Beta-adrenergic receptor kinase 2 Inhibitors (IC50, Ki)

Structure ▲ ▼	Compound Name ▲ ▼	Standard Type ▲ ▼	Standard Values (in nM) ▲ ▼
	Balanol	IC50	47.0 [1]
	CID 11677079	IC50	5.4 [1]
	6-(2,4-Difluorophenyl)sulfonyl-2-(1H-indol-5-ylamino)-8-methylpyrido[2,3-d]pyrimidin-7-one	IC50	10000.0 [1]
	N-Benzyl-3-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methylamino]benzamide	IC50	1.8 [1]
	N-Benzyl-3-[(4-methyl-3-pyridin-4-yl-1H-pyrazol-5-yl)methylamino]benzamide	IC50	4.3 [1]
	3-(9-Oxa-3,4,6,12-tetrazatricyclo[8.4.0.02,6]tetradeca-1(10),2,4,11,13-pentaen-5-ylmethylamino)-N-[[2-(trifluoromethyl)phenyl]methyl]benzamide	IC50	0.65 [1]
	N-Benzyl-3-[(4-ethyl-5-pyridin-4-yl-1,2,4-triazol-3-yl)methylamino]benzamide	IC50	3.3 [1]
	N-Methyl-3-[(3-pyridin-4-yl-1H-1,2,4-triazol-5-yl)methylamino]benzamide	IC50	21.0 [1]
	2-(3-Chloroanilino)-N-[(E)-pyridin-4-ylmethylideneamino]acetamide	Ki	1000.0 [1]
	2-(3-Methoxyanilino)-N-[(E)-pyridin-4-ylmethylideneamino]acetamide	Ki	10.0 [1]
	3-[[2-[(2E)-2-[(3,5-Dichloropyridin-4-yl)methylidene]hydrazinyl]-2-oxoethyl]amino]-N-phenylbenzamide	Ki	10.0 [1]
	2-(3-Chloroanilino)-N-[(E)-(3,5-dichloropyridin-4-yl)methylideneamino]acetamide	Ki	1000.0 [1]
	3-[[2-Oxo-2-[(2E)-2-(pyridin-4-ylmethylidene)hydrazinyl]ethyl]amino]-N-phenylbenzamide	Ki	10.0 [1]
	3-[[2-[(2E)-2-[(3,5-Dichloropyridin-4-yl)methylidene]hydrazinyl]-2-oxoethyl]amino]-N-methylbenzamide	Ki	100.0 [1]
	3-[[2-Oxo-2-[(2E)-2-(1-pyridin-4-ylethylidene)hydrazinyl]ethyl]amino]-N-phenylbenzamide	Ki	100.0 [1]
	N-Methyl-3-[[2-oxo-2-[(2E)-2-(pyridin-4-ylmethylidene)hydrazinyl]ethyl]amino]benzamide	Ki	100.0 [1]
	3-[[2-Oxo-2-[(2E)-2-(pyridin-4-ylmethylidene)hydrazinyl]ethyl]amino]benzamide	Ki	10.0 [1]
	N-[(E)-Pyridin-4-ylmethylideneamino]-2-(3-sulfamoylanilino)acetamide	Ki	1000.0 [1]
	N-[(E)-(3,5-Dichloropyridin-4-yl)methylideneamino]-2-(3-fluoroanilino)acetamide	Ki	1000.0 [1]
	N-[(E)-(3,5-Dichloropyridin-4-yl)methylideneamino]-2-(3-phenoxyanilino)acetamide	Ki	100.0 [1]
	2-(3-Methylsulfanylanilino)-N-[(E)-pyridin-4-ylmethylideneamino]acetamide	Ki	100.0 [1]
	N-[(E)-(3,5-Dichloropyridin-4-yl)methylideneamino]-2-(3-sulfamoylanilino)acetamide	Ki	1000.0 [1]
	2-(3-Fluoroanilino)-N-[(E)-pyridin-4-ylmethylideneamino]acetamide	Ki	1000.0 [1]
	2-(3-Phenoxyanilino)-N-[(E)-pyridin-4-ylmethylideneamino]acetamide	Ki	100.0 [1]
	N-[(E)-(3,5-Dichloropyridin-4-yl)methylideneamino]-2-(3-phenylmethoxyanilino)acetamide	Ki	100.0 [1]
	2-(3-Phenoxyanilino)-N-[(E)-1-pyridin-4-ylethylideneamino]acetamide	Ki	100.0 [1]
	2-(3-Methoxyanilino)-N-[(E)-1-pyridin-4-ylethylideneamino]acetamide	Ki	100.0 [1]
	2-(3-Phenylmethoxyanilino)-N-[(E)-1-pyridin-4-ylethylideneamino]acetamide	Ki	100.0 [1]
	N-[(E)-(3,5-Dichloropyridin-4-yl)methylideneamino]-2-(3-methylsulfanylanilino)acetamide	Ki	100.0 [1]
	N-[(E)-(3,5-Dichloropyridin-4-yl)methylideneamino]-2-(3-ethoxyanilino)acetamide	Ki	10000.0 [1]
	N-[(E)-(3,5-Dichloropyridin-4-yl)methylideneamino]-2-(3-methoxyanilino)acetamide	Ki	10.0 [1]
	2-(3-Phenylmethoxyanilino)-N-[(E)-pyridin-4-ylmethylideneamino]acetamide	Ki	100.0 [1]

Entire TableStructureCompound NameStandard TypeStandard Values (in nM)

Items per page: 510All1 - 10 of 32 ⟨⟩

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References

This online tool may be cited as follows

MLA	"Quest Database™ Beta-adrenergic receptor kinase 2 Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Nov. 2024, https://www.aatbio.com/data-sets/beta-adrenergic-receptor-kinase-2-inhibitors-ic50-ki.
APA	AAT Bioquest, Inc. (2024, November 21). Quest Database™ Beta-adrenergic receptor kinase 2 Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/beta-adrenergic-receptor-kinase-2-inhibitors-ic50-ki.
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