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Beta-3 adrenergic receptor Inhibitors (IC50, Ki)

Structure
▲
▼
Compound Name
▲
▼
Standard Type
▲
▼
Standard Values (in nM)
▲
▼
2-(4-((2R)-2-(((2R)-2-(3-Chlorophenyl)-2-hydroxyethyl)amino)propyl)phenoxy)acetic acidKi660.0 [1], 960.0 [2]
2-(Methylsulfonylamino)-4-[(R)-1-hydroxy-2-[bis(4-methoxyphenyl)methylamino]ethyl]phenolKi81.0 [1]
[3-[(2R)-2-[[(2R)-2-Hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl] methanesulfonateKi4.0 [1]
1-(4-Methoxyphenoxy)-3-(1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-ylamino)propan-2-olKi378.0 [1], 460.0 [2]
N-[5-[(1R)-2-[[(1R)-1-[4-(Difluoromethoxy)phenyl]-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamideKi21.0 [1]
(2S)-2-[[(2R)-2-Hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-(4-methoxyphenyl)-N-phenylacetamideKi77.0 [1], 370.0 [2]
2-(Methylsulfonylamino)-4-[1-hydroxy-2-[1-(4-methoxyphenyl)-2-phenylethylamino]ethyl]phenolKi44.0 [1]
2-(Methylsulfonylamino)-4-[1-hydroxy-2-(alpha-phenylphenethylamino)ethyl]phenolKi360.0 [1]
N-[5-[(1R)-2-[[(1R)-1-(3,4-Dimethoxyphenyl)-2-phenylethyl]amino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamideKi11.0 [1]
1-[4-(Hydroxymethyl)phenoxy]-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propan-2-olIC50162.0 [1]
1-[4-(Hydroxymethyl)phenoxy]-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propan-2-olKi290.0 [1]
2-[[1-[2-Hydroxy-3-(5-methyl-2-propan-2-ylphenoxy)propyl]piperidin-4-yl]methyl]benzo[de]isoquinoline-1,3-dioneIC501474.0 [1]
2-[[1-[2-Hydroxy-3-(5-methyl-2-propan-2-ylphenoxy)propyl]piperidin-4-yl]methyl]benzo[de]isoquinoline-1,3-dioneKi411.0 [1]
N-[3-[2-Hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]phenyl]acetamideIC50107.0 [1]
N-[3-[2-Hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]phenyl]acetamideKi85.0 [1]
3-[2-Hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]-N-methylbenzamideIC50402.0 [1]
3-[2-Hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]-N-methylbenzamideKi331.0 [1]
1-(4-Ethylphenoxy)-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propan-2-olIC508064.0 [1]
1-(4-Ethylphenoxy)-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propan-2-olKi107.0 [1]
(6Ar,7R)-1,2-dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-7-olIC50240.0 [1]
(6Ar,7R)-1,2-dimethoxy-5,6,6a,7-tetrahydro-4H-dibenzo[de,g]quinolin-7-olKi308.0 [1]
PropranololKi99.0 [1]
IsoprenalineKi18620.87 [1]
TamoxifenKi5778.0 [1]
AmiodaroneKi31761.0 [1]
CelecoxibKi12093.0 [1]
ClomipheneKi4254.0 [1]
FenofibrateKi92959.0 [1]
CarvedilolKi3.12 [1]
PindololKi66.0 [1]
CandesartanKi3200.0 [1]
TimololKi339.0 [1]
DanazolKi12765.0 [1]
MiconazoleKi4111.0 [1]
ClotrimazoleKi5406.0 [1]
NelfinavirKi25566.0 [1]
FluphenazineKi22116.0 [1]
PropafenoneKi318.0 [1]
MontelukastKi3200.0 [1]
