | 7210000.0 [1] |
| Guvacine | IC50 | 1870000.0 [1] |
| 1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid | IC50 | 208000.0 [1] |
| (R)-Piperidine-3-carboxylic acid | IC50 | 2310000.0 [1] |
| CI-966 Free base | IC50 | 300000.0 [1] |
| (S)-Piperidine-3-carboxylic acid | IC50 | 6410000.0 [1] |
| N-(1-Benzylpiperidin-4-yl)benzamide | IC50 | 290000.0 [1] |
| 1-(3-(9H-Carbazol-9-yl)propyl)-4-(4-methoxyphenyl)piperidin-4-ol | Ki | 1600.0 [1] |
| 2-Ethoxy-N-[1-(phenylmethyl)-4-piperidinyl]benzamide | IC50 | 180000.0 [1] |
| 1-{2-[9-(4-Methoxy-phenyl)-9H-fluoren-9-yloxy]-ethyl}-piperidine-3-carboxylic acid | IC50 | 27000.0 [1] |
| N-(1-Benzylpiperidin-4-yl)-2,3-dimethoxybenzamide | IC50 | 91000.0 [1] |
| N-(1-Benzylpiperidine-4-yl)-2-naphthamide | Ki | 15000.0 [1] |
| 1-(4,4-Diphenyl-but-3-enyl)-piperidine-3-carboxylic acid | IC50 | 7210000.0 [1] |
| N-(1-Benzylpiperidin-4-yl)-4-fluorobenzamide | IC50 | 100000.0 [1] |
| 1-[2-[[4-Methoxy-3-(trifluoromethyl)phenyl]-phenyl-[3-(trifluoromethyl)phenyl]methoxy]ethyl]piperidine-3-carboxylic acid | IC50 | 201000.0 [1] |
| 1-{2-[Tris-(4-fluoro-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid | IC50 | 1270000.0 [1] |
| 1-[2-[Bis(4-fluorophenyl)-(4-methoxyphenyl)methoxy]ethyl]piperidine-3-carboxylic acid | IC50 | 151000.0 [1] |
| 1-{2-[Bis-(4-methoxy-phenyl)-phenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid | IC50 | 382000.0 [1] |
| 1-[2-(9-Phenyl-9H-xanthen-9-yloxy)-ethyl]-piperidine-3-carboxylic acid | IC50 | 920000.0 [1] |
| 1-{2-[(4-Methoxy-phenyl)-diphenyl-methoxy]-ethyl}-piperidine-3-carboxylic acid | IC50 | 655000.0 [1] |
| 1-[2-[(4-Methoxyphenyl)-bis(4-methylphenyl)methoxy]ethyl]piperidine-3-carboxylic acid | IC50 | 109000.0 [1] |
| 1-[2-[Bis(4-chlorophenyl)-(4-methoxyphenyl)methoxy]ethyl]piperidine-3-carboxylic acid | IC50 | 88000.0 [1] |
| 1-(2-Tritylsulfanyl-ethyl)-piperidine-3-carboxylic acid | IC50 | 435000.0 [1] |
| CID 118711599 | IC50 | 590.0 [1] |
| 2,4-Dichloro-N-[1-(pyridin-3-ylmethyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
| 2,4-Dichloro-N-[1-[(4-nitrophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 100000.0 [1] |
| 2,4-Dichloro-N-(1-phenacylpiperidin-4-yl)benzamide | IC50 | 100000.0 [1] |
| 2,4-Dichloro-N-[1-[(E)-3-phenylprop-2-enyl]piperidin-4-yl]benzamide | IC50 | 100000.0 [1] |
| 2,4-Dichloro-N-[1-(naphthalen-2-ylmethyl)piperidin-4-yl]benzamide | IC50 | 50000.0 [1] |
| 2,4-Dichloro-N-[1-[(4-iodophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 100000.0 [1] |
| 2,4-Dichloro-N-[1-(3-diethoxyphosphorylpropyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
| Methyl 4-[[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]methyl]benzoate | IC50 | 100000.0 [1] |
| 2,4-Dichloro-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
| 2,4-Dichloro-N-[1-(3-cyanopropyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
| Tert-butyl 2-[4-[(2,4-dichlorobenzoyl)amino]piperidin-1-yl]acetate | IC50 | 1000000.0 [1] |
| 2,4-Dichloro-N-(1-prop-2-ynylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
| 2-[4-[(2,4-Dichlorobenzoyl)amino]piperidin-1-yl]acetic acid | IC50 | 1000000.0 [1] |
| 2,4-Dichloro-N-[1-[(2-cyanophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 50000.0 [1] |
| 2,4-Dichloro-N-[1-[(2-nitrophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 100000.0 [1] |
| 2,4-Dichloro-N-[1-[(4-cyanophenyl)methyl]piperidin-4-yl]benzamide | IC50 | 50000.0 [1] |
| 2,4-Dichloro-N-[1-(quinolin-2-ylmethyl)piperidin-4-yl]benzamide | IC50 | 50000.0 [1] |
| N-(1-Benzylpiperidin-4-yl)-2-methylpropanamide | IC50 | 1000000.0 [1] |
| 2,4-Dichloro-N-(1-propylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
| 2,4-Dichloro-N-(1-ethylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
| N-(1-Benzylpiperidin-4-yl)-3-(trifluoromethyl)benzamide | IC50 | 170000.0 [1] |
| CID 43345728 | IC50 | 1000000.0 [1] |
| 2,4-Dichloro-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]benzamide | IC50 | 1000000.0 [1] |
| (3R)-1-[(E)-4-(2-Fluorophenyl)-4-(2-methylphenyl)but-3-enyl]piperidine-3-carboxylic acid | IC50 | 100000.0 [1] |
| 2-[(1S,2S)-2-Aminocyclopropyl]acetic acid | IC50 | 5480.0 [1] |
| 2,4-Dichloro-N-(1-methylpiperidin-4-yl)benzamide | IC50 | 1000000.0 [1] |
| (R)-1-{2-[Tris-(4-methoxy-phenyl)-methoxy]-ethyl}-piperidine-3-carboxylic acid | IC50 | 630000.0 [1] |
| 2-[(1S,2R)-2-Aminocyclopropyl]acetic acid;hydrochloride | IC50 | 5480.0 [1] |
| N-(1-Benzyl-4-piperidinyl)-1,3-benzodioxole-5-carboxamide | Ki | 42000.0 [1] |
| N,N-Dimethyl-2-[(1,7,7-trimethyl-2-phenyl-2-bicyclo[2.2.1]heptanyl)oxy]ethanamine | IC50 | 39000.0 [1] |
| 1-[2-[Tris(4-methoxyphenyl)methoxy]ethyl]-3,6-dihydro-2H-pyridine-5-carboxylic acid | IC50 | 2660000.0 [1] |
| (3S)-8-Benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid | IC50 | 335000.0 [1] |
| (3R,8R)-8-Benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid | IC50 | 2900000.0 [1] |
| (3S,8R)-8-Benzhydryl-2,3,4,6,7,8,9,9a-octahydro-1H-quinolizine-3-carboxylic acid | IC50 | 809000.0 [1] |
| (3R)-8-Benzhydrylidene-1,2,3,4,6,7,9,9a-octahydroquinolizine-3-carboxylic acid | IC50 | 436000.0 [1] |