4-NonylphenolKi3142.0 [1]
AstemizoleKi6045.0 [1]
EconazoleKi4612.0 [1]
CiglitazoneKi13403.0 [1]
EbastineKi1909.1 [1]
LevobunololKi255.0 [1]
1-(Isopropylamino)-3-(1-naphthyloxy)-2-propanolKi124.0 [1]
Cl-316243 Free diacidKi20000.0 [1]
PenfluridolKi515.0 [1]
1-[(3,4,5-Trimethoxyphenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-6,7-diolKi3715.35 [1]
BopindololKi344.0 [1]
(1S,2R)-2-(Octylamino)-1-[4-(propan-2-ylthio)phenyl]-1-propanolKi3747.2 [1]
alpha-ErgocryptineKi1872.0 [1]
(S)-2-(2-Benzoylphenylamino)-3-(4-(2-(methyl(pyridin-2-yl)amino)ethoxy)phenyl)propanoic acidKi16564.0 [1]
alpha-MethyltryptamineKi10000.0 [1]
OxiconazoleKi3558.7 [1]
CipargaminIC5030000.0 [1]
(4-{(R)-2-[(R)-2-(3-Chloro-phenyl)-2-hydroxy-ethylamino]-propyl}-phenoxy)-acetic acid methyl esterKi1150.0 [1]
(S)-(-)-PindololKi36.0 [1]
Dihydroergocristine mesylateKi2481.0 [1]
SoterenolKi4100.0 [1]
N,N-Diallyl-5-methoxytryptamineKi10000.0 [1]
L-796568 Free baseIC5046.0 [1]
ThalictruberineKi10000.0 [1]
2-[4-[2-[[(2S)-2-Hydroxy-3-phenoxypropyl]amino]ethoxy]phenoxy]acetic acidKi520.0 [1]
1-(2-Allylphenoxy)-3-morpholinopropan-2-olKi4960.0 [1]
1-(3,5-Diiodo-4-methoxybenzyl)-1,2,3,4-tetrahydroisoquinoline-6,7-diolKi21.38 [1]
4-[4-(3-Cyclopentylpropyl)-5-oxotetrazol-1-yl]-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamideIC5092.0 [1]
N,N-Dimethyl-1-(3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(18),7,9,11,14,16-hexaen-4-yl)methanamineIC501862.09 [1]
(2R)-2-[3-[[3-(4-Chlorobenzoyl)-2-methyl-6-(trifluoromethoxy)indol-1-yl]methyl]phenoxy]propanoic acidIC504860.0 [1]
3-((2-Fluorothiazol-4-yl)ethynyl)-5-fluorobenzonitrileKi10000.0 [1]
Unii-93zdv2P17IKi160.0 [1]
N,N-Dimethyl-1-(3-oxa-2,17-diazatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)methanamineIC501000.0 [1]
1-(17-Chloro-3-oxa-2-azatetracyclo[12.4.0.02,6.07,12]octadeca-1(14),7,9,11,15,17-hexaen-4-yl)-N,N-dimethylmethanamineIC50870.96 [1]
2-[4-[4-(7-(111C)Methoxynaphthalen-1-yl)piperazin-1-yl]butyl]-4-methyl-1,2,4-triazine-3,5-dioneKi10000.0 [1]
4-[4-(3,4-Difluorophenyl)-1,3-thiazol-2-yl]-N-[4-[2-[[(2R)-2-hydroxy-2-pyridin-3-ylethyl]amino]ethyl]phenyl]benzenesulfonamideIC5020.0 [1]
(1S,2R,3S,4R,5S)-4-[2-[2-(5-Chlorothiophen-2-yl)ethynyl]-6-(propylamino)purin-9-yl]-2,3-dihydroxy-N-methylbicyclo[3.1.0]hexane-1-carboxamideKi1440.0 [1]
4-Fluoro-N-methyl-N-(4-(6-(methylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl)benzamideKi10000.0 [1]
2-(Hydroxymethyl)-4-[2-hydroxy-3-[[1-(5-phenylthieno[2,3-d]pyrimidin-4-yl)piperidin-4-yl]amino]propoxy]phenolKi7.3 [1]
N-[5-[(1R)-2-[1,1-Bis[4-(difluoromethoxy)phenyl]ethylamino]-1-hydroxyethyl]-2-hydroxyphenyl]methanesulfonamideKi81.0 [1]
N-[3-[(1R)-1-Hydroxy-2-[[(2R)-1-(1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamideKi30.0 [1]
2-[[3-[(2R)-2-[[(2R)-2-Hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]propyl]-1H-indol-7-yl]oxy]acetic acidKi17.0 [1]
N-[3-[(1R)-1-Hydroxy-2-[[(2R)-1-(7-methoxy-1H-indol-3-yl)propan-2-yl]amino]ethyl]phenyl]thiophene-2-sulfonamideKi14.0 [1]
[3-[2-[[(2R)-2-Hydroxy-2-[3-(thiophen-2-ylsulfonylamino)phenyl]ethyl]amino]ethyl]-1H-indol-7-yl] methanesulfonateKi33.0 [1]
1-(10H-Phenothiazin-10-yl)-2-phenylpropan-1-oneKi2500.0 [1]
1-(10H-Phenothiazin-10-yl)-4-phenylbutan-1-oneKi1700.0 [1]
(2S)-N-(4-Diethoxyphosphorylphenyl)-2-[[(2R)-2-hydroxy-2-[4-hydroxy-3-(methanesulfonamido)phenyl]ethyl]amino]-2-(4-methoxyphenyl)propanamideKi93.0 [1]
(1-(4-Fluorophenethyl)piperidin-4-yl)(3-(2-fluoroethoxy)-2-methoxyphenyl)methanolKi10000.0 [1]
5-Methyl-1,5-diazapentacyclo[10.8.1.02,7.08,21.013,18]henicosa-2(7),8(21),9,11,13,15,17-heptaeneKi10000.0 [1]
(4-Fluorophenyl)(2-(2-((2R)-2-methyl-1-pyrrolidinyl)ethyl)-1-benzofuran-5-yl)methanoneKi10000.0 [1]
4-(3,5-Diiodo-4-methoxybenzyl)-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridine-2-amineKi1479.11 [1]
N-[5-[(2R)-3-[[(1R)-1-(3,4-Dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamideKi25.0 [1]
N-[5-[(2S)-3-[[(1R)-2-(4-Chlorophenyl)-1-(3,4-dimethoxyphenyl)ethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamideKi24.0 [1]
N-[2-Hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamideKi53.0 [1]
N-[2-Hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(3-hydroxy-4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamideKi8.0 [1]
N-[2-Hydroxy-5-[(2S)-2-hydroxy-3-[[(1R)-1-(3-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamideKi110.0 [1]
N-[5-[(2S)-3-[[(1R)-2-(2-Chlorophenyl)-1-(3,4-dimethoxyphenyl)ethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamideKi7.0 [1]
N-[5-[(2S)-3-[[(1S)-1-(3,4-Dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamideKi9.0 [1]
N-[5-[(2R)-3-[[(1S)-1-(3,4-Dimethoxyphenyl)-2-phenylethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamideKi150.0 [1]
N-[2-Hydroxy-5-[(2R)-2-hydroxy-3-[[(1R)-1-(4-methoxyphenyl)-2-phenylethyl]amino]propyl]phenyl]methanesulfonamideKi460.0 [1]
N-[5-[(2S)-3-[[(1R)-2-(3-Chlorophenyl)-1-(3,4-dimethoxyphenyl)ethyl]amino]-2-hydroxypropyl]-2-hydroxyphenyl]methanesulfonamideKi6.0 [1]
Items per page: 1 - 10 of 100
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References

This online tool may be cited as follows

MLA

"Quest Database™ Beta-3 adrenergic receptor Inhibitors (IC50, Ki)." AAT Bioquest, Inc., 21 Feb. 2025, https://www.aatbio.com/data-sets/beta-3-adrenergic-receptor-inhibitors-ic50-ki.

APA

AAT Bioquest, Inc. (2025, February 21). Quest Database™ Beta-3 adrenergic receptor Inhibitors (IC50, Ki). AAT Bioquest. https://www.aatbio.com/data-sets/beta-3-adrenergic-receptor-inhibitors-ic50-ki.
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